Citations (49)
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Mateusz Kciuk, Adrianna Gielecińska, Somdutt Mujwar, Mariusz Mojzych, Beata Marciniak, Rafał Drozda & Renata Kontek. (2022) Targeting carbonic anhydrase IX and XII isoforms with small molecule inhibitors and monoclonal antibodies. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 1278-1298.
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Alessio Nocentini, Andrea Angeli, Fabrizio Carta, Jean-Yves Winum, Raivis Zalubovskis, Simone Carradori, Clemente Capasso, William A. Donald & Claudiu T. Supuran. (2021) Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 561-580.
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Claudiu T Supuran. (2020) Experimental Carbonic Anhydrase Inhibitors for the Treatment of Hypoxic Tumors. Journal of Experimental Pharmacology 12, pages 603-617.
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Claudiu T. Supuran. (2020) An update on drug interaction considerations in the therapeutic use of carbonic anhydrase inhibitors. Expert Opinion on Drug Metabolism & Toxicology 16:4, pages 297-307.
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Silvia Peppicelli, Elena Andreucci, Jessica Ruzzolini, Francesca Bianchini, Chiara Nediani, Claudiu T. Supuran & Lido Calorini. (2020) The Carbonic Anhydrase IX inhibitor SLC-0111 as emerging agent against the mesenchymal stem cell-derived pro-survival effects on melanoma cells. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1185-1193.
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Emanuela Berrino & Claudiu T. Supuran. (2019) Novel approaches for designing drugs that interfere with pH regulation. Expert Opinion on Drug Discovery 14:3, pages 231-248.
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Mariantonia Logozzi, Clemente Capasso, Rossella Di Raimo, Sonia Del Prete, Davide Mizzoni, Mario Falchi, Claudiu T. Supuran & Stefano Fais. (2019) Prostate cancer cells and exosomes in acidic condition show increased carbonic anhydrase IX expression and activity. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 272-278.
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Claudiu T. Supuran. (2018) Carbonic anhydrase inhibitors as emerging agents for the treatment and imaging of hypoxic tumors. Expert Opinion on Investigational Drugs 27:12, pages 963-970.
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Özlen Güzel-Akdemir, Andrea Angeli, Kübra Demir, Claudiu T. Supuran & Atilla Akdemir. (2018) Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 1299-1308.
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Morteza Abdoli, Andrea Angeli, Murat Bozdag, Fabrizio Carta, Ali Kakanejadifard, Hamid Saeidian & Claudiu T. Supuran. (2017) Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo[d]thiazole-5- and 6-sulfonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1071-1078.
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Murat Bozdag, Silvia Bua, Sameh M. Osman, Zeid AlOthman & Claudiu T. Supuran. (2017) Carbonic anhydrase I, II, IV and IX inhibition with a series of 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 885-892.
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Zhengxing Zhang, Joseph Lau, Chengcheng Zhang, Nadine Colpo, Alessio Nocentini, Claudiu T. Supuran, François Bénard & Kuo-Shyan Lin. (2017) Design, synthesis and evaluation of 18F-labeled cationic carbonic anhydrase IX inhibitors for PET imaging. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 722-730.
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Marco Bragagni, Fabrizio Carta, Sameh M. Osman, Zeid AlOthman & Claudiu T. Supuran. (2017) Synthesis of an acridine orange sulfonamide derivative with potent carbonic anhydrase IX inhibitory action. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 701-706.
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Articles from other publishers (36)
Rong A, Haoyu Wang, Chaoqun Nie, Zhaoguo Han, Meifang Zhou, Olagbaju Oluwatosin Atinuke, Kaiqi Wang, Xiance Wang, Shuang Liu, Jingshi Zhao, Wenju Qiao, Xiaohong Sun, Lina Wu & Xilin Sun. (2023) Glycerol-weighted chemical exchange saturation transfer nanoprobes allow 19F/1H dual-modality magnetic resonance imaging-guided cancer radiotherapy. Nature Communications 14:1.
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Jing Cui, Huizhe Xu, Ji Shi, Kun Fang, Jia Liu, Feng Liu, Yi Chen, Haiyang Liang, Ye Zhang & Haozhe Piao. (2023) Carbonic anhydrase IX inhibitor S4 triggers release of DAMPs related to immunogenic cell death in glioma cells via endoplasmic reticulum stress pathway. Cell Communication and Signaling 21:1.
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Reham M. M. El-Hazek, Nashwa H. Zaher, Hagar E. S. Emam, Marwa G. El-Gazzar & Amira Khalil. (2023) Pyrazole-sulfonamide scaffold featuring dual-tail strategy as apoptosis inducers in colon cancer. Scientific Reports 13:1.
