Advanced search
Publication Cover
Journal of Enzyme Inhibition and Medicinal Chemistry Volume 21, 2006 - Issue 4
Submit an article Journal homepage
948
Views
36
CrossRef citations to date
0
Altmetric
Research Article

PTP1B inhibitory activity of kaurane diterpenes isolated from Siegesbeckia glabrescens

Sohee Kim Korea Research Institute of Bioscience and Biotechnology (KRIBB), 52 Eoun-dong, Yuseong-gu, Daejeon, 305-333, KoreaSouth Korea
,
Minkyun Na Korea Research Institute of Bioscience and Biotechnology (KRIBB), 52 Eoun-dong, Yuseong-gu, Daejeon, 305-333, KoreaSouth Korea
,
Hyuncheol Oh MCBI & College of Natural Sciences, Silla University, San 1-1, Gwaebeop-dong, Sasang-gu, Busan, 617-736, KoreaSouth Korea
,
Junpil Jang Korea Research Institute of Bioscience and Biotechnology (KRIBB), 52 Eoun-dong, Yuseong-gu, Daejeon, 305-333, KoreaSouth Korea
,
Cheon Bae Sohn Department of Food and Nutrition, Chungnam National University, 220 Gung-dong, Yuseong-gu, Daejeon, 305-764, KoreaSouth Korea
,
Bo Yeon Kim Korea Research Institute of Bioscience and Biotechnology (KRIBB), 52 Eoun-dong, Yuseong-gu, Daejeon, 305-333, KoreaSouth Korea
,
Won Keun Oh Korea Research Institute of Bioscience and Biotechnology (KRIBB), 52 Eoun-dong, Yuseong-gu, Daejeon, 305-333, KoreaSouth Korea
&
Jong Seog Ahn Korea Research Institute of Bioscience and Biotechnology (KRIBB), 52 Eoun-dong, Yuseong-gu, Daejeon, 305-333, KoreaSouth Korea
 show all
Pages 379-383 | Received 08 Feb 2006, Accepted 10 Mar 2006, Published online: 04 Oct 2008

Citations (36)

Keep up to date with the latest research on this topic with citation updates for this article.

Subscribe to citation updates

Read on this site (3)

Jianbin Wang, Kehui Xie, Qing Wang, Wenchao Li & Hongzheng Fu. (2021) Isolation and characterization of ent-pimarane diterpenoids from Sigesbeckia pubescens. Natural Product Research 35:9, pages 1510-1517.
Read now
Akhilesh Kumar Tamrakar, Chandan K Maurya & Amit K Rai. (2014) PTP1B inhibitors for type 2 diabetes treatment: a patent review (2011 – 2014). Expert Opinion on Therapeutic Patents 24:10, pages 1101-1115.
Read now
Minkyun Na, Bo Yeon Kim, Hiroyuki Osada & Jong Seog Ahn. (2009) Inhibition of protein tyrosine phosphatase 1B by lupeol and lupenone isolated from Sorbus commixta. Journal of Enzyme Inhibition and Medicinal Chemistry 24:4, pages 1056-1059.
Read now

Articles from other publishers (33)

