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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 35, 2020 - Issue 1
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Short Communication

Synthesis of thiazolidin-4-ones and thiazinan-4-ones from 1-(2-aminoethyl)pyrrolidine as acetylcholinesterase inhibitors

Adriana M. das Nevesa Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
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Gabriele A. Berwaldta Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
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Cinara T. Avilaa Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
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Taís B. Goularta Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
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Bruna C. Moreiraa Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
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Taís P. Ferreiraa Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
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Mayara S. P. Soaresb Laboratório de Neuroquímica, Inflamação e Câncer, Centro de Ciências Químicas Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
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Nathalia S. Pedrab Laboratório de Neuroquímica, Inflamação e Câncer, Centro de Ciências Químicas Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
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Luiza Spohrb Laboratório de Neuroquímica, Inflamação e Câncer, Centro de Ciências Químicas Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
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Anita A. A. dE Souzab Laboratório de Neuroquímica, Inflamação e Câncer, Centro de Ciências Químicas Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
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Roselia M. Spanevellob Laboratório de Neuroquímica, Inflamação e Câncer, Centro de Ciências Químicas Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilCorrespondence[email protected]
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Wilson Cunicoa Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilCorrespondence[email protected],br [email protected]
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Pages 31-41 | Received 18 Jul 2019, Accepted 30 Sep 2019, Published online: 23 Oct 2019

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Kshipra S. Karnik, Aniket P. Sarkate, Deepak K. Lokwani, Shailee V. Tiwari, Rajaram Azad & Pravin S. Wakte. (2023) Molecular dynamic simulations based discovery and development of thiazolidin-4-one derivatives as EGFR inhibitors targeting resistance in non-small cell lung cancer (NSCLC). Journal of Biomolecular Structure and Dynamics 41:10, pages 4696-4710.
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Shagufta Naz, Lina Tariq Al Kury, Humaira Nadeem, Fawad Ali Shah, Aman Ullah, Rehan Zafar Paracha, Muhammad Imran & Shupeng Li. (2022) Synthesis, In Silico and Pharmacological Evaluation of New Thiazolidine-4-Carboxylic Acid Derivatives Against Ethanol-Induced Neurodegeneration and Memory Impairment. Journal of Inflammation Research 15, pages 3643-3660.
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Asmaa H. Mohamed, Sara M. Mostafa, Ashraf A. Aly, Alaa A. Hassan, Esraa M. Osman, AbdElAziz A. Nayl, Alan B. Brown & Elshimaa M. N. Abdelhafez. (2023) Novel quinoline/thiazinan-4-one hybrids; design, synthesis, and molecular docking studies as potential anti-bacterial candidates against MRSA. RSC Advances 13:21, pages 14631-14640.
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Veniamin Grigorev, Oleg Tinkov, Ludmila Grigoreva & Alexander Rasdolsky. (2022) Structural fractal analysis of the active sites of acetylcholinesterase from various organisms. Journal of Molecular Graphics and Modelling 116, pages 108265.
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Hetal I. Soni, Navin B. Patel, Rahul B. Parmar, Manuel J. Chan-Bacab & Gildardo Rivera. (2022) Microwave Irradiated Synthesis of Pyrimidine Containing, Thiazolidin-4- ones: Antimicrobial, Anti-Tuberculosis, Antimalarial and Anti-Protozoa Evaluation. Letters in Organic Chemistry 19:9, pages 731-738.
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Ayhan Yıldırım & Serkan Öztürk. (2022) An Efficient Ni(II) Laurate Promoted Heterocyclization of Symmetrical Thioureas with Maleic Anhydride and Mechanistic Approach toward Higher Substituted Thiazolidine‐4‐one‐5‐acetic Acids. ChemistrySelect 7:26.
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Emel Karakılıç, Zuhal Alım, Aslıhan Günel & Arif Baran. (2022) A versatile study of novel A3B-type unsymmetric zinc(II) phthalocyanines containing thiazolidin-4-one: Their, carbonic anhydrase I, II isoenzymes, and xanthine oxidase inhibitors evaluation. Journal of Molecular Structure 1257, pages 132630.
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Marlon P. Almeida, Flávio V.C. Kock, Hugo C.R. de Jesus, Rose M. Carlos & Tiago Venâncio. (2021) Probing the acetylcholinesterase inhibitory activity of a novel Ru(II) polypyridyl complex and the supramolecular interaction by (STD)-NMR. Journal of Inorganic Biochemistry 224, pages 111560.
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Nazlı Turan Yücel, Derya Osmaniye, Ümmühan Kandemir, Asaf Evrim Evren, Özgür Devrim Can & Ümide Demir Özkay. (2021) Synthesis and Antinociceptive Effect of Some Thiazole-Piperazine Derivatives: Involvement of Opioidergic System in the Activity. Molecules 26:11, pages 3350.
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