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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 33, 2018 - Issue 1
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Research Paper

Carbonic anhydrase inhibition with a series of novel benzenesulfonamide-triazole conjugates

Marwa G. El-GazzarDepartment of Drug Radiation Research, National Center for Radiation Research and Technology (NCRRT), Egyptian Atomic Energy Authority (EAEA), Cairo, Egypt; Correspondence[email protected]
,
Nessma H. NafieDepartment of Drug Radiation Research, National Center for Radiation Research and Technology (NCRRT), Egyptian Atomic Energy Authority (EAEA), Cairo, Egypt;
,
Alessio NocentiniNEUROFARBA Department, Pharmaceutical and Nutraceutical Sciences Section, University of Florence, Firenze, Italy
,
Mostafa M. GhorabDepartment of Drug Radiation Research, National Center for Radiation Research and Technology (NCRRT), Egyptian Atomic Energy Authority (EAEA), Cairo, Egypt;
,
Helmi I. HeibaDepartment of Drug Radiation Research, National Center for Radiation Research and Technology (NCRRT), Egyptian Atomic Energy Authority (EAEA), Cairo, Egypt;
&
Claudiu T. SupuranNEUROFARBA Department, Pharmaceutical and Nutraceutical Sciences Section, University of Florence, Firenze, ItalyCorrespondence[email protected]
ORCID Iconhttp://orcid.org/0000-0003-4262-0323
ORCID Icon
Pages 1565-1574 | Received 27 Jul 2018, Accepted 16 Aug 2018, Published online: 02 Oct 2018

