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Citations (51)
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Anastasija Balašova, Aleksandrs Pustenko, Alessio Nocentini, Daniela Vullo, Claudiu T. Supuran & Raivis Žalubovskis. (2023) Aryl derivatives of 3H-1,2-benzoxaphosphepine 2-oxides as inhibitors of cancer-related carbonic anhydrase isoforms IX and XII. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Simone Giovannuzzi, Viviana De Luca, Clemente Capasso & Claudiu T. Supuran. (2023) Inhibition studies with simple and complex (in)organic anions of the γ-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri, MscCAγ. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Andrea Angeli & Claudiu T. Supuran. (2023) Click chemistry approaches for developing carbonic anhydrase inhibitors and their applications. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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G. B. Venkatesh, S. HariPrasad & A. S. Jeevan Chakravarthy. (2023) One-pot synthesis of a new class of alkynyl anionic synthons: the 4-(2',2-trimethylsilylethynylphenoxymethyl)-2H-chromen-2-ones. Phosphorus, Sulfur, and Silicon and the Related Elements 198:4, pages 330-335.
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Mehmet Onyılmaz, Murat Koca, Alessandro Bonardi, Mustafa Degirmenci & Claudiu T. Supuran. (2022) Isocoumarins: a new class of selective carbonic anhydrase IX and XII inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 743-748.
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Simone Giovannuzzi, Viviana De Luca, Alessio Nocentini, Clemente Capasso & Claudiu T. Supuran. (2022) Coumarins inhibit η-class carbonic anhydrase from Plasmodium falciparum. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 680-685.
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Wagdy M. Eldehna, Mohammed S. Taghour, Tarfah Al-Warhi, Alessio Nocentini, Mostafa M. Elbadawi, Hazem A. Mahdy, Mohamed A. Abdelrahman, Ohoud J. Alotaibi, Nada Aljaeed, Diaaeldin M. Elimam, Kamyar Afarinkia, Hatem A. Abdel-Aziz & Claudiu T. Supuran. (2022) Discovery of 2,4-thiazolidinedione-tethered coumarins as novel selective inhibitors for carbonic anhydrase IX and XII isoforms. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 531-541.
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Yinbo Pan, Teng Liu, Xiaojing Wang & Jie Sun. (2022) Research progress of coumarins and their derivatives in the treatment of diabetes. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 616-628.
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Simone Giovannuzzi, Chad S. Hewitt, Alessio Nocentini, Clemente Capasso, Daniel P. Flaherty & Claudiu T. Supuran. (2022) Coumarins effectively inhibit bacterial α-carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 333-338.
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Alma Fuentes-Aguilar, Penélope Merino-Montiel, Sara Montiel-Smith, Socorro Meza-Reyes, José Luis Vega-Báez, Adrián Puerta, Miguel X. Fernandes, José M. Padrón, Andrea Petreni, Alessio Nocentini, Claudiu T. Supuran, Óscar López & José G. Fernández-Bolaños. (2022) 2-Aminobenzoxazole-appended coumarins as potent and selective inhibitors of tumour-associated carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 168-177.
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Claudiu T. Supuran, Alessio Nocentini, Elena Yakubova, Nikolay Savchuk, Stanislav Kalinin & Mikhail Krasavin. (2021) Biochemical profiling of anti-HIV prodrug Elsulfavirine (Elpida®) and its active form VM1500A against a panel of twelve human carbonic anhydrase isoforms. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 1056-1060.
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Rita Meleddu, Serenella Deplano, Elias Maccioni, Francesco Ortuso, Filippo Cottiglia, Daniela Secci, Alessia Onali, Erica Sanna, Andrea Angeli, Rossella Angius, Stefano Alcaro, Claudiu T. Supuran & Simona Distinto. (2021) Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 685-692.
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Alessio Nocentini, Andrea Angeli, Fabrizio Carta, Jean-Yves Winum, Raivis Zalubovskis, Simone Carradori, Clemente Capasso, William A. Donald & Claudiu T. Supuran. (2021) Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 561-580.
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Heping Zhu, Shilong Ying, Bingluo Zhou, Xinyang Hu, Xiao Liang, Wangyu Li, Dungai Wang, Hongchuan Jin & Yuanjiang Pan. (2021) Design, synthesis, and evaluation of novel coumarin-dithiocarbamate derivatives (IDs) as anti-colorectal cancer agents. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 593-604.