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Marta Venturella, Alessandro Falsini, Federica Coppola, Gaia Giuntini, Fabio Carraro, Davide Zocco, Antonio Chiesi & Antonella Naldini. (2023) CA-IX-Expressing Small Extracellular Vesicles (sEVs) Are Released by Melanoma Cells under Hypoxia and in the Blood of Advanced Melanoma Patients. International Journal of Molecular Sciences 24:7, pages 6122.
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Tomas Koltai, Larry Fliegel, Fátima Baltazar, Stephan J. Reshkin, Khalid O. Alfarouk, Rosa Angela Cardone & Julieta Afonso. 2023. pH Deregulation as the Eleventh Hallmark of Cancer. pH Deregulation as the Eleventh Hallmark of Cancer
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Alessandro Giuliani & Stefano Fais. (2022) Proposal to Consider Chemical/Physical Microenvironment as a New Therapeutic Off-Target Approach. Pharmaceutics 14:10, pages 2084.
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Ying Li, Ju Zhang, Jie Xu & Shanglong Liu. (2021) The Metabolism Symbiosis Between Pancreatic Cancer and Tumor Microenvironment. Frontiers in Oncology 11.
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Stanislav Kalinin, Anna Malkova, Tatiana Sharonova, Vladimir Sharoyko, Alexander Bunev, Claudiu T. Supuran & Mikhail Krasavin. (2021) Carbonic Anhydrase IX Inhibitors as Candidates for Combination Therapy of Solid Tumors. International Journal of Molecular Sciences 22:24, pages 13405.
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Wen Li, Baofang Zhang & Zilin Chen. (2021) Screening carbonic anhydrase IX inhibitors in traditional Chinese medicine based on electrophoretically mediated microanalysis. Talanta 232, pages 122444.
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Sonia E. Trojan, Paulina Dudzik, Justyna Totoń-Żurańska, Piotr Laidler & Kinga A. Kocemba-Pilarczyk. (2021) Expression of Alternative Splice Variants of 6-Phosphofructo-2-kinase/Fructose-2,6-bisphosphatase-4 in Normoxic and Hypoxic Melanoma Cells. International Journal of Molecular Sciences 22:16, pages 8848.
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Edgar Pérez-Herrero & Alberto Fernández-Medarde. (2021) The reversed intra- and extracellular pH in tumors as a unified strategy to chemotherapeutic delivery using targeted nanocarriers. Acta Pharmaceutica Sinica B 11:8, pages 2243-2264.
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Zhoulei Li, Peng He, Yali Long, Gang Yuan, Wanqing Shen, Zhifeng Chen, Bing Zhang, Yue Wang, Dianchao Yue, Christof Seidl & Xiangsong Zhang. (2021) Drug Repurposing of Pantoprazole and Vitamin C Targeting Tumor Microenvironment Conditions Improves Anticancer Effect in Metastatic Castration-Resistant Prostate Cancer. Frontiers in Oncology 11.
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Justina Kazokaitė-Adomaitienė, Holger M. Becker, Joana Smirnovienė, Ludwig J. Dubois & Daumantas Matulis. (2021) Experimental Approaches to Identify Selective Picomolar Inhibitors for Carbonic Anhydrase IX. Current Medicinal Chemistry 28:17, pages 3361-3384.
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Shiori Hiromoto, Takehiro Kawashiri, Natsumi Yamanaka, Daisuke Kobayashi, Keisuke Mine, Mizuki Inoue, Mayako Uchida & Takao Shimazoe. (2021) Use of omeprazole, the proton pump inhibitor, as a potential therapy for the capecitabine-induced hand-foot syndrome. Scientific Reports 11:1.
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Peter W. Halcrow, Jonathan D. Geiger & Xuesong Chen. (2021) Overcoming Chemoresistance: Altering pH of Cellular Compartments by Chloroquine and Hydroxychloroquine. Frontiers in Cell and Developmental Biology 9.
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Tomas Koltai, Stephan J. Reshkin, Fátima Baltazar & Larry Fliegel. 2021. Prostate Cancer Metabolism. Prostate Cancer Metabolism
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Tomas Koltai. (2020) Targeting the pH Paradigm at the Bedside: A Practical Approach. International Journal of Molecular Sciences 21:23, pages 9221.
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Lisa Annabel Weber, Anne Funtan, Reinhard Paschke, Julien Delarocque, Jutta Kalbitz, Jessica Meißner, Karsten Feige, Manfred Kietzmann & Jessika-Maximiliane V. Cavalleri. (2020) In vitro assessment of triterpenoids NVX-207 and betulinyl-bis-sulfamate as a topical treatment for equine skin cancer. PLOS ONE 15:11, pages e0241448.
