3,223
Views
181
CrossRef citations to date
0
Altmetric
Research Article

Synthesis of 4-benzyl-1,3-thiazole derivatives as potential anti-inflammatory agents: An analogue-based drug design approach

, , , &
Pages 890-897 | Received 27 Jun 2008, Accepted 09 Sep 2008, Published online: 01 Jun 2009

Keep up to date with the latest research on this topic with citation updates for this article.

Read on this site (22)

Muhammad Taha, Fazal Rahim, Ihsan Ullah Khan, Nizam Uddin, Rai Khalid Farooq, Abdul Wadood, Ashfaq Ur Rehman & Khalid Mohammed Khan. (2023) Synthesis of thiazole-based-thiourea analogs: as anticancer, antiglycation and antioxidant agents, structure activity relationship analysis and docking study. Journal of Biomolecular Structure and Dynamics 41:21, pages 12077-12092.
Read now
Soufiane Benreka, Fatima-Zohra Zradni, Fatiha Madi, Gilbert Kirsch & Souad Kasmi-Mir. (2022) Synthesis of thiazolylidenethiazoloquinazolinone hybrids from monocarbonyl curcumin analogues. Characterization, bio-evaluation and DFT study. Journal of Sulfur Chemistry 43:1, pages 53-77.
Read now
Huda K. Mahmoud, Ashraf A. Abbas & Sobhi M. Gomha. (2021) Synthesis, Antimicrobial Evaluation and Molecular Docking of New Functionalized Bis(1,3,4-Thiadiazole) and Bis(Thiazole) Derivatives. Polycyclic Aromatic Compounds 41:9, pages 2029-2041.
Read now
Hossein Shahbazi-Alavi, Ali Kareem Abbas & Javad Safaei-Ghomi. (2021) Synthesis of Thiazoles Catalyzed by Dichlorotriazine Attached to Graphene Oxide. Organic Preparations and Procedures International 53:4, pages 426-430.
Read now
Rayees Ahmad Naikoo, Rupesh Kumar, Vipan Kumar & Gaurav Bhargava. (2021) Recent developments in the synthesis of tricyclic condensed pyrimidinones. Synthetic Communications 51:10, pages 1451-1477.
Read now
Olesia G. Kulyk, Dmytro A. Biloborodov, Maksim A. Cherevatenko, Yevhen Y. Shyriakin, Alexander Yu. Lyapunov, Alexander V. Mazepa, Valerii V. Vashchenko, Valeriy D. Orlov & Maksim A. Kolosov. (2020) Versatile approaches to a library of building blocks based on 5-acylthiazole skeleton. Synthetic Communications 50:23, pages 3616-3628.
Read now
Manisha R. Bhosle, Sayali A. Kharote, Giribala M. Bondle & Jyotirling R. Mali. (2019) Tromethamine organocatalyzed efficient tandem-multicomponent synthesis of new thiazolyl-4-thiazolidinones in aqueous medium. Synthetic Communications 49:10, pages 1286-1300.
Read now
Mosaad S. Mohamed, Yara E. Mansour, Hatem K. Amin & Moustafa E. El-Araby. (2018) Molecular modelling insights into a physiologically favourable approach to eicosanoid biosynthesis inhibition through novel thieno[2,3-b]pyridine derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 755-767.
Read now
Abdou O. Abdelhamid & Sobhi M. Gomha. (2017) Synthesis and characterization of new pyrazole-based thiazoles. Synthetic Communications 47:15, pages 1409-1414.
Read now
Sabine Grösch, Ellen Niederberger & Gerd Geisslinger. (2017) Investigational drugs targeting the prostaglandin E2 signaling pathway for the treatment of inflammatory pain. Expert Opinion on Investigational Drugs 26:1, pages 51-61.
Read now
Shaik Thaslim Basha, Hasti Sudhamani, Syed Rasheed, Nagam Venkateswarlu, Tartte Vijaya & Chamarthi Naga Raju. (2016) Microwave-assisted neat synthesis of α-aminophosphonate/phosphinate derivatives of 2-(2-aminophenyl)benzothiazole as potent antimicrobial and antioxidant agents. Phosphorus, Sulfur, and Silicon and the Related Elements 191:10, pages 1339-1343.
Read now
Ahmed A. Fadda, Afnan M. El-badraw, Hala M. Refat & Ehab Abdel-Latif. (2016) Synthesis of some new 2-substituted-4-sulfamoylphenylazo-thiophene and/or thiazole derivatives as antibacterial agents. Phosphorus, Sulfur, and Silicon and the Related Elements 191:5, pages 778-785.
Read now
F. Ghanbari Pirbasti, Nosrat O. Mahmoodi & Jafar Abbasi Shiran. (2016) Synthesis and evaluation of biological activities of 4-cyclopropyl-5-(2-fluorophenyl) arylhydrazono-2,3-dihydrothiazoles as potent antioxidant agents. Journal of Sulfur Chemistry 37:2, pages 196-210.
Read now
Sunil Kumar, Ranjana Aggarwal & Chetan Sharma. (2015) Synthesis of Some 2-(3-Alkyl/aryl-5-trifluoromethylpyrazol-1-yl)-4-(coumarin-3-yl)thiazoles as Novel Antibacterial Agents. Synthetic Communications 45:17, pages 2022-2029.
Read now
Mungara Anil Kumar, Tran Nguyen Minh An, In Ja Lee, Soonheum Park & Kap Duk Lee. (2015) Synthesis and Bioactivity of Novel Phenothiazine-Based Thiazole Derivatives. Phosphorus, Sulfur, and Silicon and the Related Elements 190:7, pages 1160-1168.
Read now
Ravibabu Velpula, Ramesh Gondru, Yashodhara Velivela & Rajitha Bavantula. (2015) Synthesis and Antibacterial Evaluation of Novel 3,6-Disubstituted Coumarin Derivatives. Synthetic Communications 45:5, pages 578-585.
Read now
Minh An Tran Nguyen, Anil Kumar Mungara, Jung-Ae Kim, Kap Duk Lee & Soonheum Park. (2015) Synthesis, Anticancer and Antioxidant Activity of Novel Carbazole-based Thiazole Derivatives. Phosphorus, Sulfur, and Silicon and the Related Elements 190:2, pages 191-199.
Read now
Moustafa A. Gouda, Yousery El-Sayed Sherif & Mohamed S. Elsherbini. (2014) Synthesis, Anti-Inflammatory, and Analgesic Evaluation of Some 2-Amino-5-Selenothiazoles. Phosphorus, Sulfur, and Silicon and the Related Elements 189:11, pages 1633-1643.
Read now
ManojN. Bhoi, MayuriA. Borad & HiteshD. Patel. (2014) Synthetic Strategies for Fused Benzothiazoles: Past, Present, and Future. Synthetic Communications 44:17, pages 2427-2457.
Read now
NosratO. Mahmoodi, Niloufar Safari & Bahman Sharifzadeh. (2014) One-Pot Synthesis of Novel 2-(Thiazol-2-yl)-4,5-dihydropyridazin-3(2H)-one Derivatives Catalyzed by Activated KSF. Synthetic Communications 44:2, pages 245-250.
Read now

Articles from other publishers (159)

Refaie M Kassab, Sami A Al-Hussain, Aboubakr H Abdelmonsef, Magdi EA Zaki, Sobhi M Gomha & Zeinab A Muhammad. (2023) Novel xylenyl-spaced bis-thiazoles/thiazines: synthesis, biological profile as herpes simplex virus type 1 inhibitors and in silico simulations . Future Medicinal Chemistry.
Crossref
Nutan V. Sadgir, Vishnu A. Adole, Sunil L. Dhonnar & Bapu S. Jagdale. (2023) Synthesis and biological evaluation of coumarin appended thiazole hybrid heterocycles: Antibacterial and antifungal study. Journal of Molecular Structure 1293, pages 136229.
Crossref
Hayat Ullah, Aisha Rab Nawaz, Muhammad Nabi, Ayesha Nawaz, Fazal Rahim, Fahad Khan & Amjad Hussain. (2023) Design, synthesis, in vitro urease inhibitory potential and in silico molecular docking study of substituted thiazole bearing thiourea hybrid analogues. Chemical Data Collections 48, pages 101086.
