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Research Article

Development of a new nanovesicle formulation as transdermal carrier: Formulation, physicochemical characterization, permeation studies and anti-inflammatory activity

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Pages 323-330 | Received 26 Jun 2013, Accepted 17 Jul 2013, Published online: 15 Aug 2013

References

  • Aguiar AJ, Weiner MA. 1969. Percutaneous absorption studies of chloramphenicol solutions. J Pharm Sci 58:210–215.
  • Akhter S, Jain GK, Ahmad FJ, Khar RK, Khan ZI, Talegaonkar S. 2008. Investigation of nanoemulsion system for transdermal delivery of domperidone: Ex-vivo and in vivo studies. Curr Nanosci 4: 381–390.
  • An K, Sun Y, Xu L, Cui X. 2011. Preparation and in vitro evaluation of simvastatin ethosome. Artif Cells Blood Substit Immobil Biotechnol 39:347–350.
  • Anne P, Ilkka K, Jouko Y, Per R. 2000. Controlled release injectable liposomal gel of ibuprofen for epidural analgesia. Int J Pharm 199:85–93.
  • Antal E, Wright C, Brown B, Albert K, Aman L, Levin N. 1986. The influence of hemodialysis on the pharmacokinetics of ibuprofen and its major metabolites. J Clin Pharmacol 26:184.
  • Arifin DR, Palmer AF. 2005. Stability of liposome encapsulated hemoglobin dispersions. Artif Cells Blood Substit Immobil Biotechnol 33:113–136.
  • Dragicevic-Curic N, Scheglmann D, Albrecht V, Fahr A. 2008. Temoporfin-loaded invasomes: Development, characterization and in vitro skin permeation studies. J Control Release 127:59–69.
  • Dugard PH (Ed). 1976. Advanccs in Modern Toxicology, vol. 4. New York: Wiley.
  • Durrheim H, Flynn GL, Higuchi WI, Behl CR. 1980. Permeation of hairless mouse skin I: Experimental methods and comparison with human epidermal permeation by alkanols. J Pharm Sci 69:781–786.
  • El-Leithy ES, Shaker DS, Ghorab MK, Abdel-Rashid RS. 2010. Evaluation of mucoadhesive hydrogels loaded with diclofenac sodium-chitosan microspheres for rectal administration. AAPS PharmSciTech 11:1695–1702.
  • Evans AM, Nation RL, Sansom LN, Bochner F, Somogyi AA. 1989. Stereoselective plasma protein binding of ibuprofen enantiomers. Eur J Clin Pharmacol 36:283–290.
  • Fresta M, Puglisi G. 1996. Application of liposomes as potential cutaneous drug delivery systems. In vitro and in vivo investigation with radioactively labelled vesicles. J Drug Target 4:95–101.
  • Furuishi T, Io T, Fukami T, Suzuki T and Tomono K. 2008. Formulation and in vitro evaluation of pentazocine transdermal delivery system. Biol Pharm Bull 31:1439–1443.
  • Gallo J, Gall E, Gillespie W, Albert K, Perrier D. 1986. Ibuprofen kinetics in plasma and synovial fluid of arthritic patients. J Clin Pharmacol 26:65.
  • Gaur PK, Mishra S, Kumar A, Panda BP. 2014a. Development and optimization of gastroretentive mucoadhesive microspheres of gabapentin by Box-Behnken design. Artif Cells Nanomed Biotechnol 42:167–177.
  • Gaur PK, Purohit S, Kumar Y, Mishra S, Bhandari A. 2014b. Development and characterization of stable nanovesicular carrier for drug delivery. Artif Cells Nanomed Biotechnol 42:296–301.
  • Gaur PK, Purohit S, Kumar Y, Mishra S, Bhandari A. 2014c. Preparation, characterization and permeation studies of a nanovesicular system containing diclofenac for transdermal delivery. Pharm Dev Technol 19:48–54.
  • Goñi FM, Alonso A. 2006. Biophysics of sphingolipids I. Membrane properties of sphingosine, ceramides and other simple sphingolipids. Biochimica Biophysica Acta. 1758:1902–1921.
