Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 29, Issue 1 (2014)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 29, Issue 1 (2014)

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Research Article

Article
Phenolic compounds with pancreatic lipase inhibitory activity from Korean yam (Dioscorea opposita)
Min Hye Yang, Young-Won Chin, Kee Dong Yoon & Jinwoong Kim
Pages: 1-6
Published online: 18 Jan 2013
AbstractforPhenolic compounds with pancreatic lipase inhibitory activity from Korean yam (Dioscorea opposita) | Full Text | References | PDF (261.7 KB)
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Article
Synthesis and biological evaluation of asymmetric indole curcumin analogs as potential anti-inflammatory and antioxidant agents
Babasaheb P. Bandgar, Santosh N. Kinkar, Hemant V. Chavan, Shivkumar S. Jalde, Rafik U. Shaikh & Rajesh N. Gacche
Pages: 7-11
Published online: 28 Jan 2013
AbstractforSynthesis and biological evaluation of asymmetric indole curcumin analogs as potential anti-inflammatory and antioxidant agents | Full Text | References | PDF (226 KB)
  • 1399 Views
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Article
Inhibitory effect of linalool-rich essential oil from Lippia alba on the peptidase and keratinase activities of dermatophytes
Danielle Cristina Machado Costa, Alane Beatriz Vermelho, Catia Amancio Almeida, Edilma Paraguai de Souza Dias, Sabrina Martins Lage Cedrola, Maria de Fátima Arrigoni-Blank, Arie Fitzgerald Blank, Celuta Sales Alviano & Daniela Sales Alviano
Pages: 12-17
Published online: 17 Jan 2013
AbstractforInhibitory effect of linalool-rich essential oil from Lippia alba on the peptidase and keratinase activities of dermatophytes | Full Text | References | PDF (481.1 KB)
  • 1255 Views
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Article
Synthesis and carbonic anhydrase inhibitory properties of novel 1,4-dihydropyrimidinone substituted diarylureas
Fatma Celik, Mustafa Arslan, Emre Yavuz, Dudu Demir & Nahit Gençer
Pages: 18-22
Published online: 16 Jan 2013
AbstractforSynthesis and carbonic anhydrase inhibitory properties of novel 1,4-dihydropyrimidinone substituted diarylureas | Full Text | References | PDF (183.9 KB)
  • 757 Views
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Article
Biochemical properties of a new α-carbonic anhydrase from the human pathogenic bacterium, Vibrio cholerae
Sonia Del Prete, Viviana De Luca, Andrea Scozzafava, Vincenzo Carginale, Claudiu T. Supuran & Clemente Capasso
Pages: 23-27
Published online: 16 Jan 2013
AbstractforBiochemical properties of a new α-carbonic anhydrase from the human pathogenic bacterium, Vibrio cholerae | Full Text | References | PDF (289 KB)
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Article
Evaluation of Geranium spp., Helleborus spp. and Hyssopus spp. polyphenolic extracts inhibitory activity against urease and α-chymotrypsin
Gabriela Paun, Simona Carmen Litescu, Elena Neagu, Andreia Tache & Gabriel Lucian Radu
Pages: 28-34
Published online: 15 Jan 2013
AbstractforEvaluation of Geranium spp., Helleborus spp. and Hyssopus spp. polyphenolic extracts inhibitory activity against urease and α-chymotrypsin | Full Text | References | PDF (584.6 KB)
  • 1385 Views
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Article
Carbonic anhydrase inhibitory properties of novel sulfonamide derivatives of aminoindanes and aminotetralins
Yusuf Akbaba, Akın Akıncıoğlu, Hülya Göçer, Süleyman Göksu, İlhami Gülçin & Claudiu T. Supuran
Pages: 35-42
Published online: 12 Jan 2013
AbstractforCarbonic anhydrase inhibitory properties of novel sulfonamide derivatives of aminoindanes and aminotetralins | Full Text | References | PDF (397.4 KB)
  • 1893 Views
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Article
Synthesis, anticandidal activity and cytotoxicity of some tetrazole derivatives
Zafer Asim Kaplancikli, Leyla Yurttaş, Ahmet Özdemir, Gülhan Turan-Zitouni, Gökalp İşcan, Gülşen Akalın & Usama Abu Mohsen
Pages: 43-48
Published online: 17 Jan 2013
AbstractforSynthesis, anticandidal activity and cytotoxicity of some tetrazole derivatives | Full Text | References | PDF (178.6 KB)
  • 1037 Views
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Article
Evaluation of the antioxidant activity of several naturally occurring coumarins and their synthesized analogues by “ferric reducing antioxidant power” assay
Zuzana Rehakova, Vit Koleckar, Ludek Jahodar, Lubomir Opletal, Katerina Macakova, Lucie Cahlikova, Daniel Jun & Kamil Kuca
Pages: 49-54
Published online: 28 Jan 2013
AbstractforEvaluation of the antioxidant activity of several naturally occurring coumarins and their synthesized analogues by “ferric reducing antioxidant power” assay | Full Text | References | PDF (502.9 KB)
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Short Communication