Crossref
Xiao Shi, Peng Liu, Yanyan Ma, Mingyuan Li, Zhenyu Zhang, Xinyue Zhang, Dahua Shi & Xinxin Si. (2023) Identification of a 2‐phenylthiazole derivative acetylcholinesterase modulator with in vitro antitumor activity in breast cancer cells. Chemical Biology & Drug Design.
Crossref
Rupali Rana, Nitish Kumar, Harmandeep Kaur Gulati, Anchal Sharma, Aanchal Khanna, Pooja, Rakshit Badhwar, Muskan Dhir, Jyoti, Jatinder Vir Singh & Preet Mohinder Singh Bedi. (2023) A comprehensive review on thiazole based conjugates as anti-cancer agents. Journal of Molecular Structure 1292, pages 136194.
Crossref
Lubna Afroz, Moinuddin Khan, H.M. Vagdevi, Mohammad Azam, Shakeel Ahmed Adhoni & Mahboob Alam. (2023) Synthesis, structural characterization, and thermal studies of 3d-metal complexes derived from a thiazole-based ligand: Multifaceted biological properties and molecular docking studies. Polyhedron 243, pages 116542.
Crossref
Mohammed Hawash, Nidal Jaradat, Rozan Sabobeh, Murad Abualhasan & Mohammed T. Qaoud. (2023) New Thiazole Carboxamide Derivatives as COX Inhibitors: Design, Synthesis, Anticancer Screening, In Silico Molecular Docking, and ADME Profile Studies. ACS Omega 8:32, pages 29512-29526.
Crossref
Sunil L. Dhonnar, Vishnu A. Adole, Rajendra H. Patil, Bhushan B. Khairnar, Thansing B. Pawar, Nutan V. Sadgir & Bapu S. Jagdale. (2023) Synthesis, Spectral, Antifungal, In Silico Molecular Docking,ADME and DFT Studies of Some 2-(2-Hydrazineyl)thiazole Derivatives: Computational and Experimental Perspective. Journal of Molecular Structure, pages 136411.
Crossref
Hayat Ullah, Saman Maqsood, Fazal Rahim, Abdullah Yahya Abdullah Alzahrani & Abdul Wadood. (2023) Synthesis, in vitro α-glucosidase, α-amylase activities and molecular docking study of hybrid thiazole-sulfonohydrazide analogues. Chemical Data Collections 46, pages 101043.
Crossref
Dandan Li, Long Chen, Yang Jin, Xiaochen Wang, Long Liu, Yilin Li, Gongyuan Chen, Guanhao Wu, Yujie Qin, Leilei Yang, Mengke Wang, Lulu Zhao, Zhihong Xu & Jiangwei Wen. (2023) An electrochemical-enabled cascaded cyclization of enaminones with potassium thiocyanate and alcohols to access 2-alkoxythiazoles. Green Chemistry 25:12, pages 4656-4661.
Crossref
Mohamed H.A. Soliman, Nashwa M. Mahmoud, Aml B. Mohamed & Howayda E. Khaled. (2023) Synthesis, anticancer evaluation, and molecular docking study of some arylidenehydrazono analogues. Canadian Journal of Chemistry 101:6, pages 353-363.
Crossref
Narges Hosseini Nasab, Hussain Raza, Young Seok Eom, Mubashir Hassan, Andrzej Kloczkowski & Song Ja Kim. (2023) Synthesis and discovery of potential tyrosinase inhibitor of new coumarin‐based thiophenyl‐pyrazolylthiazole nuclei: In vitro evaluation, cytotoxicity, kinetic, and computational studies. Chemical Biology & Drug Design 101:6, pages 1262-1272.
Crossref
Gang Li, Xiaoshan Guo, Wenkang Ren, Jiafeng Wang, Zhen Lv, Hongling Li, Mingrui Sun, Xiaoming Li, Gang Chen, Zhiguo Zhang, Wenting Zhang & Ming Bu. (2023) Novel Endoperoxide Steroid Derivatives Containing Thiazole Moiety as Potential Antitumor Agents: Design, Synthesis, and Cytotoxic Evaluation. Natural Product Communications 18:5, pages 1934578X2311755.
Crossref
Mohammed Hawash, Nidal Jaradat, Murad Abualhasan, Murat Kadır Şüküroğlu, Mohammed T. Qaoud, Deniz Cansen Kahraman, Heba Daraghmeh, Leen Maslamani, Mais Sawafta, Ala Ratrout & Linda Issa. (2023) Design, synthesis, molecular docking studies and biological evaluation of thiazole carboxamide derivatives as COX inhibitors. BMC Chemistry 17:1.
Crossref
. (2023) Systematic Review on Thiazole Compounds as Nanoparticles: Chemistry, Synthesis, Antimicrobial Activities, Therapeutic Investigation. Nanosistemi, Nanomateriali, Nanotehnologii 21:1.
Crossref
Ghaidaa H. Alfaifi, Thoraya A. Farghaly & Magda H. Abdellattif. (2023) Indenyl-thiazole and indenyl-formazan derivatives: Synthesis, anticancer screening studies, molecular-docking, and pharmacokinetic/ molin-spiration properties. PLOS ONE 18:3, pages e0274459.
Crossref
Shahnawaz Khan, Monish Arbaz Ansari & Maya Shankar Singh. (2023) Access to Functionalized Thiazolothiadiazoles via the Chemoselective Cascade Heteroannulation of Thioamides with Hypervalent Iodine Reagents. Organic Letters 25:4, pages 642-646.
Crossref
Rafaqat Hussain, Fazal Rahim, Wajid Rehman, Syed Adnan Ali Shah, Shoaib Khan, Imran Khan, Liaqat Rasheed, Syahrul Imran, Abdul Wadood & Magda H. Abdellatif. (2023) Benzoxazole based thiazole hybrid analogs: Synthesis, in vitro cholinesterase inhibition, and molecular docking studies. Computational Toxicology 25, pages 100253.
Crossref
Rayees Ahmad Naikoo, Rashmi Sharma, Rupesh Kumar & Gaurav Bhargava. (2023) A new entrant in ketene family: Generation of 2‐(3‐Oxo‐allyl)‐isoindole‐1,3‐dione and their [4+2] Cycloadditions with 1,3‐Diazabuta‐1,3‐dienes. Asian Journal of Organic Chemistry 12:2.
Crossref
S. B. Bakare. (2023) Synthesis and Mass Spectra of Thiazole and Thiohydantoin Derivatives. Russian Journal of Organic Chemistry 59:1, pages 93-98.
Crossref
Rajia Sultana, Md. Din Islam, Fazria Tanjum, Mohammad Mostafizur Rahman & Md. Aminul Haque. (2022) Antioxidant, Antibacterial and Antifungal Properties of Black Pepper Essential Oil (Piper nigrum Linn) and Molecular Docking and Pharmacokinetic Studies of Its’ Major Component. Oriental Journal Of Chemistry 38:6, pages 1554-1560.
Crossref
Inas G. Shahin, Khaled O. Mohamed, Azza T. Taher, Abdelrahman S. Mayhoub & Asmaa E. Kassab. (2022) The Anti-MRSA Activity of Phenylthiazoles: A Comprehensive Review. Current Pharmaceutical Design 28:43, pages 3469-3477.
Crossref
Narges Hosseini Nasab, Fereshteh Azimian, Hendrik G. Kruger & Song Ja Kim. (2022) Acetylcoumarin in cyclic and heterocyclic-containing coumarins: Synthesis and biological applications. Tetrahedron 129, pages 133158.
Crossref
Said Rammali, Lahoucine Hilali, Khadija Dari, Bouchaib Bencharki, Abdellatif Rahim, Mohammed Timinouni, Fatima Gaboune, Mohamed El Aalaoui & Abdelkrim khattabi. (2022) Antimicrobial and antioxidant activities of Streptomyces species from soils of three different cold sites in the Fez-Meknes region Morocco. Scientific Reports 12:1.
Crossref
Sajid Ali Channar, Pervaiz Ali Channar, Aamer Saeed, Aisha A. Alsfouk, Syeda Abida Ejaz, Rabail Ujan, Razia Noor, Muhammad Sajjad Bilal, Qamar Abbas, Zahid Hussain, Bilal Ahmad Khan, Hussain Raza, Hafiz Abdul Bari Indher & Parvez Ali Mahesar. (2022) Exploring thiazole-linked thioureas using alkaline phosphatase assay, biochemical evaluation, computational analysis and structure–activity relationship (SAR) studies. Medicinal Chemistry Research 31:10, pages 1792-1802.
