Citations (71)
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Claudiu T. Supuran & Clemente Capasso. (2020) Antibacterial carbonic anhydrase inhibitors: an update on the recent literature. Expert Opinion on Therapeutic Patents 30:12, pages 963-982.
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Hasan Küçükbay, Zeynep Gönül, F. Zehra Küçükbay, Andrea Angeli, Gianluca Bartolucci & Claudiu T. Supuran. (2020) Preparation, carbonic anhydrase enzyme inhibition and antioxidant activity of novel 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives incorporating mono or dipeptide moiety. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1021-1026.
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Hasan Küçükbay, Nesrin Buğday, F. Zehra Küçükbay, Andrea Ageli, Gianluca Bartolucci & Claudiu T. Supuran. (2020) Synthesis and human carbonic anhydrase I, II, VA, and XII inhibition with novel amino acid–sulphonamide conjugates. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 489-497.
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Ashok Aspatwar, Milka Hammaren, Mataleena Parikka, Seppo Parkkila, Fabrizio Carta, Murat Bozdag, Daniela Vullo & Claudiu T. Supuran. (2020) In vitro inhibition of Mycobacterium tuberculosis β-carbonic anhydrase 3 with Mono- and dithiocarbamates and evaluation of their toxicity using zebrafish developing embryos. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 65-71.
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Deniz Üzeroğlu Payaz, F. Zehra Küçükbay, Hasan Küçükbay, Andrea Angeli & Claudiu T. Supuran. (2019) Synthesis carbonic anhydrase enzyme inhibition and antioxidant activity of novel benzothiazole derivatives incorporating glycine, methionine, alanine, and phenylalanine moieties. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 343-349.
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Claudiu T. Supuran. (2017) Advances in structure-based drug discovery of carbonic anhydrase inhibitors. Expert Opinion on Drug Discovery 12:1, pages 61-88.
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P. V. Sri Ramya, Srinivas Angapelly, Andrea Angeli, Chander Singh Digwal, Mohammed Arifuddin, Bathini Nagendra Babu, Claudiu T. Supuran & Ahmed Kamal. (2017) Discovery of curcumin inspired sulfonamide derivatives as a new class of carbonic anhydrase isoforms I, II, IX, and XII inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1274-1281.
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Rajiv Kumar, Vikas Sharma, Silvia Bua, Claudiu T. Supuran & Pawan K. Sharma. (2017) Synthesis and biological evaluation of benzenesulphonamide-bearing 1,4,5-trisubstituted-1,2,3-triazoles possessing human carbonic anhydrase I, II, IV, and IX inhibitory activity. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1187-1194.
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Erol Licsandru, Muhammet Tanc, Istvan Kocsis, Mihail Barboiu & Claudiu T. Supuran. (2017) A class of carbonic anhydrase I – selective activators. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 37-46.
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Süleyman Yılmaz, Yusuf Akbaba, Bünyamin Özgeriş, Leyla Polat Köse, Süleyman Göksu, İlhami Gülçin, Saleh H. Alwasel & Claudiu T. Supuran. (2016) Synthesis and inhibitory properties of some carbamates on carbonic anhydrase and acetylcholine esterase. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1484-1491.
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F. Zehra Küçükbay, Hasan Küçükbay, Muhammet Tanc & Claudiu T. Supuran. (2016) Synthesis and carbonic anhydrase I, II, IV and XII inhibitory properties of N-protected amino acid – sulfonamide conjugates. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1476-1483.
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Leyla Polat Kose, İlhami Gulcin, Alper Yıldırım, Ufuk Atmaca, Murat Çelik, Saleh H. Alwasel & Claudiu T. Supuran. (2016) The human carbonic anhydrase isoenzymes I and II inhibitory effects of some hydroperoxides, alcohols, and acetates. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1248-1253.
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Marta Abellán-Flos, Muhammet Tanç, Claudiu T. Supuran & Stéphane P. Vincent. (2016) Multimeric xanthates as carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 946-952.
