Citations (44)
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Emma Baglini, Rahul Ravichandran, Emanuela Berrino, Silvia Salerno, Elisabetta Barresi, Anna Maria Marini, Monica Viviano, Sabrina Castellano, Federico Da Settimo, Claudiu T. Supuran, Sandro Cosconati & Sabrina Taliani. (2021) Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 1874-1883.
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Paolo Guglielmi, Giulia Rotondi, Daniela Secci, Andrea Angeli, Paola Chimenti, Alessio Nocentini, Alessandro Bonardi, Paola Gratteri, Simone Carradori & Claudiu T. Supuran. (2020) Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1891-1905.
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Siham A. Alissa, Hanan A. Alghulikah, Zeid A. ALOthman, Sameh M. Osman, Sonia Del Prete, Clemente Capasso, Alessio Nocentini & Claudiu T. Supuran. (2020) Inhibition survey with phenolic compounds against the δ- and η-class carbonic anhydrases from the marine diatom thalassiosira weissflogii and protozoan Plasmodium falciparum. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 377-382.
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Ali Irfan, Fozia Batool, Syeda Andleeb Zahra Naqvi, Amjad Islam, Sameh M. Osman, Alessio Nocentini, Siham A. Alissa & Claudiu T. Supuran. (2020) Benzothiazole derivatives as anticancer agents. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 265-279.
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Siham A. Alissa, Hanan A. Alghulikah, Zeid A. Alothman, Sameh M. Osman, Sonia Del Prete, Clemente Capasso, Alessio Nocentini & Claudiu T. Supuran. (2020) Phosphonamidates are the first phosphorus-based zinc binding motif to show inhibition of β-class carbonic anhydrases from bacteria, fungi, and protozoa. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 59-64.
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Emanuela Berrino & Claudiu T. Supuran. (2019) Novel approaches for designing drugs that interfere with pH regulation. Expert Opinion on Drug Discovery 14:3, pages 231-248.
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Mohammad M. Al-Sanea, Ahmed Elkamhawy, Sora Paik, Silvia Bua, So Ha Lee, Mohamed A. Abdelgawad, Eun Joo Roh, Wagdy M. Eldehna & Claudiu T. Supuran. (2019) Synthesis and biological evaluation of novel 3-(quinolin-4-ylamino)benzenesulfonamides as carbonic anhydrase isoforms I and II inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1457-1464.
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Giulia Rotondi, Paolo Guglielmi, Simone Carradori, Daniela Secci, Celeste De Monte, Barbara De Filippis, Cristina Maccallini, Rosa Amoroso, Roberto Cirilli, Atilla Akdemir, Andrea Angeli & Claudiu T. Supuran. (2019) Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1400-1413.
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Suleyman Akocak, Nabih Lolak, Silvia Bua, Alessio Nocentini & Claudiu T. Supuran. (2019) Activation of human α-carbonic anhydrase isoforms I, II, IV and VII with bis-histamine schiff bases and bis-spinaceamine substituted derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1193-1198.
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Baijayantimala Swain, Andrea Angeli, Srinivas Angapelly, Pavitra S. Thacker, Priti Singh, Claudiu T. Supuran & Mohammed Arifuddin. (2019) Synthesis of a new series of 3-functionalised-1-phenyl-1,2,3-triazole sulfamoylbenzamides as carbonic anhydrase I, II, IV and IX inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1199-1209.
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Alessandra Ammazzalorso, Simone Carradori, Andrea Angeli, Atilla Akdemir, Barbara De Filippis, Marialuigia Fantacuzzi, Letizia Giampietro, Cristina Maccallini, Rosa Amoroso & Claudiu T. Supuran. (2019) Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1051-1061.
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Özlen Güzel-Akdemir, Andrea Angeli, Kübra Demir, Claudiu T. Supuran & Atilla Akdemir. (2018) Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 1299-1308.
