Advanced search
Publication Cover
Journal of Enzyme Inhibition and Medicinal Chemistry Volume 35, 2020 - Issue 1
Submit an article Journal homepage
2,441
Views
10
CrossRef citations to date
0
Altmetric
Short Communication

Synthesis of thiazolidin-4-ones and thiazinan-4-ones from 1-(2-aminoethyl)pyrrolidine as acetylcholinesterase inhibitors

Adriana M. das Nevesa Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
,
Gabriele A. Berwaldta Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
,
Cinara T. Avilaa Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
,
Taís B. Goularta Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
,
Bruna C. Moreiraa Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
,
Taís P. Ferreiraa Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
,
Mayara S. P. Soaresb Laboratório de Neuroquímica, Inflamação e Câncer, Centro de Ciências Químicas Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
,
Nathalia S. Pedrab Laboratório de Neuroquímica, Inflamação e Câncer, Centro de Ciências Químicas Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
,
Luiza Spohrb Laboratório de Neuroquímica, Inflamação e Câncer, Centro de Ciências Químicas Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
,
Anita A. A. dE Souzab Laboratório de Neuroquímica, Inflamação e Câncer, Centro de Ciências Químicas Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilView further author information
,
Roselia M. Spanevellob Laboratório de Neuroquímica, Inflamação e Câncer, Centro de Ciências Químicas Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilCorrespondence[email protected]
View further author information
&
Wilson Cunicoa Laboratório de Química Aplicada a Bioativos, Centro Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas, Capão do Leão, BrazilCorrespondence[email protected],br [email protected]
View further author information
 show all
Pages 31-41 | Received 18 Jul 2019, Accepted 30 Sep 2019, Published online: 23 Oct 2019

Related Research Data

Miniperspective
Source: American Chemical Society (ACS)
Synthesis and evaluation of antibacterial and antifungal activities of 4-thiazolidinones and 2-azetidinones derivatives from chalcone
Source: Springer Science and Business Media LLC
Thiazolidin-4-one and thiazinan-4-one derivatives analogous to rosiglitazone as potential antihyperglycemic and antidyslipidemic agents
Source: Elsevier BV
Drug treatments in Alzheimer's disease.
Source: Royal College of Physicians
Synthesis of Novel Thiazolidin‐4‐ones and Thiazinan‐4‐ones Analogous to Rosiglitazone
Source: Wiley
Acetylcholinesterases – the structural similarities and differences
Source: Informa UK Limited
Recent developments in structural studies on acetylcholinesterase.
Source: Wiley
Thiazolidin-4-ones from 4-(methylthio)benzaldehyde and 4-(methylsulfonyl)benzaldehyde: Synthesis, antiglioma activity and cytotoxicity.
Source: Elsevier BV
Synthesis of tacrine-lophine hybrids via one-pot four component reaction and biological evaluation as acetyl- and butyrylcholinesterase inhibitors.
Source: Elsevier BV
THIAZOLIDIN-4-ONES AND THIAZINAN-4-ONES
Source: Wiley
Synthesis and antimalarial activity evaluation of 3-(3-(7-chloroquinolin-4-ylamino)propyl)-1,3-thiazinan-4-one derivatives
Source: Elsevier
The antinociceptive evaluation of 2,3-substituted-1,3-thiazolidin-4-ones through thermal stimulation in mice
Source: Springer Science and Business Media LLC
Derivatives of oxoisoaporphine alkaloids: a novel class of selective acetylcholinesterase inhibitors.
Source: Elsevier BV
A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding
Source: Elsevier BV
Synthesis of aminoalkyl-substituted coumarin derivatives as acetylcholinesterase inhibitors
Source: Elsevier BV
Deep Learning in Alzheimer's Disease: Diagnostic Classification and Prognostic Prediction Using Neuroimaging Data
Source: Frontiers Media SA
Current and novel therapeutic molecules and targets in Alzheimer's disease.
Source: Elsevier BV
5,6,7,8-Tetrahydronaphthalen-1-amine as Precursor for Thiazolidi­nones and Benzothiazepinones: Synthesis and Atropisomeric Relationship
Source: Georg Thieme Verlag KG
Amyloid-beta immunotherapy: the hope for Alzheimer disease?
Source: Universidad del Valle

Linking provided by 

Related research

People also read lists articles that other readers of this article have read.

Recommended articles lists articles that we recommend and is powered by our AI driven recommendation engine.

Cited by lists all citing articles based on Crossref citations.
Articles with the Crossref icon will open in a new tab.