Article
Synthesis and activity of proteasome inhibitors
Derek Dunn, Mohamed Iqbal & Sankar Chatterjee
Pages: 55-58
Published online: 23 Jan 2013
AbstractforSynthesis and activity of proteasome inhibitors | Full Text | References | PDF (318.4 KB)
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Research Article

Article
Phenolic phytochemical displaying SARS-CoV papain-like protease inhibition from the seeds of Psoralea corylifolia
Dae Wook Kim, Kyung Hye Seo, Marcus J. Curtis-Long, Kyeong Yeol Oh, Jong-Won Oh, Jung Keun Cho, Kon Ho Lee & Ki Hun Park
Pages: 59-63
Published online: 16 Jan 2013
AbstractforPhenolic phytochemical displaying SARS-CoV papain-like protease inhibition from the seeds of Psoralea corylifolia | Full Text | References | PDF (255.8 KB)
  • 5121 Views
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Article
Microwave-assisted synthesis of new benzimidazole derivatives with lipase inhibition activity
Emre Menteşe, Hakan Bektaş, Serdar Ülker, Olcay Bekircan & Bahittin Kahveci
Pages: 64-68
Published online: 18 Jan 2013
AbstractforMicrowave-assisted synthesis of new benzimidazole derivatives with lipase inhibition activity | Full Text | References | PDF (225 KB)
  • 1822 Views
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Article
Ligand-based pharmacophore modeling and Bayesian approaches to identify c-Src inhibitors
Sugunadevi Sakkiah, Venkatesh Arullaperumal, Swan Hwang & Keun Woo Lee
Pages: 69-80
Published online: 25 Feb 2013
AbstractforLigand-based pharmacophore modeling and Bayesian approaches to identify c-Src inhibitors | Full Text | References | PDF (3.4 MB)
  • 1590 Views
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Article
Quantum chemical modeling of the inhibition mechanism of monoamine oxidase by oxazolidinone and analogous heterocyclic compounds
Safiye Sağ Erdem, Gül Altınbaş Özpınar & Ümüt Boz
Pages: 81-86
Published online: 17 Jan 2013
AbstractforQuantum chemical modeling of the inhibition mechanism of monoamine oxidase by oxazolidinone and analogous heterocyclic compounds | Full Text | References | PDF (402.7 KB)
  • 782 Views
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Article
Carbonic anhydrase in minor salivary glands of quail: histochemistry versus immunohistochemistry
Maria Gabriella Gabrielli & Daniele Tomassoni
Pages: 87-91
Published online: 16 Jan 2013
AbstractforCarbonic anhydrase in minor salivary glands of quail: histochemistry versus immunohistochemistry | Full Text | References | PDF (1.6 MB)
  • 827 Views
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Article
On the interpretation of tyrosinase inhibition kinetics
Wei Sun, Michael Wendt, Gerhard Klebe & Klaus-Heinrich Röhm
Pages: 92-99
Published online: 17 Jan 2013
AbstractforOn the interpretation of tyrosinase inhibition kinetics | Full Text | References | PDF (235.8 KB)
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Article
Design, synthesis, antimicrobial activity and anti-HIV activity evaluation of novel hybrid quinazoline–triazine derivatives
Rahul P. Modh, Erik De Clercq, Christophe Pannecouque & Kishor H. Chikhalia
Pages: 100-108
Published online: 18 Jan 2013
AbstractforDesign, synthesis, antimicrobial activity and anti-HIV activity evaluation of novel hybrid quinazoline–triazine derivatives | Full Text | References | PDF (739.1 KB)