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Articles from other publishers (32)
Morteza Abdoli, Viviana De Luca, Clemente Capasso, Claudiu T. Supuran & Raivis Žalubovskis. (2023) Inhibition Studies on Carbonic Anhydrase Isoforms I, II, IX, and XII with a Series of Sulfaguanidines. ChemMedChem 18:6.
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Amber Ata, Uzma Salar, Faiza Saleem, Mehreen Lateef, Salman Ali Khan, Khalid Mohammed Khan, Muhammed Taha, Syed Moazzam Haider & Zaheer Ul-Haq. (2023) Identification of potential urease inhibitors and antioxidants based on saccharin derived analogs: Synthesis, in vitro, and in silico studies. Journal of Molecular Structure 1274, pages 134376.
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Ayoub El Mahmoudi, Hamza Tachallait, Zakaria Moutaoukil, Suhana Arshad, Khalid Karrouchi, Rachid Benhida & Khalid Bougrin. (2022)
Ultrasound‐Assisted Green Synthesis of 3,5‐Disubstituted Isoxazole Secondary Sulfonamides via One‐Pot Five‐Component Reaction using CaCl
2
/K
2
CO
3
as Pre‐Catalyst in Water
. ChemistrySelect 7:45.
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Amit Kumar, Kiran Siwach, Claudiu T. Supuran & Pawan K. Sharma. (2022) A decade of tail-approach based design of selective as well as potent tumor associated carbonic anhydrase inhibitors. Bioorganic Chemistry 126, pages 105920.
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Krishna K. Chinchilli, Venkata N. Royyala, Pavitra S. Thacker, Andrea Angeli, Srikanth Danaboina, Priti Singh, Srinivas Nanduri, Claudiu T. Supuran & Mohammed Arifuddin. (2022) Design, synthesis, SAR, and biological evaluation of saccharin‐based hybrids as carbonic anhydrase inhibitors. Archiv der Pharmazie 355:8.
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Yukimi Sugisaka, Shiori Aoyama, Konoka Kumagai, Makoto Ihara & Kazuhiko Matsuda. (2022)
TcGLIP GDSL Lipase Substrate Specificity Co-determines the Pyrethrin Composition in
Tanacetum cinerariifolium
. Journal of Agricultural and Food Chemistry 70:28, pages 8645-8652.
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Virginia Pontecorvi, Mattia Mori, Francesca Picarazzi, Susi Zara, Simone Carradori, Amelia Cataldi, Andrea Angeli, Emanuela Berrino, Paola Chimenti, Alessia Ciogli, Daniela Secci, Paolo Guglielmi & Claudiu T. Supuran. (2022) Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies. International Journal of Molecular Sciences 23:14, pages 7950.
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Derya Aktas Anil, Busra Ozturk Aydin, Yeliz Demir & Burcin Turkmenoglu. (2022) Design, synthesis, biological evaluation and molecular docking studies of novel 1H-1,2,3-Triazole derivatives as potent inhibitors of carbonic anhydrase, acetylcholinesterase and aldose reductase. Journal of Molecular Structure 1257, pages 132613.
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Lokman Durmaz, Adem Erturk, Mehmet Akyüz, Leyla Polat Kose, Eda Mehtap Uc, Zeynebe Bingol, Ruya Saglamtas, Saleh Alwasel & İlhami Gulcin. (2022) Screening of Carbonic Anhydrase, Acetylcholinesterase, Butyrylcholinesterase, and α-Glycosidase Enzyme Inhibition Effects and Antioxidant Activity of Coumestrol. Molecules 27:10, pages 3091.
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Kashif Rafiq, Najeeb Ur Rehman, Sobia Ahsan Halim, Majid Khan, Ajmal Khan & Ahmed Al-Harrasi. (2022) Design, Synthesis and Molecular Docking Study of Novel 3-Phenyl-β-Alanine-Based Oxadiazole Analogues as Potent Carbonic Anhydrase II Inhibitors. Molecules 27:3, pages 816.
