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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 30, 2015 - Issue 3
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Research Article

Synthesis and biological evaluation of 5-benzylidenerhodanine-3-acetic acid derivatives as AChE and 15-LOX inhibitors

Negah ShafiiTehran University of Medical Sciences, International Campus (TUMS-IC), Tehran, Iran,
,
Mehdi KhoobiDepartment of Medicinal Chemistry, Faculty of Pharmacy and Pharmaceutical Sciences Research Center, Tehran University of Medical Sciences, Tehran, Iran,
,
Mohsen AminiDepartment of Medicinal Chemistry, Faculty of Pharmacy and Pharmaceutical Sciences Research Center, Tehran University of Medical Sciences, Tehran, Iran,
,
Amirhossein SakhtemanDepartment of Medicinal Chemistry, Faculty of Pharmacy, Shahid Sadoughi University of Medical Sciences, Yazd, Iran, and
,
Hamid NadriDepartment of Medicinal Chemistry, Faculty of Pharmacy, Shahid Sadoughi University of Medical Sciences, Yazd, Iran, and
,
Alireza MoradiDepartment of Medicinal Chemistry, Faculty of Pharmacy, Shahid Sadoughi University of Medical Sciences, Yazd, Iran, and
,
Saeed EmamiDepartment of Medicinal Chemistry and Pharmaceutical Sciences Research Center, Faculty of Pharmacy, Mazanderan University of Medical Sciences, Sari, Iran
,
Ebrahim Saeedian MoghadamDepartment of Medicinal Chemistry, Faculty of Pharmacy and Pharmaceutical Sciences Research Center, Tehran University of Medical Sciences, Tehran, Iran,
,
Alireza ForoumadiDepartment of Medicinal Chemistry, Faculty of Pharmacy and Pharmaceutical Sciences Research Center, Tehran University of Medical Sciences, Tehran, Iran,
&
Abbas ShafieeTehran University of Medical Sciences, International Campus (TUMS-IC), Tehran, Iran, ;Department of Medicinal Chemistry, Faculty of Pharmacy and Pharmaceutical Sciences Research Center, Tehran University of Medical Sciences, Tehran, Iran, Correspondence[email protected]
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Pages 389-395 | Received 14 May 2014, Accepted 30 Jun 2014, Published online: 22 Jun 2015

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Duc-Thuan Nguyen, Ngoc-Khoi Pham, Xuan-Triet Nguyen, Thi Xuan Thi Luu & Quynh-Nhi Nguyen Luong. (2023) Ultrasound accelerated solvent-free condensation reaction of rhodanines and carbonyls using Amberlyst 26 as a green and efficient base catalyst. Journal of Sulfur Chemistry 44:4, pages 447-461.
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Ebrahim Saeedian Moghadam, Maryam Hosseinpour Tehrani, Raid Abdel-Jalil, Mohammad Ali Faramarzi & Mohsen Amini. (2022) Design, Synthesis and Bioactivity Investigation of Novel 2,3-Diarylthiazolidine-4-Ones as Potent α-Glucosidase Inhibitors. Polycyclic Aromatic Compounds 42:8, pages 5748-5766.
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T. Bensafi, D. Hadji, A. Yahiaoui, K. Argoub, A. Hachemaoui, A. Kenane, B. Baroudi, K. Toubal, A. Djafri & A. M. Benkouider. (2021) Synthesis, characterization and DFT calculations of linear and NLO properties of novel (Z)-5-benzylidene-3-N(4-methylphenyl)-2-thioxothiazolidin-4-one. Journal of Sulfur Chemistry 42:6, pages 645-663.
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Ebrahim Saeedian Moghadam, Bilqees Sameem, Raid Abdel-Jalil, Mohammad Ali Faramarzi & Mohsen Amini. (2021) 5-Benzylidene-2,3-diarylthiazolidine-4-ones: Design, synthesis, spectroscopic characterization, in vitro biological and computational evaluation. Synthetic Communications 51:17, pages 2668-2683.
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Suresh Maddila, Sridevi Gorle & Sreekantha B Jonnalagadda. (2020) Drug screening of rhodanine derivatives for antibacterial activity. Expert Opinion on Drug Discovery 15:2, pages 203-229.
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Seyyed Mojtaba Mousavi, Maryam Zarei, Seyyed Alireza Hashemi, Aziz Babapoor & Ali Mohammad Amani. (2019) A conceptual review of rhodanine: current applications of antiviral drugs, anticancer and antimicrobial activities. Artificial Cells, Nanomedicine, and Biotechnology 47:1, pages 1132-1148.
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R. Baharfar, M. Tarahomi & R. Azimi. (2019) Efficient Multicomponent Synthesis of Novel Rhodanine Based Amide Derivatives. Organic Preparations and Procedures International 51:6, pages 595-601.
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Abhishek Chaurasyia, Pooja Chawla, Vikramdeep Monga & Gurpreet Singh. (2022) Rhodanine derivatives: An insight into the synthetic and medicinal perspectives as antimicrobial and antiviral agents. Chemical Biology & Drug Design 101:3, pages 500-549.
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Du Ri Jo, Young-Ok Kim, Ran Kim, Young-Cheol Chang, DuBok Choi & Hoon Cho. (2018) Novel rhodanine derivatives are selective algicides against Microcystis aeruginosa. Biotechnology and Bioprocess Engineering 22:6, pages 748-757.
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Martin Krátký, Šárka Štěpánková, Katarína Vorčáková & Jarmila Vinšová. (2016) Synthesis and in vitro evaluation of novel rhodanine derivatives as potential cholinesterase inhibitors. Bioorganic Chemistry 68, pages 23-29.
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Simiao Gao, Yu Zhang, Jun Dong, Ning Chen & Jiaxi Xu. (2016) Synthesis of functionalized 5-substituted thiazolidine-2-thiones via adscititious xanthate-promoted radical cyclization of allyl(alkyl/aryl)dithiocarbamates. Organic & Biomolecular Chemistry 14:3, pages 1002-1012.
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