Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 30, Issue 2 (2015)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 30, Issue 2 (2015)

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Original Article

Article
Synthesis and potent antistaphylococcal activity of some new 2-[4-(3,4-dimethoxyphenoxy)phenyl]-1,N-disubstituted-1H-benzimidazole-5-carboxamidines
M. Orhan Püsküllü, Sulhiye Yıldız, Yalçın Duydu, Aylin Üstündağ & Hakan Göker
Pages: 173-179
Published online: 25 Mar 2014
AbstractforSynthesis and potent antistaphylococcal activity of some new 2-[4-(3,4-dimethoxyphenoxy)phenyl]-1,N-disubstituted-1H-benzimidazole-5-carboxamidines | Full Text | References | PDF (201.1 KB)
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Research Article

Article
Biologically active carbazole derivatives: focus on oxazinocarbazoles and related compounds
Zouhair Bouaziz, Samar Issa, Jacques Gentili, Andreas Gratz, Andre Bollacke, Matthias Kassack, Joachim Jose, Lars Herfindal, Gro Gausdal, Stein Ove Døskeland, Catherine Mullié, Pascal Sonnet, Camille Desgrouas, Nicolas Taudon, Glaucio Valdameri, Attilio Di Pietro, Milad Baitiche & Marc Le Borgne
Pages: 180-188
Published online: 03 Apr 2014
AbstractforBiologically active carbazole derivatives: focus on oxazinocarbazoles and related compounds | Full Text | References | PDF (419.5 KB)
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Original Articles

Article
Design, synthesis, and antitumor screening of certain novel tetrahydroquinoline sulfonamides
Ahmed M. Alafeefy
Pages: 189-194
Published online: 25 Mar 2014
AbstractforDesign, synthesis, and antitumor screening of certain novel tetrahydroquinoline sulfonamides | Full Text | References | PDF (191.6 KB)
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Research Article

Article
Synthesis and characterization of complexes of a novel proton transfer salt and their inhibition studies on carbonic anhydrase isoenzymes
Halil İlkimen, Cengiz Yenikaya, Musa Sarı, Metin Bülbül, Ekrem Tunca, Hakan Dal & Metin Baş
Pages: 195-203
Published online: 23 Apr 2014
AbstractforSynthesis and characterization of complexes of a novel proton transfer salt and their inhibition studies on carbonic anhydrase isoenzymes | Full Text | References | PDF (1.4 MB) | Supplemental
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Original Articles

Article
Intrinsic thermodynamics of sulfonamide inhibitor binding to human carbonic anhydrases I and II
Vaida Morkūnaitė, Joana Gylytė, Asta Zubrienė, Lina Baranauskienė, Miglė Kišonaitė, Vilma Michailovienė, Vaida Juozapaitienė, Matthew J. Todd & Daumantas Matulis
Pages: 204-211
Published online: 23 Apr 2014
AbstractforIntrinsic thermodynamics of sulfonamide inhibitor binding to human carbonic anhydrases I and II | Full Text | References | PDF (369.8 KB)
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Original Article

Article
Catalase, carbonic anhydrase and xanthine oxidase activities in patients with mycosis fungoides
Fatma Pelin Cengiz, Serap Beyaztas, Basak Gokce, Oktay Arslan & Ozen Ozensoy Guler
Pages: 212-215
Published online: 25 Apr 2014
AbstractforCatalase, carbonic anhydrase and xanthine oxidase activities in patients with mycosis fungoides | Full Text | References | PDF (183.8 KB) | Supplemental
  • 751 Views
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Research Article

Article
5-Membered cyclic hydroxamic acids as HDAC inhibitors
Ilze Mutule, Diana Borovika, Elina Rozenberga, Nadezhda Romanchikova, Raivis Zalubovskis, Irina Shestakova & Peteris Trapencieris
Pages: 216-223
Published online: 18 Jun 2014
Abstractfor5-Membered cyclic hydroxamic acids as HDAC inhibitors | Full Text | References | PDF (658.3 KB)
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Original Article