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Silvia Salerno, Giorgio Amendola, Andrea Angeli, Emma Baglini, Elisabetta Barresi, Anna Maria Marini, Rahul Ravichandran, Monica Viviano, Sabrina Castellano, Ettore Novellino, Federico Da Settimo, Claudiu T. Supuran, Sandro Cosconati & Sabrina Taliani. (2021) Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold. European Journal of Medicinal Chemistry 220, pages 113490.
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Kashif Rafiq, Majid Khan, Niaz Muhammed, Ajmal Khan, Najeeb Ur Rehman, Balqees Essa Mohammad Al-Yahyaei, Mohammed Khiat, Sobia Ahsan Halim, Zarbad Shah, Rene Csuk & Ahmed Al-Harrasi. (2021) New amino acid clubbed Schiff bases inhibit carbonic anhydrase II, α-glucosidase, and urease enzymes: in silico and in vitro. Medicinal Chemistry Research 30:3, pages 712-728.
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Simone Carradori & Claudiu T. Supuran. 2021. pH-Interfering Agents as Chemosensitizers in Cancer Therapy. pH-Interfering Agents as Chemosensitizers in Cancer Therapy
79
94
.
Fabrizio Carta, Daniela Vullo & Andrea Angeli. 2021. pH-Interfering Agents as Chemosensitizers in Cancer Therapy. pH-Interfering Agents as Chemosensitizers in Cancer Therapy
63
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Shovan Mondal & Suniti Malakar. (2020) Synthesis of sulfonamide and their synthetic and therapeutic applications: Recent advances. Tetrahedron 76:48, pages 131662.
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Chandra B. Mishra, Manisha Tiwari & Claudiu T. Supuran. (2020) Progress in the development of human carbonic anhydrase inhibitors and their pharmacological applications: Where are we today?. Medicinal Research Reviews 40:6, pages 2485-2565.
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Kübra Demir-Yazıcı, Özlen Güzel-Akdemir, Andrea Angeli, Claudiu T. Supuran & Atilla Akdemir. (2020) Novel Indole-Based Hydrazones as Potent Inhibitors of the α-class Carbonic Anhydrase from Pathogenic Bacterium Vibrio cholerae. International Journal of Molecular Sciences 21:9, pages 3131.
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Melissa D’Ascenzio, Daniela Secci, Simone Carradori, Susi Zara, Paolo Guglielmi, Roberto Cirilli, Marco Pierini, Giulio Poli, Tiziano Tuccinardi, Andrea Angeli & Claudiu T. Supuran. (2020) 1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors. Journal of Medicinal Chemistry 63:5, pages 2470-2488.
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Alessio Nocentini, Sameh M. Osman, Sonia Del Prete, Clemente Capasso, Zeid A. ALOthman & Claudiu T. Supuran. (2019) Extending the γ-class carbonic anhydrases inhibition profiles with phenolic compounds. Bioorganic Chemistry 93, pages 103336.
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Begüm Nurpelin Sağlık, Ulviye Acar Çevik, Derya Osmaniye, Serkan Levent, Betul Kaya Çavuşoğlu, Yeliz Demir, Sinem Ilgın, Yusuf Özkay, Ali Savaş Koparal, Şükrü Beydemir & Zafer Asım Kaplancıklı. (2019) Synthesis, molecular docking analysis and carbonic anhydrase I-II inhibitory evaluation of new sulfonamide derivatives. Bioorganic Chemistry 91, pages 103153.
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Belma Zengin Kurt, Aydan Dag, Berna Doğan, Serdar Durdagi, Andrea Angeli, Alessio Nocentini, Claudiu T. Supuran & Fatih Sonmez. (2019) Synthesis, biological activity and multiscale molecular modeling studies of bis-coumarins as selective carbonic anhydrase IX and XII inhibitors with effective cytotoxicity against hepatocellular carcinoma. Bioorganic Chemistry 87, pages 838-850.
