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Acetazolamide for the treatment of idiopathic intracranial hypertension

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Andrea Angeli & Claudiu T. Supuran. (2023) Click chemistry approaches for developing carbonic anhydrase inhibitors and their applications. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Maan T. Khayat, Hany E. A. Ahmed, Abdelsattar M. Omar, Yosra A. Muhammad, Khadijah A. Mohammad, Azizah M. Malebari, Ahdab N. Khayyat, Ahmed H. Halawa, Hamada S. Abulkhair, Ahmed A. Al-Karmalawy, Mohammed Almaghrabi, Majed Alharbi, Anfal S. Aljahdali & Ahmed M. El-Agrody. (2023) A novel class of phenylpyrazolone-sulphonamides rigid synthetic anticancer molecules selectively inhibit the isoform IX of carbonic anhydrases guided by molecular docking and orbital analyses. Journal of Biomolecular Structure and Dynamics 0:0, pages 1-19.
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Mahmoud F. Abo-Ashour, Hadia Almahli, Alessandro Bonardi, Amira Khalil, Tarfah Al-Warhi, Sara T. Al-Rashood, Hatem A. Abdel-Aziz, Alessio Nocentini, Claudiu T. Supuran & Wagdy M. Eldehna. (2022) Enaminone-based carboxylic acids as novel non-classical carbonic anhydrases inhibitors: design, synthesis and in vitro biological assessment. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 2256-2264.
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Tatiana Sharonova, Petr Zhmurov, Stanislav Kalinin, Alessio Nocentini, Andrea Angeli, Marta Ferraroni, Mikhail Korsakov, Claudiu T. Supuran & Mikhail Krasavin. (2022) Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 857-865.
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Mona F. Said, Riham F. George, Andrea Petreni, Claudiu T. Supuran & Nada M. Mohamed. (2022) Synthesis, molecular modelling and QSAR study of new N-phenylacetamide-2-oxoindole benzensulfonamide conjugates as carbonic anhydrase inhibitors with antiproliferative activity. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 701-717.
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Silvia Mussi, Sara Rezzola, Paola Chiodelli, Alessio Nocentini, Claudiu T. Supuran & Roberto Ronca. (2022) Antiproliferative effects of sulphonamide carbonic anhydrase inhibitors C18, SLC-0111 and acetazolamide on bladder, glioblastoma and pancreatic cancer cell lines. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 280-286.
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Gustavo Provensi, Alessio Nocentini, Maria Beatrice Passani, Patrizio Blandina & Claudiu T. Supuran. (2021) Activation of carbonic anhydrase isoforms involved in modulation of emotional memory and cognitive disorders with histamine agonists, antagonists and derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 719-726.
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Alessio Nocentini, Andrea Angeli, Fabrizio Carta, Jean-Yves Winum, Raivis Zalubovskis, Simone Carradori, Clemente Capasso, William A. Donald & Claudiu T. Supuran. (2021) Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 561-580.
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Claudiu T. Supuran. (2020) Exploring the multiple binding modes of inhibitors to carbonic anhydrases for novel drug discovery. Expert Opinion on Drug Discovery 15:6, pages 671-686.
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Claudiu T. Supuran. (2020) An update on drug interaction considerations in the therapeutic use of carbonic anhydrase inhibitors. Expert Opinion on Drug Metabolism & Toxicology 16:4, pages 297-307.
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Claudiu T. Supuran. (2020) Coumarin carbonic anhydrase inhibitors from natural sources. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1462-1470.
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Patrizio Blandina, Gustavo Provensi, Maria Beatrice Passani, Clemente Capasso & Claudiu T. Supuran. (2020) Carbonic anhydrase modulation of emotional memory. Implications for the treatment of cognitive disorders. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1206-1214.
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Hasan Küçükbay, Zeynep Gönül, F. Zehra Küçükbay, Andrea Angeli, Gianluca Bartolucci & Claudiu T. Supuran. (2020) Preparation, carbonic anhydrase enzyme inhibition and antioxidant activity of novel 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives incorporating mono or dipeptide moiety. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1021-1026.
