Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 19, Issue 6 (2004)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 19, Issue 6 (2004)

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Editorial

Editorial
12th European Conference of GP2A—La Rochelle 2003
Marc Le Borgne
Page: 449
Published online: 03 Oct 2008
Citationfor12th European Conference of GP2A—La Rochelle 2003 | PDF (34.2 KB)
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Research Article

Article
Synthesis and Antileishmanial Activity of 3-Imidazolylalkylindoles. Part I
Young Min Na, Nicolas Lebouvier, Marc Le Borgne, Fabrice Pagniez, Nidia Alvarez, Patrice Le Pape & Guillaume Le Baut
Pages: 451-457
Published online: 03 Oct 2008
AbstractforSynthesis and Antileishmanial Activity of 3-Imidazolylalkylindoles. Part I | References | PDF (136.6 KB)
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Article
Synthesis and Evaluation of Disubstituted N1- and N3-Imidazolidin-2-ones Acting as Potential Immunosuppressive Agents
Caroline Sabourin, Jean-Michel H. Robert, Sylvie Robert-Piessard, Delphine Carbonnelle & Francois Lang
Pages: 459-465
Published online: 03 Oct 2008
AbstractforSynthesis and Evaluation of Disubstituted N1- and N3-Imidazolidin-2-ones Acting as Potential Immunosuppressive Agents | References | PDF (127.3 KB)
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Article
Microwave-assisted Synthesis of Novel Thiazolocarbazoles and Evaluation as Potential Anticancer Agents. Part III
Alexandra Testard, Laurent Picot, Ingrid Fruitier-Arnaudin, Jean-Marie Piot, Hadjila Chabane, Lisianne Domon, Valerie Thiery & Thierry Besson
Pages: 467-473
Published online: 03 Oct 2008
AbstractforMicrowave-assisted Synthesis of Novel Thiazolocarbazoles and Evaluation as Potential Anticancer Agents. Part III | References | PDF (177.4 KB)
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Article
Synthesis and Potential Anti-Inflammatory Activity of Some Tetrahydrophthalazinones
Nicolas Gouault, Benoit Pinel, Jean-Francois Cupif, Alexandra Depince, Corinne A.E. Martin-Chouly, Chantal Belleguic & Michele David
Pages: 475-480
Published online: 03 Oct 2008
AbstractforSynthesis and Potential Anti-Inflammatory Activity of Some Tetrahydrophthalazinones | References | PDF (219.9 KB)
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Article
Synthesis and Antiviral Effect against Herpes Simplex Type 1 of 12-substituted Benzo[c]phenanthridinium Salts
Enguerran Vanquelef, Maryvonne Amoros, Joel Boustie, Michael A. Lynch, Roger D. Waigh & Olivier Duval
Pages: 481-487
Published online: 03 Oct 2008
AbstractforSynthesis and Antiviral Effect against Herpes Simplex Type 1 of 12-substituted Benzo[c]phenanthridinium Salts | References | PDF (126 KB)
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Article
Synthesis and PreliminaryIn Vitro Evaluation of Antimycobacterial Activity of New Pyrrolo[1,2-a]quinoxaline-carboxylic Acid Hydrazide Derivatives
Jean Guillon, Robert C. Reynolds, Jean-Michel Leger, Marie-Aude Guie, Stephane Massip, Patrick Dallemagne & Christian Jarry
Pages: 489-495
Published online: 03 Oct 2008
AbstractforSynthesis and PreliminaryIn Vitro Evaluation of Antimycobacterial Activity of New Pyrrolo[1,2-a]quinoxaline-carboxylic Acid Hydrazide Derivatives | References | PDF (127.5 KB)
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Article
Synthesis and Anti-HIV Activity of Some [Nucleoside Reverse Transcriptase Inhibitor]-C5′-Linker-[Integrase Inhibitor] Heterodimers as Inhibitors of HIV Replication
Elena Sugeac, Christine Fossey, Daniel Ladurée, Sylvie Schmidt, Geraldine Laumond & Anne-Marie Aubertin
Pages: 497-509
Published online: 03 Oct 2008