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Stefano Fais & Yoshinori Marunaka. (2020) The Acidic Microenvironment: Is It a Phenotype of All Cancers? A Focus on Multiple Myeloma and Some Analogies with Diabetes Mellitus. Cancers 12:11, pages 3226.
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Andrea Angeli, Fabrizio Carta, Alessio Nocentini, Jean-Yves Winum, Raivis Zalubovskis, Atilla Akdemir, Valentina Onnis, Wagdy M. Eldehna, Clemente Capasso, Giuseppina De Simone, Simona Maria Monti, Simone Carradori, William A. Donald, Shoukat Dedhar & Claudiu T. Supuran. (2020) Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment. Metabolites 10:10, pages 412.
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Salvador Harguindey, Khalid Alfarouk, Julián Polo Orozco, Stefano Fais & Jesús Devesa. (2020) Towards an Integral Therapeutic Protocol for Breast Cancer Based upon the New H+-Centered Anticancer Paradigm of the Late Post-Warburg Era. International Journal of Molecular Sciences 21:20, pages 7475.
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Stefano Burgio, Leila Noori, Antonella Marino Gammazza, Claudia Campanella, Mariantonia Logozzi, Stefano Fais, Fabio Bucchieri, Francesco Cappello & Celeste Caruso Bavisotto. (2020) Extracellular Vesicles-Based Drug Delivery Systems: A New Challenge and the Exemplum of Malignant Pleural Mesothelioma. International Journal of Molecular Sciences 21:15, pages 5432.
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Tomas Koltai, Stephan J. Reshkin & Salvador Harguindey. 2020. An Innovative Approach to Understanding and Treating Cancer: Targeting pH. An Innovative Approach to Understanding and Treating Cancer: Targeting pH
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Kaye J. Williams & Roben G. Gieling. (2019) Preclinical Evaluation of Ureidosulfamate Carbonic Anhydrase IX/XII Inhibitors in the Treatment of Cancers. International Journal of Molecular Sciences 20:23, pages 6080.
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Alberto Foletti & Stefano Fais. (2019) Unexpected Discoveries Should Be Reconsidered in Science—A Look to the Past?. International Journal of Molecular Sciences 20:16, pages 3973.
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Mariantonia Logozzi, Enrico Spugnini, Davide Mizzoni, Rossella Di Raimo & Stefano Fais. (2019) Extracellular acidity and increased exosome release as key phenotypes of malignant tumors. Cancer and Metastasis Reviews 38:1-2, pages 93-101.
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A. Koch & A. Schwab. (2019) Cutaneous pH landscape as a facilitator of melanoma initiation and progression. Acta Physiologica 225:1, pages e13105.
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Justina Kazokaitė, Holger M. Becker, Harlan R. Barker, Ashok Aspatwar, Seppo Parkkila, Ludwig J. Dubois & Daumantas Matulis. 2019. Carbonic Anhydrase as Drug Target. Carbonic Anhydrase as Drug Target
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Antonio Mazzocca, Giovanni Ferraro, Giovanni Misciagna & Stefano Fais. (2018) Moving the systemic evolutionary approach to cancer forward: Therapeutic implications. Medical Hypotheses 121, pages 80-87.
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Claudiu Supuran. (2018) Carbonic Anhydrases and Metabolism. Metabolites 8:2, pages 25.
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Elisabetta Iessi, Mariantonia Logozzi, Davide Mizzoni, Rossella Di Raimo, Claudiu Supuran & Stefano Fais. (2017) Rethinking the Combination of Proton Exchanger Inhibitors in Cancer Therapy. Metabolites 8:1, pages 2.
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Claudiu T. Supuran. (2017) Carbonic Anhydrase Inhibition and the Management of Hypoxic Tumors. Metabolites 7:3, pages 48.
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Enrica Balza, Patrizia Castellani, Paola Sanchez Moreno, Patrizia Piccioli, Iria Medraño-Fernandez, Claudia Semino & Anna Rubartelli. (2017) Restoring microenvironmental redox and pH homeostasis inhibits neoplastic cell growth and migration: therapeutic efficacy of esomeprazole plus sulfasalazine on 3-MCA-induced sarcoma. Oncotarget 8:40, pages 67482-67496.
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Suleyman Akocak, Nabih Lolak, Alessio Nocentini, Gulcin Karakoc, Anzel Tufan & Claudiu T. Supuran. (2017) Synthesis and biological evaluation of novel aromatic and heterocyclic bis-sulfonamide Schiff bases as carbonic anhydrase I, II, VII and IX inhibitors. Bioorganic & Medicinal Chemistry 25:12, pages 3093-3097.
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