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Barbara Kaproń, Robert Czarnomysy, Mariusz Wysokiński, Rudolf Andrys, Kamil Musilek, Andrea Angeli, Claudiu T. Supuran & Tomasz Plech. (2020) 1,2,4-Triazole-based anticonvulsant agents with additional ROS scavenging activity are effective in a model of pharmacoresistant epilepsy. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 993-1002.
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Jeremie Brichet, Rodrigo Arancibia, Emanuela Berrino & Claudiu T. Supuran. (2020) Bioorganometallic derivatives of 4-hydrazino-benzenesulphonamide as carbonic anhydrase inhibitors: synthesis, characterisation and biological evaluation. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 622-628.
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Manuel A. Llanos, María L. Sbaraglini, María L. Villalba, María D. Ruiz, Carolina Carrillo, Catalina Alba Soto, Alan Talevi, Andrea Angeli, Seppo Parkkila, Claudiu T. Supuran & Luciana Gavernet. (2020) A structure-based approach towards the identification of novel antichagasic compounds: Trypanosoma cruzi carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 21-30.
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Alessio Nocentini & Claudiu T. Supuran. (2019) Advances in the structural annotation of human carbonic anhydrases and impact on future drug discovery. Expert Opinion on Drug Discovery 14:11, pages 1175-1197.
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Deborah I. Friedman. (2019) Contemporary management of the pseudotumor cerebri syndrome. Expert Review of Neurotherapeutics 19:9, pages 881-893.
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Mohammad M. Al-Sanea, Ahmed Elkamhawy, Sora Paik, Silvia Bua, So Ha Lee, Mohamed A. Abdelgawad, Eun Joo Roh, Wagdy M. Eldehna & Claudiu T. Supuran. (2019) Synthesis and biological evaluation of novel 3-(quinolin-4-ylamino)benzenesulfonamides as carbonic anhydrase isoforms I and II inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1457-1464.
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Pavitra S. Thacker, Pirpasha Shaikh, Andrea Angeli, Mohammed Arifuddin & Claudiu T. Supuran. (2019) Synthesis and biological evaluation of novel 8-substituted quinoline-2-carboxamides as carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1172-1177.
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Claudiu T. Supuran. (2018) Carbonic anhydrase inhibitors as emerging agents for the treatment and imaging of hypoxic tumors. Expert Opinion on Investigational Drugs 27:12, pages 963-970.
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Claudiu T. Supuran. (2018) Carbonic anhydrase inhibitors and their potential in a range of therapeutic areas. Expert Opinion on Therapeutic Patents 28:10, pages 709-712.
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Claudiu T. Supuran. (2018) Applications of carbonic anhydrases inhibitors in renal and central nervous system diseases. Expert Opinion on Therapeutic Patents 28:10, pages 713-721.
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Claudiu T. Supuran & Clemente Capasso. (2018) Biomedical applications of prokaryotic carbonic anhydrases. Expert Opinion on Therapeutic Patents 28:10, pages 745-754.
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Claudiu T. Supuran. (2018) Carbon- versus sulphur-based zinc binding groups for carbonic anhydrase inhibitors?. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 485-495.
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Vincenzo Alterio, Davide Esposito, Simona Maria Monti, Claudiu T. Supuran & Giuseppina De Simone. (2018) Crystal structure of the human carbonic anhydrase II adduct with 1-(4-sulfamoylphenyl-ethyl)-2,4,6-triphenylpyridinium perchlorate, a membrane-impermeant, isoform selective inhibitor. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 151-157.
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Daniela Vullo, R. Siva Sai Kumar, Andrea Scozzafava, James G. Ferry & Claudiu T. Supuran. (2018) Sulphonamide inhibition studies of the β-carbonic anhydrase from the bacterial pathogen Clostridium perfringens. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 31-36.
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Claudiu T. Supuran. (2017) Advances in structure-based drug discovery of carbonic anhydrase inhibitors. Expert Opinion on Drug Discovery 12:1, pages 61-88.
