Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 27, Issue 6 (2012)

Browse this journal
Sample our Bioscience journals, sign in here to start your access, Latest two full volumes FREE to you for 14 days

Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 27, Issue 6 (2012)

See all volumes and issues
Vol 39, 2024 Vol 38, 2023 Vol 37, 2022 Vol 36, 2021 Vol 35, 2020 Vol 34, 2019 Vol 33, 2018 Vol 32, 2017 Vol 31, 2016 Vol 30, 2015 Vol 29, 2014 Vol 28, 2013 Volume 27, 2012 Vol 26, 2011 Vol 25, 2010 Vol 24, 2009 Vol 23, 2008 Vol 22, 2007 Vol 21, 2006 Vol 20, 2005 Vol 19, 2004 Vol 18, 2003 Vol 17, 2002 Vol 16, 2001 Vol 15, 1999-2000 Vol 14, 1998-1999 Vol 13, 1998 Vol 12, 1997 Vol 11, 1996-1997 Vol 10, 1995-1996 Vol 9, 1995 Vol 8, 1994-1995 Vol 7, 1993 Vol 6, 1992-1993 Vol 5, 1991 Vol 4, 1990-1991 Vol 3, 1989-1990 Vol 2, 1987-1989 Vol 1, 1985-1987
Download citations Download PDFs Download issue

Review Article

Review Article
Structure-based drug discovery of carbonic anhydrase inhibitors
Claudiu T. Supuran
Pages: 759-772
Published online: 02 Apr 2012
AbstractforStructure-based drug discovery of carbonic anhydrase inhibitors | Full Text | References | PDF (982.8 KB)
  • 9424 Views
  • 536 CrossRef citations
  • 0Altmetric
Free Access
Review Article
Heterocyclic compounds as carbonic anhydrase inhibitor
Asif Husain & Diwakar Madhesia
Pages: 773-783
Published online: 10 Oct 2011
AbstractforHeterocyclic compounds as carbonic anhydrase inhibitor | Full Text | References | PDF (967.2 KB)
  • 1750 Views
  • 16 CrossRef citations
  • 0Altmetric
Free Access