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Yuhang Miao, Jie Yang, Yinling Yun, Jie Sun & Xiaojing Wang. (2021) Synthesis and anti-rheumatoid arthritis activities of 3-(4-aminophenyl)-coumarin derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 450-461.
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Articles from other publishers (36)
Claudiu T. Supuran. 2024. Metalloenzymes. Metalloenzymes
139
156
.
Dilipkumar Pal, Kamal Bareth, Priyanka Rani, Chandi Charan Kandar & Abhishek Mishra. 2024. Anti-Viral Metabolites from Medicinal Plants. Anti-Viral Metabolites from Medicinal Plants
1039
1065
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Aleksandrs Pustenko, Anastasija Balašova, Alessio Nocentini, Claudiu T. Supuran & Raivis Žalubovskis. (2022)
3
H
-1,2-Benzoxaphosphepine 2-oxides as selective inhibitors of carbonic anhydrase IX and XII
. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1, pages 216-224.
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Emanuela Berrino, Simone Carradori, Fabrizio Carta, Francesco Melfi, Marialucia Gallorini, Giulio Poli, Tiziano Tuccinardi, José G. Fernández-Bolaños, Óscar López, Jacobus P. Petzer, Anél Petzer, Paolo Guglielmi, Daniela Secci & Claudiu T. Supuran. (2023) A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration. Antioxidants 12:12, pages 2044.
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Ayşe Çiçek Kaya, Hilal Özbek, Hafize Yuca, Gülderen Yılmaz, Zeynebe Bingöl, Cavit Kazaz, İlhami Gülçin & Zühal Güvenalp. (2023) Phytochemical content and enzyme inhibitory effect of Heptaptera triquetra (Vent.) Tutin fruit against acetylcholinesterase and carbonic anhydrase I and II isoenzymes. Chemical Papers 77:10, pages 5829-5837.
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Claudiu T. Supuran. (2023) A simple yet multifaceted 90 years old, evergreen enzyme: Carbonic anhydrase, its inhibition and activation. Bioorganic & Medicinal Chemistry Letters 93, pages 129411.
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Eman M. Radwan, Eman Abo-Elabass, Atef E. Abd El-Baky, Hussah Abdullah Alshwyeh, Riyad A. Almaimani, Ghassan Almaimani, Ibrahim Abdel Aziz Ibrahim, Abdulaziz Albogami, Mariusz Jaremko, Samar Z. Alshawwa & Essa M. Saied. (2023) Unveiling the antitumor potential of novel N-(substituted-phenyl)-8-methoxycoumarin-3-carboxamides as dual inhibitors of VEGFR2 kinase and cytochrome P450 for targeted treatment of hepatocellular carcinoma. Frontiers in Chemistry 11.
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Cătălina Mareş, Ana-Maria Udrea, Nicoleta Anca Şuţan & Speranţa Avram. (2023) Bioinformatics Tools for the Analysis of Active Compounds Identified in Ranunculaceae Species. Pharmaceuticals 16:6, pages 842.
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Aditi Redij, Simone Carradori, Andrea Petreni, Claudiu T. Supuran & Mrunmayee P. Toraskar. (2023) Coumarin-pyrazoline Hybrids as Selective Inhibitors of the Tumor-associated
Carbonic Anhydrase IX and XII. Anti-Cancer Agents in Medicinal Chemistry 23:10, pages 1217-1223.
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Ayça Aktaş Karaçelik & Gözde Yalçın Özkat. (2023) Mentha longifolia ssp. longifolia Essential Oil Components as Novel Carbonic
Anhydrase Isoform II and IX Inhibitors: Biological and Molecular
Docking Studies. Letters in Drug Design & Discovery 20:6, pages 767-778.
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Bader I. Huwaimel, Sravan K. Jonnalagadda, Shirisha Jonnalagadda, Shikha Kumari, Alessio Nocentini, Claudiu T. Supuran & Paul C. Trippier. (2023) Selective carbonic anhydrase IX and XII inhibitors based around a functionalized coumarin scaffold. Drug Development Research 84:4, pages 681-702.