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Claudiu T. Supuran. (2016) How many carbonic anhydrase inhibition mechanisms exist?. Journal of Enzyme Inhibition and Medicinal Chemistry 31:3, pages 345-360.
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Ondrej Holas, Pavel Ondrejcek & Martin Dolezal. (2015) Mycobacterium tuberculosis enoyl-acyl carrier protein reductase inhibitors as potential antituberculotics: development in the past decade. Journal of Enzyme Inhibition and Medicinal Chemistry 30:4, pages 629-648.
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Anna Di Fiore, Viviana De Luca, Emma Langella, Alessio Nocentini, Martina Buonanno, Simona Maria Monti, Claudiu T. Supuran, Clemente Capasso & Giuseppina De Simone. (2022) Biochemical, structural, and computational studies of a γ-carbonic anhydrase from the pathogenic bacterium Burkholderia pseudomallei. Computational and Structural Biotechnology Journal 20, pages 4185-4194.
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Alka Pawar, Prakash Jha, Madhu Chopra, Uma Chaudhry & Daman Saluja. (2020) Screening of natural compounds that targets glutamate racemase of Mycobacterium tuberculosis reveals the anti-tubercular potential of flavonoids. Scientific Reports 10:1.
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Aspatwar, Kairys, Rala, Parikka, Bozdag, Carta, Supuran & Parkkila. (2019) Mycobacterium tuberculosis β-Carbonic Anhydrases: Novel Targets for Developing Antituberculosis Drugs. International Journal of Molecular Sciences 20:20, pages 5153.
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Hasan Küçükbay, Nesrin Buğday, F. Zehra Küçükbay, Emanuela Berrino, Gianluca Bartolucci, Sonia Del Prete, Clemente Capasso & Claudiu T. Supuran. (2019) Synthesis and carbonic anhydrase inhibitory properties of novel 4-(2-aminoethyl)benzenesulfonamide-dipeptide conjugates. Bioorganic Chemistry 83, pages 414-423.
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Nesrin Buğday, F. Zehra Küçükbay, Hasan Küçükbay, Silvia Bua, Gianluca Bartolucci, Janis Leitans, Andris Kazaks, Kaspars Tars & Claudiu T. Supuran. (2018) Synthesis of novel dipeptide sulfonamide conjugates with effective carbonic anhydrase I, II, IX, and XII inhibitory properties. Bioorganic Chemistry 81, pages 311-318.
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Ashok Aspatwar, Jean-Yves Winum, Fabrizio Carta, Claudiu Supuran, Milka Hammaren, Mataleena Parikka & Seppo Parkkila. (2018) Carbonic Anhydrase Inhibitors as Novel Drugs against Mycobacterial β-Carbonic Anhydrases: An Update on In Vitro and In Vivo Studies. Molecules 23:11, pages 2911.
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Carrie L. Lomelino, Jacob T. Andring & Robert McKenna. (2018) Crystallography and Its Impact on Carbonic Anhydrase Research. International Journal of Medicinal Chemistry 2018, pages 1-21.
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Srinivas Angapelly, P.V. Sri Ramya, Andrea Angeli, Sonia Del Prete, Clemente Capasso, Mohammed Arifuddin & Claudiu T. Supuran. (2017) Development of sulfonamides incorporating phenylacrylamido functionalities as carbonic anhydrase isoforms I, II, IX and XII inhibitors. Bioorganic & Medicinal Chemistry 25:20, pages 5726-5732.
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Fabrizio Carta, Alexander Birkmann, Tamara Pfaff, Helmut Buschmann, Wilfried Schwab, Holger Zimmermann, Alfonso Maresca & Claudiu T. Supuran. (2017) Lead Development of Thiazolylsulfonamides with Carbonic Anhydrase Inhibitory Action. Journal of Medicinal Chemistry 60:7, pages 3154-3164.
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Benjamin K. Johnson & Robert B. Abramovitch. (2017) Small Molecules That Sabotage Bacterial Virulence. Trends in Pharmacological Sciences 38:4, pages 339-362.