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Morteza Abdoli, Andrea Angeli, Murat Bozdag, Fabrizio Carta, Ali Kakanejadifard, Hamid Saeidian & Claudiu T. Supuran. (2017) Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo[d]thiazole-5- and 6-sulfonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1071-1078.
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Murat Bozdag, Silvia Bua, Sameh M. Osman, Zeid AlOthman & Claudiu T. Supuran. (2017) Carbonic anhydrase I, II, IV and IX inhibition with a series of 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 885-892.
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Aleksandrs Pustenko, Dmitrijs Stepanovs, Raivis Žalubovskis, Daniela Vullo, Andris Kazaks, Janis Leitans, Kaspars Tars & Claudiu T. Supuran. (2017) 3H-1,2-benzoxathiepine 2,2-dioxides: a new class of isoform-selective carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 767-775.
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Marco Bragagni, Fabrizio Carta, Sameh M. Osman, Zeid AlOthman & Claudiu T. Supuran. (2017) Synthesis of an acridine orange sulfonamide derivative with potent carbonic anhydrase IX inhibitory action. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 701-706.
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Erol Licsandru, Muhammet Tanc, Istvan Kocsis, Mihail Barboiu & Claudiu T. Supuran. (2017) A class of carbonic anhydrase I – selective activators. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 37-46.
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Chandra Bhushan Mishra, Shikha Kumari, Andrea Angeli, Simona Maria Monti, Martina Buonanno, Amresh Prakash, Manisha Tiwari & Claudiu T. Supuran. (2016) Design, synthesis and biological evaluation of N-(5-methyl-isoxazol-3-yl/1,3,4-thiadiazol-2-yl)-4-(3-substitutedphenylureido) benzenesulfonamides as human carbonic anhydrase isoenzymes I, II, VII and XII inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 31:sup2, pages 174-179.
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F. Zehra Küçükbay, Hasan Küçükbay, Muhammet Tanc & Claudiu T. Supuran. (2016) Synthesis and carbonic anhydrase I, II, IV and XII inhibitory properties of N-protected amino acid – sulfonamide conjugates. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1476-1483.
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Claudiu T. Supuran & Clemente Capasso. (2016) New light on bacterial carbonic anhydrases phylogeny based on the analysis of signal peptide sequences. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1254-1260.
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Claudiu T. Supuran. (2016) Carbonic anhydrase inhibition and the management of neuropathic pain. Expert Review of Neurotherapeutics 16:8, pages 961-968.
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Claudiu T. Supuran. (2016) How many carbonic anhydrase inhibition mechanisms exist?. Journal of Enzyme Inhibition and Medicinal Chemistry 31:3, pages 345-360.
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Claudiu T. Supuran. (2016) Drug interaction considerations in the therapeutic use of carbonic anhydrase inhibitors. Expert Opinion on Drug Metabolism & Toxicology 12:4, pages 423-431.
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Yarden Bulkowstein, Adi Nitzan‑Luques, Aviad Schnapp, Noa Barnoy, Shimon Reif, Tal Gilboa & Oded Volovesky. (2023) The manifestations of metabolic acidosis during acetazolamide treatment in a cohort of pediatric idiopathic intracranial hypertension. Pediatric Nephrology 39:1, pages 185-191.
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Benjamin J. Umlauf, Gabriel Frampton, Alexis Cooper & Hannah-Faith Greene. (2023) A novel strategy to increase the therapeutic potency of GBM chemotherapy via altering parenchymal/cerebral spinal fluid clearance rate. Journal of Controlled Release 364, pages 195-205.
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Darya Fayzullina, Semyon Yakushov, Kamilla Kantserova, Elizaveta Belyaeva, Denis Aniskin, Sergey Tsibulnikov, Nafisa Fayzullina, Stanislav Kalinin, Olga Romantsova, Peter S. Timashev, Brett A. Schroeder & Ilya V. Ulasov. (2023) Carbonic Anhydrase Inhibitors Induce Ferroptosis through Inhibition of AKT/FTH1 Signaling in Ewing Sarcoma Tumor Cells. Cancers 15:21, pages 5225.
