Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 23, Issue 1 (2008)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 23, Issue 1 (2008)

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Research Article

Article
Quantitative structure-activity relationship study of ATP-sensitive potassium channel openers: Derivatives of 3-alkylamino-4H-1,2,4-benzothiadiazine 1,1-dioxide
B. K. Sharma, S. K. Sharma, P. Singh & Susheela Sharma
Pages: 1-6
Published online: 04 Oct 2008
AbstractforQuantitative structure-activity relationship study of ATP-sensitive potassium channel openers: Derivatives of 3-alkylamino-4H-1,2,4-benzothiadiazine 1,1-dioxide | Full Text | References | PDF (100.2 KB)
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Article
Kinetic analysis of urea-inactivation of β-galactosidase in the presence of galactose
Ferdinand C. Chilaka & Charles O. Nwamba
Pages: 7-15
Published online: 04 Oct 2008
AbstractforKinetic analysis of urea-inactivation of β-galactosidase in the presence of galactose | Full Text | References | PDF (212.3 KB)
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Article
pH-dependent inhibition of mushroom tyrosinase by N-substituted N-nitrosohydroxylamines
Mitsuhiro Shiino, Yumi Watanabe & Kazuo Umezawa
Pages: 16-20
Published online: 04 Oct 2008
AbstractforpH-dependent inhibition of mushroom tyrosinase by N-substituted N-nitrosohydroxylamines | Full Text | References | PDF (145.3 KB)
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Article
Irreversible inhibition of aldolase by a phosphorylated α-dicarbonyl compound
Nicolas Chabot, Virginie Vinatier, Thierry Gefflaut, Cecile Baudoin, Frederic Rodriguez, Casimir Blonski & Pascal Hoffmann
Pages: 21-27
Published online: 04 Oct 2008
AbstractforIrreversible inhibition of aldolase by a phosphorylated α-dicarbonyl compound | Full Text | References | PDF (153 KB)
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Article
In-vitro evaluation of selected chalcones for antioxidant activity
R. N. Gacche, N. A. Dhole, S. G. Kamble & B. P. Bandgar
Pages: 28-31
Published online: 04 Oct 2008
AbstractforIn-vitro evaluation of selected chalcones for antioxidant activity | Full Text | References | PDF (84.6 KB)
  • 1932 Views
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Article
In vitro inhibition of cytosolic carbonic anhydrases I and II by some new dihydroxycoumarin compounds
Ismet Basaran, Selma Sinan, Umit Cakir, Mustafa Bulut, Oktay Arslan & Ozen Ozensoy
Pages: 32-36
Published online: 04 Oct 2008
AbstractforIn vitro inhibition of cytosolic carbonic anhydrases I and II by some new dihydroxycoumarin compounds | Full Text | References | PDF (103.3 KB)
  • 440 Views
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Article
Some benzoxazoles and benzimidazoles as DNA topoisomerase I and II inhibitors
Emine Oksuzoglu, Betul Tekiner-Gulbas, Sabiha Alper, Ozlem Temiz-Arpaci, Tugba Ertan, Ilkay Yildiz, Nuran Diril, Esin Sener-Aki & Ismail Yalcin
Pages: 37-42
Published online: 04 Oct 2008
AbstractforSome benzoxazoles and benzimidazoles as DNA topoisomerase I and II inhibitors | Full Text | References | PDF (199.3 KB)
  • 1956 Views
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Article
Synthesis and biological evaluation of novel angular fused Pyrrolocoumarins
Christos Kontogiorgis, Konstantinos E. Litinas, Aristea Makri, Demetrios N. Nicolaides, Anastasia Vronteli, Dimitra J. Hadjipavlou-Litina, Eleni Pontiki & Asimoula Siohou
Pages: 43-49
Published online: 04 Oct 2008
AbstractforSynthesis and biological evaluation of novel angular fused Pyrrolocoumarins | Full Text | References | PDF (131.6 KB)
  • 717 Views
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Article