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Tiphaine Rogez-Florent, Catherine Foulon, Anne-Sophie Drucbert, Nadège Schifano, Perrine Six, Stéphanie Devassine, Patrick Depreux, Pierre-Marie Danzé, Laurence Goossens, Cécile Danel & Jean-François Goossens. (2017) Chiral separation of new sulfonamide derivatives and evaluation of their enantioselective affinity for human carbonic anhydrase II by microscale thermophoresis and surface plasmon resonance. Journal of Pharmaceutical and Biomedical Analysis 137, pages 113-122.
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Mustafa Durgun, Hasan Turkmen, Gulay Zengin, Huseyin Zengin, Mehmet Koyunsever & Ismail Koyuncu. (2017) Synthesis, characterization, in vitro cytotoxicity and antimicrobial investigation and evaluation of physicochemical properties of novel 4-(2-methylacetamide)benzenesulfonamide derivatives. Bioorganic Chemistry 70, pages 163-172.
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Srinivas Angapelly, P.V. Sri Ramya, Andrea Angeli, Simona Maria Monti, Martina Buonanno, Mallika Alvala, Cladiu T. Supuran & Mohammed Arifuddin. (2017) Discovery of 4-sulfamoyl-phenyl-β-lactams as a new class of potent carbonic anhydrase isoforms I, II, IV and VII inhibitors: The first example of subnanomolar CA IV inhibitors. Bioorganic & Medicinal Chemistry 25:2, pages 539-544.
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Giannamaria Annunziato, Andrea Angeli, Francesca D'Alba, Agostino Bruno, Marco Pieroni, Daniela Vullo, Viviana De Luca, Clemente Capasso, Claudiu T. Supuran & Gabriele Costantino. (2016) Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches. ChemMedChem 11:17, pages 1904-1914.
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Ramazan Ulus, Burak Aday, Muhammet Tanç, Claudiu T. Supuran & Muharrem Kaya. (2016) Microwave assisted synthesis of novel acridine–acetazolamide conjugates and investigation of their inhibition effects on human carbonic anhydrase isoforms hCA I, II, IV and VII. Bioorganic & Medicinal Chemistry 24:16, pages 3548-3555.
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Haydar Göksu, Meryem Topal, Ali Keskin, Mehmet S. Gültekin, Murat Çelik, İlhami Gülçin, Muhammet Tanc & Claudiu T. Supuran. (2016)
9,10-Dibromo-
N
-aryl-9,10-dihydro-9,10-[3,4]epipyrroloanthracene-12,14-diones: Synthesis and Investigation of Their Effects on Carbonic Anhydrase Isozymes I, II, IX, and XII
. Archiv der Pharmazie 349:6, pages 466-474.
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Tekin Artunç, Yasin Çetinkaya, Hülya Göçer, İlhami Gülçin, Abdullah Menzek, Ertan Şahin & Claudiu T. Supuran. (2016) Synthesis of 4-[2-(3,4-dimethoxybenzyl)cyclopentyl]-1,2-dimethoxybenzene Derivatives and Evaluations of Their Carbonic Anhydrase Isoenzymes Inhibitory Effects. Chemical Biology & Drug Design 87:4, pages 594-607.
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Wagdy M. Eldehna, Mohamed Fares, Mariangela Ceruso, Hazem A. Ghabbour, Sahar M. Abou-Seri, Hatem A. Abdel-Aziz, Dalal A. Abou El Ella & Claudiu T. Supuran. (2016) Amido/ureidosubstituted benzenesulfonamides-isatin conjugates as low nanomolar/subnanomolar inhibitors of the tumor-associated carbonic anhydrase isoform XII. European Journal of Medicinal Chemistry 110, pages 259-266.
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Daniela Vullo, Sonia Del Prete, Viviana De Luca, Vincenzo Carginale, Marta Ferraroni, Nurcan Dedeoglu, Sameh M. Osman, Zeid AlOthman, Clemente Capasso & Claudiu T. Supuran. (2016) Anion inhibition studies of the β-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae. Bioorganic & Medicinal Chemistry Letters 26:5, pages 1406-1410.