Adriana R. Dutra‐Nobre, Wesley J. Olivier, Bianca J. Deans, Nathan L. Kilah, Fernando Maya Alejandro, Jason A. Smith & Alex C. Bissember. (2023) Intraspecific Variation in the Terpene Profiles of Dodonaea viscosa . Asian Journal of Organic Chemistry 12:4.
Crossref
Aminu Mohammed, Nasir Tajuddeen, Mohammed Auwal Ibrahim, Murtala Bindawa Isah, Abubakar Babando Aliyu & Md. Shahidul Islam. (2022) Potential of diterpenes as antidiabetic agents: Evidence from clinical and pre-clinical studies. Pharmacological Research 179, pages 106158.
Crossref
Sukhbir Singh, Ajmer Singh Grewal, Rupanshi Grover, Neelam Sharma, Bhawna Chopra, Ashwani Kumar Dhingra, Sandeep Arora, Sonika Redhu & Viney Lather. (2022) Recent updates on development of protein-tyrosine phosphatase 1B inhibitors for treatment of diabetes, obesity and related disorders. Bioorganic Chemistry 121, pages 105626.
Crossref
Sudhakar Dattatray Tanpure, Tung-Chun Kuo, Mu-Jeng Cheng & Rai-Shung Liu. (2021) Gold(I)-Catalyzed Highly Diastereo- and Enantioselective Constructions of Bicyclo[3.2.1]oct-6-ene Frameworks via (4 + 3)-Cycloadditions. ACS Catalysis 12:1, pages 536-543.
Crossref
Qi Wang, Yi-Yu Liang, Kun-Wei Li, Ying Li, Feng-Jv Niu, Sheng-Jun Zhou, Hao-Cheng Wei & Chang-Zheng Zhou. (2021) Herba Siegesbeckiae: A review on its traditional uses, chemical constituents, pharmacological activities and clinical studies. Journal of Ethnopharmacology 275, pages 114117.
Crossref
Hong Xun Tao, Guan Ding Zhao, Ke Gang Linghu, Wei Xiong, Wei Sang, Yu Peng, Yitao Wang & Hua Yu. (2020) Botany, traditional use, phytochemistry, pharmacology and toxicology of Sigesbeckiae Herba (Xixiancao): a review. Phytochemistry Reviews 20:3, pages 569-587.
Crossref
Sun-Yup Shim, Ye Eun Lee & Mina Lee. (2021) Antioxidant Compounds, Kirenol and Methyl ent-16α, 17-dihydroxy-kauran-19-oate Bioactivity-Guided Isolated from Siegesbeckia glabrescens Attenuates MITF-Mediated Melanogenesis via Inhibition of Intracellular ROS Production. Molecules 26:7, pages 1940.
Crossref
Suchitra K. Panigrahy, Renu Bhatt & Awanish Kumar. (2020) Targeting type II diabetes with plant terpenes: the new and promising antidiabetic therapeutics. Biologia 76:1, pages 241-254.
Crossref
Muhammad Torequl Islam, Eunus S. Ali & Mohammad S. Mubarak. (2020) Anti‐obesity effect of plant diterpenes and their derivatives: A review. Phytotherapy Research 34:6, pages 1216-1225.
Crossref
Pranav K. Prabhakar & Ponnurengam M. Sivakumar. (2019) Protein Tyrosine Phosphatase 1B Inhibitors: A Novel Therapeutic Strategy for the Management of type 2 Diabetes Mellitus. Current Pharmaceutical Design 25:23, pages 2526-2539.
Crossref
Nguyen Van Quan, Tran Dang Xuan, Hoang-Dung Tran, Ateeque Ahmad, Tran Dang Khanh & Tran Dang Dat. (2019) Contribution of momilactones A and B to diabetes inhibitory potential of rice bran: Evidence from in vitro assays. Saudi Pharmaceutical Journal 27:5, pages 643-649.
Crossref
Phaedra Eleftheriou, Athina Geronikaki & Anthi Petrou. (2019) PTP1b Inhibition, A Promising Approach for the Treatment of Diabetes Type II. Current Topics in Medicinal Chemistry 19:4, pages 246-263.
Crossref
Bing Tian Zhao, Duc Hung Nguyen, Duc Dat Le, Jae Sue Choi, Byung Sun Min & Mi Hee Woo. (2017) Protein tyrosine phosphatase 1B inhibitors from natural sources. Archives of Pharmacal Research 41:2, pages 130-161.
Crossref
Da Hye Kim, Pradeep Paudel, Ting Yu, Thi Men Ngo, Jeong Ah Kim, Hyun Ah Jung, Takako Yokozawa & Jae Sue Choi. (2017) Characterization of the inhibitory activity of natural tanshinones from Salvia miltiorrhiza roots on protein tyrosine phosphatase 1B. Chemico-Biological Interactions 278, pages 65-73.
Crossref
Qing-Qing Yuan, Wei-Bin Song, Wen-Qiong Wang, Jiao-Jiao Wei, Jun Li, Yi Liu & Li-Jiang Xuan. (2017) New ent -kaurane and ent -pimarane diterpenoids from Siegesbeckia pubescens. Phytochemistry Letters 21, pages 273-277.
Crossref
Qiao-Qiao Tao, Ke Ma, Li Bao, Kai Wang, Jun-Jie Han, Jin-Xia Zhang, Chen-Yang Huang & Hong-Wei Liu. (2016) New sesquiterpenoids from the edible mushroom Pleurotus cystidiosus and their inhibitory activity against α-glucosidase and PTP1B. Fitoterapia 111, pages 29-35.
Crossref
Chang-Ling Hu, Juan Xiong, Li-Xin Gao, Jia Li, Huaqiang Zeng, Yike Zou & Jin-Feng Hu. (2016) Diterpenoids from the shed trunk barks of the endangered plant Pinus dabeshanensis and their PTP1B inhibitory effects. RSC Advances 6:65, pages 60467-60478.
Crossref