Quantitative structure-activity relationship study of novel rhinacanthins and related naphthoquinone esters as anticancer agents
B. K. Sharma, P. Singh, R. Kumar & Susheela Sharma
Pages: 50-55
Published online: 04 Oct 2008
AbstractforQuantitative structure-activity relationship study of novel rhinacanthins and related naphthoquinone esters as anticancer agents | Full Text | References | PDF (100.8 KB)
  • 461 Views
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Article
6-Azathymidine-4′-thionucleosides: synthesis and antiviral evaluation
Malina Jasamai, Jan Balzarini & Claire Simons
Pages: 56-61
Published online: 04 Oct 2008
Abstractfor6-Azathymidine-4′-thionucleosides: synthesis and antiviral evaluation | Full Text | References | PDF (160.2 KB)
  • 517 Views
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Article
Mild and efficient synthesis of new tetraketones as lipoxygenase inhibitors and antioxidants
Ghulam M. Maharvi, Samar Ali, Naheed Riaz, Nighat Afza, Abdul Malik, Muhammad Ashraf, Lubna Iqbal & Mehreen Lateef
Pages: 62-69
Published online: 04 Oct 2008
AbstractforMild and efficient synthesis of new tetraketones as lipoxygenase inhibitors and antioxidants | Full Text | References | PDF (137.5 KB)
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Article
Synthesis of monooxime-monocarbamoyl bispyridinium compounds bearing (E)-but-2-ene linker and evaluation of their reactivation activity against tabun- and paraoxon-inhibited acetylcholinesterase
Kamil Musilek, Ondrej Holas, Kamil Kuca, Daniel Jun, Vlastimil Dohnal, Veronika Opletalova & Martin Dolezal
Pages: 70-76
Published online: 04 Oct 2008
AbstractforSynthesis of monooxime-monocarbamoyl bispyridinium compounds bearing (E)-but-2-ene linker and evaluation of their reactivation activity against tabun- and paraoxon-inhibited acetylcholinesterase | Full Text | References | PDF (153.6 KB)
  • 684 Views
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Article
Synthesis and in vitro antimicrobial studies of some new 3-[phenyldiazenyl] benzaldehyde N-phenyl thiosemicarbazones
Anand K. Halve, Bhuwan Bhashkar, Vasudha Sharma, Raman Bhadauria, Amit Kankoriya, Ajay Soni & Kiran Tiwari
Pages: 77-81
Published online: 04 Oct 2008
AbstractforSynthesis and in vitro antimicrobial studies of some new 3-[phenyldiazenyl] benzaldehyde N-phenyl thiosemicarbazones | Full Text | References | PDF (93.4 KB)
  • 897 Views
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Article
A novel synthesis and antimicrobial activity of 1-[(Substituted-phenyl) sulfonyl]pyrrolidin-2-ones
Muhammad Zareef, Rashid Iqbal & Muhammad Arfan
Pages: 82-86
Published online: 04 Oct 2008
AbstractforA novel synthesis and antimicrobial activity of 1-[(Substituted-phenyl) sulfonyl]pyrrolidin-2-ones | Full Text | References | PDF (106.8 KB)
  • 394 Views
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Article
Three components coupling catalysed by NaHSO4.Sio2 – A convenient synthesis, antibacterial and antifungal activities of novel 6-Aryl-1,2,4,5-tetrazinan-3-ones
M. Gopalakrishnan, P. Sureshkumar, J. Thanusu & V. Kanagarajan
Pages: 87-93
Published online: 04 Oct 2008
AbstractforThree components coupling catalysed by NaHSO4.Sio2 – A convenient synthesis, antibacterial and antifungal activities of novel 6-Aryl-1,2,4,5-tetrazinan-3-ones | Full Text | References | PDF (216.7 KB)
  • 491 Views
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Article
Targeting human DNA polymerase α for the inhibition of keratinocyte proliferation. Part 1. Homology model, active site architecture and ligand binding
Anja Richartz, Monika Höltje, Birte Brandt, Monika Schäfer-Korting & Hans-Dieter Höltje
Pages: 94-100
Published online: 04 Oct 2008