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Abhishek Goyal & Katherine Zarroli. (2023) Should topiramate be initial therapy in the management of idiopathic intracranial hypertension?: A literature review. Medicine 102:42, pages e35545.
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Ayse Er. (2023) Various Carbonic Anhydrases in Physiopathological Events, Carbonic Anhydrase Inhibitors, and Hybrid Compounds. Letters in Drug Design & Discovery 20:10, pages 1427-1436.
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Claudiu T. Supuran. (2023) A simple yet multifaceted 90 years old, evergreen enzyme: Carbonic anhydrase, its inhibition and activation. Bioorganic & Medicinal Chemistry Letters 93, pages 129411.
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Inês T. Tavares, Ramón Rivero, José P. Sales‐Luís, Carlo G. Vaudano, Sérgio D. Correia, Juan Alberto Corbera & Jose Raduan Jaber. (2023) Premedication with acetazolamide: Is its use for postoperative pain and stress control after laparoscopic ovariectomy in dogs ruled out?. Veterinary Medicine and Science.
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Alexey Lukin, Lyubov Vinogradova, Kristina Komarova, Stanislav Kalinin & Mikhail Krasavin. (2023) Synthesis of 1-oxa-9-azaspiro[5.5]undecane-9-sulfonamides bearing a diverse molecular periphery and a rare zinc-binding group for carbonic anhydrase interrogation. Mendeleev Communications 33:2, pages 191-193.
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Nikolina Sibinčić, Stanislav Kalinin, Vladimir Sharoyko, Julia Efimova, Olga A. Gasilina, Mikhail Korsakov, Maxim Gureev & Mikhail Krasavin. (2023) A Series of Trifluoromethylisoxazolyl- and Trifluoromethylpyrazolyl- Substituted (Hetero)aromatic Sulfonamide Carbonic Anhydrase Inhibitors: Synthesis, and Convenient Prioritization Workflow for Further In Vivo Studies. Medicinal Chemistry 19:2, pages 193-210.
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Melisa E. Gantner, Denis N. Prada Gori, Manuel A. Llanos, Alan Talevi, Andrea Angeli, Daniela Vullo, Claudiu T. Supuran & Luciana Gavernet. (2022) Identification of New Carbonic Anhydrase VII Inhibitors by Structure-Based Virtual Screening. Journal of Chemical Information and Modeling 62:19, pages 4760-4770.
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Khadija Karim, Abderrahman Lamaoui & Aziz Amine. (2022) Acetazolamide smartphone-based detection via its competition with sulfamethoxazole on molecularly imprinted polymer: A proof-of-concept. Journal of Pharmaceutical and Biomedical Analysis 219, pages 114954.
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Fatemeh Dabbagh, Horst Schroten & Christian Schwerk. (2022) In Vitro Models of the Blood–Cerebrospinal Fluid Barrier and Their Applications in the Development and Research of (Neuro)Pharmaceuticals. Pharmaceutics 14:8, pages 1729.
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Francesco P. Busardò, Alfredo F. Lo Faro, Ascanio Sirignano, Raffaele Giorgetti & Jeremy Carlier. (2022) In silico, in vitro, and in vivo human metabolism of acetazolamide, a carbonic anhydrase inhibitor and common “diuretic and masking agent” in doping. Archives of Toxicology 96:7, pages 1989-2001.
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Miriam C. A. Kehrenberg & Hagen S. Bachmann. (2022) Diuretics: a contemporary pharmacological classification?. Naunyn-Schmiedeberg's Archives of Pharmacology 395:6, pages 619-627.
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Pengcheng Lv, Yinyi Cai, Jiayi Luo & Kun Chen. (2022) Recent Advances in the Design and Synthesis of Small Molecule Carbonic Anhydrase IX Inhibitors. Current Topics in Medicinal Chemistry 22:7, pages 550-560.
