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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 23, 2008 - Issue 1
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Research Article

Carbonic anhydrase inhibitors. Inhibition of the cytosolic and tumor-associated carbonic anhydrase isozymes I, II and IX with some 1,3,4-oxadiazole- and 1,2,4-triazole-thiols

Gabriela Laura Almajan Organic Chemistry Departament, Faculty of Pharmacy, Traian Vuia Street 6, 020956, Bucharest, Romania
,
Stefania-Felicia Barbuceanu Organic Chemistry Departament, Faculty of Pharmacy, Traian Vuia Street 6, 020956, Bucharest, Romania
,
Alessio innocenti Polo Scientifico, Laboratorio di Chimica Bioinorganica, Università degli Studi di Firenze, Rm. 188, Via della Lastruccia 3, 50019, Sesto Fiorentino (Florence, Italy
,
Andrea Scozzafava Polo Scientifico, Laboratorio di Chimica Bioinorganica, Università degli Studi di Firenze, Rm. 188, Via della Lastruccia 3, 50019, Sesto Fiorentino (Florence, Italy
&
Claudiu T. Supuran Polo Scientifico, Laboratorio di Chimica Bioinorganica, Università degli Studi di Firenze, Rm. 188, Via della Lastruccia 3, 50019, Sesto Fiorentino (Florence, Italy
Pages 101-107 | Received 09 Nov 2006, Accepted 13 Feb 2007, Published online: 04 Oct 2008

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Bhavesh N. Socha, Sachin B. Pandya, Bhavin R. Chavda, Kaushik P. Chaudhary, Taruna J. Padariya, Mohammed Dawood Alalawy, Rahul P. Dubey, Urmila H. Patel & R. H. Patel. (2021) Gas-phase DFT studies, quantum chemical calculation and 3D energy framework analysis of novel copper complex of sulfadimethoxine in the presence of secondary ligand 3-methyl pyridine. Inorganic and Nano-Metal Chemistry 51:12, pages 1822-1830.
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Claudiu T. Supuran. (2017) Advances in structure-based drug discovery of carbonic anhydrase inhibitors. Expert Opinion on Drug Discovery 12:1, pages 61-88.
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Emir Alper Türkoğlu, Murat Şentürk, Claudiu T. Supuran & Deniz Ekinci. (2017) Carbonic anhydrase inhibitory properties of some uracil derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 74-77.
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Asif Husain & Diwakar Madhesia. (2012) Heterocyclic compounds as carbonic anhydrase inhibitor. Journal of Enzyme Inhibition and Medicinal Chemistry 27:6, pages 773-783.
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Articles from other publishers (17)