Article
A new affinity gel for the purification of α-carbonic anhdrases
Aysegul Sahin, Semra Isık, Oktay Arslan, Claudiu T. Supuran & Ozen Ozensoy Guler
Pages: 224-228
Published online: 17 Jun 2014
AbstractforA new affinity gel for the purification of α-carbonic anhdrases | Full Text | References | PDF (276.4 KB)
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Article
Implication of novel thiazolo-thiophene derivative (MCD-KV-10) for management of asthma
Dhiraj Patil, Ranjeet Prasad Dash, Sandeep Kumar Thakur, Amit N. Pandya, P. Venkatesh, Kamala K. Vasu & Manish Nivsarkar
Pages: 229-239
Published online: 18 Jun 2014
AbstractforImplication of novel thiazolo-thiophene derivative (MCD-KV-10) for management of asthma | Full Text | References | PDF (1.6 MB) | Supplemental
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Research Article

Article
Synthesis of a novel affinity gel for the purification of carbonic anhydrases
Murat Bozdag, Semra Isik, Serap Beyaztas, Oktay Arslan & Claudiu T. Supuran
Pages: 240-244
Published online: 18 Jun 2014
AbstractforSynthesis of a novel affinity gel for the purification of carbonic anhydrases | Full Text | References | PDF (458.5 KB)
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Article
Antidepressant and antipsychotic drugs differentially affect PON1 enzyme activity
Ayla Solmaz Avcikurt, Selma Sinan & Feray Kockar
Pages: 245-249
Published online: 17 Jun 2014
AbstractforAntidepressant and antipsychotic drugs differentially affect PON1 enzyme activity | Full Text | References | PDF (505.4 KB)
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Original Article

Article
Prophylactic and curative anti-ulcerative colitis activity and the possible mechanisms of action of some desert plants
Reham M. El-Meligy, Amani S. Awaad, Gamal A. Soliman, Abir B. Bacha, Ahmed M. Alafeefy & Sanaa A. Kenawy
Pages: 250-258
Published online: 09 May 2014
AbstractforProphylactic and curative anti-ulcerative colitis activity and the possible mechanisms of action of some desert plants | Full Text | References | PDF (799.2 KB)
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Article
3-Benzylidene-4-chromanones: a novel cluster of anti-tubercular agents
Umashankar Das, Tamas Lorand, Stephen G. Dimmock, Pal Perjesi & Jonathan R. Dimmock
Pages: 259-263
Published online: 18 Jun 2014
Abstractfor3-Benzylidene-4-chromanones: a novel cluster of anti-tubercular agents | Full Text | References | PDF (282.8 KB)
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Research Article

Article
Pistachio (Pistacia vera L.) Gum: a potent inhibitor of reactive oxygen species
M. Hilal Sehitoglu, Hatice Han, Pınar Kalin, İlhami Gülçin, Ali Ozkan & Hassan Y. Aboul-Enein
Pages: 264-269
Published online: 18 Jun 2014
AbstractforPistachio (Pistacia vera L.) Gum: a potent inhibitor of reactive oxygen species | Full Text | References | PDF (267.4 KB)
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Article
Synthesis and biological evaluation of certain 3-substituted benzylideneamino-2-(4-nitrophenyl)quinazolin-4(3H)-one derivatives
Ahmed M. Alafeefy, Amani S. Awaad, Hatem A. Abdel-Aziz, Reham M. El-Meligy, Mohamed E. Zain, Mounerah R. Al-Outhman & Abir B. Bacha
Pages: 270-276
Published online: 18 Jun 2014
AbstractforSynthesis and biological evaluation of certain 3-substituted benzylideneamino-2-(4-nitrophenyl)quinazolin-4(3H)-one derivatives | Full Text | References | PDF (361.9 KB)
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Original Article

Article
Protonography, a new technique for the analysis of carbonic anhydrase activity
Viviana De Luca, Sonia Del Prete, Claudiu T. Supuran & Clemente Capasso
Pages: 277-282
Published online: 09 Jul 2014
AbstractforProtonography, a new technique for the analysis of carbonic anhydrase activity | Full Text | References | PDF (737.8 KB)
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Research Article

Article
Pattern recognition of HER-1 in biological fluids using stochastic sensing
Raluca-Ioana Stefan-van Staden, Iuliana Moldoveanu & Camelia Stanciu Gavan
Pages: 283-285
Published online: 25 Jun 2014
AbstractforPattern recognition of HER-1 in biological fluids using stochastic sensing | Full Text | References | PDF (179 KB)
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Original Articles

