Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 25, Issue 4 (2010)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 25, Issue 4 (2010)

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Research Article

Article
Synthesis and antileishmanial and antimicrobial activities of some 2,3-disubstituted 3H-quinazolin-4-ones
Muhammad Arfan, Rasool Khan, Murad Ali Khan, Shazia Anjum, Muhammad Iqbal Choudhary & Manzoor Ahmad
Pages: 451-458
Published online: 17 Mar 2010
AbstractforSynthesis and antileishmanial and antimicrobial activities of some 2,3-disubstituted 3H-quinazolin-4-ones | Full Text | References | PDF (748.2 KB)
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Article
Molecular modeling and biological effects of peptidomimetic inhibitors of TACE activity
Wen-fang Feng, Yun-bin Zhao, Wei Huang & Yu-zhen Yang
Pages: 459-466
Published online: 01 Dec 2009
AbstractforMolecular modeling and biological effects of peptidomimetic inhibitors of TACE activity | Full Text | References | PDF (1.1 MB)
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Original Article

Article
Antioxidant effect of functionalized alkyl-organotellurides: a study in vitro
Bibiana M. Gay, Cristiane Luchese, Cristina W. Nogueira, P. Wendler, Alexandra Macedo & Alcindo A. Dos Santos
Pages: 467-475
Published online: 17 Mar 2010
AbstractforAntioxidant effect of functionalized alkyl-organotellurides: a study in vitro | Full Text | References | PDF (766.7 KB)
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Article
Effects of some drugs on human erythrocyte 6-phosphogluconate dehydrogenase: an in vitro study
Ebru Akkemik, Harun Budak & Mehmet Ciftci
Pages: 476-479
Published online: 17 Mar 2010
AbstractforEffects of some drugs on human erythrocyte 6-phosphogluconate dehydrogenase: an in vitro study | Full Text | References | PDF (633.4 KB)
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Article
A comparison of reactivating and therapeutic efficacy of the oxime K203 and its fluorinated analog (KR-22836) with currently available oximes (obidoxime, trimedoxime, HI-6) against tabun in rats and mice
Jiri Kassa, Jana Zdarova Karasova, Filip Caisberger, Kamil Musilek, Kamil Kuca & Young-Sik Jung
Pages: 480-484
Published online: 16 Mar 2010
AbstractforA comparison of reactivating and therapeutic efficacy of the oxime K203 and its fluorinated analog (KR-22836) with currently available oximes (obidoxime, trimedoxime, HI-6) against tabun in rats and mice | Full Text | References | PDF (598.7 KB)
  • 618 Views
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Article
Sulfonamide derivatives of thiazolidin-4-ones with anticonvulsant activity against two seizure models: synthesis and pharmacological evaluation
Nadeem Siddiqui, M. Faiz Arshad, Suroor A. Khan & Waquar Ahsan
Pages: 485-491
Published online: 16 Mar 2010
AbstractforSulfonamide derivatives of thiazolidin-4-ones with anticonvulsant activity against two seizure models: synthesis and pharmacological evaluation | Full Text | References | PDF (658.3 KB)
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Article
Design, synthesis, and pharmacological evaluation of novel oxadiazole and oxadiazoline analogs as anti-inflammatory agents
Harish Rajak, Ravichandran Veerasamy, Murlidhar Kharya & Pradeep Mishra
Pages: 492-501
Published online: 26 Oct 2009
AbstractforDesign, synthesis, and pharmacological evaluation of novel oxadiazole and oxadiazoline analogs as anti-inflammatory agents | Full Text | References | PDF (703.4 KB)
  • 618 Views
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Article
Synthesis, characterization, cytotoxicity, and DNA binding of some new platinum(II) and platinum(IV) complexes with benzimidazole ligands
Semra Utku, Fatma Gumus, Seda Tezcan, Mehmet Sami Serin & Aykut Ozkul
Pages: 502-508
Published online: 16 Mar 2010
AbstractforSynthesis, characterization, cytotoxicity, and DNA binding of some new platinum(II) and platinum(IV) complexes with benzimidazole ligands | Full Text | References | PDF (726.4 KB)
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Article
Oxime K027: novel low-toxic candidate for the universal reactivator of nerve agent- and pesticide-inhibited acetylcholinesterase
Kamil Kuca, Kamil Musilek, Daniel Jun, Miroslav Pohanka, Kallol Kumar Ghosh & Martina Hrabinova
Pages: 509-512
Published online: 23 Feb 2010
AbstractforOxime K027: novel low-toxic candidate for the universal reactivator of nerve agent- and pesticide-inhibited acetylcholinesterase | Full Text | References | PDF (574.1 KB)
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Article
Synthesis, antineoplastic and cytotoxic activities of some mononuclear Ru(II) complexes
Sreekanth Thota, Subhas S. Karki, K. N. Jayaveera, Jan Balzarini & Erik De Clercq
Pages: 513-519
Published online: 03 Feb 2010
AbstractforSynthesis, antineoplastic and cytotoxic activities of some mononuclear Ru(II) complexes | Full Text | References | PDF (721.8 KB)
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Article
