Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 17, Issue 3 (2002)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 17, Issue 3 (2002)

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Research Article

Article
Experiments Towards the Synthesis of the Ergot Alkaloids and Related Structures. Part 8.17 The Total Synthesis of 4-Methyl-2,3,4,4a,5,6-hexahydro-benzo[f]quinoline-2-carbonitrile Hydrochloride Hemihydrate, an Immediate Precursor of the Despyrrole Analogues of Lysergic Acid and Its Amides
Mark A.E. Bowman, Ralph E. Bowman, Roy V. Davies, Gerry Haran, Paul J. Harris, H. John Smith, Robert W. Steele, Nigel Walker & Keith Whiting
Pages: 137-154
Published online: 30 Sep 2008
AbstractforExperiments Towards the Synthesis of the Ergot Alkaloids and Related Structures. Part 8.17 The Total Synthesis of 4-Methyl-2,3,4,4a,5,6-hexahydro-benzo[f]quinoline-2-carbonitrile Hydrochloride Hemihydrate, an Immediate Precursor of the Despyrrole Analogues of Lysergic Acid and Its Amides | References | PDF (528.5 KB)
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Article
Androsterone Derivatives Substituted at Position 16: Chemical Synthesis, Inhibition of Type 3 17β-hydroxysteroid Dehydrogenase, Binding Affinity for Steroid Receptors and Proliferative/antiproliferative Activity on Shionogi (AR +) Cells
Béatrice Tchédam-Ngatcha, Van Luu-The & Donald Poirier
Pages: 155-165
Published online: 30 Sep 2008
AbstractforAndrosterone Derivatives Substituted at Position 16: Chemical Synthesis, Inhibition of Type 3 17β-hydroxysteroid Dehydrogenase, Binding Affinity for Steroid Receptors and Proliferative/antiproliferative Activity on Shionogi (AR +) Cells | References | PDF (317.7 KB)
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Article
Database Searching for Thymidine and Thymidylate Kinase Inhibitors Using Three-dimensional Structure-based Methods
David T. Manallack, Will R. Pitt, Piet Herdewijn, Jan Balzarini, Erik De Clercq, Mark R. Sanderson, Maninder Sohi, Frank Wien, Helene Munier-Lehmann, Ahmed Haouz & Marc Delarue
Pages: 167-174
Published online: 30 Sep 2008
AbstractforDatabase Searching for Thymidine and Thymidylate Kinase Inhibitors Using Three-dimensional Structure-based Methods | References | PDF (243.7 KB)
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Article
Synthesis of Potential Anti-HIV GP120 Inhibitors Using a Lysine Template
Valerie E. Doyle, Thomas Klimkait, Naheed Mahmood, Martin Slater, Richard J. Hazen & Ian H. Gilbert
Pages: 175-182
Published online: 30 Sep 2008
AbstractforSynthesis of Potential Anti-HIV GP120 Inhibitors Using a Lysine Template | References | PDF (217.5 KB)
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Article
Inhibition of Hyaluronidases and Chondroitinases by Fatty Acids
Keitarou Suzuki, Yoshikazu Terasaki & Masaru Uyeda
Pages: 183-186
Published online: 30 Sep 2008
AbstractforInhibition of Hyaluronidases and Chondroitinases by Fatty Acids | References | PDF (122.3 KB)
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Article
N -substituted 4-(4-carboxyphenoxy)benzamides. Synthesis and Evaluation as Inhibitors of Steroid-5α-reductase Type 1 and 2
Franck Picard & Rolf W. Hartmann
Pages: 187-196
Published online: 30 Sep 2008
AbstractforN -substituted 4-(4-carboxyphenoxy)benzamides. Synthesis and Evaluation as Inhibitors of Steroid-5α-reductase Type 1 and 2 | References | PDF (234.8 KB)
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Article
Inhibition of Butyrylcholinesterase by Phenothiazine Derivatives
Jean Debord, Louis Merle, Jean-Claude Bollinger & Thierry Dantoine
Pages: 197-202
Published online: 30 Sep 2008
AbstractforInhibition of Butyrylcholinesterase by Phenothiazine Derivatives | References | PDF (151 KB)
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Article
Product Inhibition Study on Carbonic Anhydrase Using Spectroscopy and Calorimetry
N.S. Sarraf, A.A. Saboury & A.A. Moosavi-Movahedi
Pages: 203-206
Published online: 30 Sep 2008
AbstractforProduct Inhibition Study on Carbonic Anhydrase Using Spectroscopy and Calorimetry | References | PDF (132.6 KB)
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