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Original Articles

The Preparation of Ternary Solid Dispersions of an Herbal Drug via Spray Drying of Liquid Feed

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Pages 412-421 | Published online: 09 Mar 2010

Keep up to date with the latest research on this topic with citation updates for this article.

Read on this site (16)

Xin Wang, Yijian Zhu, Xudong Zhao, Shurong Zhang, Meiting Cao, Xiaoyue Wang & Wei Li. (2022) Development and characterization of an amorphous curcumin-Eudragit®E100 solid dispersions with improved solubility, stability, and pharmacokinetic properties. Pharmaceutical Development and Technology 27:9, pages 965-974.
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Ashok Mahajan, Naazneen Surti, Priyal Patel, Naziya Gheewala, Ashwini Patel & Dimal Shah. (2022) Optimization of formulation and process variables using central composite design for the production of nevirapine spray dried solid dispersion. Drying Technology 40:9, pages 1745-1757.
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L. A. Vázquez-León, J. A. Olguín-Rojas, D. E. Páramo-Calderón, Gerardo F. Barbero, M. A. Salgado-Cervantes, Miguel Palma, M. A. García-Alvarado & G. C. Rodríguez-Jimenes. (2021) Closed-loop spray drying with N2 of Moringa oleifera leaf ethanolic extracts: Effects on bioactive compounds and antiradical activity. Drying Technology 39:14, pages 2092-2104.
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Shambhavi Borde, Sagar Kumar Paul & Harsh Chauhan. (2021) Ternary solid dispersions: classification and formulation considerations. Drug Development and Industrial Pharmacy 47:7, pages 1011-1028.
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Debborah Gonçalves Bezerra, Ivano Alessandro Devilla, Edemilson Cardoso da Conceição, Cecília Czepak, Karina C. Albernaz Godinho, Samantha Salomão Caramori, Roberto Campos Portela & Joelma Abadia Marciano de Paula. (2021) Microencapsulated extracts from Azadirachta indica seeds: Acquisition, characterization, and use in controlling Helicoverpa armigera. Drying Technology 39:10, pages 1325-1338.
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Vandita Kakkar, Indu Pal Kaur, Amrit Pal Kaur, Komal Saini & Kamalinder K. Singh. (2018) Topical delivery of tetrahydrocurcumin lipid nanoparticles effectively inhibits skin inflammation: in vitro and in vivo study. Drug Development and Industrial Pharmacy 44:10, pages 1701-1712.
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Simone Vieira Pereira, Fábio Belotti Colombo, Rodrigo Molina Martins & Luis Alexandre Pedro de Freitas. (2014) Spray Cooling Process Factors and Quality Interactions During the Preparation of Microparticles Containing an Active Pharmaceutical Ingredient. Drying Technology 32:10, pages 1188-1199.
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Rodrigo Molina Martins, Silvia Siqueira, Marcela Olaia Machado & Luis Alexandre Pedro Freitas. (2013) The effect of homogenization method on the properties of carbamazepine microparticles prepared by spray congealing. Journal of Microencapsulation 30:7, pages 692-700.
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R.M. Martins, M.O. Machado, S.V. Pereira, A.B. F. L. Nosari, L.A. Tacon & L.A. P. Freitas. (2012) Engineering Active Pharmaceutical Ingredients by Spray Drying: Effects on Physical Properties and In Vitro Dissolution. Drying Technology 30:9, pages 905-913.
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R.M. Martins, M.O. Machado, S.V. Pereira, A.B. F. L. Nosari, L.A. Tacon & L.A. P. Freitas. (2012) Microparticulated Hydrochlorothiazide Solid Dispersion: Enhancing Dissolution Properties via Spray Drying. Drying Technology 30:9, pages 959-967.
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Rodrigo Molina Martins, Silvia Siqueira & Luis Alexandre Pedro Freitas. (2012) Spray Congealing of Pharmaceuticals: Study on Production of Solid Dispersions Using Box-Behnken Design. Drying Technology 30:9, pages 935-945.