Crossref
Murtaza Madni, Muhammad Naeem Ahmed, Ghazala Abbasi, Shahid Hameed, Mahmoud A. A. Ibrahim, Muhammad N. Tahir, Muhammad Ashfaq, Diego M. Gil, Rosa M. Gomila & Antonio Frontera. (2022) Synthesis and X‐ray Characterization of 4,5‐Dihydropyrazolyl‐Thiazoles Bearing a Coumarin Moiety: On the Importance of Antiparallel π‐Stacking. ChemistrySelect 7:36.
Crossref
Fernando Mejía Zarate, Maribel Arroyo Carranza, Hugo Torrens Miquel, Adán Bazán-Jiménez, Marco A. García-Revilla & Juan Luis Bautista Martínez. (2022) Synthesis and computational characterization of aryl-fluorinated thiazoles: Experimental, DFT and molecular coupling studies. Journal of Fluorine Chemistry 261-262, pages 110024.
Crossref
N. P. Novichikhina, Z. E. Ashrafova, N. V. Stolpovskaya, I. V. Ledenyova, M. G. Kholyavka, N. A. Podoplelova, M. A. Panteleev & Kh. S. Shikhaliev. (2022) Synthesis and properties of novel hybrid molecules bearing 4H-pyrrolo[3,2,1-ij]quinolin-2-one and thiazole moieties. Russian Chemical Bulletin 71:9, pages 1969-1975.
Crossref
Nazli Farajzadeh, Sadin Özdemir, Serpil Gonca, Göknur Yaşa Atmaca, Ali Erdoğmuş, Zehra Altuntaş Bayır & Makbule Burkut Koçak. (2021) Photophysicochemical and Biological Properties of New Phthalocyanines Bearing 4‐(trifluoromethoxy)phenoxy and 2‐(4‐methylthiazol‐5‐yl)ethoxy Groups on Peripheral Positions. Photochemistry and Photobiology 98:4, pages 894-906.
Crossref
Rais Ahmad Khan, Seham Suliman Alterary, Ibtisam I. BinSharfan, Huda Alsaeedi, Amal AlFawaz, Mohd. Shahnawaz Khan, Mohammad H Jaafar, Yanshu Shi, Hadi D. Arman & Ali Alsalme. (2022) Piano-stool type (η6-p-cymene)ruthenium(II) thiazole-derived motifs complexes: Synthesis, crystal structures, DFT studies, molecular docking and in-vitro binding studies with HSA and cytotoxicity. Inorganica Chimica Acta 537, pages 120925.
Crossref
Salah A. Abdel‐Aziz, Ehab S. Taher, Ping Lan, Nawal A. El‐Koussi, Ola I. A. Salem, Hesham A. M. Gomaa & Bahaa G. M. Youssif. (2022) New pyrimidine/thiazole hybrids endowed with analgesic, anti‐inflammatory, and lower cardiotoxic activities: Design, synthesis, and COX‐2/sEH dual inhibition. Archiv der Pharmazie 355:7.
Crossref
Pradip Bera, Abhishek Aher, Paula Brandao, Utsab Debnath, Varun Dewaker, Sunil Kr. Manna, Abhimanyu Jana, Chandana Pramanik, Basudev Mandal & Pulakesh Bera. (2022) Instigating the In Vitro Anticancer Activity of New Pyridine–Thiazole-Based Co(III), Mn(II), and Ni(II) Complexes: Synthesis, Structure, DFT, Docking, and MD Simulation Studies . Journal of Chemical Information and Modeling 62:6, pages 1437-1457.
Crossref
Lakshmi Haritha Bharathi Maganti, Deepthi Ramesh, Balaji Gowrivel Vijayakumar, Mohd Imran K. Khan, Arunkumar Dhayalan, Jayabal Kamalraja & Tharanikkarasu Kannan. (2022) Acetylene containing 2-(2-hydrazinyl)thiazole derivatives: design, synthesis, and in vitro and in silico evaluation of antimycobacterial activity against Mycobacterium tuberculosis . RSC Advances 12:14, pages 8771-8782.
Crossref
Rasha Z. Batran, Sherien M. El‐Daly, Walaa A. El‐Kashak & Eman Y. Ahmed. (2022) Design, synthesis, and molecular modeling of quinoline‐based derivatives as anti‐breast cancer agents targeting EGFR/AKT signaling pathway. Chemical Biology & Drug Design 99:3, pages 470-482.
Crossref
Vishal Srivastava, Pravin K. Singh, Shraddha Tivari & Praveen P. Singh. (2022) Visible light photocatalysis in the synthesis of pharmaceutically relevant heterocyclic scaffolds. Organic Chemistry Frontiers 9:5, pages 1485-1507.
Crossref
Rabail Ujan, Hafiz Mohammad Kashif Mahmood, Pervaiz Ali Channar, Syeda Abida Ejaz, Shomaila Saeed, Aamer Saeed, Amna Saeed, Mamoona Rafiq, Kashif Ali Channar, Hafiz Abdul Bari Indher & Hammad Ismail. (2022) N-(5-acetyl-4-methylthiazol-2-yl)arylamide derivatives as multi-target-directed ligands: design, synthesis, biochemical evaluation and computational analysis. Journal of Chemical Sciences 134:1.
Crossref
Rambabu Palabindela Rambabu PalabindelaPrabhakar MyadaraveniaRajashekar Korra Rajashekar KorraHimabindu Mekala Himabindu Mekala, Mamatha Kasula Mamatha Kasula & DEVENDAR BANOTHU DEVENDAR BANOTHU. (2022) Anthracene and 1,8-napthalimide aminothiazole hybrids: Synthesis, Antimicrobial activity and Molecular Docking Studies. Oriental Journal Of Chemistry 38:1, pages 137-143.
Crossref
Baji Baba Shaik, Pule Seboletswe, Sachin Balaso Mohite, Naresh Kumar KatariMuhammad D. Bala, Rajshekhar Karpoormath & Parvesh Singh. (2022) Lemon Juice: A Versatile Biocatalyst and Green Solvent in Organic Transformations. ChemistrySelect 7:5.
Crossref
Heba Mohamed, Mohamed AL-Ghareeb & Raghda Abd-Allah. (2022) Pharmacological Evaluation of Novel 1,2,4-triazine Derivatives Containing Thiazole Ring against Hepatocellular Carcinoma. Current Bioactive Compounds 18:2.
Crossref
Siddhant V. Kokate & Sachin V. Patil. (2022) Synthesis and Antimicrobial Screening of Some New Thiazole Substituted 1,3,4-Oxadiazole Derivatives. Synthesis and Antimicrobial Screening of Some New Thiazole Substituted 1,3,4-Oxadiazole Derivatives.
Rayees Ahmad Naikoo, Rupesh Kumar, Vipan Kumar & Gaurav Bhargava. (2022) Recent Developments in the Synthesis of Bicyclic Condensed Pyrimidinones. Current Organic Chemistry 26:2, pages 122-161.
Crossref
S. AGGARWAL, M. DEVGUN, R. NARANG, S. LAL, A.C. RANA & R. GOYAL. (2022) Thiazolopyrimidines: A Retrospective Study of Synthesis, Structure-Activity Relationship and Diverse Pharmacological Actions. Asian Journal of Chemistry 34:3, pages 519-530.
Crossref
Md. Shahazada Shah, Mohammad Mostafizur Rahman, Md. Din Islam, Abdullah Al-Macktuf, Junaid Uddin Ahmed, Hiroshi Nishino & Md. Aminul Haque. (2022) Synthesis, antimicrobial and antioxidant evaluation with in silico studies of new thiazole Schiff base derivatives. Journal of Molecular Structure 1248, pages 131465.
Crossref
Minakshi A. Meshram, Utkarsha O. Bhise, Priyanka N. Makhal & Venkata Rao Kaki. (2021) Synthetically-tailored and nature-derived dual COX-2/5-LOX inhibitors: Structural aspects and SAR. European Journal of Medicinal Chemistry 225, pages 113804.
