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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 34, 2019 - Issue 1
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Research Paper

Synthesis carbonic anhydrase enzyme inhibition and antioxidant activity of novel benzothiazole derivatives incorporating glycine, methionine, alanine, and phenylalanine moieties

Deniz Üzeroğlu PayazDepartment of Chemistry, Faculty of Arts and Sciences, İnönü University, Malatya, Turkey; ORCID Iconhttp://orcid.org/0000-0002-4160-5669View further author information
ORCID Icon,
F. Zehra KüçükbayDepartment of Basic Pharmaceutical Sciences, Faculty of Pharmacy, İnönü University, Malatya, Turkey; ORCID Iconhttp://orcid.org/0000-0002-5471-3933View further author information
ORCID Icon,
Hasan KüçükbayDepartment of Chemistry, Faculty of Arts and Sciences, İnönü University, Malatya, Turkey; Correspondence[email protected] [email protected]
ORCID Iconhttp://orcid.org/0000-0002-7180-9486View further author information
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Andrea AngeliDipartimento Neurofarba, Sezione Di Scienze Farmaceutiche E Nutraceutiche e Laboratorio Di Chimica Bioinorganica, Universita` Degli Studi Di Firenze, Florence, ItalyORCID Iconhttp://orcid.org/0000-0002-1470-7192View further author information
ORCID Icon &
Claudiu T. SupuranDipartimento Neurofarba, Sezione Di Scienze Farmaceutiche E Nutraceutiche e Laboratorio Di Chimica Bioinorganica, Universita` Degli Studi Di Firenze, Florence, ItalyCorrespondence[email protected] [email protected]
ORCID Iconhttp://orcid.org/0000-0003-4262-0323View further author information
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Pages 343-349 | Received 24 Oct 2018, Accepted 22 Nov 2018, Published online: 27 Dec 2018

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Zhongcheng Cao, Xingyue Wang, Tianlong Zhang, Xianwu Fu, Fan Zhang & Jiang Zhu. (2023) Discovery of novel 2-(4-(benzyloxy)-5-(hydroxyl) phenyl) benzothiazole derivatives as multifunctional MAO-B inhibitors for the treatment of Parkinson’s disease. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Morteza Abdoli, Alessandro Bonardi, Claudiu T. Supuran & Raivis Žalubovskis. (2023) Investigation of novel alkyl/benzyl (4-sulphamoylphenyl)carbamimidothioates as carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Hasan Küçükbay, Zeynep Gönül, F. Zehra Küçükbay, Andrea Angeli, Gianluca Bartolucci & Claudiu T. Supuran. (2020) Preparation, carbonic anhydrase enzyme inhibition and antioxidant activity of novel 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives incorporating mono or dipeptide moiety. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1021-1026.
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Ali Irfan, Fozia Batool, Syeda Andleeb Zahra Naqvi, Amjad Islam, Sameh M. Osman, Alessio Nocentini, Siham A. Alissa & Claudiu T. Supuran. (2020) Benzothiazole derivatives as anticancer agents. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 265-279.
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Articles from other publishers (15)