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Katarina Koruza, Brian P. Mahon, Matthew P. Blakeley, Andreas Ostermann, Tobias E. Schrader, Robert McKenna, Wolfgang Knecht & S. Zoë Fisher. (2019) Using neutron crystallography to elucidate the basis of selective inhibition of carbonic anhydrase by saccharin and a derivative. Journal of Structural Biology 205:2, pages 147-154.
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Marc A. Ilies & Jean-Yves Winum. 2019. Carbonic Anhydrases. Carbonic Anhydrases
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Simone Carradori & Paolo Guglielmi. 2019. Carbonic Anhydrases. Carbonic Anhydrases
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Daniela Vullo & Fabrizio Carta. 2019. Carbonic Anhydrases. Carbonic Anhydrases
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Claudiu T. Supuran, Vincenzo Alterio, Anna Di Fiore, Katia D’ Ambrosio, Fabrizio Carta, Simona Maria Monti & Giuseppina De Simone. (2018) Inhibition of carbonic anhydrase IX targets primary tumors, metastases, and cancer stem cells: Three for the price of one. Medicinal Research Reviews 38:6, pages 1799-1836.
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Srishti Singh, Carrie Lomelino, Mam Mboge, Susan Frost & Robert McKenna. (2018) Cancer Drug Development of Carbonic Anhydrase Inhibitors beyond the Active Site. Molecules 23:5, pages 1045.
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Ylenia Cau, Daniela Vullo, Mattia Mori, Elena Dreassi, Claudiu Supuran & Maurizio Botta. (2017) Potent and Selective Carboxylic Acid Inhibitors of Tumor-Associated Carbonic Anhydrases IX and XII. Molecules 23:1, pages 17.
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Wagdy M. Eldehna, Mahmoud F. Abo-Ashour, Alessio Nocentini, Paola Gratteri, Ibrahim H. Eissa, Mohamed Fares, Omnia E. Ismael, Hazem A. Ghabbour, Mahmoud M. Elaasser, Hatem A. Abdel-Aziz & Claudiu T. Supuran. (2017) Novel 4/3-((4-oxo-5-(2-oxoindolin-3-ylidene)thiazolidin-2-ylidene)amino) benzenesulfonamides: Synthesis, carbonic anhydrase inhibitory activity, anticancer activity and molecular modelling studies. European Journal of Medicinal Chemistry 139, pages 250-262.
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Giulia Bianco, Rita Meleddu, Simona Distinto, Filippo Cottiglia, Marco Gaspari, Claudia Melis, Angela Corona, Rossella Angius, Andrea Angeli, Domenico Taverna, Stefano Alcaro, Janis Leitans, Andris Kazaks, Kaspars Tars, Claudiu T. Supuran & Elias Maccioni. (2017)
N
-Acylbenzenesulfonamide Dihydro-1,3,4-oxadiazole Hybrids: Seeking Selectivity toward Carbonic Anhydrase Isoforms
. ACS Medicinal Chemistry Letters 8:8, pages 792-796.
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Jekaterīna Ivanova, Fabrizio Carta, Daniela Vullo, Janis Leitans, Andris Kazaks, Kaspars Tars, Raivis Žalubovskis & Claudiu T. Supuran. (2017) N -Substituted and ring opened saccharin derivatives selectively inhibit transmembrane, tumor-associated carbonic anhydrases IX and XII. Bioorganic & Medicinal Chemistry 25:13, pages 3583-3589.
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Feng-Ran Li, Zhan-Fang Fan, Su-Jiao Qi, Yan-Shi Wang, Jian Wang, Yang Liu & Mao-Sheng Cheng. (2017) Design, Synthesis, Molecular Docking Analysis, and Carbonic Anhydrase IX Inhibitory Evaluations of Novel N-Substituted-β-d-Glucosamine Derivatives that Incorporate Benzenesulfonamides. Molecules 22:5, pages 785.
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