Citations (48)
Keep up to date with the latest research on this topic with citation updates for this article.
Read on this site (12)
Christian Battipaglia, Lia Feliciello, Alessandro D. Genazzani, Fabio Facchinetti & Giovanni Grandi. (2023) Combined oral contraceptive with estetrol plus drospirenone: from pharmacokinetics to clinical applications. Expert Opinion on Drug Metabolism & Toxicology 0:0, pages 1-9.
Read now
Read now
Darakhshan Parveen, Anwesha Das, Shaista Amin, M. Mumtaz Alam, Mymoona Akhter, Mohammad Ahmed Khan, Ruhi Ali, Tarique Anwer, Khursheed A. Sheikh, Faizul Azam & M. Shaquiquzzaman. (2023) Effectiveness of estrogen and its derivatives over dexamethasone in the treatment of COVID-19. Journal of Biomolecular Structure and Dynamics 0:0, pages 1-17.
Read now
Read now
Kristina Gemzell-Danielsson, Angelo Cagnacci, Nathalie Chabbert-Buffet, Jonathan Douxfils, Jean-Michel Foidart, Ali Kubba, Luis Ignacio Lete Lasa, Diana Mansour, Joseph Neulen, Jaoquim Neves, Fátima Palma, Thomas Römer, Robert Spaczyński & Vera Tóth. (2022) A novel estetrol-containing combined oral contraceptive: European expert panel review. The European Journal of Contraception & Reproductive Health Care 27:5, pages 373-383.
Read now
Read now
Céline Gérard, Jean-François Arnal, Maud Jost, Jonathan Douxfils, Françoise Lenfant, Coralie Fontaine, René Houtman, David F. Archer, Robert L. Reid, Rogerio A. Lobo, Ulysse Gaspard, Herjan J.T. Coelingh Bennink, Mitchell D. Creinin & Jean-Michel Foidart. (2022) Profile of estetrol, a promising native estrogen for oral contraception and the relief of climacteric symptoms of menopause. Expert Review of Clinical Pharmacology 15:2, pages 121-137.
Read now
Read now
Andrea R. Genazzani, Ulysse Gaspard & Jean-Michel Foidart. (2019) Oral investigational drugs currently in phase I or phase II for the amelioration
of menopausal symptoms. Expert Opinion on Investigational Drugs 28:3, pages 235-247.
Read now
Read now
H. J. T. Coelingh Bennink, C. Verhoeven, Y. Zimmerman, M. Visser, J-M. Foidart & K. Gemzell-Danielsson. (2017) Pharmacokinetics of the fetal estrogen estetrol in a multiple-rising-dose study in postmenopausal women. Climacteric 20:3, pages 285-289.
Read now
Read now
Marie Mawet, Catherine Maillard, Christine Klipping, Yvette Zimmerman, Jean-Michel Foidart & Herjan J.T. Coelingh Bennink. (2015) Unique effects on hepatic function, lipid metabolism, bone and growth endocrine parameters of estetrol in combined oral contraceptives. The European Journal of Contraception & Reproductive Health Care 20:6, pages 463-475.
Read now
Read now
A. Nath & R. Sitruk-Ware. (2009) Pharmacology and clinical applications of selective estrogen receptor modulators. Climacteric 12:3, pages 188-205.
Read now
Read now
H. J. T. Coelingh Bennink, C. F. Holinka & E. Diczfalusy. (2008) Estetrol review: profile and potential clinical applications. Climacteric 11:sup1, pages 47-58.
Read now
Read now
M. Visser, C. F. Holinka & H. J. T. Coelingh Bennink. (2008) First human exposure to exogenous single-dose oral estetrol in early postmenopausal women. Climacteric 11:sup1, pages 31-40.
Read now
Read now
A.-M. Heegaard, C. F. Holinka, P. Kenemans & H. J. T. Coelingh Bennink. (2008) Estrogenic uterovaginal effects of oral estetrol in the modified Allen–Doisy test. Climacteric 11:sup1, pages 22-28.
Read now
Read now
C. F. Holinka, M. Brincat & H. J. T. Coelingh Bennink. (2008) Preventive effect of oral estetrol in a menopausal hot flush model. Climacteric 11:sup1, pages 15-21.
Read now
Read now
Articles from other publishers (36)
Catherine de Bournonville, Philippine Lemoine, Jean‐Michel Foidart, Jean‐François Arnal, Françoise Lenfant & Charlotte A. Cornil. (2023)
Role of membrane estrogen receptor alpha (
ERα
) in the rapid regulation of male sexual behavior
. Journal of Neuroendocrinology 35:10.