Eida S. Al‐Farraj & Ahmed Fetoh. (2023) Synthesis of new Fe(III), Co(II), and Cr(III) complexes of N ‐(benzo[ d ]thiazol‐2‐ylcarbamothioyl)benzamide (H 2 L 2 ): Structural characterization and biological activities . Applied Organometallic Chemistry.
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Alexander Zubenko, Victor Kartsev, Anthi Petrou, Athina Geronikaki, Marija Ivanov, Jasmina Glamočlija, Marina Soković, Lyudmila Divaeva, Anatolii Morkovnik & Alexander Klimenko. (2022) Experimental and In Silico Evaluation of New Heteroaryl Benzothiazole Derivatives as Antimicrobial Agents. Antibiotics 11:11, pages 1654.
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Priti Singh, Dilep Kumar Sigalapalli, Nerella Sridhar Goud, Baijayantimala Swain, Santosh Kumar Sahoo, Andrea Angeli, Afzal B. Shaik, Venkata Madhavi Yaddanapudi, Claudiu T. Supuran & Mohammed Arifuddin. (2021) Ureidosulfocoumarin Derivatives As Selective and Potent Carbonic Anhydrase IX and XII Inhibitors. ChemMedChem 17:5.
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Ahmad H. Abdullah, Jalal A. Zahra, Salim S. Sabri, Firas F. Awwadi, Mohammed M. Abadleh, Qasem M. Abdallah & Mustafa M. El-Abadelah. (2022) Thiophene Ring-opening Reactions III: One-Pot Synthesis and Antitumor Activity of 1,3,4-Thiadiazoline–Benzothiazolo[3,2-b]pyridazine Hybrids†. Current Organic Synthesis 19:2, pages 279-290.
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Asmaa M. Fahim, Hala. E.M. Tolan & Wael A. El-Sayed. (2022) Synthesis of novel 1,2,3-triazole based acridine and benzothiazole scaffold N-glycosides with anti-proliferative activity, docking studies, and comparative computational studies. Journal of Molecular Structure 1251, pages 131941.
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Kashif Rafiq, Najeeb Ur Rehman, Sobia Ahsan Halim, Majid Khan, Ajmal Khan & Ahmed Al-Harrasi. (2022) Design, Synthesis and Molecular Docking Study of Novel 3-Phenyl-β-Alanine-Based Oxadiazole Analogues as Potent Carbonic Anhydrase II Inhibitors. Molecules 27:3, pages 816.
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Derya OSMANİYE & Begüm Nurpelin SAGLİK. (2022) Synthesis and Characterization of New Series Benzothiazole-Dithiocarbamate Derivatives As Potential Antifungal Agents. Deu Muhendislik Fakultesi Fen ve Muhendislik 24:70, pages 105-110.
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Meenakshi Duhan, Parvin Kumar, Jayant Sindhu, Rahul Singh, Meena Devi, Ashwani Kumar, Ramesh Kumar & Sohan Lal. (2021) Exploring biological efficacy of novel benzothiazole linked 2,5-disubstituted-1,3,4-oxadiazole hybrids as efficient α-amylase inhibitors: Synthesis, characterization, inhibition, molecular docking, molecular dynamics and Monte Carlo based QSAR studies. Computers in Biology and Medicine 138, pages 104876.
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Hasan Küçükbay, Zeynep Gönül, Fatümetüzzehra Zehra Küçükbay, Zehra Tekin, Andrea Angeli, Gianluca Bartolucci, Claudiu T. Supuran, Eray Tatlıcı, Elif Apohan & Özfer Yeşilada. (2021) Synthesis of new 7‐amino‐3,4‐dihydroquinolin‐2(1 H )‐one‐peptide derivatives and their carbonic anhydrase enzyme inhibition, antioxidant, and cytotoxic activities . Archiv der Pharmazie 354:11.
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Pınar Güller, Ziya Dağalan, Uğur Güller, Ulaş Çalışır & Bilal Nişancı. (2021) Enzymes inhibition profiles and antibacterial activities of benzylidenemalononitrile derivatives. Journal of Molecular Structure 1239, pages 130498.
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Yousef Mardani, Zahed Karimi-Jaberi & Mohammad Jaafar Soltanian Fard. (2021) One-pot synthesis of 1-(benzothiazolylamino)aryl methyl-2-naphthols and 3-benzothiazolyl 2,3-dihydroquinazolinones using a magnetically recoverable core–shell nanocomposite as catalyst. Zeitschrift für Naturforschung B 76:6-7, pages 385-393.
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Rahul Singh, Jayant Sindhu, Meena Devi, Ashwani Kumar, Ramesh Kumar, Khalid Hussain & Parvin Kumar. (2021) Solid‐Supported Materials‐Based Synthesis of 2‐Substituted Benzothiazoles: Recent Developments and Sanguine Future. ChemistrySelect 6:25, pages 6388-6449.
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Mahmoud Nassiri & Forough Jalili Milani. (2020) Simple, novel, and efficient synthesis of ethyl 2-(2-(1 H -indol-3-yl)benzo[ d ]thiazol-3(2 H )-yl)-2-cyanoacetate or acetate via a three-component reaction . Journal of Chemical Research 45:5-6, pages 526-530.
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Gundluru Mohan, Sumit Kuma, Murali Sudileti, Chadive Sridevi, Pannuru Venkatesu & Cirandur Suresh Reddy. (2020) Excellency of pyrimidinyl moieties containing α-aminophosphonates over benzthiazolyl moieties for thermal and structural stability of stem bromelain. International Journal of Biological Macromolecules 165, pages 2010-2021.
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James A. Ezugwu, Uchechukwu C. Okoro, Mercy A. Ezeokonkwo, China R. Bhimapaka, Sunday N. Okafor, David I. Ugwu, Ogechi C. Ekoh & Solomon I. Attah. (2020) Novel Leu-Val Based Dipeptide as Antimicrobial and Antimalarial Agents: Synthesis and Molecular Docking. Frontiers in Chemistry 8.
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