Shoaib Ahmad. 2006. Reviews in Cell Biology and Molecular Medicine. Reviews in Cell Biology and Molecular Medicine 276 309 .
Qian Wu, Hua Li, So Lee, Hwa Lee & Jae-Ha Ryu. (2015) New Cytotoxic Sesquiterpenoids from Siegesbeckia glabrescens. Molecules 20:2, pages 2850-2856.
Crossref
Jacqueline Takahashi, Dhionne Gomes, Fernanda Lyra, Gabriel dos Santos & Leonardo Martins. (2014) The Remarkable Structural Diversity Achieved in ent-Kaurane Diterpenes by Fungal Biotransformations. Molecules 19:2, pages 1856-1886.
Crossref
Kyungjin Lee, Jinho Jung, Gabsik Yang, Inhye Ham, Youngmin Bu, Hocheol Kim & Ho‐Young Choi. (2012) Endothelium‐Independent Vasorelaxation Effects of Sigesbeckia glabrescens (Makino) Makino on Isolated Rat Thoracic Aorta . Phytotherapy Research 27:9, pages 1308-1312.
Crossref
Hyun Ah Jung, Yoon Sook Cho, Sang Ho Oh, Sanghyuk Lee, Byung-Sun Min, Kyung Ho Moon & Jae Sue Choi. (2013) Kinetics and molecular docking studies of pimarane-type diterpenes as protein tyrosine phosphatase (PTP1B) inhibitors from Aralia continentalis roots. Archives of Pharmacal Research 36:8, pages 957-965.
Crossref
Cheng-shi Jiang, Lin-fu Liang & Yue-wei Guo. (2012) Natural products possessing protein tyrosine phosphatase 1B (PTP1B) inhibitory activity found in the last decades. Acta Pharmacologica Sinica 33:10, pages 1217-1245.
Crossref
Hee Jin Jung, Hyun Ah Jung, Sam Sik Kang, Je-Hyun Lee, Yoon Sook Cho, Kyong Ho Moon & Jae Sue Choi. (2012) Inhibitory activity of Aralia continentalis roots on protein tyrosine phosphatase 1B and rat lens aldose reductase. Archives of Pharmacal Research 35:10, pages 1771-1777.
Crossref
Suresh Thareja, Saurabh Aggarwal, T. R. Bhardwaj & Manoj Kumar. (2010) Protein Tyrosine Phosphatase 1B Inhibitors: A Molecular Level Legitimate Approach for the Management of Diabetes Mellitus. Medicinal Research Reviews 32:3, pages 459-517.
Crossref
Ya Li, Tong-Tong Wang, Jie Zhao, Xiang Shi, Shu-Chen Hu & Kun Gao. (2012) Norditerpenoids from Agathis macrophylla. Food Chemistry 131:3, pages 972-976.
Crossref
S.-H. Sung, S.-H. Park, S.-Y. Song, S.-J. Lee, H.-W. Lee, S.-H. Kim, M. A Lee, I.-S. Yoon, D.-D. Kim, S. Kang & J.-H. Sung. (2011) Epidermal regeneration by ent-16α, 17-dihydroxy-kauran-19-oic acid isolated from Siegesbeckia pubescens. Cell Proliferation 44:6, pages 527-536.
Crossref
Hua Li, Jae Yeon Kim, Jinseong Hyeon, Hwa Jin Lee & Jae‐Ha Ryu. (2011) In Vitro Antiinflammatory Activity of a New Sesquiterpene Lactone Isolated from Siegesbeckia glabrescens . Phytotherapy Research 25:9, pages 1323-1327.
Crossref
Ran Joo Choi, Eun Myoung Shin, Hyun Ah Jung, Jae Sue Choi & Yeong Shik Kim. (2011) Inhibitory effects of kaurenoic acid from Aralia continentalis on LPS-induced inflammatory response in RAW264.7 macrophages. Phytomedicine 18:8-9, pages 677-682.
Crossref
Zhen Jiang, Qing-Hong Yu, Yan Cheng & Xing-Jie Guo. (2011) Simultaneous quantification of eight major constituents in Herba Siegesbeckiae by liquid chromatography coupled with electrospray ionization time-of-flight tandem mass spectrometry. Journal of Pharmaceutical and Biomedical Analysis 55:3, pages 452-457.
Crossref
Hyun Ah Jung, Eun Ju Lee, Ju Sun Kim, Sam Sik Kang, Je-Hyun Lee, Byung-Sun Min & Jae Sue Choi. (2009) Cholinesterase and BACE1 inhibitory diterpenoids from Aralia cordata. Archives of Pharmacal Research 32:10, pages 1399-1408.
Crossref
JunPil JangMinKyun NaPhuong Thien Thuong, Dieudonné Njamen, Joseph Tanyi Mbafor, Zacharias Tanee Fomum, Eun-Rhan Woo & Won Keun Oh. (2008) Prenylated Flavonoids with PTP1B Inhibitory Activity from the Root Bark of Erythrina mildbraedii. Chemical and Pharmaceutical Bulletin 56:1, pages 85-88.
Crossref
Pablo Garcia, Alaide De Oliveira & Ronan Batista. (2007) Occurrence, Biological Activities and Synthesis of Kaurane Diterpenes and their Glycosides. Molecules 12:3, pages 455-483.
Crossref

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Order Reprints Request Corporate Permissions

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

Request Academic Permissions

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.

Related research

People also read lists articles that other readers of this article have read.

Recommended articles lists articles that we recommend and is powered by our AI driven recommendation engine.

Cited by lists all citing articles based on Crossref citations.
Articles with the Crossref icon will open in a new tab.