  • 2190 Views
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Article
Synthesis and biological evaluation of modified purine homo-N-nucleosides containing pyrazole or 2-pyrazoline moiety
Andreas Thalassitis, Anna-Maria Katsori, Konstantinos Dimas, Dimitra J. Hadjipavlou-Litina, Fokion Pyleris, Nikolaos Sakellaridis & Konstantinos E. Litinas
Pages: 109-117
Published online: 23 Jan 2013
AbstractforSynthesis and biological evaluation of modified purine homo-N-nucleosides containing pyrazole or 2-pyrazoline moiety | Full Text | References | PDF (301.6 KB)
  • 790 Views
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Article
In vitro inhibition effect and structure–activity relationships of some saccharin derivatives on erythrocyte carbonic anhydrase I and II
Fatih Sonmez, Cigdem Bilen, Sinem Sumersan, Nahit Gencer, Semra Isik, Oktay Arslan & Mustafa Kucukislamoglu
Pages: 118-123
Published online: 23 Jan 2013
AbstractforIn vitro inhibition effect and structure–activity relationships of some saccharin derivatives on erythrocyte carbonic anhydrase I and II | Full Text | References | PDF (433.8 KB)
  • 864 Views
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Article
Benzenesulfonamides with benzimidazole moieties as inhibitors of carbonic anhydrases I, II, VII, XII and XIII
Asta Zubrienė, Edita Čapkauskaitė, Joana Gylytė, Miglė Kišonaitė, Sigitas Tumkevičius & Daumantas Matulis
Pages: 124-131
Published online: 28 Jan 2013
AbstractforBenzenesulfonamides with benzimidazole moieties as inhibitors of carbonic anhydrases I, II, VII, XII and XIII | Full Text | References | PDF (454.1 KB)
  • 983 Views
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Article
Synthesis and carbonic anhydrase inhibitory properties of 1,3-dicarbonyl derivatives of methylaminobenzene-sulfonamide
Tuna Demirci, Mustafa Arslan, Çiğdem Bilen, Dudu Demir, Nahit Gençer & Oktay Arslan
Pages: 132-136
Published online: 28 Jan 2013
AbstractforSynthesis and carbonic anhydrase inhibitory properties of 1,3-dicarbonyl derivatives of methylaminobenzene-sulfonamide | Full Text | References | PDF (169.7 KB)
  • 625 Views
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Article
Aminopurine derivatives as putative SopE inhibitors
Gizem Ozbuyukkaya, Elif Ozkirimli Olmez & Kutlu Ozergin Ulgen
Pages: 137-145
Published online: 30 Jan 2013
AbstractforAminopurine derivatives as putative SopE inhibitors | Full Text | References | PDF (1.9 MB)
  • 650 Views
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Article
Biomimetic CO2 capture using a highly thermostable bacterial α-carbonic anhydrase immobilized on a polyurethane foam
Fortunato Migliardini, Viviana De Luca, Vincenzo Carginale, Mosè Rossi, Pasquale Corbo, Claudiu T. Supuran & Clemente Capasso
Pages: 146-150
Published online: 15 Feb 2013
AbstractforBiomimetic CO2 capture using a highly thermostable bacterial α-carbonic anhydrase immobilized on a polyurethane foam | Full Text | References | PDF (407.2 KB)
  • 3573 Views
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Errata

Correction
Corrigendum
Page: 151
Published online: 06 Sep 2013
CitationforCorrigendum | Full Text | PDF (139.9 KB)
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