Crossref
Crossref
Anne Gallez, Gwenaël Nys, Vincent Wuidar, Isabelle Dias Da Silva, Mélanie Taziaux, Virginie Kinet, Ekaterine Tskitishvili, Agnès Noel, Jean-Michel Foidart, Géraldine Piel, Marianne Fillet & Christel Péqueux. (2023) Comparison of Estetrol Exposure between Women and Mice to Model Preclinical Experiments and Anticipate Human Treatment. International Journal of Molecular Sciences 24:11, pages 9718.
Crossref
Crossref
Céline Gérard & Jean-Michel Foidart. (2023) Estetrol: From Preclinical to Clinical Pharmacology and Advances in the Understanding of the Molecular Mechanism of Action. Drugs in R&D 23:2, pages 77-92.
Crossref
Crossref
Daniel Patiño-García, Jaime Palomino, Cristián Pomés, Claudia Celle, Verónica Torres-Estay & Renán Orellana. (2023) Estetrol Increases Progesterone Genetic Response without Triggering Common Estrogenic Effects in Endometriotic Cell Lines and Primary Cultures. Biomedicines 11:4, pages 1169.
Crossref
Crossref
Aida U. Hamadyanova, Afzal H. Tuhtaboev, Venera A. Shafieva, Elena A. Kolodyazhnaya, Julia R. Mansurova, Aliya A. Muratova, Arina A. Andreeva & Julia A. Muzafarova. (2023) Estetrol: a new estrogen component in combined oral contraceptives: A review. Gynecology 24:6, pages 459-464.
Crossref
Crossref
Herjan J T Coelingh Bennink, Jan Krijgh, Jan F M Egberts, Maria Slootweg, Harm H E van Melick, Erik P M Roos, Diederik M Somford, Yvette Zimmerman, Iman J Schultz, Noel W Clarke, R Jeroen A van Moorselaar & Frans M J Debruyne. (2022) Maintaining bone health by estrogen therapy in patients with advanced prostate cancer: a narrative review. Endocrine Connections 11:12.
Crossref
Crossref
Yvette Zimmerman, Mark Frydenberg, Hendrik van Poppel, R. Jeroen A. van Moorselaar, Erik P.M. Roos, Diederik M. Somford, Ton A. Roeleveld, Tjard D. de Haan, Harm H.E. van Melick, Yacov Reisman, Jan Krijgh, Frans M.J. Debruyne & Herjan J.T. Coelingh Bennink. (2022) Estetrol Prevents Hot Flushes and Improves Quality of Life in Patients with Advanced Prostate Cancer Treated with Androgen Deprivation Therapy: The PCombi Study. European Urology Open Science 45, pages 59-67.
Crossref
Crossref
Priya Yawale, Neelam Upadhyay, Sangita Ganguly & Singh KumarAshishAshish. (2022) A comprehensive review on recent novel food and industrial applications of flaxseed: 2014 onwards. Food and Feed Research 49:2, pages 67-95.
Crossref
Crossref
Priya Yawale, Neelam Upadhyay, Sangita Ganguly & Singh KumarAshishAshish. (2022) A comprehensive review on recent novel food and industrial applications of flaxseed: 2014 onwards. Food and Feed Research:00, pages 16-16.
Crossref
Crossref
Teresa Navarrete Horta, Francisco Javier Guerrero Carreño, Paulina Valdés Aguerrebere & Leopoldo Alejandro Vázquez Estrada. (2022) Estetrol: ¿un nuevo paradigma en terapia ginecológica?. Acta Médica Grupo Ángeles 20:1, pages 50-57.
Crossref
Crossref
T.N. Bebneva, M.B. Khamoshina & V.E. Radzinsky. (2022) Estetrol is a new estrogen with selective tissue activity in the composition of a combined oral contraceptive. Problemy reproduktsii 28:6, pages 133.
Crossref
Crossref
Franca Fruzzetti, Tiziana Fidecicchi, Maria Magdalena Montt Guevara & Tommaso Simoncini. (2021) Estetrol: A New Choice for Contraception. Journal of Clinical Medicine 10:23, pages 5625.
Crossref
Crossref
Anne Gallez, Isabelle Dias Da Silva, Vincent Wuidar, Jean-Michel Foidart & Christel Péqueux. (2021) Estetrol and Mammary Gland: Friends or Foes?. Journal of Mammary Gland Biology and Neoplasia 26:3, pages 297-308.
Crossref
Crossref
Herjan J.T. Coelingh Bennink, Jeroen A. van Moorselaar, E. David Crawford, Erik P.M. Roos, Diederik M. Somford, Ton A. Roeleveld, Tjard D. de Haan, Harm H.E. van Melick, Yacov Reisman, Yvette Zimmerman, Gonnie van Osta, Jan Krijgh, Neal D. Shore, Fred Saad, Andrew V. Schally & Frans M.J. Debruyne. (2021) Estetrol Cotreatment of Androgen Deprivation Therapy in Infiltrating or Metastatic, Castration-sensitive Prostate Cancer: A Randomized, Double-blind, Phase II Trial (PCombi). European Urology Open Science 28, pages 52-61.
