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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 34, 2019 - Issue 1
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Research Paper

Appraisal of anti-protozoan activity of nitroaromatic benzenesulfonamides inhibiting carbonic anhydrases from Trypanosoma cruzi and Leishmania donovani

Alessio NocentiniDepartment of Neuroscience, Psychology, Drug Research and Child's Health, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Sesto Fiorentino, Italy; View further author information
,
Sameh M. OsmanDepartment of Chemistry, College of Science, King Saud University, Riyadh, Saudi Arabia; View further author information
,
Igor A. RodriguesDepartment of Natural Products and Food, School of Pharmacy, Federal University of Rio de Janeiro, Rio de Janeiro, Brazil; View further author information
,
Veronica S. CardosoBIOINOVAR – Biotechnology Laboratories: Biocatalysis, Bioproducts and Bioenergy, Institute of Microbiology Paulo de Góes, Federal University of Rio de Janeiro, Rio de Janeiro, BrazilView further author information
,
Fatmah Ali S. AlasmaryDepartment of Chemistry, College of Science, King Saud University, Riyadh, Saudi Arabia; View further author information
,
Zeid AlOthmanDepartment of Chemistry, College of Science, King Saud University, Riyadh, Saudi Arabia; View further author information
,
Alane B. VermelhoBIOINOVAR – Biotechnology Laboratories: Biocatalysis, Bioproducts and Bioenergy, Institute of Microbiology Paulo de Góes, Federal University of Rio de Janeiro, Rio de Janeiro, BrazilORCID Iconhttp://orcid.org/0000-0001-5926-4172View further author information
ORCID Icon,
Paola GratteriDepartment of Neuroscience, Psychology, Drug Research and Child's Health, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Sesto Fiorentino, Italy; Correspondence[email protected]
View further author information
&
Claudiu T. SupuranDepartment of Neuroscience, Psychology, Drug Research and Child's Health, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Sesto Fiorentino, Italy; Correspondence[email protected]
ORCID Iconhttp://orcid.org/0000-0003-4262-0323View further author information
ORCID Icon show all
Pages 1164-1171 | Received 28 Apr 2019, Accepted 28 May 2019, Published online: 20 Jun 2019

Citations (18)

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Read on this site (8)

Clemente Capasso & Claudiu T. Supuran. (2023) The management of Babesia, amoeba and other zoonotic diseases provoked by protozoa. Expert Opinion on Therapeutic Patents 33:3, pages 179-192.
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Alessandro Bonardi, Seppo Parkkila & Claudiu T. Supuran. (2022) Inhibition studies of the protozoan α-carbonic anhydrase from Trypanosoma cruzi with phenols. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 2417-2422.
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Alane Beatriz Vermelho, Giseli Capaci Rodrigues, Alessio Nocentini, Felipe R. P. Mansoldo & Claudiu T. Supuran. (2022) Discovery of novel drugs for Chagas disease: is carbonic anhydrase a target for antiprotozoal drugs?. Expert Opinion on Drug Discovery 17:10, pages 1147-1158.
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Andrea Angeli, Linda J. Urbański, Vesa P. Hytönen, Seppo Parkkila & Claudiu T. Supuran. (2021) Activation of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with amines and amino acids. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 758-763.
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Andrea Petreni, Viviana De Luca, Andrea Scaloni, Alessio Nocentini, Clemente Capasso & Claudiu T. Supuran. (2021) Anion inhibition studies of the Zn(II)-bound ι-carbonic anhydrase from the Gram-negative bacterium Burkholderia territorii. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 372-376.
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Linda J. Urbański, Andrea Angeli, Vesa P. Hytönen, Anna Di Fiore, Giuseppina De Simone, Seppo Parkkila & Claudiu T. Supuran. (2021) Inhibition of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with sulphonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 330-335.
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Claudiu T. Supuran. (2020) Exploring the multiple binding modes of inhibitors to carbonic anhydrases for novel drug discovery. Expert Opinion on Drug Discovery 15:6, pages 671-686.
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Claudiu T. Supuran. (2020) Coumarin carbonic anhydrase inhibitors from natural sources. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1462-1470.
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Claudiu T. Supuran. 2024. Metalloenzymes. Metalloenzymes 139 156 .
Miguel Gallardo, Rodrigo Arancibia, Claudio Jiménez, Shane Wilkinson, Patricia M. Toro, Pascal Roussel & Natacha Henry. (2023) Ferrocene-based nitroheterocyclic sulfonylhydrazones: design, synthesis, characterization and trypanocidal properties. JBIC Journal of Biological Inorganic Chemistry 28:6, pages 549-558.
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Andreina Henriquez-Figuereo, Cristina Morán-Serradilla, Eduardo Angulo-Elizari, Carmen Sanmartín & Daniel Plano. (2023) Small molecules containing chalcogen elements (S, Se, Te) as new warhead to fight neglected tropical diseases. European Journal of Medicinal Chemistry 246, pages 115002.
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Joana D’Arc S. Trindade, Célio Geraldo Freire-de-Lima, Suzana Côrte-Real, Debora Decote-Ricardo & Marco Edilson Freire de Lima. (2021) Drug repurposing for Chagas disease: In vitro assessment of nimesulide against Trypanosoma cruzi and insights on its mechanisms of action. PLOS ONE 16:10, pages e0258292.
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Alessio Nocentini, Alane B. Vermelho & Claudiu T. Supuran. 2022. Antiprotozoal Drug Development and Delivery. Antiprotozoal Drug Development and Delivery 83 111 .
Linda J. Urbański, Andrea Angeli, Vesa P. Hytönen, Anna Di Fiore, Seppo Parkkila, Giuseppina De Simone & Claudiu T. Supuran. (2020) Inhibition of the newly discovered β‑carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with inorganic anions and small molecules. Journal of Inorganic Biochemistry 213, pages 111274.
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Ana Paula dos Santos Matos, Deise Cristina Drummond Xavier Paes Lopes, Maria Luíza Honório Peixoto, Veronica da Silva Cardoso, Alane Beatriz Vermelho, Ralph Santos-Oliveira, Alessandra Lifsitch Viçosa, Carla Holandino & Eduardo Ricci-Júnior. (2020) Development, characterization, and anti-leishmanial activity of topical amphotericin B nanoemulsions. Drug Delivery and Translational Research 10:6, pages 1552-1570.
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Freddy A. Bernal, Marcel Kaiser, Bernhard Wünsch & Thomas J. Schmidt. (2019) Structure−Activity Relationships of Cinnamate Ester Analogues as Potent Antiprotozoal Agents. ChemMedChem 15:1, pages 68-78.
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Freddy A. Bernal & Thomas J. Schmidt. (2019) A Comprehensive QSAR Study on Antileishmanial and Antitrypanosomal Cinnamate Ester Analogues. Molecules 24:23, pages 4358.
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Aspatwar, Kairys, Rala, Parikka, Bozdag, Carta, Supuran & Parkkila. (2019) Mycobacterium tuberculosis β-Carbonic Anhydrases: Novel Targets for Developing Antituberculosis Drugs. International Journal of Molecular Sciences 20:20, pages 5153.
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