  • Haigh JM, Beyssac E, Chanet L, Aiache JM. 1998. In vitro permeation of progesterone from a gel through the shed skin of three different snake species. Int J Pharm 170:151–156.
  • Higuchi T. 1960. Physical chemical analysis of percutaneous absorption process from creams and ointments. J Soc Cosmet Chem 11:85–97.
  • Ishida T, Takanashi Y, Doi H, Yamamoto I, Kiwada H. 2002. Encapsulation of an antivasospastic drug, fasudil, into liposomes, and in vitro stability of the fasudil-loaded liposomes. Int J Pharm 232:59–67.
  • Jukanti R, Sheela S, Bandari S, Veerareddy PR. 2011. Enhanced bioavailability of exemestane via proliposomes based transdermal delivery. J Pharm Sci 100:3208–3222.
  • Kitagawa S, Yokochi N, Murooka N. 1995. pH-Dependence of phase transition of the lipid bilayer of liposomes of stratum corneum lipids. Int J Pharm 126:49–56.
  • Kobayashi N, Saitoh I. 1999. Development of a test method for in vitro drug release from soluble and crystal dispersion type ointments. Chem Pharm Bull 47:199–202.
  • Lee E, Williams K, Day R, Graham G, Champion D. 2004. Stereoselective disposition of ibuprofen enantiomers in man. Br J Clin Pharmacol 58:S759–S764.
  • Manconi M, Caddeo C, Sinico C, Valenti D, Mostallino MC, Biggio G, Fadda AM. 2011. Ex vivo skin delivery of diclofenac by transcutol containing liposomes and suggested mechanism of vesicle-skin interaction. Eur J Pharm Biopharm 78:27–35.
  • Manosroi A, Jantrawut P, Manosroi J. 2008. Anti-inflammatory activity of gel containing novel elastic niosomes entrapped with diclofenac diethylammonium. Int J Pharm 360:156–163.
  • Mishra D, Garg M, Dubey V, Jain S, Jain NK. 2007. Elastic liposomes mediated transdermal delivery of an anti-hypertensive agent: propranolol hydrochloride. J Pharm Sci 96:147–155.
  • Patel NA, Patel NJ, Patel RP. 2009. Formulation and evaluation of curcumin gel for topical application. Pharm Dev Technol 14:80–89.
  • Paudel KS, Milewski M, Swadley CL, Brogden NK, Ghosh P, Stinchcomb AL. 2010. Challenges and opportunities in dermal/transdermal delivery. Ther Deliv 1:109–131.
  • Sinico C, Manconi M, Valenti M, Fadda AM. 2005. Liposomes as carriers for dermal delivery of tretinoin: in vitro evaluation of drug permeation and vesicle-skin interaction. J Control Release 103:123–136.
  • Touitou E, Dayan N, Bergelson L, Godin B, Eliaz M. 2000. Ethosomes – novel vesicular carriers for enhanced delivery: characterization and skin permeation properties. J Control Release 65:403–418.
  • Vasiljevic D, Parojcic J, Primorac M, Vuleta G. 2006. An investigation into the characteristics and drug release properties ofmultiple W/O/W emulsion systems containing low concentration of lipophilic polymeric emulsifier. Int J Pharm 309:171–177.
  • Walters KA, Roberts MS (Eds). 2002. The Structure and Function of Skin. New York: Marcel Dekker INC.
  • Wartewig S, Neubert RH. 2007. Properties of ceramides and their impact on the stratum corneum structure: a review. Skin Pharmacol Physiol 20:220–229.
  • Yardley HL, Summerly R. 1981. Lipid composition and metabolism in normal and diseased epidermis. Pharmacol Ther 13:357–383.
  • Zellmer S, Zimmermann I, Selle C, Sternberg B, Pohle W, Lasch J. 1998. Physicochemical characterisation of human stratum corneum lipid liposomes. Chem Phys Lipids 94:97–108.

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