Crossref
Crossref
Marcus Schmidt, Hans Lenhard, Arnd Hoenig, Yvette Zimmerman, Jan Krijgh, Monique Jansen & Herjan J. T. Coelingh Bennink. (2020) Tumor suppression, dose-limiting toxicity and wellbeing with the fetal estrogen estetrol in patients with advanced breast cancer. Journal of Cancer Research and Clinical Oncology 147:6, pages 1833-1842.
Crossref
Crossref
Anne Gallez, Silvia Blacher, Erik Maquoi, Erika Konradowski, Marc Joiret, Irina Primac, Céline Gérard, Mélanie Taziaux, René Houtman, Liesbet Geris, Françoise Lenfant, Elisabetta Marangoni, Nor Eddine Sounni, Jean-Michel Foidart, Agnès Noël & Christel Péqueux. (2021) Estetrol Combined to Progestogen for Menopause or Contraception Indication Is Neutral on Breast Cancer. Cancers 13:10, pages 2486.
Crossref
Crossref
Emmanuelle Noirrit-Esclassan, Marie-Cécile Valera, Florence Tremollieres, Jean-Francois Arnal, Françoise Lenfant, Coralie Fontaine & Alexia Vinel. (2021) Critical Role of Estrogens on Bone Homeostasis in Both Male and Female: From Physiology to Medical Implications. International Journal of Molecular Sciences 22:4, pages 1568.
Crossref
Crossref
Ulysse Gaspard, Mélanie Taziaux, Marie Mawet, Maud Jost, Valérie Gordenne, Herjan J.T. Coelingh Bennink, Rogerio A. Lobo, Wulf H. UtianJean-Michel Foidart. (2020) A multicenter, randomized study to select the minimum effective dose of estetrol (E4) in postmenopausal women (E4Relief): part 1. Vasomotor symptoms and overall safety. Menopause 27:8, pages 848-857.
Crossref
Crossref
Marie-Cécile Valéra, Coralie Fontaine, Emmanuelle Noirrit-Esclassan, Pierre Gourdy, Françoise Lenfant & Jean-François Arnal. 2019. La Ménopause en Pratique. La Ménopause en Pratique
157
168
.
Marie-Cécile Valéra, Coralie Fontaine, Emmanuelle Noirrit-Esclassan, Frédéric Boudou, Melissa Buscato, Marine Adlanmerini, Florence Trémollières, Pierre Gourdy, Françoise Lenfant & Jean-François Arnal. (2019) Vers une optimisation de la modulation du récepteur des œstrogènes dans le traitement hormonal de la ménopause. médecine/sciences 34:12, pages 1056-1062.
Crossref
Crossref
Marie-Cécile Valéra, Emmanuelle Noirrit-Esclassan, Marion Dupuis, Coralie Fontaine, Françoise Lenfant, Anne Briaux, Cendrine Cabou, Cedric Garcia, Olivier Lairez, Jean-Michel Foidart, Bernard Payrastre & Jean-François Arnal. (2018) Effect of estetrol, a selective nuclear estrogen receptor modulator, in mouse models of arterial and venous thrombosis. Molecular and Cellular Endocrinology 477, pages 132-139.
Crossref
Crossref
Marie-Cécile Valéra, Coralie Fontaine, Marion Dupuis, Emmanuelle Noirrit-Esclassan, Alexia Vinel, Maeva Guillaume, Pierre Gourdy, Françoise Lenfant & Jean-François Arnal. (2018) Towards optimization of estrogen receptor modulation in medicine. Pharmacology & Therapeutics 189, pages 123-129.
Crossref
Crossref
I. V. Kuznetsova, L. V. Evsyukova & V. A. Konovalov. (2018) Combined oral contraception: is there a resource for increased use?. Medical Council:12, pages 146-151.
Crossref
Crossref
Herjan J.T. Coelingh Bennink, Carole Verhoeven, Yvette Zimmerman, Monique Visser, Jean-Michel Foidart & Kristina Gemzell-Danielsson. (2017) Pharmacodynamic effects of the fetal estrogen estetrol in postmenopausal women: results from a multiple-rising-dose study. Menopause 24:6, pages 677-685.