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Luiz C. Di Stasi. (2023) Natural Coumarin Derivatives Activating Nrf2 Signaling Pathway as Lead Compounds for the Design and Synthesis of Intestinal Anti-Inflammatory Drugs. Pharmaceuticals 16:4, pages 511.
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Belma Zengin Kurt, Gulsen Celebi, Dilek Ozturk Civelek, Andrea Angeli, Atilla Akdemir, Fatih Sonmez & Claudiu T. Supuran. (2023) Tail-Approach-Based Design and Synthesis of Coumarin-Monoterpenes as Carbonic Anhydrase Inhibitors and Anticancer Agents. ACS Omega 8:6, pages 5787-5807.
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Emanuela Berrino, Laura Micheli, Simone Carradori, Lorenzo di Cesare Mannelli, Paolo Guglielmi, Alessandro De Luca, Fabrizio Carta, Carla Ghelardini, Daniela Secci & Claudiu T. Supuran. (2023) Novel Insights on CAI–CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis. Journal of Medicinal Chemistry 66:3, pages 1892-1908.
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Kanchanlata Tungare, Ameyota De, Shreya Das, Vaishnavi Kesarkar, Mustansir Bhori & Renitta Jobby. 2023. Microbial Biofilms. Microbial Biofilms
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Tinuccia Dettori, Giuseppina Sanna, Andrea Cocco, Gabriele Serreli, Monica Deiana, Vanessa Palmas, Valentina Onnis, Luca Pilia, Nicola Melis, Davide Moi, Paola Caria & Francesco Secci. (2022) Synthesis and Antiproliferative Effect of Halogenated Coumarin Derivatives. Molecules 27:24, pages 8897.
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Claudiu T. Supuran. 2022. Flavonoids and Phenolics. Flavonoids and Phenolics
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329
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Claudiu T. Supuran. (2022) Carbonic Anhydrase Inhibitors from Marine Natural Products. Marine Drugs 20:11, pages 721.
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Aarfa Queen, Humaira Naaz Bhutto, Mohd Yousuf, Mansoor Ali Syed & Md. Imtaiyaz Hassan. (2022) Carbonic anhydrase IX: A tumor acidification switch in heterogeneity and chemokine regulation. Seminars in Cancer Biology 86, pages 899-913.
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Ayşe ÇİÇEK KAYA, Hilal ÖZBEK, Hafize YUCA, Gülderen YILMAZ, Zeynebe BİNGÖL, Cavit KAZAZ, İlhami GÜLÇİN & Zuhal GÜVENALP. (2022) Phytochemical Analysis and Screening of Acetylcholinesterase and Carbonic Anhydrase I and II Isoenzymes Inhibitory Effect of Heptaptera triquetra (Vent.) Tutin Root. Fabad Journal of Pharmaceutical Sciences.
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Virginia Pontecorvi, Mattia Mori, Francesca Picarazzi, Susi Zara, Simone Carradori, Amelia Cataldi, Andrea Angeli, Emanuela Berrino, Paola Chimenti, Alessia Ciogli, Daniela Secci, Paolo Guglielmi & Claudiu T. Supuran. (2022) Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies. International Journal of Molecular Sciences 23:14, pages 7950.
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Giulia Arrighi, Adrián Puerta, Andrea Petrini, Francisco J. Hicke, Alessio Nocentini, Miguel X. Fernandes, José M. Padrón, Claudiu T. Supuran, José G. Fernández-Bolaños & Óscar López. (2022) Squaramide-Tethered Sulfonamides and Coumarins: Synthesis, Inhibition of Tumor-Associated CAs IX and XII and Docking Simulations. International Journal of Molecular Sciences 23:14, pages 7685.
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Priti Singh, Dilep Kumar Sigalapalli, Nerella Sridhar Goud, Baijayantimala Swain, Santosh Kumar Sahoo, Andrea Angeli, Afzal B. Shaik, Venkata Madhavi Yaddanapudi, Claudiu T. Supuran & Mohammed Arifuddin. (2021) Ureidosulfocoumarin Derivatives As Selective and Potent Carbonic Anhydrase IX and XII Inhibitors. ChemMedChem 17:5.
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Laila Rubab, Sumbal Afroz, Sajjad Ahmad, Saddam Hussain, Iram Nawaz, Ali Irfan, Fozia Batool, Katarzyna Kotwica-Mojzych & Mariusz Mojzych. (2022) An Update on Synthesis of Coumarin Sulfonamides as Enzyme Inhibitors and Anticancer Agents. Molecules 27:5, pages 1604.
