Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 21, Issue 4 (2006)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 21, Issue 4 (2006)

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Research Article

Article
Novel tight binding PETT, HEPT and DABO-based non-nucleoside inhibitors of HIV-1 reverse transcriptase
Review
Osmond J. D'cruz & Fatih M. Uckun
Pages: 329-350
Published online: 04 Oct 2008
AbstractforNovel tight binding PETT, HEPT and DABO-based non-nucleoside inhibitors of HIV-1 reverse transcriptase | Full Text | References | PDF (1.1 MB)
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Article
Carbonic anhydrase inhibitors. Inhibition of human tumor-associated isozymes IX and cytosolic isozymes I and II with some 1,3,4-oxadiazole-thiols
Muhammad Zareef, Alessio Innocenti, Rashid Iqbal, Javid H. Zaidi, Muhammad Arfan, Andrea Scozzafava & Claudiu T. Supuran
Pages: 351-359
Published online: 04 Oct 2008
AbstractforCarbonic anhydrase inhibitors. Inhibition of human tumor-associated isozymes IX and cytosolic isozymes I and II with some 1,3,4-oxadiazole-thiols | Full Text | References | PDF (184.7 KB)
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Article
Homology Model of Human Retinoic Acid Metabolising Enzyme Cytochrome P450 26A1 (CYP26A1): Active Site Architecture and Ligand Binding
Mohamed Sayed Gomaa, Sook Wah Yee, Ceri Elizabeth Milbourne, Maria Chiara Barbera, Claire Simons & Andrea Brancale
Pages: 361-369
Published online: 04 Oct 2008
AbstractforHomology Model of Human Retinoic Acid Metabolising Enzyme Cytochrome P450 26A1 (CYP26A1): Active Site Architecture and Ligand Binding | Full Text | References | PDF (678.3 KB)
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Article
New progesterone derivatives as inhibitors of 5α-reductase enzyme and prostate cancer cell growth
Marisa Cabeza, Eugene Bratoeff, Ivonne Heuze, Arely Rojas, Nayely Terán, Martha' Ochoa, Ma Teresa Ramírez-Apan, Elena Ramírez, Victor Pérez & Isabel Gracia
Pages: 371-378
Published online: 04 Oct 2008
AbstractforNew progesterone derivatives as inhibitors of 5α-reductase enzyme and prostate cancer cell growth | Full Text | References | PDF (199.7 KB)
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Article
PTP1B inhibitory activity of kaurane diterpenes isolated from Siegesbeckia glabrescens
Sohee Kim, Minkyun Na, Hyuncheol Oh, Junpil Jang, Cheon Bae Sohn, Bo Yeon Kim, Won Keun Oh & Jong Seog Ahn
Pages: 379-383
Published online: 04 Oct 2008
AbstractforPTP1B inhibitory activity of kaurane diterpenes isolated from Siegesbeckia glabrescens | Full Text | References | PDF (115.4 KB)
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Article
Lipophilicity Relationships in Inhibitors of CYP2C9 and CYP2C19 Enzymes
David F.V. Lewis, Brian G. Lake, Yuko Ito & Maurice Dickins
Pages: 385-389
Published online: 04 Oct 2008
AbstractforLipophilicity Relationships in Inhibitors of CYP2C9 and CYP2C19 Enzymes | Full Text | References | PDF (120.1 KB)
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Article
New lipophilic phthalimido- and 3-phenoxybenzyl sulfonates: Inhibition of antigen 85C mycolyltransferase activity and cytotoxicity
Andreja Kovač, Rosalind A. Wilson, Gurdyal S. Besra, Metka Filipič, Danijel Kikelj & Stanislav Gobec
Pages: 391-397
Published online: 04 Oct 2008
AbstractforNew lipophilic phthalimido- and 3-phenoxybenzyl sulfonates: Inhibition of antigen 85C mycolyltransferase activity and cytotoxicity | Full Text | References | PDF (124.5 KB)
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Article
Synthesis and antioxidant evaluation of novel silybin analogues
Leixiang Yang, Jingxu Gong, Feng Wang, Yongmin Zhang, Yanguang Wang, Xiaojiang Hao, Xiumei Wu, Hua Bai, Joachim Stöckigt & Yu Zhao
Pages: 399-404
Published online: 04 Oct 2008
AbstractforSynthesis and antioxidant evaluation of novel silybin analogues | Full Text | References | PDF (179 KB)
  • 668 Views
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Article
Investigation of the in vitro antioxidant behaviour of some 2-phenylindole derivatives: discussion on possible antioxidant mechanisms and comparison with melatonin
Sibel Suzen, Pinar Bozkaya, Tulay Coban & Doğu Nebioğlu
Pages: 405-411
Published online: 04 Oct 2008
AbstractforInvestigation of the in vitro antioxidant behaviour of some 2-phenylindole derivatives: discussion on possible antioxidant mechanisms and comparison with melatonin | Full Text | References | PDF (187.3 KB)
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Article
Inhibitory effects of fluorobenzaldehydes on the activity of mushroom tyrosinase
Xiao-Hong Huang, Qing-Xi Chen, Min-sheng You, Qin Wang, Kang-Kang Song, Jun Wang, Li Sha & Xiong Guan