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Paolo Guglielmi, Giulia Rotondi, Daniela Secci, Andrea Angeli, Paola Chimenti, Alessio Nocentini, Alessandro Bonardi, Paola Gratteri, Simone Carradori & Claudiu T. Supuran. (2020) Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1891-1905.
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Jeremie Brichet, Rodrigo Arancibia, Emanuela Berrino & Claudiu T. Supuran. (2020) Bioorganometallic derivatives of 4-hydrazino-benzenesulphonamide as carbonic anhydrase inhibitors: synthesis, characterisation and biological evaluation. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 622-628.
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Aleksandrs Pustenko, Alessio Nocentini, Anastasija Balašova, Mikhail Krasavin, Raivis Žalubovskis & Claudiu T. Supuran. (2020) 7-Acylamino-3H-1,2-benzoxathiepine 2,2-dioxides as new isoform-selective carbonic anhydrase IX and XII inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 650-656.
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Rakia Abd Alhameed, Emanuela Berrino, Zainab Almarhoon, Ayman El-Faham & Claudiu T. Supuran. (2020) A class of carbonic anhydrase IX/XII – selective carboxylate inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 549-554.
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Benedetta Fois, Simona Distinto, Rita Meleddu, Serenella Deplano, Elias Maccioni, Costantino Floris, Antonella Rosa, Mariella Nieddu, Pierluigi Caboni, Claudia Sissi, Andrea Angeli, Claudiu T. Supuran & Filippo Cottiglia. (2020) Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 539-548.
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Siham A. Alissa, Hanan A. Alghulikah, Zeid A. ALOthman, Sameh M. Osman, Sonia Del Prete, Clemente Capasso, Alessio Nocentini & Claudiu T. Supuran. (2020) Inhibition survey with phenolic compounds against the δ- and η-class carbonic anhydrases from the marine diatom thalassiosira weissflogii and protozoan Plasmodium falciparum. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 377-382.
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Ali Irfan, Fozia Batool, Syeda Andleeb Zahra Naqvi, Amjad Islam, Sameh M. Osman, Alessio Nocentini, Siham A. Alissa & Claudiu T. Supuran. (2020) Benzothiazole derivatives as anticancer agents. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 265-279.
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Siham A. Alissa, Hanan A. Alghulikah, Zeid A. Alothman, Sameh M. Osman, Sonia Del Prete, Clemente Capasso, Alessio Nocentini & Claudiu T. Supuran. (2020) Phosphonamidates are the first phosphorus-based zinc binding motif to show inhibition of β-class carbonic anhydrases from bacteria, fungi, and protozoa. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 59-64.
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Suleyman Akocak, Nabih Lolak, Silvia Bua, Alessio Nocentini & Claudiu T. Supuran. (2019) Activation of human α-carbonic anhydrase isoforms I, II, IV and VII with bis-histamine schiff bases and bis-spinaceamine substituted derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1193-1198.
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Baijayantimala Swain, Andrea Angeli, Srinivas Angapelly, Pavitra S. Thacker, Priti Singh, Claudiu T. Supuran & Mohammed Arifuddin. (2019) Synthesis of a new series of 3-functionalised-1-phenyl-1,2,3-triazole sulfamoylbenzamides as carbonic anhydrase I, II, IV and IX inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1199-1209.
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Reihane Ghomashi, Shakila Ghomashi, Hamidreza Aghaei, Samineh Massah & Ahmad Reza Massah. (2023) Recent Advances in Biological Active Sulfonamide based Hybrid Compounds Part C: Multicomponent Sulfonamide Hybrids. Current Medicinal Chemistry 30:37, pages 4181-4255.
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Chander, Monika, Pawan K. Sharma & Sita Ram. (2023) Recent advances in triazole-benzenesulfonamide hybrids and their biological activities. Medicinal Chemistry Research 32:5, pages 777-801.
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Serghei Pogrebnoi, Oleg Radul, Eugenia Stingaci, Lucian Lupascu, Vladimir Valica, Livia Uncu, Anastasia Smetanscaia, Anthi Petrou, Ana Ćirić, Jasmina Glamočlija, Marina Soković, Athina Geronikaki & Fliur Z. Macaev. (2022) The Synthesis of Triazolium Salts as Antifungal Agents: A Biological and In Silico Evaluation. Antibiotics 11:5, pages 588.
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Ali Irfan, Sajjad Ahmad, Saddam Hussain, Fozia Batool, Haseeba Riaz, Rehman Zafar, Katarzyna Kotwica-Mojzych & Mariusz Mojzych. (2021) Recent Updates on the Synthesis of Bioactive Quinoxaline-Containing Sulfonamides. Applied Sciences 11:12, pages 5702.
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S. A. El‐Sebaey. (2020) Recent Advances in 1,2,4‐Triazole Scaffolds as Antiviral Agents. ChemistrySelect 5:37, pages 11654-11680.
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Ahmed H. Halawa, Walid E. Elgammal, Saber M. Hassan, Ahmed H. Hassan, Hesham S. Nassar, Hassan Y. Ebrahim, Ahmed B.M. Mehany & Ahmed M. El-Agrody. (2020) Synthesis, anticancer evaluation and molecular docking studies of new heterocycles linked to sulfonamide moiety as novel human topoisomerase types I and II poisons. Bioorganic Chemistry 98, pages 103725.
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Ghouse Khan, Swamy Sreenivasa, Shivaraja Govindaiah, Vivek Chandramohan & Raghurama Shetty P. (2020) Synthesis, biological screening, in silico study and fingerprint applications of novel 1, 2, 4‐triazole derivatives. Journal of Heterocyclic Chemistry 57:4, pages 2010-2023.
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Nashwa M. Saleh, Marwa G. El-Gazzar, Hala M. Aly & Rana A. Othman. (2020) Novel Anticancer Fused Pyrazole Derivatives as EGFR and VEGFR-2 Dual TK Inhibitors. Frontiers in Chemistry 7.
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Mohamed A. Said, Wagdy M. Eldehna, Alessio Nocentini, Alessandro Bonardi, Samar H. Fahim, Silvia Bua, Dalia H. Soliman, Hatem A. Abdel-Aziz, Paola Gratteri, Sahar M. Abou-Seri & Claudiu T. Supuran. (2020) Synthesis, biological and molecular dynamics investigations with a series of triazolopyrimidine/triazole-based benzenesulfonamides as novel carbonic anhydrase inhibitors. European Journal of Medicinal Chemistry 185, pages 111843.
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Alessio Nocentini, Sameh M. Osman, Sonia Del Prete, Clemente Capasso, Zeid A. ALOthman & Claudiu T. Supuran. (2019) Extending the γ-class carbonic anhydrases inhibition profiles with phenolic compounds. Bioorganic Chemistry 93, pages 103336.
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Immo Serbian, Philipp Schwarzenberger, Anne Loesche, Sophie Hoenke, Ahmed Al-Harrasi & René Csuk. (2019) Ureidobenzenesulfonamides as efficient inhibitors of carbonic anhydrase II. Bioorganic Chemistry 91, pages 103123.
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Süleyman AKOCAK, Mehmet BOGA, Nabih LOLAK, Muhammed TUNEG & Rajesh K K SANKU. (2019) Design, synthesis and biological evaluation of 1,3-diaryltriazenesubstituted sulfonamides as antioxidant, acetylcholinesterase and butyrylcholinesterase inhibitors. Journal of the Turkish Chemical Society Section A: Chemistry 6:1, pages 63-70.
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Marc A. Ilies & Jean-Yves Winum. 2019. Carbonic Anhydrases. Carbonic Anhydrases 331 365 .
Emanuela Masini, Silvia Sgambellone & Laura Lucarini. 2019. Carbonic Anhydrases. Carbonic Anhydrases 269 285 .

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