Crossref
Diksha Sharma, Vishal Sharma, Archana Sharma, Rajat Goyal, Rajiv K. Tonk, Vijay Kumar Thakur & Prabodh C. Sharma. (2021) Green chemistry approaches for thiazole containing compounds as a potential scaffold for cancer therapy. Sustainable Chemistry and Pharmacy 23, pages 100496.
Crossref
P. Akhileshwari, K.R. Kiran, M.A. Sridhar, M.P. Sadashiva & N.K. Lokanath. (2021) Synthesis, crystal structure characterization, Hirshfeld surface analysis, and Quantum chemical computations of Ethyl 5-(thiophene-2-carbonyl)thiazole-4-carboxylate. Journal of Molecular Structure 1242, pages 130747.
Crossref
L. K. Durgeswari, Ravi Kumar Ganta & Y. L. N. Murthy. (2021) Synthesis, Characterization, and Antioxidant Properties of Novel 1-(4-Aryl-1,3-thiazol-2-yl)-2-{[1-(3-methylbut-2-en-1-yl)-1H-indol-3-yl]methylidene}hydrazines. Russian Journal of Organic Chemistry 57:9, pages 1552-1558.
Crossref
Amerah M. Al-Soliemy, Thoraya A. Farghaly, Eman M.H. Abbas, Mohamed R. Shaaban, Mohie E.M. Zayed & Tarek B.A. El-Naggar. (2021) Synthesis of Thiazolyl-N-phenylmorpholine Derivatives and their Biological Activities. Medicinal Chemistry 17:7, pages 790-805.
Crossref
O. Benali, M. Zebida & U. Maschke. (2021) Synthesis and inhibition corrosion effect of two thiazole derivatives for carbon steel in 1 ​M HCl. Journal of the Indian Chemical Society 98:8, pages 100113.
Crossref
Mamdouh A. Sofan, Ahmed El‐Mekabaty, Ali M. Hasel & Samy B. Said. (2021) Synthesis, cytotoxicity assessment and antioxidant activity of some new thiazol‐2‐yl carboxamides. Journal of Heterocyclic Chemistry 58:8, pages 1645-1655.
Crossref
Sraa Abu-Melha, Sobhi Gomha, Amr Abouzied, Mastoura Edrees, Ahmed Abo Dena & Zeinab Muhammad. (2021) Microwave-Assisted One Pot Three-Component Synthesis of Novel Bioactive Thiazolyl-Pyridazinediones as Potential Antimicrobial Agents against Antibiotic-Resistant Bacteria. Molecules 26:14, pages 4260.
Crossref
Sherif M. H. Sanad, Ahmed E. M. Mekky, Ahmed Y. Said & Mohamed A. A. Elneairy. (2021) Pyridine‐2( 1 H )‐thiones: Versatile precursors for one‐pot synthesis of new nicotinonitrile‐thiazole hybrids . Journal of Heterocyclic Chemistry 58:7, pages 1461-1471.
Crossref
Seham A. Ibrahim & Hala F. Rizk. 2021. Azoles - Synthesis, Properties, Applications and Perspectives. Azoles - Synthesis, Properties, Applications and Perspectives.
Saraa Abu-Melha, Zeinab A. Muhammad, Amr S. Abouzid, Mastoura M. Edrees, Ahmed S. Abo Dena, Sara Nabil & Sobhi M. Gomha. (2021) Multicomponent synthesis, DFT calculations and molecular docking studies of novel thiazolyl-pyridazinones as potential antimicrobial agents against antibiotic-resistant bacteria. Journal of Molecular Structure 1234, pages 130180.
Crossref
Somaia S. Abd El-Karim, Hanaa S. Mohamed, Mohamed F. Abdelhameed, Abd El-Galil E. Amr, Abdulrahman A. Almehizia & Eman S. Nossier. (2021) Design, synthesis and molecular docking of new pyrazole-thiazolidinones as potent anti-inflammatory and analgesic agents with TNF-α inhibitory activity. Bioorganic Chemistry 111, pages 104827.
Crossref
Rizk E. Khidre & Ibrahim Ali M. Radini. (2021) Design, synthesis and docking studies of novel thiazole derivatives incorporating pyridine moiety and assessment as antimicrobial agents. Scientific Reports 11:1.
Crossref
Akhil Bansal, Alka Bali & Ajitesh Balaini. (2020) Synthesis and Evaluation of Substituted Aryl Thiazoles With Antioxidant Potential as Gastro-sparing Anti-inflammatory Agents. Letters in Drug Design & Discovery 17:12, pages 1566-1578.
Crossref
Abdullah S. Al‐Bogami, Tamer S. Saleh & Adel H. Al‐Shareef. (2020) Mechanochemical synthesis of 5‐acetylthiazole: A step toward green and sustainable chemistry. Journal of Heterocyclic Chemistry 57:10, pages 3605-3611.
Crossref
Murtaza Madni, Muhammad Naeem Ahmed, Muhammad Hafeez, Muhammad Ashfaq, Muhammad Nawaz Tahir, Diego M. Gil, Bartomeu Galmés, Shahid Hameed & Antonio Frontera. (2020) Recurrent π–π stacking motifs in three new 4,5-dihydropyrazolyl–thiazole–coumarin hybrids: X-ray characterization, Hirshfeld surface analysis and DFT calculations. New Journal of Chemistry 44:34, pages 14592-14603.
Crossref
Jaismy Jacob P & S.L. Manju. (2020) Identification and development of thiazole leads as COX-2/5-LOX inhibitors through in-vitro and in-vivo biological evaluation for anti-inflammatory activity. Bioorganic Chemistry 100, pages 103882.
Crossref
Mahesh Hublikar, Vikas Kadu, Jitender Kumar Dublad, Dattatraya Raut, Sachin Shirame, Parameshwar Makam & Raghunath Bhosale. (2020) ( E )‐2‐(2‐Allylidenehydrazinyl)thiazole derivatives: Design, green synthesis, in silico and in vitro antimycobacterial and radical scavenging studies . Archiv der Pharmazie 353:7.
Crossref
E. O. Hamed, M. G. Assy & M. M. Galahom. (2020) Heterocyclization of Aromatic Amino Acids: Novel Syntheses and Antibacterial Activity of Fused, Non-fused, and Spiro Polyheterocyclic Derivatives. Russian Journal of Organic Chemistry 56:6, pages 1062-1069.
Crossref
Tran Nguyen Minh An, Pham Thai Phuong, Nguyen Minh Quang, Nguyen Van Son, Nguyen Van Cuong, Le Van Tan, Mai Dinh Tri, Mahboob Alam & Pham Van Tat. (2020) Synthesis, Docking Study, Cytotoxicity, Antioxidant, and Anti-microbial Activities of Novel 2,4-Disubstituted Thiazoles Based on Phenothiazine. Current Organic Synthesis 17:2, pages 151-159.
Crossref
Pradip Bera, Abhishek Aher, Paula Brandao, Sunil Kumar Manna, Gopinath Mondal, Abhimanyu Jana, Ananyakumari Santra, Harekrishna Jana & Pulakesh Bera. (2020) Induced apoptosis against U937 cancer cells by Fe(II), Co(III) and Ni(II) complexes with a pyrazine-thiazole ligand: Synthesis, structure and biological evaluation. Polyhedron 182, pages 114503.
Crossref
Ashraf A. AlyProfProf, Asmaa H. Mohamed & Mohamed Ramadan. (2020) Synthesis and colon anticancer activity of some novel thiazole/-2-quinolone derivatives. Journal of Molecular Structure 1207, pages 127798.
Crossref
Mohammed T.-E. Maghraby, Ola M.F. Abou-Ghadir, Samia G. Abdel-Moty, Asmaa Y. Ali & Ola I.A. Salem. (2020) Novel class of benzimidazole-thiazole hybrids: The privileged scaffolds of potent anti-inflammatory activity with dual inhibition of cyclooxygenase and 15-lipoxygenase enzymes. Bioorganic & Medicinal Chemistry 28:7, pages 115403.
Crossref
Muhammad Haroon, Muhammad Khalid, Tashfeen Akhtar, Muhammad Nawaz Tahir, Muhammad Usman Khan, Shabbir Muhammad, Abdullah G. Al-Sehemi & Shahid Hameed. (2020) Synthesis, crystal structure, spectroscopic, electronic and nonlinear optical properties of potent thiazole based derivatives: Joint experimental and computational insight. Journal of Molecular Structure 1202, pages 127354.