Crossref
Crossref
Gwenaël Nys, Anne Gallez, Miranda G.M. Kok, Gaël Cobraiville, Anne-Catherine Servais, Géraldine Piel, Christel Pequeux & Marianne Fillet. (2017) Whole blood microsampling for the quantitation of estetrol without derivatization by liquid chromatography-tandem mass spectrometry. Journal of Pharmaceutical and Biomedical Analysis 140, pages 258-265.
Crossref
Crossref
Herjan J.T. Coelingh Bennink, Carole Verhoeven, Yvette Zimmerman, Monique Visser, Jean-Michel Foidart & Kristina Gemzell-Danielsson. (2016) Clinical effects of the fetal estrogen estetrol in a multiple-rising-dose study in postmenopausal women. Maturitas 91, pages 93-100.
Crossref
Crossref
Maria Magdalena Montt-Guevara, Maria Silvia Giretti, Eleonora Russo, Andrea Giannini, Paolo Mannella, Andrea Riccardo Genazzani, Alessandro David Genazzani & Tommaso Simoncini. (2015) Estetrol Modulates Endothelial Nitric Oxide Synthesis in Human Endothelial Cells. Frontiers in Endocrinology 6.
Crossref
Crossref
N. Pluchino, P. Drakopoulos, E. Casarosa, L. Freschi, P. Petignat, M. Yaron & A.R. Genazzani. (2015) Effect of estetrol on Beta-Endorphin level in female rats. Steroids 95, pages 104-110.
Crossref
Crossref
C Gérard, S Blacher, L Communal, A Courtin, E Tskitishvili, M Mestdagt, C Munaut, A Noel, A Gompel, C Péqueux & J M Foidart. (2015) Estetrol is a weak estrogen antagonizing estradiol-dependent mammary gland proliferation. Journal of Endocrinology 224:1, pages 85-95.
Crossref
Crossref
C. F. Singer, H. J. T. C. Bennink, C. Natter, S. Steurer, M. Rudas, F. Moinfar, N. Appels, M. Visser & E. Kubista. (2014) Antiestrogenic effects of the fetal estrogen estetrol in women with estrogen-receptor positive early breast cancer. Carcinogenesis 35:11, pages 2447-2451.
Crossref
Crossref
Anne Abot, Coralie Fontaine, Mélissa Buscato, Romain Solinhac, Gilles Flouriot, Aurélie Fabre, Anne Drougard, Shyamala Rajan, Muriel Laine, Alain Milon, Isabelle Muller, Daniel Henrion, Marine Adlanmerini, Marie‐Cécile Valéra, Anne Gompel, Céline Gerard, Christel Péqueux, Mélanie Mestdagt, Isabelle Raymond‐Letron, Claude Knauf, François Ferriere, Philippe Valet, Pierre Gourdy, Benita S Katzenellenbogen, John A Katzenellenbogen, Françoise Lenfant, Geoffrey L Greene, Jean‐Michel Foidart & Jean‐François Arnal. (2014) The uterine and vascular actions of estetrol delineate a distinctive profile of estrogen receptor α modulation, uncoupling nuclear and membrane activation. EMBO Molecular Medicine 6:10, pages 1328-1346.
Crossref
Crossref
N. Pluchino, A.N. Santoro, E. Casarosa, A. Giannini, A. Genazzani, M. Russo, N. Russo, P. Petignat & A.R. Genazzani. (2014) Effect of estetrol administration on brain and serum allopregnanolone in intact and ovariectomized rats. The Journal of Steroid Biochemistry and Molecular Biology 143, pages 285-290.
Crossref
Crossref
Maria Silvia Giretti, Maria Magdalena Montt Guevara, Elena Cecchi, Paolo Mannella, Giulia Palla, Stefania Spina, Guja Bernacchi, Silvia Di Bello, Andrea Riccardo Genazzani, Alessandro D. Genazzani & Tommaso Simoncini. (2014) Effects of Estetrol on Migration and Invasion in T47-D Breast Cancer Cells through the Actin Cytoskeleton. Frontiers in Endocrinology 5.
Crossref
Crossref
Dana Seidlova-Wuttke, David Christel, Priya Kapur, Ba Tiep Nguyen, Hubertus Jarry & Wolfgang Wuttke. (2010) β-Ecdysone has bone protective but no estrogenic effects in ovariectomized rats. Phytomedicine 17:11, pages 884-889.
Crossref
Crossref
Monique Visser & Herjan J.T. Coelingh Bennink. (2009) Clinical applications for estetrol. The Journal of Steroid Biochemistry and Molecular Biology 114:1-2, pages 85-89.
Crossref
Crossref
Herjan J.T. Coelingh Bennink, Sven Skouby, Philippe Bouchard & Christian F. Holinka. (2008) Ovulation inhibition by estetrol in an in vivo model. Contraception 77:3, pages 186-190.
Crossref
Crossref