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LucianaA. Tacon & LuisA. P. Freitas. (2011) Paste Residence Time in a Spouted Bed Dryer. IV: Effect of the Inert Particle Size Distribution. Drying Technology 29:14, pages 1662-1672.
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R.O. Couto, R.R. Araújo, L.A. Tacon, E.C. Conceição, M. T. F. Bara, J.R. Paula & L. A. P. Freitas. (2011) Development of a Phytopharmaceutical Intermediate Product via Spray Drying. Drying Technology 29:6, pages 709-718.
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Wei-Qiang Tang, Di-Cai Li, Yang-Xiao Lv & Jian-Guo Jiang. (2011) Concentration and Drying of Tea Polyphenols Extracted from Green Tea Using Molecular Distillation and Spray Drying. Drying Technology 29:5, pages 584-590.
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C. C. C. Teixeira, G.A. Teixeira & L. A. P. Freitas. (2011) Spray Drying of Extracts from Red Yeast Fermentation Broth. Drying Technology 29:3, pages 342-350.
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Matheus Gabriel de Oliveira, Guilherme Gomes Moreira, Andressa Tuane Santana Paz, Thiago Levi Silva Oliveira, Luís Antônio Dantas Silva, Edemilson Cardoso da Conceição, Leonardo Luiz Borges, Vinicius Barreto da Silva & José Realino de Paula. (2023) Process optimization of physicochemical properties of spray-dried Hydrocotyle umbellata L. extract. Brazilian Journal of Pharmaceutical Sciences 59.
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Bárbara Verônica Cardoso de Souza, Mariana de Morais Sousa, José Augusto Gasparotto Sattler, Ana Cristina Sousa Gramoza Vilarinho Santana, Rusbene Bruno Fonseca de Carvalho, José de Sousa Lima Neto, Fernando de Matos Borges, Iramaia Angelica Neri Numa, Alessandra Braga Ribeiro & Lívio César Cunha Nunes. (2022) Nanoencapsulation and bioaccessibility of polyphenols of aqueous extracts from Bauhinia forficata link. Food Chemistry: Molecular Sciences 5, pages 100144.
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Saurabh Shankar Patel, Heartwin A. Pushpadass, Magdaline Eljeeva Emerald Franklin, Surendra Nath Battula & Palanimuthu Vellingiri. (2021) Microencapsulation of curcumin by spray drying: Characterization and fortification of milk. Journal of Food Science and Technology 59:4, pages 1326-1340.
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Gangqi Han, Bing Wang, Mengli Jia, Shuxin Ding, Wenxuan Qiu, Yuxuan Mi, Zhimei Mi, Yuhao Qin, Wenxing Zhu, Xinli Liu & Wei Li. (2022) Optimization and evaluation of resveratrol amorphous solid dispersions with a novel polymeric system. Mathematical Biosciences and Engineering 19:8, pages 8019-8034.
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Christina Winarti & Titi Candra Sunarti. (2022) Effect of Heating on the Stability of Curcumin on Temulawak Oleoresin Encapsulated in Arrowroot Starch Nanoparticles. E3S Web of Conferences 361, pages 04005.
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Jelena Mudrić, Katarina Šavikin, Ljiljana Đekić, Stefan Pavlović, Ivana Kurćubić, Svetlana Ibrić & Jelena Đuriš. (2021) Development of Lipid-Based Gastroretentive Delivery System for Gentian Extract by Double Emulsion–Melt Dispersion Technique. Pharmaceutics 13:12, pages 2095.
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Thi Sinh VO, Tran Thi Bich Chau VO, Tran Thi Thu Ngoc VO & Thi Ngoc Huyen LAİ. (2021) Turmeric (Curcuma longa L.): Chemical Components and Their Effective Clinical Applications. Journal of the Turkish Chemical Society Section A: Chemistry 8:3, pages 883-898.