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Aamer Saeed, Syeda Abida Ejaz, Anwar Ul-Hamid, Hesham R. El-Seedi & Jamshed Iqbal. (2021) Synthesis of and molecular docking studies of azomethine- tethered sulfonamides as carbonic anhydrase II & 15-lipoxygenase inhibitors. Journal of Molecular Structure 1243, pages 130821.
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Camilla de Laurentis, Paola Cristaldi, Andrea Arighi, Clarissa Cavandoli, Andrea Trezza, Erik P. Sganzerla, Carlo G. Giussani & Andrea Di Cristofori. (2020) Role of aquaporins in hydrocephalus: what do we know and where do we stand? A systematic review. Journal of Neurology 268:11, pages 4078-4094.
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Hasan Küçükbay, Zeynep Gönül, Fatümetüzzehra Zehra Küçükbay, Zehra Tekin, Andrea Angeli, Gianluca Bartolucci, Claudiu T. Supuran, Eray Tatlıcı, Elif Apohan & Özfer Yeşilada. (2021) Synthesis of new 7‐amino‐3,4‐dihydroquinolin‐2(1 H )‐one‐peptide derivatives and their carbonic anhydrase enzyme inhibition, antioxidant, and cytotoxic activities . Archiv der Pharmazie 354:11.
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Burak Kuzu, Meltem Tan, İlhami Gülçin & Nurettin Menges. (2021) A novel class for carbonic anhydrases inhibitors and evaluation of their non‐zinc binding. Archiv der Pharmazie 354:10.
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Steven W. Bothwell, Daniel Omileke, Adjanie Patabendige & Neil J. Spratt. (2021) CSF Secretion Is Not Altered by NKCC1 Nor TRPV4 Antagonism in Healthy Rats. Brain Sciences 11:9, pages 1117.
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Claudiu T. Supuran. (2021) Emerging role of carbonic anhydrase inhibitors. Clinical Science 135:10, pages 1233-1249.
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Vincent Rossi, Scott Wait, Sarah Jernigan, Mark Van Poppel, Deborah Pfortmiller, Daniel Zeitouni & Martin M. Henegar. (2021) Preoperative Acetazolamide Challenge in Pediatric Chiari I Malformation. Pediatric Neurosurgery 56:4, pages 328-333.
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Inae Hwang & Marta Ugarte. (2021) Morning glory disc anomaly-associated maculopathy: multimodal imaging. BMJ Case Reports 14:1, pages e237462.
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Andrea Angeli, Fabrizio Carta, Alessio Nocentini, Jean-Yves Winum, Raivis Zalubovskis, Atilla Akdemir, Valentina Onnis, Wagdy M. Eldehna, Clemente Capasso, Giuseppina De Simone, Simona Maria Monti, Simone Carradori, William A. Donald, Shoukat Dedhar & Claudiu T. Supuran. (2020) Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment. Metabolites 10:10, pages 412.
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Aiten M. Soliman, Mostafa M. Ghorab, Silvia Bua & Claudiu T. Supuran. (2020) Iodoquinazolinones bearing benzenesulfonamide as human carbonic anhydrase I, II, IX and XII inhibitors: Synthesis, biological evaluation and radiosensitizing activity. European Journal of Medicinal Chemistry 200, pages 112449.
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Nicolai A. Aksenov, Nikolai A. Arutiunov, Nikita K. Kirillov, Dmitrii A. Aksenov, Alexander V. Aksenov & Michael Rubin. (2020) Preparation of 1,3,4-oxadiazoles and 1,3,4-thiadiazoles via chemoselective сyclocondensation of electrophilically activated nitroalkanes to (thio)semicarbazides or thiohydrazides. Chemistry of Heterocyclic Compounds 56:8, pages 1067-1072.
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Allison R. Loiselle, Emile de Kleine, Pim van Dijk & Nomdo M. Jansonius. (2020) Intraocular and intracranial pressure in glaucoma patients taking acetazolamide. PLOS ONE 15:6, pages e0234690.
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Jyoti Singh Tomar & Jun Shen. (2020) Characterization of Carbonic Anhydrase In Vivo Using Magnetic Resonance Spectroscopy. International Journal of Molecular Sciences 21:7, pages 2442.
