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Original Research

An optimized probucol microencapsulated formulation integrating a secondary bile acid (deoxycholic acid) as a permeation enhancer

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Pages 1673-1683 | Published online: 29 Sep 2014

Keep up to date with the latest research on this topic with citation updates for this article.

Read on this site (10)

Armin Mooranian, Thomas Foster, Corina M Ionescu, Louise Carey, Daniel Walker, Melissa Jones, Susbin Raj Wagle, Bozica Kovacevic, Jacqueline Chester, Edan Johnstone, Jafri Kuthubutheen, Daniel Brown, Marcus D Atlas, Momir Mikov & Hani Al-Salami. (2021) The Effects of Primary Unconjugated Bile Acids on Nanoencapsulated Pharmaceutical Formulation of Hydrophilic Drugs: Pharmacological Implications. Drug Design, Development and Therapy 15, pages 4423-4434.
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Armin Mooranian, Nassim Zamani, Momir Mikov, Svetlana Goločorbin-Kon, Goran Stojanovic, Frank Arfuso, Bozica Kovacevic & Hani Al-Salami. (2020) Bio Micro-Nano Technologies of Antioxidants Optimised Their Pharmacological and Cellular Effects, ex vivo, in Pancreatic β-Cells. Nanotechnology, Science and Applications 13, pages 1-9.
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Susbin Raj Wagle, Bozica Kovacevic, Daniel Walker, Corina Mihaela Ionescu, Umar Shah, Goran Stojanovic, Sanja Kojic, Armin Mooranian & Hani Al-Salami. (2020) Alginate-based drug oral targeting using bio-micro/nano encapsulation technologies. Expert Opinion on Drug Delivery 17:10, pages 1361-1376.
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Armin Mooranian, Nassim Zamani, Giuseppe Luna, Hesham Al-Sallami, Momir Mikov, Svetlana Goločorbin-Kon, Goran Stojanovic, Frank Arfuso, Bozica Kovacevic & Hani Al-Salami. (2019) Bile acid-polymer-probucol microparticles: protective effect on pancreatic β-cells and decrease in type 1 diabetes development in a murine model. Pharmaceutical Development and Technology 24:10, pages 1272-1277.
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Armin Mooranian, Nassim Zamani, Momir Mikov, Svetlana Goločorbin-Kon, Goran Stojanovic, Frank Arfuso & Hani Al-Salami. (2018) Novel nano-encapsulation of probucol in microgels: scanning electron micrograph characterizations, buoyancy profiling, and antioxidant assay analyses. Artificial Cells, Nanomedicine, and Biotechnology 46:sup3, pages 741-747.
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Armin Mooranian, Rebecca Negrulj, Frank Arfuso & Hani Al-Salami. (2016) Multicompartmental, multilayered probucol microcapsules for diabetes mellitus: Formulation characterization and effects on production of insulin and inflammation in a pancreatic β-cell line. Artificial Cells, Nanomedicine, and Biotechnology 44:7, pages 1642-1653.
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Sangeetha Mathavan, Nigel Chen-Tan, Frank Arfuso & Hani Al-Salami. (2016) The role of the bile acid chenodeoxycholic acid in the targeted oral delivery of the anti-diabetic drug gliclazide, and its applications in type 1 diabetes. Artificial Cells, Nanomedicine, and Biotechnology 44:6, pages 1508-1519.
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Armin Mooranian, Rebecca Negrulj, Momir Mikov, Svetlana Golocorbin-Kon, Frank Arfuso & Hani Al-Salami. (2015) Novel chenodeoxycholic acid–sodium alginate matrix in the microencapsulation of the potential antidiabetic drug, probucol. An in vitro study. Journal of Microencapsulation 32:6, pages 589-597.
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Articles from other publishers (10)

ShiQuan Wu, LiMin Lu, Li Li, QiQi Liang, HuaXu Gao, TianYu Tang & YanLin Tang. (2023) Density functional studies of probucol excited states and spectral properties. The European Physical Journal D 77:1.
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Branislava Teofilovic, Svetlana Golocorbin-Kon, Nebojsa Stilinovic, Nevena Grujic-Letic, Aleksandar Raškovic, Armin Mooranian, Hani Al-Salami & Momir Mikov. (2021) Pharmacological effects of novel microvesicles of basil, on blood glucose and the lipid profile: a preclinical study. Scientific Reports 11:1.
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Susbin Raj Wagle, Bozica Kovacevic, Corina Mihaela Ionescu, Daniel Walker, Melissa Jones, Louise Carey, Ryusuke Takechi, Momir Mikov, Armin Mooranian & Hani Al-Salami. (2021) Pharmacological and Biological Study of Microencapsulated Probucol-Secondary Bile Acid in a Diseased Mouse Model. Pharmaceutics 13:8, pages 1223.
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Armin Mooranian, Thomas Foster, Corina M. Ionescu, Daniel Walker, Melissa Jones, Susbin Raj Wagle, Bozica Kovacevic, Jacqueline Chester, Edan Johnston, Elaine Wong, Marcus D. Atlas, Momir Mikov & Hani Al-Salami. (2021) Enhanced Bilosomal Properties Resulted in Optimum Pharmacological Effects by Increased Acidification Pathways. Pharmaceutics 13:8, pages 1184.
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Jacqueline Chester, Edan Johnston, Daniel Walker, Melissa Jones, Corina Mihaela Ionescu, Susbin Raj Wagle, Božica Kovacevic, Daniel Brown, Momir Mikov, Armin Mooranian & Hani Al-Salami. (2021) A Review on Recent Advancement on Age-Related Hearing Loss: The Applications of Nanotechnology, Drug Pharmacology, and Biotechnology. Pharmaceutics 13:7, pages 1041.
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Armin Mooranian, Nassim Zamani, Corina M. Ionescu, Ryu Takechi, Giuseppe Luna, Momir Mikov, Svetlana Goločorbin-Kon, Božica Kovačević & Hani Al-Salami. (2020) Oral gavage of nano-encapsulated conjugated acrylic acid-bile acid formulation in type 1 diabetes altered pharmacological profile of bile acids, and improved glycaemia and suppressed inflammation. Pharmacological Reports 72:2, pages 368-378.
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Nebojša Pavlović, Svetlana Goločorbin-Kon, Maja Ðanić, Bojan Stanimirov, Hani Al-Salami, Karmen Stankov & Momir Mikov. (2018) Bile Acids and Their Derivatives as Potential Modifiers of Drug Release and Pharmacokinetic Profiles. Frontiers in Pharmacology 9.
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Armin Mooranian, Rebecca Negrulj, Ryu Takechi, John Mamo, Hesham Al-Sallami & Hani Al-Salami. (2018) The biological effects of the hypolipidaemic drug probucol microcapsules fed daily for 4 weeks, to an insulin-resistant mouse model: potential hypoglycaemic and anti-inflammatory effects. Drug Delivery and Translational Research 8:3, pages 543-551.
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Armin Mooranian, Rebecca Negrulj, Ryu Takechi, Emma Jamieson, Grant Morahan & Hani Al-Salami. (2017) New Biotechnological Microencapsulating Methodology Utilizing Individualized Gradient-Screened Jet Laminar Flow Techniques for Pancreatic β-Cell Delivery: Bile Acids Support Cell Energy-Generating Mechanisms. Molecular Pharmaceutics 14:8, pages 2711-2718.
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Armin Mooranian, Rebecca Negrulj & Hani Al-Salami. (2016) Primary Bile Acid Chenodeoxycholic Acid-Based Microcapsules to Examine β-cell Survival and the Inflammatory Response. BioNanoScience 6:2, pages 103-109.
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