Pages: 413-418
Published online: 04 Oct 2008
AbstractforInhibitory effects of fluorobenzaldehydes on the activity of mushroom tyrosinase | Full Text | References | PDF (100.1 KB)
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Article
Differential effects of flavonoids on bovine kidney low molecular mass protein tyrosine phosphatase
Márcio A. Miranda, André K. Okamoto, Carmen V. Ferreira, Thelma L. Silva, José M. Granjeiro & Hiroshi Aoyama
Pages: 419-425
Published online: 04 Oct 2008
AbstractforDifferential effects of flavonoids on bovine kidney low molecular mass protein tyrosine phosphatase | Full Text | References | PDF (224.6 KB)
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Article
Tests with Daphnia magna: A new approach to prescreen toxicity of newly synthesized acetylcholinesterase reactivators
Sarka Vesela, Vlastimil Ondruska, Kamil Kuca & Jiri Patocka
Pages: 427-432
Published online: 04 Oct 2008
AbstractforTests with Daphnia magna: A new approach to prescreen toxicity of newly synthesized acetylcholinesterase reactivators | Full Text | References | PDF (197.4 KB)
  • 701 Views
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Article
Purification and characterisation of an inhibitor of a cathepsin B-like proteinase from sunflower seed
Xin-Chang Zhang, Hong-Lian Shao, Jin-Xing Wang & Xiao-Fan Zhao
Pages: 433-439
Published online: 04 Oct 2008
AbstractforPurification and characterisation of an inhibitor of a cathepsin B-like proteinase from sunflower seed | Full Text | References | PDF (250.9 KB)
  • 558 Views
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Article
Metalloantibiotics: Synthesis, characterization and in-vitro antibacterial studies on cobalt (ii), copper (ii), nickel (ii) and zinc (ii) complexes with cloxacillin
Zahid H. Chohan & Claudiu T. Supuran
Pages: 441-448
Published online: 04 Oct 2008
AbstractforMetalloantibiotics: Synthesis, characterization and in-vitro antibacterial studies on cobalt (ii), copper (ii), nickel (ii) and zinc (ii) complexes with cloxacillin | Full Text | References | PDF (155.8 KB)
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Article
Inhibition activities of colchicum luteum baker on lipoxygenase and other enzymes
Bashir Ahmad, Haroon Khan, Shumaila Bashir, M. Nisar & M. Hassan
Pages: 449-452
Published online: 04 Oct 2008
AbstractforInhibition activities of colchicum luteum baker on lipoxygenase and other enzymes | Full Text | References | PDF (103.6 KB)
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Article
In-vitro biological evaluation of some ONS and NS donor Schiff's bases and their metal complexes
Pragnesh K. Panchal, Pramod B. Pansuriya & M. N. Patel
Pages: 453-458
Published online: 04 Oct 2008
AbstractforIn-vitro biological evaluation of some ONS and NS donor Schiff's bases and their metal complexes | Full Text | References | PDF (191.2 KB)
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Article
Interaction of some Pd(II) complexes with Na+/K+-ATPase: Inhibition, kinetics, prevention and recovery
Katarina S. Krinulović & Vesna M. Vasić
Pages: 459-465
Published online: 04 Oct 2008
AbstractforInteraction of some Pd(II) complexes with Na+/K+-ATPase: Inhibition, kinetics, prevention and recovery | Full Text | References | PDF (249.3 KB)
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Article
Boric acid and boronic acids inhibition of pigeonpea urease
K. Ravi Charan Reddy & Arvind M. Kayastha
Pages: 467-470
Published online: 04 Oct 2008
AbstractforBoric acid and boronic acids inhibition of pigeonpea urease | Full Text | References | PDF (126.7 KB)
  • 1073 Views
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Article
The influence of potassium ion (K+) on digoxin-induced inhibition of porcine cerebral cortex Na+/K+-ATPase
Danijela Krstić, Nenad Tomić, Katarina Krinulović & Vesna Vasić
Pages: 471-475
Published online: 04 Oct 2008
AbstractforThe influence of potassium ion (K+) on digoxin-induced inhibition of porcine cerebral cortex Na+/K+-ATPase | Full Text | References | PDF (89.7 KB)
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Article
Carbonic anhydrase inhibitors. N-Cyanomethylsulfonamides—a new zinc binding group in the design of inhibitors targeting cytosolic and membrane-anchored isoforms
Jean-Yves Winum, Alessandro Cecchi, Achour Seridi, Andrea Scozzafava, Jean-Louis Montero & Claudiu T. Supuran
Pages: 477-481
Published online: 04 Oct 2008
AbstractforCarbonic anhydrase inhibitors. N-Cyanomethylsulfonamides—a new zinc binding group in the design of inhibitors targeting cytosolic and membrane-anchored isoforms | Full Text | References | PDF (80.4 KB)
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