Research Article

Article
Synthesis and evaluation of substrate analogue inhibitors of trypanothione reductase
Michael H. Duyzend, Christopher T. Clark, Shayna L. Simmons, Wade B. Johnson, Anna M. Larson, Aaron M. Leconte, Andrew W. Wills, Matthew Ginder-Vogel, April K. Wilhelm, Josephine A. Czechowicz & David G. Alberg
Pages: 784-794
Published online: 15 Nov 2011
AbstractforSynthesis and evaluation of substrate analogue inhibitors of trypanothione reductase | Full Text | References | PDF (919.4 KB)
  • 775 Views
  • 10 CrossRef citations
  • 0Altmetric
Free Access
Article
Purification of carbonic anhydrase-II from sheep liver and inhibitory effects of some heavy metals on enzyme activity
Ramazan Demirdag, Emrah Yerlikaya & Omer Irfan Kufrevioglu
Pages: 795-799
Published online: 10 Oct 2011
AbstractforPurification of carbonic anhydrase-II from sheep liver and inhibitory effects of some heavy metals on enzyme activity | Full Text | References | PDF (596.6 KB)
  • 597 Views
  • 6 CrossRef citations
  • 0Altmetric
Free Access
Article
Polyphenol fatty acid esters as serine protease inhibitors: a quantum-chemical QSAR analysis
Jana Viskupicova, Martina Danihelova, Magdalena Majekova, Tibor Liptaj & Ernest Sturdik
Pages: 800-809
Published online: 10 Oct 2011
AbstractforPolyphenol fatty acid esters as serine protease inhibitors: a quantum-chemical QSAR analysis | Full Text | References | PDF (739 KB)
  • 1293 Views
  • 16 CrossRef citations
  • 0Altmetric
Free Access
Article
Evaluation of the oxidation of 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine (MPTP) to toxic pyridinium cations by monoamine oxidase (MAO) enzymes and its use to search for new MAO inhibitors and protective agents
Tomás Herraiz
Pages: 810-817
Published online: 12 Oct 2011
AbstractforEvaluation of the oxidation of 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine (MPTP) to toxic pyridinium cations by monoamine oxidase (MAO) enzymes and its use to search for new MAO inhibitors and protective agents | Full Text | References | PDF (825.3 KB)
  • 1154 Views
  • 17 CrossRef citations
  • 0Altmetric
Free Access
Article
Sulfapyridine-like benzenesulfonamide derivatives as inhibitors of carbonic anhydrase isoenzymes I, II and VI
Cemalettin Alp, Şeyda Özsoy, Nurdan Alcan Alp, Deryanur Erdem, Mehmet Serdar Gültekin, Ömer İrfan Küfrevioğlu, Murat Şentürk & Claudiu T. Supuran
Pages: 818-824
Published online: 22 Dec 2011
AbstractforSulfapyridine-like benzenesulfonamide derivatives as inhibitors of carbonic anhydrase isoenzymes I, II and VI | Full Text | References | PDF (645.5 KB)
  • 2541 Views
  • 49 CrossRef citations
  • 0Altmetric
Free Access
Article
Synthesis and anticonvulsant activity of some 2-(2-{1-[substituted phenyl]ethylidene}hydrazinyl)-4-(4-methoxy-phenyl)-6-oxo-1,6-dihydro-pyrimidine-5-carbonitrile
Mohammad Shaquiquzzaman, Suroor Ahmad Khan, Mohammad Amir & Mohammad Mumtaz Alam
Pages: 825-831
Published online: 10 Oct 2011
AbstractforSynthesis and anticonvulsant activity of some 2-(2-{1-[substituted phenyl]ethylidene}hydrazinyl)-4-(4-methoxy-phenyl)-6-oxo-1,6-dihydro-pyrimidine-5-carbonitrile | Full Text | References | PDF (759.5 KB)
  • 746 Views
  • 8 CrossRef citations
  • 0Altmetric
Free Access
Article
Prediction of estrogen receptor β ligands potency and selectivity by docking and MM-GBSA scoring methods using three different scaffolds
B. Balaji & M. Ramanathan
Pages: 832-844
Published online: 14 Oct 2011
AbstractforPrediction of estrogen receptor β ligands potency and selectivity by docking and MM-GBSA scoring methods using three different scaffolds | Full Text | References | PDF (820.7 KB) | Supplemental
  • 1555 Views
  • 15 CrossRef citations
  • 0Altmetric
Free Access
Article
Carbonic anhydrase inhibitors: inhibition of human and bovine isoenzymes by benzenesulphonamides, cyclitols and phenolic compounds
Deniz Ekinci, Namudar I. Kurbanoglu, Emine Salamcı, Murat Şentürk & Claudiu T. Supuran
Pages: 845-848
Published online: 14 Oct 2011
AbstractforCarbonic anhydrase inhibitors: inhibition of human and bovine isoenzymes by benzenesulphonamides, cyclitols and phenolic compounds | Full Text | References | PDF (612.1 KB)
  • 1109 Views
  • 72 CrossRef citations
  • 0Altmetric