Crossref
Prabodh Chander Sharma, Kushal Kumar Bansal, Archana Sharma, Diksha Sharma & Aakash Deep. (2020) Thiazole-containing compounds as therapeutic targets for cancer therapy. European Journal of Medicinal Chemistry 188, pages 112016.
Crossref
Madavi Sunitha, G. Venkateshappa, G. Ramesh, Jayanna Kengaiah, G. Shivaraja, Vivek Chandramohan, M. Shet Prakash & M.K. Shivananda. (2020) Antioxidant, Antimicrobial, Molecular Docking Studies of Novel 2,6-bis(1,3-Thiazol-2-yl)-4-(3,4,5-trimethoxyphenyl)pyridine and its Cu(II) and Ni(II) Complexes. Asian Journal of Organic & Medicinal Chemistry 5:2, pages 103-108.
Crossref
Pathki Uma, Firasath Unnisa, Pallati Naresh, Sai Prakash, P. R. Sushma & Kamatala Chinna Rajanna. Synthesis, characterization and biological activity of benzothiazoles derivatives. Synthesis, characterization and biological activity of benzothiazoles derivatives.
Ahmed H. Halawa, Essam M. Eliwa, Ahmed A. Hassan, Hesham S. Nassar, R.A. El-Eisawy, Mohamed Ismail, Marcel Frese, Mohamed Shaaban, Ahmed M. El-Agrody, Ahmed H. Bedair & Norbert Sewald. (2020) Synthesis, in vitro cytotoxicity activity against the human cervix carcinoma cell line and in silico computational predictions of new 4-arylamino-3-nitrocoumarin analogues. Journal of Molecular Structure 1200, pages 127047.
Crossref
Sumana Y. Kotian, Chakrabhavi Dhananjaya Mohan, Aloir A. Merlo, Shobith Rangappa, S. Chandra Nayak, K.M. Lokanatha Rai & Kanchugarakoppal S. Rangappa. (2020) Small molecule based five-membered heterocycles: A view of liquid crystalline properties beyond the biological applications. Journal of Molecular Liquids 297, pages 111686.
Crossref
Hossein Shahbazi-Alavi, Sheida Khojasteh-Khosro, Javad Safaei-Ghomi & Maryam Tavazo. (2019) Crosslinked sulfonated polyacrylamide (Cross-PAA-SO3H) tethered to nano-Fe3O4 as a superior catalyst for the synthesis of 1,3-thiazoles. BMC Chemistry 13:1.
Crossref
Abdou O. Abdelhamid, Ibrahim E. El Sayed, Yasser H. Zaki, Ahmed M. Hussein, Mangoud M. Mangoud & Mona A. Hosny. (2019) Utility of 5-(furan-2-yl)-3-(p-tolyl)-4,5-dihydro-1H-pyrazole-1-carbothioamide in the synthesis of heterocyclic compounds with antimicrobial activity. BMC Chemistry 13:1.
Crossref
Deepika Sharma, Sanjiv Kumar, Balasubramanian Narasimhan, Kalavathy Ramasamy, Siong Meng Lim, Syed Adnan Ali Shah & Vasudevan Mani. (2019) Synthesis, molecular modelling and biological significance of N-(4-(4-bromophenyl) thiazol-2-yl)-2-chloroacetamide derivatives as prospective antimicrobial and antiproliferative agents. BMC Chemistry 13:1.
Crossref
Hui Li, Juan Zhang, Yanqiu Zhang, Jiayi Wang & Gonghua Song. (2019) A novel metal-free synthesis of thiazole-substituted α-hydroxy carbonyl compounds and 2-alkenylthiazoles from thiazole N-oxides and olefins. Tetrahedron Letters 60:51, pages 150825.
Crossref
Shulei Pan, Binqiang Wu, Jinjin Hu, Ruigang Xu, Min Jiang, Xiaofei Zeng & Guofu Zhong. (2019) Palladium-Catalyzed Allylic Substitution Reaction of Benzothiazolylacetamide with Allylic Alcohols in Water. The Journal of Organic Chemistry 84:16, pages 10111-10119.
Crossref
Adileh Ayati, Saeed Emami, Setareh Moghimi & Alireza Foroumadi. (2019) Thiazole in the targeted anticancer drug discovery. Future Medicinal Chemistry 11:15, pages 1929-1952.
Crossref
Nurcan BERBER. (2019) Synthesis of Certain New Morpholine Derivatives Bearing a Thiazole Moiety. Sakarya University Journal of Science 23:4, pages 554-558.
Crossref
Sahar Majnooni, Joseph Duffield, Jessica Price, Ahmad Reza Khosropour, Hassan Zali-Boeini & Hudson Beyzavi. (2019) Aryliodoazide Synthons: A Different Approach for Diversified Synthesis of 2-Aminothiazole, 1,3-Thiazole, and 1,3-Selenazole Scaffolds. ACS Combinatorial Science 21:7, pages 516-521.
Crossref
Birutė Grybaitė, Rita Vaickelionienė, Maryna Stasevych, Olena Komarovska‐Porokhnyavets, Kristina Kantminienė, Volodymyr Novikov & Vytautas Mickevičius. (2019) Synthesis and Antimicrobial Activity of Novel Thiazoles with Reactive Functional Groups. ChemistrySelect 4:23, pages 6965-6970.
Crossref
Ye-Ji Kim, Hye-Jin Kwon, Si-Yeon Han & Young-Dae Gong. (2019) Synthesis of 2-Amino-5-Carboxamide Thiazole Derivatives via Dehydrative Cyclization of Thiourea Intermediate Resin on Solid Phase. ACS Combinatorial Science 21:5, pages 380-388.
Crossref
Sobhi M. Gomha, Hassan M. Abdel-aziz, Mohamed G. Badrey & Mohamed M. Abdulla. (2019) Efficient Synthesis of Some New 1,3,4‐Thiadiazoles and 1,2,4‐Triazoles Linked to Pyrazolylcoumarin Ring System as Potent 5α‐Reductase Inhibitors. Journal of Heterocyclic Chemistry 56:4, pages 1275-1282.
Crossref
Ibrahim F. Nassar, Dina S. El kady, Hanem M. Awad & Wael A. El‐Sayed. (2019) Design, Synthesis, and Anticancer Activity of New Oxadiazolyl‐Linked and Thiazolyl‐Linked Benzimidazole Arylidines, Thioglycoside, and Acyclic Analogs. Journal of Heterocyclic Chemistry 56:3, pages 1086-1100.
Crossref
Manal M. Alsharekh, Ismail I. Althagafi, Mohamed R. Shaaban & Thoraya A. Farghaly. (2018) Microwave-assisted and thermal synthesis of nanosized thiazolyl-phenothiazine derivatives and their biological activities. Research on Chemical Intermediates 45:2, pages 127-154.
Crossref
Runjhun Tandon, Iqubal Singh, Vijay Luxami, Nitin Tandon & Kamaldeep Paul. (2018) Recent Advances and Developments of in vitro Evaluation of Heterocyclic Moieties on Cancer Cell Lines . The Chemical Record 19:2-3, pages 362-393.
Crossref
Arshi Naqvi. (2018) Synthesis, Characterization and Drug-Likeness Predictions of 1,3-Thiazole and Benzothiazole Derivatives. Oriental Journal of Chemistry 34:6, pages 3134-3139.
Crossref
Yasser H. Zaki, Marwa S. Al-Gendey & Abdou O. Abdelhamid. (2018) A facile synthesis, and antimicrobial and anticancer activities of some pyridines, thioamides, thiazole, urea, quinazoline, β-naphthyl carbamate, and pyrano[2,3-d]thiazole derivatives. Chemistry Central Journal 12:1.
Crossref
Pramod K. Sahu, Praveen K. Sahu, Manvendra S. Kaurav, Mouslim Messali, Saud M. Almutairi, Puran L. Sahu & Dau D. Agarwal. (2018) Metal-Free Construction of Fused Pyrimidines via Consecutive C–C and C–N Bond Formation in Water. ACS Omega 3:11, pages 15035-15042.
