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Lipid nanoparticles: state of the art, new preparation methods and challenges in drug delivery

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Pages 497-508 | Published online: 22 Mar 2012

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Wenhui Xue, Tingting Li, Ying Gu, Shaowei Li & Ningshao Xia. (2023) Molecular engineering tools for the development of vaccines against infectious diseases: current status and future directions. Expert Review of Vaccines 22:1, pages 563-578.
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Mohamed Fawzi Kabil, Osama A. Badary, Frank Bier, Shaker A. Mousa & Ibrahim M. El-Sherbiny. (2023) A comprehensive review on lipid nanocarrier systems for cancer treatment: fabrication, future prospects and clinical trials. Journal of Liposome Research 0:0, pages 1-43.
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Aisha Aziz, Urushi Rehman, Afsana Sheikh, Mohammed A. S. Abourehab & Prashant Kesharwani. (2023) Lipid-based nanocarrier mediated CRISPR/Cas9 delivery for cancer therapy. Journal of Biomaterials Science, Polymer Edition 34:3, pages 398-418.
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Andrea Perrelli, Parisa Fatehbasharzad, Valerio Benedetti, Chiara Ferraris, Marco Fontanella, Elisa De Luca, Mauro Moglianetti, Luigi Battaglia & Saverio Francesco Retta. (2021) Towards precision nanomedicine for cerebrovascular diseases with emphasis on Cerebral Cavernous Malformation (CCM). Expert Opinion on Drug Delivery 18:7, pages 849-876.
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Fatin Hannani Zakarial Ansar, Saiful Yazan Latifah, Wan Hamirul Bahrin Wan Kamal, Khei Choong Khong, Yen Ng, Jia Ning Foong, Banulata Gopalsamy, Wei Keat Ng, Chee Wun How, Yong Sze Ong, Rasedee Abdullah & Mohd Yusmaidie Aziz. (2020) Pharmacokinetics and Biodistribution of Thymoquinone-loaded Nanostructured Lipid Carrier After Oral and Intravenous Administration into Rats. International Journal of Nanomedicine 15, pages 7703-7717.
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Silvia Mannucci, Federico Boschi, Barbara Cisterna, Elisabetta Esposito, Rita Cortesi, Claudio Nastruzzi, Enrica Cappellozza, Paolo Bernardi, Andrea Sbarbati, Manuela Malatesta & Laura Calderan. (2020) A Correlative Imaging Study of in vivo and ex vivo Biodistribution of Solid Lipid Nanoparticles. International Journal of Nanomedicine 15, pages 1745-1758.
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Victor Hugo Sousa Araujo, Jonatas Lobato Duarte, Gabriela Corrêa Carvalho, Amanda Letícia Polli Silvestre, Bruno Fonseca-Santos, Gabriel Davi Marena, Tais de Cassia Ribeiro, Matheus Aparecido dos Santos Ramos, Taís Maria Bauab & Marlus Chorilli. (2020) Nanosystems against candidiasis: a review of studies performed over the last two decades. Critical Reviews in Microbiology 46:5, pages 508-547.
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Eliana B. Souto, Iara Baldim, Wanderley P. Oliveira, Rekha Rao, Nitesh Yadav, Francisco M. Gama & Sheefali Mahant. (2020) SLN and NLC for topical, dermal, and transdermal drug delivery. Expert Opinion on Drug Delivery 17:3, pages 357-377.
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Rishi Paliwal, Shivani Rai Paliwal, Rameshroo Kenwat, Balak Das Kurmi & Mukesh Kumar Sahu. (2020) Solid lipid nanoparticles: a review on recent perspectives and patents. Expert Opinion on Therapeutic Patents 30:3, pages 179-194.
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Qingming Ma, Yang Gao, Wentao Sun, Jie Cao, Yan Liang, Shangcong Han, Xinyu Wang & Yong Sun. (2020) Self-Assembled chitosan/phospholipid nanoparticles: from fundamentals to preparation for advanced drug delivery. Drug Delivery 27:1, pages 200-215.
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Daniela Lopes-de-Campos, Rita M Pinto, Sofia A Costa Lima, Tiago Santos, Bruno Sarmento, Cláudia Nunes & Salette Reis. (2019) Delivering amoxicillin at the infection site – a rational design through lipid nanoparticles. International Journal of Nanomedicine 14, pages 2781-2795.
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Chiara Bianca Maria Platania, Michele Dei Cas, Simona Cianciolo, Annamaria Fidilio, Francesca Lazzara, Rita Paroni, Rosario Pignatello, Enrica Strettoi, Riccardo Ghidoni, Filippo Drago & Claudio Bucolo. (2019) Novel ophthalmic formulation of myriocin: implications in retinitis pigmentosa. Drug Delivery 26:1, pages 237-243.
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Luigi Battaglia, Pier Paolo Panciani, Elisabetta Muntoni, Maria Teresa Capucchio, Elena Biasibetti, Pasquale De Bonis, Silvia Mioletti, Marco Fontanella & Shankar Swaminathan. (2018) Lipid nanoparticles for intranasal administration: application to nose-to-brain delivery. Expert Opinion on Drug Delivery 15:4, pages 369-378.
