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Research Article

Synthesis and biological screening of some pyridine derivatives as anti-malarial agents

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Pages 69-77 | Received 23 Jun 2010, Accepted 22 Mar 2011, Published online: 25 May 2011

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D Ashok, M Ram Reddy, Ravinder Dharavath, Nalaparaju Nagaraju, Katta Ramakrishna, Srinivas Gundu & M Sarasija. (2021) One-pot three-component condensation for the synthesis of 2,4,6-triarylpyridines and evaluation of their antimicrobial activity. Journal of Chemical Sciences 133:1.
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Piotr Pomarański, Piotr Roszkowski, Jan K. Maurin & Zbigniew Czarnocki. (2019) Regio-and atropselective synthesis of selected ortho-phenyl substituted arylpyridine derivatives. Journal of Molecular Structure 1177, pages 564-570.
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Sherine N. Khattab, Hosam H. Khalil, Adnan A. Bekhit, Mohamed M. Abd El‐Rahman, Beatriz G. de la Torre, Ayman El‐Faham & Fernando Albericio. (2018) 1,3,5‐Triazino Peptide Derivatives: Synthesis, Characterization, and Preliminary Antileishmanial Activity. ChemMedChem 13:7, pages 725-735.
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Sandeep Jain, Ajay Kumar & Deepika Saini. (2018) Novel arylidene derivatives of quinoline based thiazolidinones: Synthesis, in vitro, in vivo and in silico study as antimalarials. Experimental Parasitology 185, pages 107-114.
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Kamal Fahmy Mohamed Atta, Tamer Mohamed Ibrahim, Omaima Osman Mahmoud Farahat, Tareq Qasem Al-Shargabi, Mohamed Gaber Marei, Adnan Ahmed Bekhit & El Sayed Helmy El Ashry. (2017) Synthesis, modeling and biological evaluation of hybrids from pyrazolo[1,5c]pyrimidine as antileishmanial agents. Future Medicinal Chemistry 9:16, pages 1913-1929.
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Sherine Nabil Khattab, Nesreen Saied Haiba, Ahmed Mosaad Asal, Adnan A. Bekhit, Aida A. Guemei, Adel Amer & Ayman El-Faham. (2017) Study of antileishmanial activity of 2-aminobenzoyl amino acid hydrazides and their quinazoline derivatives. Bioorganic & Medicinal Chemistry Letters 27:4, pages 918-921.
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Adnan A. Bekhit, Ahmed M.M. Hassan, Heba A. Abd El Razik, Mostafa M.M. El-Miligy, Eman J. El-Agroudy & Alaa El-Din A. Bekhit. (2015) New heterocyclic hybrids of pyrazole and its bioisosteres: Design, synthesis and biological evaluation as dual acting antimalarial-antileishmanial agents. European Journal of Medicinal Chemistry 94, pages 30-44.
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Xing‐Hai Liu, Zhao‐Hui Sun, Ming‐Yan Yang, Cheng‐Xia Tan, Jian‐Quan Weng, Yong‐Gang Zhang & Yi Ma. (2014) Microwave Assistant One Pot Synthesis, Crystal Structure, Antifungal Activities and 3D‐ QSAR of Novel 1,2,4‐Triazolo[4,3‐ a ]pyridines . Chemical Biology & Drug Design 84:3, pages 342-347.
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Shahzad Ahmed, Muhammad Sharif, Khurram Shoaib, Sebastian Reimann, Jamshed Iqbal, Tamás Patonay, Anke Spannenberg & Peter Langer. (2013) Synthesis of 2,6-diaryl-3-(trifluoromethyl)pyridines by regioselective Suzuki–Miyaura reactions of 2,6-dichloro-3-(trifluoromethyl)pyridine. Tetrahedron Letters 54:13, pages 1669-1672.
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. (2012) Current World Literature. Current Opinion in Infectious Diseases 25:6, pages 718-728.
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