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Marta Ferraroni, Fabrizio Carta, Andrea Scozzafava & Claudiu T. Supuran. (2015) Thioxocoumarins Show an Alternative Carbonic Anhydrase Inhibition Mechanism Compared to Coumarins. Journal of Medicinal Chemistry 59:1, pages 462-473.
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Ylenia Cau, Mattia Mori, Claudiu T. Supuran & Maurizio Botta. (2016) Mycobacterial carbonic anhydrase inhibition with phenolic acids and esters: kinetic and computational investigations. Organic & Biomolecular Chemistry 14:35, pages 8322-8330.
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Anna Di Fiore, Giuseppina De Simone, Vincenzo Alterio, Vincenzo Riccio, Jean-Yves Winum, Fabrizio Carta & Claudiu T. Supuran. (2016) The anticonvulsant sulfamide JNJ-26990990 and its S,S-dioxide analog strongly inhibit carbonic anhydrases: solution and X-ray crystallographic studies. Organic & Biomolecular Chemistry 14:21, pages 4853-4858.
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Reza Zolfaghari Emameh, Marianne Kuuslahti, Daniela Vullo, Harlan R. Barker, Claudiu T. Supuran & Seppo Parkkila. (2015) Ascaris lumbricoides β carbonic anhydrase: a potential target enzyme for treatment of ascariasis. Parasites & Vectors 8:1.
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Viviana De Luca, Sonia Del Prete, Vincenzo Carginale, Daniela Vullo, Claudiu T. Supuran & Clemente Capasso. (2015) Cloning, characterization and anion inhibition studies of a γ-carbonic anhydrase from the Antarctic cyanobacterium Nostoc commune. Bioorganic & Medicinal Chemistry Letters 25:21, pages 4970-4975.
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Hany S. Ibrahim, Sahar M. Abou-Seri, Muhammet Tanc, Mahmoud M. Elaasser, Hatem A. Abdel-Aziz & Claudiu T. Supuran. (2015) Isatin-pyrazole benzenesulfonamide hybrids potently inhibit tumor-associated carbonic anhydrase isoforms IX and XII. European Journal of Medicinal Chemistry 103, pages 583-593.
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İbrahim Esirden, Ramazan Ulus, Burak Aday, Muhammet Tanç, Claudiu T. Supuran & Muharrem Kaya. (2015) Synthesis of novel acridine bis-sulfonamides with effective inhibitory activity against the carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry 23:20, pages 6573-6580.
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Poonam Khloya, Mariangela Ceruso, Sita Ram, Claudiu T. Supuran & Pawan K. Sharma. (2015) Sulfonamide bearing pyrazolylpyrazolines as potent inhibitors of carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry Letters 25:16, pages 3208-3212.
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Ilija N. Cvijetić, Muhammet Tanç, Ivan O. Juranić, Tatjana Ž. Verbić, Claudiu T. Supuran & Branko J. Drakulić. (2015) 5-Aryl-1H-pyrazole-3-carboxylic acids as selective inhibitors of human carbonic anhydrases IX and XII. Bioorganic & Medicinal Chemistry 23:15, pages 4649-4659.
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Aiga Grandane, Muhammet Tanc, Lorenzo Di Cesare Mannelli, Fabrizio Carta, Carla Ghelardini, Raivis Žalubovskis & Claudiu T. Supuran. (2015) 6-Substituted Sulfocoumarins Are Selective Carbonic Anhdydrase IX and XII Inhibitors with Significant Cytotoxicity against Colorectal Cancer Cells. Journal of Medicinal Chemistry 58:9, pages 3975-3983.
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Leo Syrjänen, Marianne Kuuslahti, Martti Tolvanen, Daniela Vullo, Seppo Parkkila & Claudiu T. Supuran. (2015) The β-carbonic anhydrase from the malaria mosquito Anopheles gambiae is highly inhibited by sulfonamides. Bioorganic & Medicinal Chemistry 23:10, pages 2303-2309.
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Murat Bozdag, Fabrizio Carta, Daniela Vullo, Atilla Akdemir, Semra Isik, Cecilia Lanzi, Andrea Scozzafava, Emanuela Masini & Claudiu T. Supuran. (2015) Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma action. Bioorganic & Medicinal Chemistry 23:10, pages 2368-2376.
