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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 34, 2019 - Issue 1
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Research Paper

Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies

Alessandra AmmazzalorsoDepartment of Pharmacy, “G. d’Annunzio” University of Chieti-Pescara, Chieti, Italy; Correspondence[email protected]
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Simone CarradoriDepartment of Pharmacy, “G. d’Annunzio” University of Chieti-Pescara, Chieti, Italy; ORCID Iconhttp://orcid.org/0000-0002-8698-9440View further author information
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Andrea AngeliLaboratorio di Chimica Bioinorganica, Università degli Studi di Firenze, Florence, Italy; ORCID Iconhttp://orcid.org/0000-0002-1470-7192View further author information
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Atilla AkdemirDepartment of Pharmacology, Faculty of Pharmacy, Computer-Aided Drug Discovery Laboratory, Bezmialem Vakif University, Istanbul, Turkey; View further author information
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Barbara De FilippisDepartment of Pharmacy, “G. d’Annunzio” University of Chieti-Pescara, Chieti, Italy; View further author information
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Marialuigia FantacuzziDepartment of Pharmacy, “G. d’Annunzio” University of Chieti-Pescara, Chieti, Italy; View further author information
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Letizia GiampietroDepartment of Pharmacy, “G. d’Annunzio” University of Chieti-Pescara, Chieti, Italy; View further author information
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Cristina MaccalliniDepartment of Pharmacy, “G. d’Annunzio” University of Chieti-Pescara, Chieti, Italy; View further author information
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Rosa AmorosoDepartment of Pharmacy, “G. d’Annunzio” University of Chieti-Pescara, Chieti, Italy; View further author information
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Claudiu T. SupuranLaboratorio di Chimica Bioinorganica, Università degli Studi di Firenze, Florence, Italy; ;Neurofarba Department, Section of Pharmaceutical and Nutriceutical Sciences, Università degli Studi di Firenze, Florence, ItalyCorrespondence[email protected]
ORCID Iconhttp://orcid.org/0000-0003-4262-0323View further author information
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Pages 1051-1061 | Received 06 Mar 2019, Accepted 19 Apr 2019, Published online: 10 May 2019

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Emma Baglini, Rahul Ravichandran, Emanuela Berrino, Silvia Salerno, Elisabetta Barresi, Anna Maria Marini, Monica Viviano, Sabrina Castellano, Federico Da Settimo, Claudiu T. Supuran, Sandro Cosconati & Sabrina Taliani. (2021) Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 1874-1883.
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Claudiu T. Supuran. (2020) Exploring the multiple binding modes of inhibitors to carbonic anhydrases for novel drug discovery. Expert Opinion on Drug Discovery 15:6, pages 671-686.
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Mehmet Oguz, Erbay Kalay, Suleyman Akocak, Alessio Nocentini, Nebih Lolak, Mehmet Boga, Mustafa Yilmaz & Claudiu T. Supuran. (2020) Synthesis of calix[4]azacrown substituted sulphonamides with antioxidant, acetylcholinesterase, butyrylcholinesterase, tyrosinase and carbonic anhydrase inhibitory action. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1215-1223.
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Hasan Küçükbay, Zeynep Gönül, F. Zehra Küçükbay, Andrea Angeli, Gianluca Bartolucci & Claudiu T. Supuran. (2020) Preparation, carbonic anhydrase enzyme inhibition and antioxidant activity of novel 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives incorporating mono or dipeptide moiety. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1021-1026.
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Ali Irfan, Fozia Batool, Syeda Andleeb Zahra Naqvi, Amjad Islam, Sameh M. Osman, Alessio Nocentini, Siham A. Alissa & Claudiu T. Supuran. (2020) Benzothiazole derivatives as anticancer agents. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 265-279.
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Alessio Nocentini & Claudiu T. Supuran. (2019) Advances in the structural annotation of human carbonic anhydrases and impact on future drug discovery. Expert Opinion on Drug Discovery 14:11, pages 1175-1197.
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Giulia Rotondi, Paolo Guglielmi, Simone Carradori, Daniela Secci, Celeste De Monte, Barbara De Filippis, Cristina Maccallini, Rosa Amoroso, Roberto Cirilli, Atilla Akdemir, Andrea Angeli & Claudiu T. Supuran. (2019) Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1400-1413.
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Articles from other publishers (6)

Cansu Öztürk, Erbay Kalay, Serpil Gerni, Neslihan Balci, Feyzi Sinan Tokali, Osman Nuri Aslan & Emrah Polat. (2023) Sulfonamide derivatives with benzothiazole scaffold: Synthesis and carbonic anhydrase I–II inhibition properties. Biotechnology and Applied Biochemistry.
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Romain Amador, Adrien Delpal, Bruno Canard, Jean-Jacques Vasseur, Etienne Decroly, Françoise Debart, Guillaume Clavé & Michael Smietana. (2022) Facile access to 4′-( N -acylsulfonamide) modified nucleosides and evaluation of their inhibitory activity against SARS-CoV-2 RNA cap N 7-guanine-methyltransferase nsp14 . Organic & Biomolecular Chemistry 20:38, pages 7582-7586.
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Simone Carradori, Paolo Guglielmi, Grazia Luisi & Daniela Secci. 2022. Handbook of Oxidative Stress in Cancer: Mechanistic Aspects. Handbook of Oxidative Stress in Cancer: Mechanistic Aspects 2571 2588 .
Silvia Salerno, Giorgio Amendola, Andrea Angeli, Emma Baglini, Elisabetta Barresi, Anna Maria Marini, Rahul Ravichandran, Monica Viviano, Sabrina Castellano, Ettore Novellino, Federico Da Settimo, Claudiu T. Supuran, Sandro Cosconati & Sabrina Taliani. (2021) Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold. European Journal of Medicinal Chemistry 220, pages 113490.
Crossref
Simone Carradori, Paolo Guglielmi, Grazia Luisi & Daniela Secci. 2020. Handbook of Oxidative Stress in Cancer: Mechanistic Aspects. Handbook of Oxidative Stress in Cancer: Mechanistic Aspects 1 18 .
Alessandra Ammazzalorso, Simone Carradori, Rosa Amoroso & Inmaculada Fernández Fernández. (2020) 2-substituted benzothiazoles as antiproliferative agents: Novel insights on structure-activity relationships. European Journal of Medicinal Chemistry 207, pages 112762.
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