Jaya RautelaAjay Singh BishtVikash JakhmolaA. N. M. AnsoriDivya Negi. (2023) Microwave-Assisted Synthesis of New 4-Amino Acid Substituted 1,2,4-Triazole Derivative Derived from 1,2,3-Oxadiazole Nucleus and Their Anti-Bacterial and Anti-Oxidant Potential. Research Journal of Pharmacy and Technology, pages 2322-2326.
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Soumya Ranjan Kar, Priyaranjan Mohapatra & Debasis Mohanty. (2022) Green synthesis, characterisation and antibacterial activity studies of new multifunctional nano polymeric material, which may have multidimensional application in water purification. Polymer Bulletin 80:1, pages 703-723.
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Fatma AYDIN, Zeynep Aleyna KAHRAMAN, Emir Alper TÜRKOĞLU, Müslüm KUZU & Zeki SEVEROĞLU. (2021) In vitro antioxidant activity and carbonic anhydrase inhibitory features of Ferula communis extracts. International Journal of Agriculture Environment and Food Sciences 5:4, pages 592-598.
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Fatma Gülruy AYDIN, Emir Alper TÜRKOĞLU, Müslüm KUZU & Turgut TAŞKIN. (2021) In vitro Carbonic Anhydrase Inhibitory Effects of The Extracts of Satureja cuneifoliaSatureja cuneifolia Ekstraktlarının in vitro Karbonik Anhidraz İnhibitör Etkileri. Türk Tarım ve Doğa Bilimleri Dergisi 8:4, pages 1146-1150.
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Farhan M. Khan, Muhammad A. Abbasi, Aziz‐ur‐Rehman, Sabahat Z. Siddiqui, Abdul R. Sadiq Butt, Hussain Raza, Ayesha Zafar, Syed A. Ali Shah, Muhammad Shahid & Sung‐Yum Seo. (2021) Convergent synthesis of carbonic anhydrase inhibiting bi‐heterocyclic benzamides: Structure–activity relationship and mechanistic explorations through enzyme inhibition, kinetics, and computational studies. Journal of Heterocyclic Chemistry 58:5, pages 1089-1103.
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Safak Akin, Hasan Ayaloglu, Ergun Gultekin, Ahmet Colak, Olcay Bekircan & Melike Yildirim Akatin. (2019) Synthesis of 1,2,4-triazole-5-on derivatives and determination of carbonic anhydrase II isoenzyme inhibition effects. Bioorganic Chemistry 83, pages 170-179.
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Muhammad Taha, Mohd Syukri Baharudin, Nor Hadiani Ismail, Manikandan Selvaraj, Uzma Salar, Khaled A.A. Alkadi & Khalid Mohammed Khan. (2017) Synthesis and in silico studies of novel sulfonamides having oxadiazole ring: As β -glucuronidase inhibitors. Bioorganic Chemistry 71, pages 86-96.
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Ameen Shahid, Nesreen Ahmed, Tamer Saleh, Shaeel Al-Thabaiti, Sulaiman Basahel, Wilhelm Schwieger & Mohamed Mokhtar. (2017) Solvent-Free Biginelli Reactions Catalyzed by Hierarchical Zeolite Utilizing a Ball Mill Technique: A Green Sustainable Process. Catalysts 7:12, pages 84.
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Tayfun Arslan, Emir Alper Türkoğlu, Murat Şentürk & Claudiu T. Supuran. (2016) Synthesis and carbonic anhydrase inhibitory properties of novel chalcone substituted benzenesulfonamides. Bioorganic & Medicinal Chemistry Letters 26:24, pages 5867-5870.
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Shikha Kumari, Danish Idrees, Chandra Bhushan Mishra, Amresh Prakash, Wahiduzzaman, Faizan Ahmad, Md. Imtaiyaz Hassan & Manisha Tiwari. (2016) Design and synthesis of a novel class of carbonic anhydrase-IX inhibitor 1-(3-(phenyl/4-fluorophenyl)-7-imino-3H-[1,2,3]triazolo[4,5d]pyrimidin 6(7H)yl)urea. Journal of Molecular Graphics and Modelling 64, pages 101-109.
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Mohamed F. Mady, Tamer S. Saleh, Ahmed A. El-Kateb, Naglaa M. Abd El-Rahman & Sherein I. Abd El-Moez. (2015) Microwave-assisted synthesis of novel pyrazole and pyrazolo[3,4-d]pyridazine derivatives incorporating diaryl sulfone moiety as potential antimicrobial agents. Research on Chemical Intermediates 42:2, pages 753-769.
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Mohamed F. Mady, Ghada E.A. Awad & Kåre B. Jørgensen. (2014) Ultrasound-assisted synthesis of novel 1,2,3-triazoles coupled diaryl sulfone moieties by the CuAAC reaction, and biological evaluation of them as antioxidant and antimicrobial agents. European Journal of Medicinal Chemistry 84, pages 433-443.
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El Sayed H El Ashry, El Sayed H El Tamany, Mohy El Din Abdel Fattah, Mohamed R E Aly, Ahmed T A Boraei & Axel Duerkop. (2013) A new synthetic access to 2- N -(glycosyl)thiosemicarbazides from 3- N -(glycosyl)oxadiazolinethiones and the regioselectivity of the glycosylation of their oxadiazolinethione precursors . Beilstein Journal of Organic Chemistry 9, pages 135-146.
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Gilles MeesChristel VangestelRudi DierckxPatrick PauwelsJan Van MeerbeeckChristophe Van de Wiele. (2010) Carbonic Anhydrase IX Expression Correlates with FDG Uptake by Primary Non–Small Cell Lung Cancer. Cancer Biotherapy and Radiopharmaceuticals 25:2, pages 149-154.
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Haythem A. Saadeh, Ibrahim M. Mosleh, Amal G. Al-Bakri & Mohammad S. Mubarak. (2010) Synthesis and antimicrobial activity of new 1,2,4-triazole-3-thiol metronidazole derivatives. Monatshefte für Chemie - Chemical Monthly 141:4, pages 471-478.
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Khalid M. Khan, Naheed Fatima, Maimona Rasheed, Saima Jalil, Nida Ambreen, Shahnaz Perveen & M. Iqbal Choudhary. (2009) 1,3,4-Oxadiazole-2(3H)-thione and its analogues: A new class of non-competitive nucleotide pyrophosphatases/phosphodiesterases 1 inhibitors. Bioorganic & Medicinal Chemistry 17:22, pages 7816-7822.
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Alessio Innocenti, Alfonso Maresca, Andrea Scozzafava & Claudiu T. Supuran. (2008) Carbonic anhydrase inhibitors: Thioxolone versus sulfonamides for obtaining isozyme-selective inhibitors?. Bioorganic & Medicinal Chemistry Letters 18:14, pages 3938-3941.
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