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Daniela Vullo, Viviana De Luca, Sonia Del Prete, Vincenzo Carginale, Andrea Scozzafava, Clemente Capasso & Claudiu T. Supuran. (2015) Sulfonamide inhibition studies of the γ-carbonic anhydrase from the Antarctic cyanobacterium Nostoc commune. Bioorganic & Medicinal Chemistry 23:8, pages 1728-1734.
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Fabrizio Carta, Lorenzo Di Cesare Mannelli, Melissa Pinard, Carla Ghelardini, Andrea Scozzafava, Robert McKenna & Claudiu T. Supuran. (2015) A class of sulfonamide carbonic anhydrase inhibitors with neuropathic pain modulating effects. Bioorganic & Medicinal Chemistry 23:8, pages 1828-1840.
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Daniela Vullo, Sonia Del Prete, Gillian M. Fisher, Katherine T. Andrews, Sally-Ann Poulsen, Clemente Capasso & Claudiu T. Supuran. (2015) Sulfonamide inhibition studies of the η-class carbonic anhydrase from the malaria pathogen Plasmodium falciparum. Bioorganic & Medicinal Chemistry 23:3, pages 526-531.
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Murat Boztaş, Yasin Çetinkaya, Meryem Topal, İlhami Gülçin, Abdullah Menzek, Ertan Şahin, Muhammet Tanc & Claudiu T. Supuran. (2014) Synthesis and Carbonic Anhydrase Isoenzymes I, II, IX, and XII Inhibitory Effects of Dimethoxybromophenol Derivatives Incorporating Cyclopropane Moieties. Journal of Medicinal Chemistry 58:2, pages 640-650.
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Murat Bozdag, Melissa Pinard, Fabrizio Carta, Emanuela Masini, Andrea Scozzafava, Robert McKenna & Claudiu T. Supuran. (2014) A Class of 4-Sulfamoylphenyl-ω-aminoalkyl Ethers with Effective Carbonic Anhydrase Inhibitory Action and Antiglaucoma Effects. Journal of Medicinal Chemistry 57:22, pages 9673-9686.
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Murat Bozdag, Marta Ferraroni, Fabrizio Carta, Daniela Vullo, Laura Lucarini, Elisabetta Orlandini, Armando Rossello, Elisa Nuti, Andrea Scozzafava, Emanuela Masini & Claudiu T. Supuran. (2014) Structural Insights on Carbonic Anhydrase Inhibitory Action, Isoform Selectivity, and Potency of Sulfonamides and Coumarins Incorporating Arylsulfonylureido Groups. Journal of Medicinal Chemistry 57:21, pages 9152-9167.
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Alaa A.-M. Abdel-Aziz, Adel S. El-Azab, Mariangela Ceruso & Claudiu T. Supuran. (2014) Carbonic anhydrase inhibitory activity of sulfonamides and carboxylic acids incorporating cyclic imide scaffolds. Bioorganic & Medicinal Chemistry Letters 24:22, pages 5185-5189.
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Joanna Ombouma, Daniela Vullo, Claudiu T. Supuran & Jean-Yves Winum. (2014) Ferrier sulfamidoglycosylation of glycals catalyzed by nitrosonium tetrafluoroborate: Towards new carbonic anhydrase glycoinhibitors. Bioorganic & Medicinal Chemistry 22:22, pages 6353-6359.
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Clemente Capasso & Claudiu T. Supuran. 2014. Novel Antimicrobial Agents and Strategies. Novel Antimicrobial Agents and Strategies
31
46
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Jinlian Zhao, Dimitrios Evangelopoulos, Sanjib Bhakta, Alexander I. Gray & Véronique Seidel. (2014) Antitubercular activity of Arctium lappa and Tussilago farfara extracts and constituents. Journal of Ethnopharmacology 155:1, pages 796-800.