Free Access
Article
Synthesis and antibacterial activity of a new series of 3-[3-(substituted phenyl)-1-phenyl-1H-pyrazol-5-yl]-2H-chromen-2-one derivatives
Prashant Aragade, R. Venkat Narayanan, Veeresh Maddi, Pankaj Patil, Prashant Shinde & Mohan Agrawal
Pages: 849-853
Published online: 12 Oct 2011
AbstractforSynthesis and antibacterial activity of a new series of 3-[3-(substituted phenyl)-1-phenyl-1H-pyrazol-5-yl]-2H-chromen-2-one derivatives | Full Text | References | PDF (623.1 KB)
  • 876 Views
  • 6 CrossRef citations
  • 0Altmetric
Free Access
Article
The effect of angiotensin-converting enzyme inhibition by captopril on respiratory mechanics in healthy rats
Alessandro Rubini, Marco Redaelli & Andrea Parmagnani
Pages: 854-860
Published online: 16 May 2012
AbstractforThe effect of angiotensin-converting enzyme inhibition by captopril on respiratory mechanics in healthy rats | Full Text | References | PDF (676.6 KB)
  • 658 Views
  • 9 CrossRef citations
  • 0Altmetric
Free Access
Article
BPTES inhibition of hGA124–551, a truncated form of human kidney-type glutaminase
Erik W. Hartwick & Norman P. Curthoys
Pages: 861-867
Published online: 15 Oct 2011
AbstractforBPTES inhibition of hGA124–551, a truncated form of human kidney-type glutaminase | Full Text | References | PDF (798.4 KB)
  • 2007 Views
  • 31 CrossRef citations
  • 0Altmetric
Free Access
Article
Synthesis, antimicrobial activity and cytotoxicity of some new carbazole derivatives
Zafer Asim Kaplancikli, Leyla Yurttaş, Gülhan Turan-Zitouni, Ahmet Özdemir, Rasime Özic & Şafak Ulusoylar-Yıldırım
Pages: 868-874
Published online: 15 Oct 2011
AbstractforSynthesis, antimicrobial activity and cytotoxicity of some new carbazole derivatives | Full Text | References | PDF (622.3 KB)
  • 1124 Views
  • 18 CrossRef citations
  • 0Altmetric
Free Access
Article
Anti-inflammatory phenolics isolated from Juniperus rigida leaves and twigs in lipopolysaccharide-stimulated RAW264.7 macrophage cells
Eun Ju Jeong, Hanee Seo, Heejung Yang, Jinwoong Kim, Sang Hyun Sung & Young Choong Kim
Pages: 875-879
Published online: 03 Nov 2011
AbstractforAnti-inflammatory phenolics isolated from Juniperus rigida leaves and twigs in lipopolysaccharide-stimulated RAW264.7 macrophage cells | Full Text | References | PDF (792.5 KB)
  • 1277 Views
  • 23 CrossRef citations
  • 0Altmetric
Free Access
Article
Simple methanesulfonates are hydrolyzed by the sulfatase carbonic anhydrase activity
Elif Akın Kazancıoğlu, Murat Güney, Murat Şentürk & Claudiu T. Supuran
Pages: 880-885
Published online: 06 Dec 2011
AbstractforSimple methanesulfonates are hydrolyzed by the sulfatase carbonic anhydrase activity | Full Text | References | PDF (678.8 KB)
  • 1737 Views
  • 53 CrossRef citations
  • 0Altmetric
Free Access
Article
Carbonic Anhydrases inhibitory effects of new benzenesulfonamides synthesized by using superacid chemistry
Fei Liu, Agnès Martin-Mingot, F. Lecornué, Marie-Paule Jouannetaud, Alfonso Maresca, Sebastien Thibaudeau & Claudiu T. Supuran
Pages: 886-891
Published online: 14 Dec 2011
AbstractforCarbonic Anhydrases inhibitory effects of new benzenesulfonamides synthesized by using superacid chemistry | Full Text | References | PDF (716.1 KB)
  • 975 Views
  • 70 CrossRef citations
  • 0Altmetric
Free Access
Article
Biochemical properties of a novel and highly thermostable bacterial α-carbonic anhydrase from Sulfurihydrogenibium yellowstonense YO3AOP1
Clemente Capasso, Viviana De Luca, Vincenzo Carginale, Raffaele Cannio & Mosè Rossi
Pages: 892-897
Published online: 18 Jul 2012
AbstractforBiochemical properties of a novel and highly thermostable bacterial α-carbonic anhydrase from Sulfurihydrogenibium yellowstonense YO3AOP1 | Full Text | References | PDF (700.2 KB)
  • 4719 Views
  • 103 CrossRef citations
  • 0Altmetric
Free Access

Retraction

Retraction
Statement of retraction
Page: 898
Published online: 29 May 2012
CitationforStatement of retraction | Full Text | PDF (538.4 KB)
  • 847 Views
  • 0 CrossRef citations
  • 0Altmetric
Free Access

Errata

Correction
Erratum
Page: 899
Published online: 16 Oct 2012
CitationforErratum | Full Text | PDF (533.2 KB)
  • 478 Views
  • 0 CrossRef citations
  • 0Altmetric
Free Access

Explore articles