Crossref
Mir Mohammad Masood, Mohammad Irfan, Shadab Alam, Phool Hasan, Aarfa Queen, Shifa Shahid, Muhammad Zahid, Amir Azam & Mohammad Abid. (2018) Synthesis, Antimicrobial Evaluation and In silico Studies of Novel 2,4- disubstituted-1,3-thiazole Derivatives. Letters in Drug Design & Discovery 16:2, pages 160-173.
Crossref
Shweta Sinha, Mukesh Doble & S.L. Manju. (2018) Design, synthesis and identification of novel substituted 2-amino thiazole analogues as potential anti-inflammatory agents targeting 5-lipoxygenase. European Journal of Medicinal Chemistry 158, pages 34-50.
Crossref
Elsherbiny H. El-Sayed & Ahmed A. Fadda. (2018) Synthesis and Antimicrobial Activity of Some Novel bis Polyfunctional Pyridine, Pyran, and Thiazole Derivatives. Journal of Heterocyclic Chemistry 55:10, pages 2251-2260.
Crossref
Murtaza Madni, Muhammad Naeem Ahmed, Shahid Hameed, Syed Wadood Ali Shah, Umer Rashid, Khurshid Ayub, M.Nawaz Tahir & Tariq Mahmood. (2018) Synthesis, quantum chemical, in vitro acetyl cholinesterase inhibition and molecular docking studies of four new coumarin based pyrazolylthiazole nuclei. Journal of Molecular Structure 1168, pages 175-186.
Crossref
Mohamed K.S. El-Nagar, Hajjaj H.M. Abdu-Allah, Ola I.A. Salem, Abdel-Hamid N. Kafafy & Hanan S.M. Farghaly. (2018) Novel N-substituted 5-aminosalicylamides as dual inhibitors of cyclooxygenase and 5-lipoxygenase enzymes: Synthesis, biological evaluation and docking study. Bioorganic Chemistry 78, pages 80-93.
Crossref
Evangelia Tsolaki, Phaedra Eleftheriou, Victor Kartsev, Athina Geronikaki & Anil K. Saxena. (2018) Application of Docking Analysis in the Prediction and Biological Evaluation of the Lipoxygenase Inhibitory Action of Thiazolyl Derivatives of Mycophenolic Acid. Molecules 23:7, pages 1621.
Crossref
Gülhan Turan-Zitouni, Betül Kaya Çavuşoğlu, Begüm Nurpelin Sağlık & Ulviye Acar Çevik. (2018) Synthesis and antimicrobial activities of some novel thiazole compounds. Turkish Journal of Biochemistry 43:3, pages 220-227.
Crossref
Jitendra Nalawade, Pravin C. Mhaske, Abhijit Shinde, Sachin V. Patil, Prafulla B. Choudhari & Vivek D. Bobade. (2018) Synthesis, Characterization, and Antimicrobial Screening of 4″‐methyl‐2,2″‐diaryl‐4,2′:4′,5″‐terthiazole Derivatives. Journal of Heterocyclic Chemistry 55:6, pages 1366-1374.
Crossref
Sunil Kumar, Vikram Saini, Indresh K. Maurya, Jayant Sindhu, Mukesh Kumari, Ramesh Kataria & Vinod Kumar. (2018) Design, synthesis, DFT, docking studies and ADME prediction of some new coumarinyl linked pyrazolylthiazoles: Potential standalone or adjuvant antimicrobial agents. PLOS ONE 13:4, pages e0196016.
Crossref
YASSER HUSSEIN EISSA MOHAMMED & SHAUKATH ARA KHANUM. (2018) Recent progress on anti-cancer of amide appended heterocyclic and its possible therapeutic applications. A review drug progress for cancer therapeutics.. International Journal of pharma and Bio Sciences 9:2.
Crossref
Vytautas Mickevičius, Birutė Grybaitė, Rita Vaickelionienė, Maryna Stasevych, Olena Komarovska-Porokhnyavets & Volodymyr Novikov. (2018) Synthesis, Transformation of 3-[(4-Arylthiazol-2-yl)(p-tolyl)amino]propanoic Acids, Bis(thiazol-5-yl)phenyl-, Bis(thiazol-5-yl)methane Derivatives, and Their Antimicrobial Activity. HETEROCYCLES 96:1, pages 86.
Crossref
Rafat M. Mohareb, Amira E. M. Abdallah & Ebtsam A. Ahmed. (2017) Synthesis and cytotoxicity evaluation of thiazole derivatives obtained from 2-amino-4,5,6,7-tetrahydrobenzo[b]thiophene- 3-carbonitrile. Acta Pharmaceutica 67:4, pages 495-510.
Crossref
Rajitha Sadashiva, Damodara Naral, Jyothi Kudva, S. Madan Kumar, K. Byrappa, R. Mohammed Shafeeulla & Manjunatha Kumsi. (2017) Synthesis, structure characterization, in vitro and in silico biological evaluation of a new series of thiazole nucleus integrated with pyrazoline scaffolds. Journal of Molecular Structure 1145, pages 18-31.
Crossref
Wafaa S. Hamama, Mona E. Ibrahim, Hadeer A. Raoof & Hanafi H. Zoorob. (2017) Synthesis and Antimicrobial Evaluation of Some Novel 5-Phenyl-5H-thiazolo[4,3-b][1,3,4]thiadiazole Systems. Journal of Heterocyclic Chemistry 54:4, pages 2360-2366.
Crossref
Fatma A. A. El-Hag, Sobhi M. Gomha & Thoraya A. Farghaly. (2017) Hydrazonoyl Halides Precursors to Synthesis of New Thiazole, Thiadiazole, and Benzothiazepine Derivatives. Journal of Heterocyclic Chemistry 54:2, pages 1172-1177.
Crossref
Uzma Salar, Khalid Mohammed Khan, Shazia Syed, Muhammad Taha, Farman Ali, Nor Hadiani Ismail, Shahnaz Perveen, Abdul Wadood & Mehreen Ghufran. (2017) Synthesis, in vitro β -glucuronidase inhibitory activity and in silico studies of novel ( E )-4-Aryl-2-(2-(pyren-1-ylmethylene)hydrazinyl)thiazoles. Bioorganic Chemistry 70, pages 199-209.
Crossref
Hatem K. Amin, Amr M. El-Araby, Sameh Eid, Tamer Nasr, Samir Bondock, Ola Leheta & Moustafa E. Dawoud. (2017) A Thiazole Analogue Exhibits an Anti-Proliferative Effect in Different Human Carcinoma Cell Lines and Its Mechanism Based on Molecular Modeling. Advances in Biological Chemistry 07:01, pages 76-87.
Crossref
Ragavendra Butta, Sowmya Donthamsetty V, Padmaja Adivireddy & Padmavathi Venkatapuram. (2017) Synthesis and Antimicrobial Activity of Azolyl Pyrimidines. Journal of Heterocyclic Chemistry 54:1, pages 524-530.
Crossref
S. D. Jagadale, A. D. Sawant & M. B. Deshmukh. (2017) Synthesis of Dibenzothiazolyldibenzo-18-Crown-6 and its Applications in Colorimetric Recognition of Palladium and as Antimicrobial Agent. Journal of Heterocyclic Chemistry 54:1, pages 161-164.
Crossref
B. Sakram, S. Rambabu, K. Ashok, B. Sonyanaik & D. Ravi. (2017) Microwave assisted aqueous phase synthesis of benzothiazoles and benzimidazoles in the presence of Ag2O. Russian Journal of General Chemistry 86:12, pages 2737-2743.
Crossref
Mohamed S. Bekheit, Abdelbasset A. Farahat & Bakr F. Abdel-Wahab. (2016) Synthetic routes to thiazoloquinazolines. Chemistry of Heterocyclic Compounds 52:10, pages 766-772.
Crossref
M. M. Trush, V. V. Kovalishyn & V. M. Blagodatnyi. (2016) QSAR studies and antimicrobial potential of 1,3-thiazolylphosphonium salts. The Ukrainian Biochemical Journal 88:4, pages 57-65.
Crossref
Abdou Abdelhamid, Ibrahim El Sayed, Mohamed Hussein & Mangoud Mangoud. (2016) Synthesis and Antimicrobial Activity of Some New Thiadiazoles, Thioamides, 5-Arylazothiazoles and Pyrimido[4,5-d][1,2,4]triazolo[4,3-a]pyrimidines. Molecules 21:8, pages 1072.