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Mariangela Ceruso, Sonia Del Prete, Zeid AlOthman, Sameh M. Osman, Andrea Scozzafava, Clemente Capasso & Claudiu T. Supuran. (2014) Synthesis of sulfonamides with effective inhibitory action against Porphyromonas gingivalis γ-carbonic anhydrase. Bioorganic & Medicinal Chemistry Letters 24:16, pages 4006-4010.
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Kalyan K. Sethi, Saurabh M. Verma, Muhammet Tanç, Gaultier Purper, Gaetan Calafato, Fabrizio Carta & Claudiu T. Supuran. (2014) Carbonic anhydrase inhibitors: Synthesis and inhibition of the human carbonic anhydrase isoforms I, II, IX and XII with benzene sulfonamides incorporating 4- and 3-nitrophthalimide moieties. Bioorganic & Medicinal Chemistry 22:5, pages 1586-1595.
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Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Viviana De Luca, Andrea Scozzafava, Zeid AlOthman, Claudiu T. Supuran & Clemente Capasso. (2014) Sulfonamide inhibition studies of the γ-carbonic anhydrase from the oral pathogen Porphyromonas gingivalis. Bioorganic & Medicinal Chemistry Letters 24:1, pages 240-244.
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Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Viviana De Luca, Andrea Scozzafava, Zeid AlOthman, Claudiu T. Supuran & Clemente Capasso. (2014) Sulfonamide inhibition studies of the δ-carbonic anhydrase from the diatom Thalassiosira weissflogii. Bioorganic & Medicinal Chemistry Letters 24:1, pages 275-279.
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Robert McKenna & Claudiu T. Supuran. 2014. Carbonic Anhydrase: Mechanism, Regulation, Links to Disease, and Industrial Applications. Carbonic Anhydrase: Mechanism, Regulation, Links to Disease, and Industrial Applications
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323
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Simone Carradori, Celeste De Monte, Melissa D’Ascenzio, Daniela Secci, Gulsah Celik, Mariangela Ceruso, Daniela Vullo, Andrea Scozzafava & Claudiu T. Supuran. (2013) Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII—A new scaffold for designing isoform-selective inhibitors. Bioorganic & Medicinal Chemistry Letters 23:24, pages 6759-6763.
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Kalyan K. Sethi, Daniella Vullo, Saurabh M. Verma, Muhammet Tanç, Fabrizio Carta & Claudiu T. Supuran. (2013) Carbonic anhydrase inhibitors: Synthesis and inhibition of the human carbonic anhydrase isoforms I, II, VII, IX and XII with benzene sulfonamides incorporating 4,5,6,7-tetrabromophthalimide moiety. Bioorganic & Medicinal Chemistry 21:19, pages 5973-5982.
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Kalyan K. Sethi, Saurabh M. Verma, Muhammet Tanç, Fabrizio Carta & Claudiu T. Supuran. (2013) Carbonic anhydrase inhibitors: Synthesis and inhibition of the cytosolic mammalian carbonic anhydrase isoforms I, II and VII with benzene sulfonamides incorporating 4,5,6,7-tetrachlorophthalimide moiety. Bioorganic & Medicinal Chemistry 21:17, pages 5168-5174.
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Sonia Del Prete, Daniela Vullo, Viviana De Luca, Vincenzo Carginale, Andrea Scozzafava, Claudiu T. Supuran & Clemente Capasso. (2013) A highly catalytically active γ-carbonic anhydrase from the pathogenic anaerobe Porphyromonas gingivalis and its inhibition profile with anions and small molecules. Bioorganic & Medicinal Chemistry Letters 23:14, pages 4067-4071.
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Peiwen Pan, Alane Beatriz Vermelho, Giseli Capaci Rodrigues, Andrea Scozzafava, Martti E. E. Tolvanen, Seppo Parkkila, Clemente Capasso & Claudiu T. Supuran. (2013)
Cloning, Characterization, and Sulfonamide and Thiol Inhibition Studies of an α-Carbonic Anhydrase from
Trypanosoma cruzi
, the Causative Agent of Chagas Disease
. Journal of Medicinal Chemistry 56:4, pages 1761-1771.
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