Design, synthesis, and evaluation of anti-inflammatory, analgesic, ulcerogenicity, and nitric oxide releasing studies of novel indomethacin analogs as non-ulcerogenic derivatives
Shashikant V. Bhandari, Jignesh K. Parikh, Kailash G. Bothara, Trupti S. Chitre, Deepak K. Lokwani, Titiksh L. Devale, Nileema S. Modhave, Vidya S. Pawar & Santosh Panda
Pages: 520-530
Published online: 28 Jan 2010
AbstractforDesign, synthesis, and evaluation of anti-inflammatory, analgesic, ulcerogenicity, and nitric oxide releasing studies of novel indomethacin analogs as non-ulcerogenic derivatives | Full Text | References | PDF (874.4 KB)
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Article
In vivo experimental approach to treatment against tabun poisoning
Suzana Berend, Maja Katalinić, Ana Lucić Vrdoljak, Zrinka Kovarik, Kamil Kuča & Božica Radić
Pages: 531-536
Published online: 17 Mar 2010
AbstractforIn vivo experimental approach to treatment against tabun poisoning | Full Text | References | PDF (600.8 KB)
  • 629 Views
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Article
Synthesis of 1-(4-methoxybenzyl)-3-cyclopropyl-1H-pyrazol-5-amine derivatives as antimicrobial agents
H. Raju, T.S. Nagamani, S. Chandrappa, H. Ananda, K. Vinaya, N.R. Thimmegowda, S. M. Byregowda & K. S. Rangappa
Pages: 537-543
Published online: 17 Mar 2010
AbstractforSynthesis of 1-(4-methoxybenzyl)-3-cyclopropyl-1H-pyrazol-5-amine derivatives as antimicrobial agents | Full Text | References | PDF (899 KB)
  • 748 Views
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Article
Template synthesis, spectroscopic, antibacterial, and antifungal studies of trivalent transition metal ion macrocyclic complexes
D. P. Singh, Krishan Kumar, Chetan Sharma & K. R. Aneja
Pages: 544-550
Published online: 17 Mar 2010
AbstractforTemplate synthesis, spectroscopic, antibacterial, and antifungal studies of trivalent transition metal ion macrocyclic complexes | Full Text | References | PDF (868.6 KB)
  • 533 Views
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Article
Effect of lithium salts on lactate dehydrogenase, adenylate kinase, and 1-phosphofructokinase activities
Percy Russell, Anita Williams, Ami Abbott, Jessica Chadwick, Farnaz Ehya, Roxana Flores & Chanae Hardamon
Pages: 551-556
Published online: 02 Jul 2010
AbstractforEffect of lithium salts on lactate dehydrogenase, adenylate kinase, and 1-phosphofructokinase activities | Full Text | References | PDF (830.2 KB)
  • 770 Views
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Article
Synthesis, characterization, DNA interaction, and cytotoxicity of novel Pd(II) and Pt(II) complexes
Enjun Gao, Fuchun Liu, Mingchang Zhu, Lei Wang, Yun Huang, Hongyan Liu, Shuang Ma, Qunzhi Shi & Ni Wang
Pages: 557-564
Published online: 29 Dec 2009
AbstractforSynthesis, characterization, DNA interaction, and cytotoxicity of novel Pd(II) and Pt(II) complexes | Full Text | References | PDF (1 MB)
  • 557 Views
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Article
Preparation of some pyrazoline derivatives and evaluation of their antifungal activities
Ahmet Özdemir, Gülhan Turan-Zitouni, Zafer Asım Kaplancıklı, Gilbert Revial, Fatih Demirci & Gökalp İşcan
Pages: 565-571
Published online: 08 Mar 2010
AbstractforPreparation of some pyrazoline derivatives and evaluation of their antifungal activities | Full Text | References | PDF (641.9 KB)
  • 1218 Views
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Article
Design, synthesis, and urease inhibition studies of some 1,3,4-oxadiazoles and 1,2,4-triazoles derived from mandelic acid
Tashfeen Akhtar, Shahid Hameed, Khalid M. Khan, Ajmal Khan & Muhammad Iqbal Choudhary
Pages: 572-576
Published online: 17 Mar 2010
AbstractforDesign, synthesis, and urease inhibition studies of some 1,3,4-oxadiazoles and 1,2,4-triazoles derived from mandelic acid | Full Text | References | PDF (598.2 KB)
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Review Article

Review Article
Ciprofloxacin: review on developments in synthetic, analytical, and medicinal aspects
Prabodh Chander Sharma, Ankit Jain, Sandeep Jain, Rakesh Pahwa & Mohammad Shahar Yar
Pages: 577-589
Published online: 17 Mar 2010
AbstractforCiprofloxacin: review on developments in synthetic, analytical, and medicinal aspects | Full Text | References | PDF (1.3 MB)
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Short Communication

Article
Novel depsides as potential anti-inflammatory agents with potent inhibitory activity against Escherichia coli-induced interleukin-8 production
Peng-Cheng Lv, Jing Xiong, Jin Chen, Kai-Rui Wang, Wen-Jun Mao & Hai-Liang Zhu
Pages: 590-595
Published online: 17 Mar 2010
AbstractforNovel depsides as potential anti-inflammatory agents with potent inhibitory activity against Escherichia coli-induced interleukin-8 production | Full Text | References | PDF (713.1 KB)
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Errata

Correction
Erratum
Pages: 596-598
Published online: 02 Jul 2010
First Page PreviewforErratum | Full Text | PDF (614.2 KB)
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