AbstractforTargeting human DNA polymerase α for the inhibition of keratinocyte proliferation. Part 1. Homology model, active site architecture and ligand binding | Full Text | References | PDF (1.2 MB)
  • 589 Views
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Article
Carbonic anhydrase inhibitors. Inhibition of the cytosolic and tumor-associated carbonic anhydrase isozymes I, II and IX with some 1,3,4-oxadiazole- and 1,2,4-triazole-thiols
Gabriela Laura Almajan, Stefania-Felicia Barbuceanu, Alessio innocenti, Andrea Scozzafava & Claudiu T. Supuran
Pages: 101-107
Published online: 04 Oct 2008
AbstractforCarbonic anhydrase inhibitors. Inhibition of the cytosolic and tumor-associated carbonic anhydrase isozymes I, II and IX with some 1,3,4-oxadiazole- and 1,2,4-triazole-thiols | Full Text | References | PDF (150.1 KB)
  • 639 Views
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Article
Synthesis, characterization and biological aspects of novel five-coordinated dimeric-Cu(II) systems
Pramod B. Pansuriya & Mohan N. Patel
Pages: 108-119
Published online: 04 Oct 2008
AbstractforSynthesis, characterization and biological aspects of novel five-coordinated dimeric-Cu(II) systems | Full Text | References | PDF (322.6 KB)
  • 782 Views
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Article
Metal-based sulfonamides: Their preparation, characterization and in-vitro antibacterial, antifungal & cytotoxic properties. X-ray structure of 4-[(2-hydroxybenzylidene) amino] benzenesulfonamide
Zahid H. Chohan
Pages: 120-130
Published online: 04 Oct 2008
AbstractforMetal-based sulfonamides: Their preparation, characterization and in-vitro antibacterial, antifungal & cytotoxic properties. X-ray structure of 4-[(2-hydroxybenzylidene) amino] benzenesulfonamide | Full Text | References | PDF (546.7 KB)
  • 1987 Views
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Article
A microtitre plate assay for measuring glycosidase activity
Andrea L. Ball, Kirsty A. Chambers, Meera Hewinson, Sambavi Navaratnarajah, Lamia Samrin, Nesta Thomas, Abigail E. H. Tyler, Amanda J. Wall & Matthew D. Lloyd
Pages: 131-135
Published online: 04 Oct 2008
AbstractforA microtitre plate assay for measuring glycosidase activity | Full Text | References | PDF (101.8 KB)
  • 2120 Views
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Article
Antibacterial and antifungal activities of teucrium royleanum (Labiatea)
Bashir Ahmad, S. M Mukaram Shah, Shumaila Bashir & Halima Begum
Pages: 136-139
Published online: 04 Oct 2008
AbstractforAntibacterial and antifungal activities of teucrium royleanum (Labiatea) | Full Text | References | PDF (100.2 KB)
  • 627 Views
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Article
Lipoxygenase inhibiting and antioxidant iridoids from Buddleja crispa
IJAZ AHMAD, SHILIN CHEN, YONG PENG, SIBAO CHEN & LIJIA XU
Pages: 140-143
Published online: 04 Oct 2008
AbstractforLipoxygenase inhibiting and antioxidant iridoids from Buddleja crispa | Full Text | References | PDF (113.9 KB)
  • 626 Views
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Article
Effects of some antibiotics on human erythrocyte glutathione reductase: an in vitro study
Murat Senturk, O. Irfan Kufrevioglu & Mehmet Ciftci
Pages: 144-148
Published online: 04 Oct 2008
AbstractforEffects of some antibiotics on human erythrocyte glutathione reductase: an in vitro study | Full Text | References | PDF (125 KB)
  • 748 Views
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Article
In vitro prooxidant effect of caffeine
İlhami Gülçİn
Pages: 149-152
Published online: 04 Oct 2008
AbstractforIn vitro prooxidant effect of caffeine | Full Text | References | PDF (108.6 KB)
  • 973 Views
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