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Original Research

Development and characterization of self-assembling lecithin-based mixed polymeric micelles containing quercetin in cancer treatment and an in vivo pharmacokinetic study

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Pages 1557-1566 | Published online: 15 Apr 2016

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Fatma M Elsharkawy, Maha M Amin, Hesham A Shamsel-Din, Walaa Ibrahim, Ahmed B Ibrahim & Sinar Sayed. (2023) Self-Assembling Lecithin-Based Mixed Polymeric Micelles for Nose to Brain Delivery of Clozapine: In-vivo Assessment of Drug Efficacy via Radiobiological Evaluation. International Journal of Nanomedicine 18, pages 1577-1595.
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Hong-Liang Lin, Wen-Ting Cheng, Ling-Chun Chen, Hsiu-O Ho, Shyr-Yi Lin & Chien-Ming Hsieh. (2021) Honokiol/Magnolol-Loaded Self-Assembling Lecithin-Based Mixed Polymeric Micelles (lbMPMs) for Improving Solubility to Enhance Oral Bioavailability. International Journal of Nanomedicine 16, pages 651-665.
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Arjun Patra, Swaha Satpathy, Anitha K Shenoy, Jason A Bush, Mohsin Kazi & Muhammad Delwar Hussain. (2018) Formulation and evaluation of mixed polymeric micelles of quercetin for treatment of breast, ovarian, and multidrug resistant cancers. International Journal of Nanomedicine 13, pages 2869-2881.
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Ling-xin Meng, Qiang Ren, Qin Meng, Yu-xiu Zheng, Mao-lei He, Shu-yan Sun, Zhao-jun Ding, Bing-cheng Li & Hui-yun Wang. (2018) Trastuzumab modified silica nanoparticles loaded with doxorubicin for targeted and synergic therapy of breast cancer. Artificial Cells, Nanomedicine, and Biotechnology 46:sup3, pages 556-563.
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Zhen Lu, Cuiping Bu, Weicheng Hu, Hui Zhang, Mengrui Liu, Meiqi Lu & Guangxi Zhai. (2018) Preparation and in vitro and in vivo evaluation of quercetin-loaded mixed micelles for oral delivery. Bioscience, Biotechnology, and Biochemistry 82:2, pages 238-246.
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Ashil Joseph, Prasanth Shanmughan, Abhilash Balakrishnan, Balu Maliakel & Krishnakumar I M. (2022) Enhanced Bioavailability and Pharmacokinetics of a Natural Self-Emulsifying Reversible Hybrid-Hydrogel System of Quercetin: A Randomized Double-Blinded Comparative Crossover Study. ACS Omega 7:50, pages 46825-46832.
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Yating Zhang, Ruiyang Hou, Beibei Zhu, Guangwei Yin, Jian Zhang, Wenqi Zhao, Junxi Zhang, Taoran Li, Zifan Zhang, Hongwu Wang & Zheng Li. (2022) Changes on the conformational and functional properties of soybean protein isolate induced by quercetin. Frontiers in Nutrition 9.
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Miguel Ferreira, Diana Costa & Ângela Sousa. (2022) Flavonoids-Based Delivery Systems towards Cancer Therapies. Bioengineering 9:5, pages 197.
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Heba M. Aboud, Amal K. Hussein, Abdallah Z. Zayan, Tarek Saad Makram, Mona O. Sarhan & Dina M. El-Sharawy. (2022) Tailoring of Selenium-Plated Novasomes for Fine-Tuning Pharmacokinetic and Tumor Uptake of Quercetin: In Vitro Optimization and In Vivo Radiobiodistribution Assessment in Ehrlich Tumor-Bearing Mice. Pharmaceutics 14:4, pages 875.
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Joseph Thomas Ortega & Beata Jastrzebska. (2021) Neuroinflammation as a Therapeutic Target in Retinitis Pigmentosa and Quercetin as Its Potential Modulator. Pharmaceutics 13:11, pages 1935.
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Paweł Śliwa & Karolina Śliwa. (2021) Nanomicellar Extraction of Polyphenols—Methodology and Applications Review. International Journal of Molecular Sciences 22:21, pages 11392.
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Dibakar Goswami & Soumyaditya Mula. 2021. Handbook on Synthesis Strategies for Advanced Materials. Handbook on Synthesis Strategies for Advanced Materials 557 588 .
Dinh Van Thoai, Dinh Trung Nguyen, Le Hang Dang, Ngoc Hao Nguyen, Van Toan Nguyen, Phuong Doan, Bich Tram Nguyen, Le Van Thu, Nguyen Ngoc Tung & Tran Ngoc Quyen. (2020) Lipophilic effect of various pluronic-grafted gelatin copolymers on the quercetin delivery efficiency in these self-assembly nanogels. Journal of Polymer Research 27:12.
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Bahare Salehi, Laura Machin, Lianet Monzote, Javad Sharifi-Rad, Shahira M. Ezzat, Mohamed A. Salem, Rana M. Merghany, Nihal M. El Mahdy, Ceyda Sibel Kılıç, Oksana Sytar, Mehdi Sharifi-Rad, Farukh Sharopov, Natália Martins, Miquel Martorell & William C. Cho. (2020) Therapeutic Potential of Quercetin: New Insights and Perspectives for Human Health. ACS Omega 5:20, pages 11849-11872.
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S. Franklyn De Silva & Jane Alcorn. (2019) Flaxseed Lignans as Important Dietary Polyphenols for Cancer Prevention and Treatment: Chemistry, Pharmacokinetics, and Molecular Targets. Pharmaceuticals 12:2, pages 68.
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Chia-En Chang, Chien-Ming Hsieh, Sheng-Chin Huang, Chia-Yu Su, Ming-Thau Sheu & Hsiu-O. Ho. (2018) Lecithin-Stabilized Polymeric Micelles (LsbPMs) for Delivering Quercetin: Pharmacokinetic Studies and Therapeutic Effects of Quercetin Alone and in Combination with Doxorubicin. Scientific Reports 8:1.
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