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Carla J. Osigian, Daniel Gologorsky, Kara M. Cavuoto, Audina Berrocal & VM Villegas. (2020) Oral acetazolamide as a medical adjuvant to retinal surgery in optic disc pit maculopathy in a pediatric patient. American Journal of Ophthalmology Case Reports 17, pages 100599.
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Ahmed Yeddi, Pranav Shah, Omnia Awad, Mohamed A. Abdallah & Ijeoma Nnodim. (2020) Acetazolamide-Associated Hyperosmolar Hyperglycemic Nonketotic Syndrome. American Journal of Therapeutics 27:6, pages e690-e692.
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Laura Øllegaard Johnsen, Helle Hasager Damkier & Jeppe Praetorius. 2020. Ion Transport Across Epithelial Tissues and Disease. Ion Transport Across Epithelial Tissues and Disease 333 361 .
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Adel S. El-Azab, Alaa A.-M. Abdel-Aziz, Silvia Bua, Alessio Nocentini, Nawaf A. AlSaif, Abdulrahman A. Almehizia, Mohammed M. Alanazi, Mohamed M. Hefnawy & Claudiu T. Supuran. (2019) New anthranilic acid-incorporating N-benzenesulfonamidophthalimides as potent inhibitors of carbonic anhydrases I, II, IX, and XII: Synthesis, in vitro testing, and in silico assessment. European Journal of Medicinal Chemistry 181, pages 111573.
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Gustavo Provensi, Fabrizio Carta, Alessio Nocentini, Claudiu T. Supuran, Fiorella Casamenti, M. Beatrice Passani & Silvia Fossati. (2019) A New Kid on the Block? Carbonic Anhydrases as Possible New Targets in Alzheimer’s Disease. International Journal of Molecular Sciences 20:19, pages 4724.
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Andrea Angeli, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Thomas S. Peat, Gianluca Bartolucci, Marta Menicatti, Fabrizio Carta & Claudiu T. Supuran. (2019) Benzensulfonamides bearing spyrohydantoin moieties act as potent inhibitors of human carbonic anhydrases II and VII and show neuropathic pain attenuating effects. European Journal of Medicinal Chemistry 177, pages 188-197.
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M. Girod, F. Allerton, E. Vangrinsven, A.C. Tutunaru, J. de Marchin, C. Gómez-Fernández-Blanco, A. Ruiz-Nuño, A. Wojnicz, F. Farnir, K. Gommeren & D. Peeters. (2019) CSF omeprazole concentration and albumin quotient following high dose intravenous omeprazole in dogs. Research in Veterinary Science 125, pages 266-271.
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Sonia Del Prete, Silvia Bua, Fatmah Alasmary, Zeid AlOthman, Sylvie Tambutté, Didier Zoccola, Claudiu Supuran & Clemente Capasso. (2019) Comparison of the Sulfonamide Inhibition Profiles of the α-Carbonic Anhydrase Isoforms (SpiCA1, SpiCA2 and SpiCA3) Encoded by the Genome of the Scleractinian Coral Stylophora pistillata. Marine Drugs 17:3, pages 146.
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Claudiu T. Supuran, Vincenzo Alterio, Anna Di Fiore, Katia D’ Ambrosio, Fabrizio Carta, Simona Maria Monti & Giuseppina De Simone. (2018) Inhibition of carbonic anhydrase IX targets primary tumors, metastases, and cancer stem cells: Three for the price of one. Medicinal Research Reviews 38:6, pages 1799-1836.
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Samuele Cazzamalli, Barbara Ziffels, Fontaine Widmayer, Patrizia Murer, Giovanni Pellegrini, Francesca Pretto, Sarah Wulhfard & Dario Neri. (2018) Enhanced Therapeutic Activity of Non-Internalizing Small-Molecule-Drug Conjugates Targeting Carbonic Anhydrase IX in Combination with Targeted Interleukin-2. Clinical Cancer Research 24:15, pages 3656-3667.