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Maria Rosaria Lauro, Stefania Marzocco, Shara Francesca Rapa, Teresa Musumeci, Virgilio Giannone, Patrizia Picerno, Rita Patrizia Aquino & Giovanni Puglisi. (2020) Recycling of Almond By-Products for Intestinal Inflammation: Improvement of Physical-Chemical, Technological and Biological Characteristics of a Dried Almond Skins Extract. Pharmaceutics 12:9, pages 884.
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Kenji ISHIMOTO & Shinsaku NAKAGAWA. (2020) Application of Amorphous Solid Dispersion Technology for Functional Food Development機能性食品開発を目指した非晶質固体分散技術の利用法. Oleoscience 20:2, pages 53-60.
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Thi Thanh Hanh Nguyen, Changseop Seo, So-Hyung Kwak, Jeesoo Kim, Hee-Kyoung Kang, Seong-Bo Kim & Doman Kim. 2019. Enzymes in Food Biotechnology. Enzymes in Food Biotechnology 405 418 .
Cristiane C. C. Teixeira, Elias de Paiva Junior & Luis Alexandre Pedro de Freitas. (2017) Fluidized Bed Hot-Melt Granulation as a Tool to Improve Curcuminoid Solubility. AAPS PharmSciTech 19:3, pages 1061-1071.
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Marília M.S. Vieira, Rodrigo M. Martins & Luis A.P. Freitas. (2018) Characteristics of piroxicam granules prepared by fluidized bed hot melt granulation. Advanced Powder Technology 29:4, pages 934-940.
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Cristiane Cardoso Correia Teixeira, Tatiana Pereira de Freitas Cabral, Luciana Alves Tacon, Isabel Lemos Villardi, Aurea Donizete Lanchote & Luis Alexandre Pedro de Freitas. (2017) Solid state stability of polyphenols from a plant extract after fluid bed atmospheric spray-freeze-drying. Powder Technology 319, pages 494-504.
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Luiza T. Chaul, Edemilson C. Conceição, Maria Tereza F. Bara, José R. Paula & Renê O. Couto. (2017) Engineering spray-dried rosemary extracts with improved physicomechanical properties: a design of experiments issue. Revista Brasileira de Farmacognosia 27:2, pages 236-244.
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Leonardo L. Borges, Frederico S. Martins, Edemilson C. Conceição & Dâmaris Silveira. (2017) Optimization of the Spray-Drying Process for Developing Jabuticaba Waste Powder Employing Response Surface Methodology. Journal of Food Process Engineering 40:1, pages e12276.
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Maria Rosaria Lauro, Lucia Crascì, Virgilio Giannone, Gabriele Ballistreri, Simona Fabroni, Francesca Sansone, Paolo Rapisarda, Anna Maria Panico & Giovanni Puglisi. (2017) An Alginate/Cyclodextrin Spray Drying Matrix to Improve Shelf Life and Antioxidant Efficiency of a Blood Orange By-Product Extract Rich in Polyphenols: MMPs Inhibition and Antiglycation Activity in Dysmetabolic Diseases . Oxidative Medicine and Cellular Longevity 2017, pages 1-12.
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Shrawan Baghel, Helen Cathcart & Niall J. O'Reilly. (2016) Polymeric Amorphous Solid Dispersions: A Review of Amorphization, Crystallization, Stabilization, Solid-State Characterization, and Aqueous Solubilization of Biopharmaceutical Classification System Class II Drugs. Journal of Pharmaceutical Sciences 105:9, pages 2527-2544.
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Abhishek Singh & Guy Van den Mooter. (2016) Spray drying formulation of amorphous solid dispersions. Advanced Drug Delivery Reviews 100, pages 27-50.
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C. C. C. Teixeira, L. M. Mendonça, M. M. Bergamaschi, R. H. C. Queiroz, G. E. P. Souza, L. M. G. Antunes & L. A. P. Freitas. (2015) Microparticles Containing Curcumin Solid Dispersion: Stability, Bioavailability and Anti-Inflammatory Activity. AAPS PharmSciTech 17:2, pages 252-261.