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Natascia Bruni, Barbara Stella, Leonardo Giraudo, Carlo Della Pepa, Daniela Gastaldi & Franco Dosio. (2017) Nanostructured delivery systems with improved leishmanicidal activity: a critical review. International Journal of Nanomedicine 12, pages 5289-5311.
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Ahmed M Fatouh, Ahmed H Elshafeey & Ahmed Abdelbary. (2017) Intranasal agomelatine solid lipid nanoparticles to enhance brain delivery: formulation, optimization and in vivo pharmacokinetics. Drug Design, Development and Therapy 11, pages 1815-1825.
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Sally Safwat, Rania A. H. Ishak, Rania M. Hathout & Nahed D. Mortada. (2017) Nanostructured lipid carriers loaded with simvastatin: effect of PEG/glycerides on characterization, stability, cellular uptake efficiency and in vitro cytotoxicity. Drug Development and Industrial Pharmacy 43:7, pages 1112-1125.
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Rita Cortesi, Giuseppe Valacchi, Ximena Maria Muresan, Markus Drechsler, Catia Contado, Elisabetta Esposito, Alessandro Grandini, Alessandra Guerrini, Giuseppe Forlani & Gianni Sacchetti. (2017) Nanostructured lipid carriers (NLC) for the delivery of natural molecules with antimicrobial activity: production, characterisation and in vitro studies. Journal of Microencapsulation 34:1, pages 63-72.
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Ahmed M. Fatouh, Ahmed H. Elshafeey & Ahmed Abdelbary. (2017) Agomelatine-based in situ gels for brain targeting via the nasal route: statistical optimization, in vitro, and in vivo evaluation. Drug Delivery 24:1, pages 1077-1085.
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Luigi Battaglia, Loredana Serpe, Federica Foglietta, Elisabetta Muntoni, Marina Gallarate, Ana Del Pozo Rodriguez & Maria Angeles Solinis. (2016) Application of lipid nanoparticles to ocular drug delivery. Expert Opinion on Drug Delivery 13:12, pages 1743-1757.
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Stefan Lorscheidt & Alf Lamprecht. (2016) Safety assessment of nanoparticles for drug delivery by means of classic in vitro assays and beyond. Expert Opinion on Drug Delivery 13:11, pages 1545-1558.
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Débora Sgorla, Élcio J. Bunhak, Osvaldo A. Cavalcanti, Pedro Fonte & Bruno Sarmento. (2016) Exploitation of lipid-polymeric matrices at nanoscale for drug delivery applications. Expert Opinion on Drug Delivery 13:9, pages 1301-1309.
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Ibrahim Elsayed & Mohamed Hassan Hany AbouGhaly. (2016) Inhalable nanocomposite microparticles: preparation, characterization and factors affecting formulation. Expert Opinion on Drug Delivery 13:2, pages 207-222.
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Giovana Calixto, Jéssica Bernegossi, Bruno Fonseca-Santos & Marlus Chorilli. (2014) Nanotechnology-based drug delivery systems for treatment of oral cancer: a review. International Journal of Nanomedicine 9, pages 3719-3735.
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Rahul Sonawane, Harshad Harde, Mahesh Katariya, Satyam Agrawal & Sanyog Jain. (2014) Solid lipid nanoparticles-loaded topical gel containing combination drugs: an approach to offset psoriasis. Expert Opinion on Drug Delivery 11:12, pages 1833-1847.
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Wenting Xu, Soo-Jeong Lim & Mi-Kyung Lee. (2013) Cellular uptake and antitumour activity of paclitaxel incorporated into trilaurin-based solid lipid nanoparticles in ovarian cancer. Journal of Microencapsulation 30:8, pages 755-761.
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Daniele R de Araújo, Deyse C da Silva, Raquel M Barbosa, Michelle Franz-Montan, Cíntia MS Cereda, Cristina Padula, Patrizia Santi & Eneida de Paula. (2013) Strategies for delivering local anesthetics to the skin: focus on liposomes, solid lipid nanoparticles, hydrogels and patches. Expert Opinion on Drug Delivery 10:11, pages 1551-1563.
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Medha Patel, Eliana B Souto & Kamalinder K Singh. (2013) Advances in brain drug targeting and delivery: limitations and challenges of solid lipid nanoparticles. Expert Opinion on Drug Delivery 10:7, pages 889-905.
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Eneida de Paula, Cíntia MS Cereda, Leonardo F Fraceto, Daniele R de Araújo, Michelle Franz-Montan, Giovana R Tofoli, José Ranali, Maria C Volpato & Francisco C Groppo. (2012) Micro and nanosystems for delivering local anesthetics. Expert Opinion on Drug Delivery 9:12, pages 1505-1524.
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Beatriz Lasa-Saracibar, Ander Estella-Hermoso de Mendoza, Melissa Guada, Carmen Dios-Vieitez & María J Blanco-Prieto. (2012) Lipid nanoparticles for cancer therapy: state of the art and future prospects. Expert Opinion on Drug Delivery 9:10, pages 1245-1261.
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Elisabetta Esposito, Rita Cortesi, Markus Drechsler, Jie Fan, Bingmei M. Fu, Laura Calderan, Silvia Mannucci, Federico Boschi & Claudio Nastruzzi. (2017) Nanoformulations for dimethyl fumarate: Physicochemical characterization and in vitro / in vivo behavior. European Journal of Pharmaceutics and Biopharmaceutics 115, pages 285-296.
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