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Longtao Wu, Giovanna M. BernalKirk E. CahillPeter PytelCarrie A. FitzpatrickHeather MashekRalph R. Weichselbaum & Bakhtiar Yamini. (2018) BCL3 expression promotes resistance to alkylating chemotherapy in gliomas . Science Translational Medicine 10:448.
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Maciej Jakubowski, Ewa Szahidewicz-Krupska & Adrian Doroszko. (2018) The Human Carbonic Anhydrase II in Platelets: An Underestimated Field of Its Activity. BioMed Research International 2018, pages 1-10.
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Angela Jinsook Oh, Bryan Alexander Lanzman & Yaping Joyce Liao. (2018) Vertical diplopia and oscillopsia due to midbrain keyhole aqueduct syndrome associated with severe cough. American Journal of Ophthalmology Case Reports 10, pages 128-131.
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Chandra Bhushan Mishra, Shikha Kumari, Andrea Angeli, Silvia Bua, Manisha Tiwari & Claudiu T. Supuran. (2018) Discovery of Benzenesulfonamide Derivatives as Carbonic Anhydrase Inhibitors with Effective Anticonvulsant Action: Design, Synthesis, and Pharmacological Evaluation. Journal of Medicinal Chemistry 61:7, pages 3151-3165.
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Lorenzo Biancalana, Lucinda K. Batchelor, Gianluca Ciancaleoni, Stefano Zacchini, Guido Pampaloni, Paul J. Dyson & Fabio Marchetti. (2018) Versatile coordination of acetazolamide to ruthenium( ii ) p -cymene complexes and preliminary cytotoxicity studies . Dalton Transactions 47:28, pages 9367-9384.
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Marta Ferraroni, Benedetta Cornelio, Janos Sapi, Claudiu T. Supuran & Andrea Scozzafava. (2018) Sulfonamide carbonic anhydrase inhibitors: Zinc coordination and tail effects influence inhibitory efficacy and selectivity for different isoforms. Inorganica Chimica Acta 470, pages 128-132.
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Hakim Rahmoune, Nada Boutrid, Imene Gherbi, Samir Arezki, Mounira Amrane & Belkacem Bioud. (2017) Successful management of MPS hydrocephalus by acetazolamide. Child's Nervous System 33:12, pages 2075-2076.
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Claudiu Supuran & Clemente Capasso. (2017) An Overview of the Bacterial Carbonic Anhydrases. Metabolites 7:4, pages 56.
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Andrea Angeli, Alaa A.-M. Abdel-Aziz, Alessio Nocentini, Adel S. El-Azab, Paola Gratteri & Claudiu T. Supuran. (2017) Synthesis and carbonic anhydrase inhibition of polycyclic imides incorporating N-benzenesulfonamide moieties. Bioorganic & Medicinal Chemistry 25:20, pages 5373-5379.
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Claudiu Supuran & Clemente Capasso. (2017) Carbonic Anhydrase from Porphyromonas Gingivalis as a Drug Target. Pathogens 6:3, pages 30.
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David Bibi, Hafiz Mawasi, Alessio Nocentini, Claudiu T. Supuran, Bogdan Wlodarczyk, Richard H. Finnell & Meir Bialer. (2017) Design and Comparative Evaluation of the Anticonvulsant Profile, Carbonic-Anhydrate Inhibition and Teratogenicity of Novel Carbamate Derivatives of Branched Aliphatic Carboxylic Acids with 4-Aminobenzensulfonamide. Neurochemical Research 42:7, pages 1972-1982.
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Jeppe Praetorius & Helle Hasager Damkier. (2017) Transport across the choroid plexus epithelium. American Journal of Physiology-Cell Physiology 312:6, pages C673-C686.
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Zhengkuan Xu, Hao Li, Gang Chen, Fangcai Li, Shenjun Qian & Qixin Chen. (2016) Idiopathic intracranial hypertension occurred after spinal surgery: report of two rare cases and systematic review of the literature. European Spine Journal 26:S1, pages 9-16.
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