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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 32, 2017 - Issue 1
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Research Paper

Inhibition of the α-carbonic anhydrase from Vibrio cholerae with amides and sulfonamides incorporating imidazole moieties

Daniela De VitaDipartimento di Chimica e Tecnologie del Farmaco, Istituto Pasteur-Fondazione Cenci Bolognetti, Università di Roma La Sapienza, Roma, Italy; ORCID Iconhttp://orcid.org/0000-0002-0370-4244View further author information
ORCID Icon,
Andrea AngeliDipartimento Neurofarba, Sezione di Scienze Farmaceutiche e Nutraceutiche, Università degli Studi di Firenze, Florence, Italy; View further author information
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Fabiana PandolfiDipartimento di Chimica e Tecnologie del Farmaco, Istituto Pasteur-Fondazione Cenci Bolognetti, Università di Roma La Sapienza, Roma, Italy; ORCID Iconhttp://orcid.org/0000-0002-5972-851XView further author information
ORCID Icon,
Martina BortolamiDipartimento di Chimica e Tecnologie del Farmaco, Istituto Pasteur-Fondazione Cenci Bolognetti, Università di Roma La Sapienza, Roma, Italy; View further author information
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Roberta CostiDipartimento di Chimica e Tecnologie del Farmaco, Istituto Pasteur-Fondazione Cenci Bolognetti, Università di Roma La Sapienza, Roma, Italy; ORCID Iconhttp://orcid.org/0000-0002-1314-9029View further author information
ORCID Icon,
Roberto Di SantoDipartimento di Chimica e Tecnologie del Farmaco, Istituto Pasteur-Fondazione Cenci Bolognetti, Università di Roma La Sapienza, Roma, Italy; ORCID Iconhttp://orcid.org/0000-0002-4279-7666View further author information
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Elisabetta SuffrediniDipartimento di Sicurezza Alimentare, Nutrizione e Sanità Pubblica Veterinaria, Istituto Superiore di Sanità, Rome, Italy; View further author information
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Mariangela CerusoPolo Scientifico, Laboratorio di Chimica Bioinorganica, Università degli Studi di Firenze, Florence, Italy; View further author information
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Sonia Del PreteDipartimento Neurofarba, Sezione di Scienze Farmaceutiche e Nutraceutiche, Università degli Studi di Firenze, Florence, Italy; ;Istituto di Bioscienze e Biorisorse, CNR, Napoli, ItalyView further author information
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Clemente CapassoIstituto di Bioscienze e Biorisorse, CNR, Napoli, ItalyView further author information
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Luigi ScipioneDipartimento di Chimica e Tecnologie del Farmaco, Istituto Pasteur-Fondazione Cenci Bolognetti, Università di Roma La Sapienza, Roma, Italy; Correspondence[email protected]
ORCID Iconhttp://orcid.org/0000-0002-2006-7005View further author information
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Claudiu T. SupuranDipartimento Neurofarba, Sezione di Scienze Farmaceutiche e Nutraceutiche, Università degli Studi di Firenze, Florence, Italy; ;Polo Scientifico, Laboratorio di Chimica Bioinorganica, Università degli Studi di Firenze, Florence, Italy; Correspondence[email protected]
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Pages 798-804 | Received 30 Mar 2017, Accepted 28 Apr 2017, Published online: 01 Jun 2017

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Marialuigia Fantacuzzi, Ilaria D’Agostino, Simone Carradori, Francesco Liguori, Fabrizio Carta, Mariangela Agamennone, Andrea Angeli, Filomena Sannio, Jean-Denis Docquier, Clemente Capasso & Claudiu T. Supuran. (2023) Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Emanuela Berrino & Claudiu T. Supuran. (2019) Novel approaches for designing drugs that interfere with pH regulation. Expert Opinion on Drug Discovery 14:3, pages 231-248.
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Simona Maria Monti, Angela Meccariello, Mariangela Ceruso, Krzysztof Szafrański, Jarosław Sławiński & Claudiu T. Supuran. (2018) Inhibition studies of Brucella suis β-carbonic anhydrases with a series of 4-substituted pyridine-3-sulphonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 255-259.
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Andrea Angeli, Sonia Del Prete, Sameh M. Osman, Fatmah A. S. Alasmary, Zeid AlOthman, William A. Donald, Clemente Capasso & Claudiu T. Supuran. (2018) Activation studies of the α- and β-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae with amines and amino acids. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 227-233.
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