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Jin-Hai Yu, Zhi-Pu Yu, Robert J. Capon & Hua Zhang. (2022) Natural Enantiomers: Occurrence, Biogenesis and Biological Properties. Molecules 27:4, pages 1279.
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Andrea Angeli, Emanuela Berrino, Simone Carradori, Claudiu T. Supuran, Marzia Cirri, Fabrizio Carta & Gabriele Costantino. (2021) Amine- and Amino Acid-Based Compounds as Carbonic Anhydrase Activators. Molecules 26:23, pages 7331.
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Andrea Petreni, Sameh M. Osman, Fatmah A. Alasmary, Tahani M. Almutairi, Alessio Nocentini & Claudiu T. Supuran. (2021) Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. European Journal of Medicinal Chemistry 226, pages 113875.
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Burak Kuzu, Meltem Tan, İlhami Gülçin & Nurettin Menges. (2021) A novel class for carbonic anhydrases inhibitors and evaluation of their non‐zinc binding. Archiv der Pharmazie 354:10.
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Mudasir Nabi Peerzada, Ernest Hamel, Ruoli Bai, Claudiu T. Supuran & Amir Azam. (2021) Deciphering the key heterocyclic scaffolds in targeting microtubules, kinases and carbonic anhydrases for cancer drug development. Pharmacology & Therapeutics 225, pages 107860.
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Ceren Akpunar, Namık Özdemir, Mert Olgun Karataş, Bülent Alıcı & İsmail Özdemir. (2021) Synthesis, crystal structures and catalytic activities of palladium complexes with coumarin-functionalised N-heterocyclic carbene ligands. Inorganic Chemistry Communications 131, pages 108755.
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Serena Montanari, Marco Allarà, Laura Scalvini, Magdalena Kostrzewa, Federica Belluti, Silvia Gobbi, Marina Naldi, Silvia Rivara, Manuela Bartolini, Alessia Ligresti, Alessandra Bisi & Angela Rampa. (2021) New Coumarin Derivatives as Cholinergic and Cannabinoid System Modulators. Molecules 26:11, pages 3254.
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Elmas Begum Cakmak, Belma Zengin Kurt, Dilek Ozturk Civelek, Andrea Angeli, Atilla Akdemir, Fatih Sonmez, Claudiu T. Supuran & Mustafa Kucukislamoglu. (2021) Quinoline-sulfamoyl carbamates/sulfamide derivatives: Synthesis, cytotoxicity, carbonic anhydrase activity, and molecular modelling studies. Bioorganic Chemistry 110, pages 104778.
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Pavitra S. Thacker, Danaboina Srikanth, Andrea Angeli, Priti Singh, Krishna Kartheek Chinchilli, Mohammed Arifuddin & Claudiu T. Supuran. (2021) Coumarin‐Thiourea Hybrids Show Potent Carbonic Anhydrase IX and XIII Inhibitory Action. ChemMedChem 16:8, pages 1252-1256.
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Pavitra S. Thacker, Prerna L. Tiwari, Andrea Angeli, Danaboina Srikanth, Baijayantimala Swain, Mohammed Arifuddin & Claudiu T. Supuran. (2021) Synthesis and Biological Evaluation of Coumarin-Linked 4-Anilinomethyl-1,2,3-Triazoles as Potent Inhibitors of Carbonic Anhydrases IX and XIII Involved in Tumorigenesis. Metabolites 11:4, pages 225.
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R. Kanimozhi & V. Arjunan. (2021) FT-IR, FT-Raman, NMR Spectroscopic and DFT
Quantum Chemical Investigations of 6-Methylcoumarin. Asian Journal of Chemistry 33:11, pages 2715-2722.
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Andrea Angeli, Fabrizio Carta, Alessio Nocentini, Jean-Yves Winum, Raivis Zalubovskis, Atilla Akdemir, Valentina Onnis, Wagdy M. Eldehna, Clemente Capasso, Giuseppina De Simone, Simona Maria Monti, Simone Carradori, William A. Donald, Shoukat Dedhar & Claudiu T. Supuran. (2020) Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment. Metabolites 10:10, pages 412.
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