AbstractforSynthesis and Anti-HIV Activity of Some [Nucleoside Reverse Transcriptase Inhibitor]-C5′-Linker-[Integrase Inhibitor] Heterodimers as Inhibitors of HIV Replication | References | PDF (205.9 KB)
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Article
Synthesis of 5-alkynylated d4T Analogues as Potential HIV-1 Reverse Transcriptase Inhibitors
A. Ciurea, C. Fossey, D. Gavriliu, Z. Delbederi, E. Sugeac, D. Laduree, S. Schmidt, G. Laumond & A.-M. Aubertin
Pages: 511-519
Published online: 03 Oct 2008
AbstractforSynthesis of 5-alkynylated d4T Analogues as Potential HIV-1 Reverse Transcriptase Inhibitors | References | PDF (161.5 KB)
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Article
Review Article
Naphthalene Combretastatin Analogues: Synthesis, Cytotoxicity and Antitubulin Activity
Manuel Medarde, Ana B.S. Maya & Concepción Pérez-Melero
Pages: 521-540
Published online: 03 Oct 2008
AbstractforReview Article
Naphthalene Combretastatin Analogues: Synthesis, Cytotoxicity and Antitubulin Activity | References | PDF (463.6 KB)
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Article
Docking Study of Ligands into the Colchicine Binding Site of Tubulin
Amaury Farce, Cedric Loge, Sebastien Gallet, Nicolas Lebegue, Pascal Carato, Philippe Chavatte, Pascal Berthelot & Daniel Lesieur
Pages: 541-547
Published online: 03 Oct 2008
AbstractforDocking Study of Ligands into the Colchicine Binding Site of Tubulin | References | PDF (851.2 KB)
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Article
2- and 3-[(Aryl)(azolyl)methyl]indoles as Potential Non-steroidal Aromatase Inhibitors
Marie-Pierre Lézé, Marc Le Borgne, Pascal Marchand, Denis Loquet, Manuela Kogler, Guillaume Le Baut, Anja Palusczak & Rolf W. Hartmann
Pages: 549-557
Published online: 03 Oct 2008
Abstractfor2- and 3-[(Aryl)(azolyl)methyl]indoles as Potential Non-steroidal Aromatase Inhibitors | References | PDF (154.1 KB)
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Article
Synthesis and Biological Evaluation with Plant Cells of New Fosmidomycin Analogues Containing a Benzoxazolone or Oxazolopyridinone Ring
Martine Courtois, Zoia Mincheva, Françoise Andreu, Marc Rideau & Marie-Claude Viaud-Massuard
Pages: 559-565
Published online: 03 Oct 2008
AbstractforSynthesis and Biological Evaluation with Plant Cells of New Fosmidomycin Analogues Containing a Benzoxazolone or Oxazolopyridinone Ring | References | PDF (172 KB)
  • 194 Views
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Article
Synthesis and Cytotoxic Activity of Thiazolofluorenone Derivatives
Hadjila Chabane, Alain Pierre, Stephane Leonce, Bruno Pfeiffer, Pierre Renard, Valerie Thiery, Gérald Guillaumet & Thierry Besson
Pages: 567-575
Published online: 03 Oct 2008
AbstractforSynthesis and Cytotoxic Activity of Thiazolofluorenone Derivatives | References | PDF (152.6 KB)
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Article
Pharmacomodulation of a Sulfamide 5-HT6 Receptor Ligand
Jacques Renault, Aurelie Bernard, Solenn Brajeul, Pierre Verhaeghe, Sabrina Butt, Frederic Fabis, François Dauphin, Philippe Uriac & Sylvain Rault
Pages: 577-583
Published online: 03 Oct 2008
AbstractforPharmacomodulation of a Sulfamide 5-HT6 Receptor Ligand | References | PDF (315.2 KB)
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Article
Synthesis and Biological Evaluation of Thienopyrrolizines, a New Family of CDK/GSK-3 Inhibitors
Christophe Rochais, Elodie Lescot, Vincent Lisowski, Alban Lepailleur, Jana sopkova-de oliveira Santos, Ronan Bureau, Patrick Dallemagne, Laurent Meijer & Sylvain Rault
Pages: 585-593
Published online: 03 Oct 2008
AbstractforSynthesis and Biological Evaluation of Thienopyrrolizines, a New Family of CDK/GSK-3 Inhibitors | References | PDF (359.8 KB)
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