Crossref
Wafaa M. Abdou, Reham F. Barghash, Mohamed S. Bekheit & Athina Geronikaki. (2016) Cytotoxicity and Anti-inflammation Profiles of Synthesized Thiazoles-Based N -Bisphosphonates and Relevant Bisphosphonic acids . ChemistrySelect 1:13, pages 3797-3803.
Crossref
Abdou Abdelhamid, Sobhi Gomha, Nadia Abdelriheem & Saher Kandeel. (2016) Synthesis of New 3-Heteroarylindoles as Potential Anticancer Agents. Molecules 21:7, pages 929.
Crossref
Namık Özdemir. (2016) Quantum chemical study of tautomerism in 2-[(4-phenylthiazol-2-yl)hydrazonomethyl]phenol. Computational and Theoretical Chemistry 1086, pages 12-17.
Crossref
Eun-A Kim, Chang Hun Cho, Soo Young Choi, Jee-Yin Ahn, Seung-Ju Yang & Sung-Woo Cho. (2016) 2-Cyclopropylimino-3-methyl-1,3-thiazoline hydrochloride alters lipopolysaccharide-induced proinflammatory cytokines and neuronal morphology in mouse fetal brain. Neuropharmacology 102, pages 32-41.
Crossref
Sobhi M. Gomha, Mohamed G. Badrey & Mastoura M. Edrees. (2016) Heterocyclisation of 2,5-diacetyl-3,4-disubstituted-thieno[2,3-b]Thiophene Bis-Thiosemicarbazones Leading to Bis-Thiazoles and Bis-1,3,4-thiadiazoles as Anti-breast Cancer Agents. Journal of Chemical Research 40:2, pages 120-125.
Crossref
Pramod K. Sahu. (2016) Eco-friendly grinding synthesis of a double-layered nanomaterial and the correlation between its basicity, calcination and catalytic activity in the green synthesis of novel fused pyrimidines. RSC Advances 6:82, pages 78409-78423.
Crossref
Anu Mishra, Madhulika Srivastava, Pratibha Rai, Snehlata Yadav, Bhartendu Pati Tripathi, Jaya Singh & Jagdamba Singh. (2016) Visible light triggered, catalyst free approach for the synthesis of thiazoles and imidazo[2,1-b]thiazoles in EtOH : H 2 O green medium . RSC Advances 6:54, pages 49164-49172.
Crossref
Poonam Gautam, Deepika Gautam & R. P. Chaudhary. (2016) One Pot Regioselective Synthesis and Antimicrobial Studies of Some Novel Indazolyl-Thiazole Derivatives. Journal of Heterocyclic Chemistry 53:1, pages 294-302.
Crossref
Tushar Ramesh Pavase, Hong Lin, Qurat-ul-ain Shaikh & Zhenxing Li. (2015) Rapid detection methodology for inorganic mercury (Hg2+) in seafood samples using conjugated polymer (1,4-bis-(8-(4-phenylthiazole-2-thiol)-octyloxy)-benzene) (PPT) by colorimetric and fluorescence spectroscopy. Sensors and Actuators B: Chemical 220, pages 406-413.
Crossref
Chang Hun Cho, Jiae Kim, Jee-Yin Ahn, Hoh-Gyu Hahn & Sung-Woo Cho. (2015) N-adamantyl-4-methylthiazol-2-amine suppresses lipopolysaccharide-induced brain inflammation by regulating NF-κB signaling in mice. Journal of Neuroimmunology 289, pages 98-104.
Crossref
Hye Jung Ihn, Doohyun Lee, Taeho Lee, Sang-Hyun Kim, Hong-In Shin, Yong Chul Bae, Jung Min Hong & Eui Kyun Park. (2015) Inhibitory Effects of KP-A159, a Thiazolopyridine Derivative, on Osteoclast Differentiation, Function, and Inflammatory Bone Loss via Suppression of RANKL-Induced MAP Kinase Signaling Pathway. PLOS ONE 10:11, pages e0142201.
Crossref
Mehmet Akkurt, Victoria A. Smolenski, Shaaban K. Mohamed, Jerry P. Jasinski, Alaa A. Hassan & Mustafa R. Albayati. (2015) Crystal structure of methyl (2 Z )-2-[(2 Z )-2-(2-cyclopentylidenehydrazin-1-ylidene)-4-oxo-3-phenyl-1,3-thiazolidin-5-ylidene]ethanoate . Acta Crystallographica Section E Crystallographic Communications 71:10, pages o776-o777.
Crossref
Amira S. Abd El-All, Asmaa A. Magd-El-Din, Fatma A. F. Ragab, Mahmoud ElHefnawi, Mohamed M. Abdalla, Shadia A. Galal & Ahmed A. El-Rashedy. (2015) New Benzimidazoles and Their Antitumor Effects with Aurora A Kinase and KSP Inhibitory Activities. Archiv der Pharmazie 348:7, pages 475-486.
Crossref
Fernando Cagide, Fernanda Borges, Ligia R. Gomes & John Nicolson Low. (2015) Synthesis and characterisation of new 4-oxo-N-(substituted-thiazol-2-yl)-4H-chromene-2-carboxamides as potential adenosine receptor ligands. Journal of Molecular Structure 1089, pages 206-215.
Crossref
Abdul Rouf & Cihangir Tanyeli. (2015) Bioactive thiazole and benzothiazole derivatives. European Journal of Medicinal Chemistry 97, pages 911-927.
Crossref
Deepika Gautam & R.P. Chaudhary. (2015) Synthesis, X-ray, DFT and photophysical properties of some new ferrocenyl hydrazono thiazolidin-4-ones and their derivatives. Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy 143, pages 256-264.
Crossref
N. J. P. Subhashini, Jampaiah Amanaganti & Shivaraj. (2015) Synthesis and antibacterial activity of 2-(3-acylphenyl)amino-4-phenylthiazole. Russian Journal of General Chemistry 85:3, pages 686-688.
Crossref
Shaik Sharafuddin Basha, Putta Ramachandra Reddy, Adivireddy Padmaja, Venkatapuram Padmavathi, Kalla Chandra Mouli & Tartte Vijaya. (2014) Synthesis and antimicrobial activity of 3-aroyl-4-heteroaryl pyrroles and pyrazoles. Medicinal Chemistry Research 24:3, pages 954-964.
Crossref
Lizhi Gai, John Mack, Hua Lu, Tebello Nyokong, Zhifang Li, Nagao Kobayashi & Zhen Shen. (2015) Organosilicon compounds as fluorescent chemosensors for fluoride anion recognition. Coordination Chemistry Reviews 285, pages 24-51.
Crossref
Ahmad LuqmanVictoria L. BlairRajini Brammananth, Paul K. Crellin, Ross L. Coppel, Lukasz Kedzierski & Philip C. Andrews. (2015) Homoleptic and Heteroleptic Bismuth(III) Thiazole–Thiolates and the Influence of Ring Substitution on Their Antibacterial and Antileishmanial Activity. European Journal of Inorganic Chemistry 2015:4, pages 725-733.
Crossref
Sobhi Gomha, Sayed Ahmed & Abdou Abdelhamid. (2015) Synthesis and Cytotoxicity Evaluation of Some Novel Thiazoles, Thiadiazoles, and Pyrido[2,3-d][1,2,4]triazolo[4,3-a]pyrimidin-5(1H)-ones Incorporating Triazole Moiety. Molecules 20:1, pages 1357-1376.
Crossref
Abdou O. Abdelhamid, Sobhi M. Gomha & Ahmad S. Shawali. (2015) Synthesis and Antimicrobial Evaluation of Some Novel Thiazole, 1,3,4-Thiadiazole and Pyrido[2,3-d][1,2,4]triazolo[4,3-a]pyrimidine Derivatives Incorporating Pyrazole Moiety. HETEROCYCLES 91:11, pages 2126.
Crossref
Ramesh Katla, Rakhi Chowrasia, Padma Sunitha Manjari & Nelson Luís C. Domingues. (2015) An efficient aqueous phase synthesis of benzimidazoles/benzothiazoles in the presence of β-cyclodextrin. RSC Advances 5:52, pages 41716-41720.