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D.M. Cano-Higuita, C.R. Malacrida & V.R.N. Telis. (2015) Stability of Curcumin Microencapsulated by Spray and Freeze Drying in Binary and Ternary Matrices of Maltodextrin, Gum Arabic and Modified Starch. Journal of Food Processing and Preservation 39:6, pages 2049-2060.
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Avinash B. Gangurde, Harish S. Kundaikar, Sharadchandra D. Javeer, Divakar R. Jaiswar, Mariam S. Degani & Purnima D. Amin. (2015) Enhanced solubility and dissolution of curcumin by a hydrophilic polymer solid dispersion and its insilico molecular modeling studies. Journal of Drug Delivery Science and Technology 29, pages 226-237.
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Diana Maria Cano-Higuita, Harvey Alexander Villa Vélez & Vania Regina Nicoletti Telis. (2015) MICROENCAPSULATION OF TURMERIC OLEORESIN IN BINARY AND TERNARY BLENDS OF GUM ARABIC, MALTODEXTRIN AND MODIFIED STARCH. Ciência e Agrotecnologia 39:2, pages 173-182.
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Pankajkumar Yadav, Ekta Yadav, Amita Verma & Saima Amin. (2014) In vitro characterization and pharmacodynamic evaluation of furosemide loaded self nano emulsifying drug delivery systems (SNEDDS). Journal of Pharmaceutical Investigation 44:6, pages 443-453.
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M. R. V. Fernandes, A. E. C. S. Azzolini, M. L. L. Martinez, C. R. F. Souza, Y. M. Lucisano-Valim & W. P. Oliveira. (2014) Assessment of Antioxidant Activity of Spray Dried Extracts of Psidium guajava Leaves by DPPH and Chemiluminescence Inhibition in Human Neutrophils . BioMed Research International 2014, pages 1-10.
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Pankajkumar S. Yadav, Ekta Yadav, Amita Verma & Saima Amin. (2014) Development, Characterization, and Pharmacodynamic Evaluation of Hydrochlorothiazide Loaded Self-Nanoemulsifying Drug Delivery Systems. The Scientific World Journal 2014, pages 1-10.
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Amrit Paudel, Zelalem Ayenew Worku, Joke Meeus, Sandra Guns & Guy Van den Mooter. (2013) Manufacturing of solid dispersions of poorly water soluble drugs by spray drying: Formulation and process considerations. International Journal of Pharmaceutics 453:1, pages 253-284.
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Rodrigo Molina Martins, Simone Vieira Pereira, Silvia Siqueira, Wellington Fioravante Salomão & Luis Alexandre Pedro Freitas. (2013) Curcuminoid content and antioxidant activity in spray dried microparticles containing turmeric extract. Food Research International 50:2, pages 657-663.
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Luciana A. Tacon & Luis A.P. Freitas. (2013) Box-Behnken design to study the bergenin content and antioxidant activity of Endopleura uchi bark extracts obtained by dynamic maceration. Revista Brasileira de Farmacognosia 23:1, pages 65-71.
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Renê O. Couto, Frederico S. Martins, Luiza T. Chaul, Edemilson C. Conceição, Luis Alexandre P. Freitas, Maria Teresa F. Bara & José R. Paula. (2013) Spray drying of Eugenia dysenterica extract: effects of in-process parameters on product quality. Revista Brasileira de Farmacognosia 23:1, pages 115-123.
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Renê O. Couto, Edemilson C. Conceição, Luíza T. Chaul, Ezequiane M.S. Oliveira, Frederico S. Martins, Maria Teresa F. Bara, Kênnia R. Rezende, Suzana F. Alves & José R. Paula. (2012) Spray-dried rosemary extracts: Physicochemical and antioxidant properties. Food Chemistry 131:1, pages 99-105.
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Rodrigo M. Martins, Silvia Siqueira, Luciana A. Tacon & Luis A.P. Freitas. (2012) Microstructured ternary solid dispersions to improve carbamazepine solubility. Powder Technology 215-216, pages 156-165.
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