Crossref
N. C. Desai, Nayan Bhatt & Hardik Somani. (2014) Synthesis, characterization, and antimicrobial activity of some novel thiazole clubbed 1,3,4-oxadiazoles. Medicinal Chemistry Research 24:1, pages 258-266.
Crossref
Rupesh Dudhe, Pramod Kumar Sharma & Prabhakar Kumar Verma. (2014) Pyrimidine containing furanose derivative having antifungal, antioxidant, and anticancer activity. Organic and Medicinal Chemistry Letters 4:1.
Crossref
Joel T. Mague, Mehmet Akkurt, Shaaban K. Mohamed, Alaa A. Hassan & Mustafa R. Albayati. (2014) Crystal structure of 4-((1 E )-1-{(2 Z )-2-[4-(4-bromophenyl)-3-phenyl-2,3-dihydro-1,3-thiazol-2-ylidene]hydrazin-1-ylidene}ethyl)phenol hemihydrate . Acta Crystallographica Section E Structure Reports Online 70:10, pages o1124-o1125.
Crossref
Nguyen Minh An Tran, Mungara Anil Kumar, Seung Hyun Chang, Mi Yeong Kim, Jung-Ae Kim & Kap Duk Lee. (2014) Synthesis, Anticancer and Antioxidant Activity of Novel 2,4-Disubstituted Thiazoles. Bulletin of the Korean Chemical Society 35:6, pages 1619-1624.
Crossref
Joel T. Mague, Shaaban K. Mohamed, Mehmet Akkurt, Ahmed T. Abd El-Alaziz & Mustafa R. Albayati. (2014) 2-((1 E )-1-{2-[(2 Z )-4-(4-Bromophenyl)-3-phenyl-2,3-dihydro-1,3-thiazol-2-ylidene]hydrazin-1-ylidene}ethyl)pyridin-1-ium bromide monohydrate . Acta Crystallographica Section E Structure Reports Online 70:3, pages o328-o329.
Crossref
Prakash G. More, Netaji N. Karale, Anjana S. Lawand, Naina Narang & Rajendra H. Patil. (2013) Synthesis and anti-biofilm activity of thiazole Schiff bases. Medicinal Chemistry Research 23:2, pages 790-799.
Crossref
Nabhubygari Mahaboob Basha, Dandu Seenaiah, Adivireddy Padmaja, Venkatapuram Padmavathi, Desaraju Suresh Bhargav & Tartte Vijaya. (2014) Synthesis and Antioxidant Activity of Bis and Tris Heterocycles. Archiv der Pharmazie 347:1, pages 54-67.
Crossref
Yahia Nasser Mabkhot, Assem Barakat, Abdullah Mohammed Al-Majid, Saeed Alshahrani, Sammer Yousuf & M Iqbal Choudhary. (2013) Synthesis, reactions and biological activity of some new bis-heterocyclic ring compounds containing sulphur atom. Chemistry Central Journal 7:1.
Crossref
Nosrat O. Mahmoodi, Jafar Parvizi, Bahman Sharifzadeh & Mehdi Rassa. (2013) Facile Regioselective Synthesis of Novel bis -Thiazole Derivatives and Their Antimicrobial Activity . Archiv der Pharmazie 346:12, pages 860-864.
Crossref
S.V. Rajmane, V.P. Ubale, A.S. Lawand, A.M. Nalawade, N.N. Karale & P.G. More. (2013) A 4-(o-chlorophenyl)-2-aminothiazole: Microwave assisted synthesis, spectral, thermal, XRD and biological studies. Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy 115, pages 393-398.
Crossref
N.C. Desai, Nayan Bhatt, Hardik Somani & Amit Trivedi. (2013) Synthesis, antimicrobial and cytotoxic activities of some novel thiazole clubbed 1,3,4-oxadiazoles. European Journal of Medicinal Chemistry 67, pages 54-59.
Crossref
S. N. Thore, Sunil V. Gupta & Kamalkishor G. Baheti. (2012) Docking, synthesis, and pharmacological investigation of novel substituted thiazole derivatives as non-carboxylic, anti-inflammatory, and analgesic agents. Medicinal Chemistry Research 22:8, pages 3802-3811.
Crossref
Vijayta Gupta & Vinay Kant. (2013) A Review on Biological Activity of Imidazole and Thiazole Moieties and their Derivatives. Science International 1:7, pages 253-260.
Crossref
Samir Bondock, Tamer Naser & Yousry A. Ammar. (2013) Synthesis of some new 2-(3-pyridyl)-4,5-disubstituted thiazoles as potent antimicrobial agents. European Journal of Medicinal Chemistry 62, pages 270-279.
Crossref
Ranjana Aggarwal, Sunil Kumar, Pawan Kaushik, Dhirender Kaushik & Girish Kumar Gupta. (2013) Synthesis and pharmacological evaluation of some novel 2-(5-hydroxy-5-trifluoromethyl-4,5-dihydropyrazol-1-yl)-4-(coumarin-3-yl)thiazoles. European Journal of Medicinal Chemistry 62, pages 508-514.
Crossref
Channamata Shankar Naveena, Boja Poojary, Thangavelu Arulmoli, Kumshi Manjunatha, Ashwatanarayana Prabhu & Nalilu Sucheta Kumari. (2012) Synthesis and evaluation of biological and nonlinear optical properties of some novel 2,4-disubstituted [1,3]-thiazoles carrying 2-(aryloxymethyl)-phenyl moiety. Medicinal Chemistry Research 22:4, pages 1925-1937.
Crossref
Raghu Vardhan Reddy Mekala, Ravinder Reddy Danda & Hemalatha Gadegoni. (2013) Synthesis and Biological Evaluation of Some Novel [4-(1H-Benzoimidazol-2-yl)-thiazol-2-yl]-benzylidene-amines and N-[4-(1H-Benzoimidazol-2-yl)-thiazol-2-yl]-N'-benzylidene-hydrazines. Journal of the Korean Chemical Society 57:1, pages 94-98.
Crossref
Harshita Sachdeva, Diksha Dwivedi, R. R. Bhattacharjee, Sarita Khaturia & Rekha Saroj. (2013) NiO Nanoparticles: An Efficient Catalyst for the Multicomponent One-Pot Synthesis of Novel Spiro and Condensed Indole Derivatives. Journal of Chemistry 2013, pages 1-10.
Crossref
Manpreet Kaur, Jerry P. Jasinski, Amanda C. Keeley & H. S. Yathirajan. (2012) [2-(Biphenyl-4-yl)-1,3-thiazol-4-yl]methanol. Acta Crystallographica Section E Structure Reports Online 68:10, pages o2950-o2950.
Crossref
Anjali Jha, Y. L. N. Murthy, U. Sanyal & G. Durga. (2011) Rapid synthesis, characterization, anticancer and antimicrobial activity studies of substituted thiadiazoles and their dinucleating ligand metal complexes. Medicinal Chemistry Research 21:9, pages 2548-2556.
Crossref
Shiv Jee Kashyap, Vipin Kumar Garg, Pramod Kumar Sharma, Nitin Kumar, Rupesh Dudhe & Jitendra Kumar Gupta. (2011) Thiazoles: having diverse biological activities. Medicinal Chemistry Research 21:8, pages 2123-2132.
Crossref
Yahia Nasser Mabkhot, Assem Barakat, Abdullah Mohammad Al-Majid, Abdullah Saleh Alamary & Taleb T. Al-Nahary. (2012) A Novel and Expedient Approach to New Thiazoles, Thiazolo[3,2-a]pyridines, Dihydrothiophenes, and Hydrazones Incorporating Thieno[2,3-b]thiophene Moiety. International Journal of Molecular Sciences 13:4, pages 5035-5047.
Crossref
Cristina Mariana Moldovan, Ovidiu Oniga, Alina Pârvu, Brînduşa Tiperciuc, Philippe Verite, Adrian Pîrnău, Ovidiu Crişan, Marius Bojiţă & Raluca Pop. (2011) Synthesis and anti-inflammatory evaluation of some new acyl-hydrazones bearing 2-aryl-thiazole. European Journal of Medicinal Chemistry 46:2, pages 526-534.
Crossref
. (2010) Current World Literature. Current Opinion in Supportive & Palliative Care 4:2, pages 111-120.
Crossref

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.