Article
Differential in vitro inhibition studies of some cerium vanadate derivatives on xanthine oxidase
Mustafa Oğuzhan Kaya, Yeşim Kaya, Gülşah Çelik, Figen Kurtuluş, Oktay Arslan & Özen Özensoy Güler
Pages: 286-289
Published online: 25 Jun 2014
AbstractforDifferential in vitro inhibition studies of some cerium vanadate derivatives on xanthine oxidase | Full Text | References | PDF (371.9 KB)
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Original Article

Article
Synthesis and biological evaluation of new pyrimidine-4-yl-ethanol derivatives as ROS1 kinase inhibitors
Ahmed Z. Abdelazem & So Ha Lee
Pages: 290-298
Published online: 18 Jun 2014
AbstractforSynthesis and biological evaluation of new pyrimidine-4-yl-ethanol derivatives as ROS1 kinase inhibitors | Full Text | References | PDF (702.5 KB)
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Article
Synthetic compounds from an in house library as inhibitors of falcipain-2 from Plasmodium falciparum
Jean Borges Bertoldo, Louise Domeneghini Chiaradia-Delatorre, Alessandra Mascarello, Paulo César Leal, Marlon Norberto Sechini Cordeiro, Ricardo José Nunes, Emir Salas Sarduy, Philip Jon Rosenthal & Hernán Terenzi
Pages: 299-307
Published online: 25 Jun 2014
AbstractforSynthetic compounds from an in house library as inhibitors of falcipain-2 from Plasmodium falciparum | Full Text | References | PDF (1.9 MB) | Supplemental
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Original Articles

Article
Synthesis and antitumor activity of tetrahydrocarbazole hybridized with dithioate derivatives
Hala Bakr El-Nassan
Pages: 308-315
Published online: 05 Jun 2014
AbstractforSynthesis and antitumor activity of tetrahydrocarbazole hybridized with dithioate derivatives | Full Text | References | PDF (883.3 KB)
  • 2632 Views
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Research Article

Article
Carbonic anhydrase and acetylcholinesterase inhibitory effects of carbamates and sulfamoylcarbamates
Hülya Göçer, Akın Akincioğlu, Süleyman Göksu, İlhami Gülçin & Claudiu T. Supuran
Pages: 316-320
Published online: 25 Jun 2014
AbstractforCarbonic anhydrase and acetylcholinesterase inhibitory effects of carbamates and sulfamoylcarbamates | Full Text | References | PDF (202.8 KB)
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Review Article

Recent advances in the discovery of zinc-binding motifs for the development of carbonic anhydrase inhibitors
Jean-Yves Winum & Claudiu T. Supuran
Pages: 321-324
Published online: 18 Jun 2014
AbstractforRecent advances in the discovery of zinc-binding motifs for the development of carbonic anhydrase inhibitors | Full Text | References | PDF (605.6 KB)
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An overview of the alpha-, beta- and gamma-carbonic anhydrases from Bacteria: can bacterial carbonic anhydrases shed new light on evolution of bacteria?
Clemente Capasso & Claudiu T. Supuran
Pages: 325-332
Published online: 25 Apr 2014
AbstractforAn overview of the alpha-, beta- and gamma-carbonic anhydrases from Bacteria: can bacterial carbonic anhydrases shed new light on evolution of bacteria? | Full Text | References | PDF (1 MB)
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Short Communication

Further in vitro biological activity evaluation of amino-, thio- and ester-derivatives of avarol
Giuseppina Tommonaro, Boris Pejin, Carmine Iodice, Antonietta Tafuto & Salvatore De Rosa
Pages: 333-335
Published online: 18 Jun 2014
AbstractforFurther in vitro biological activity evaluation of amino-, thio- and ester-derivatives of avarol | Full Text | References | PDF (158.6 KB)
  • 679 Views
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Inhibition of human pyridoxal kinase by 2-acetyl-4-((1R,2S,3R)-1,2,3,4-tetrahydroxybutyl)imidazole (THI)
Paul W. Elsinghorst, Martino L. di Salvo, Alessia Parroni & Roberto Contestabile
Pages: 336-340
Published online: 05 Jun 2014
AbstractforInhibition of human pyridoxal kinase by 2-acetyl-4-((1R,2S,3R)-1,2,3,4-tetrahydroxybutyl)imidazole (THI) | Full Text | References | PDF (353.6 KB)
  • 1018 Views
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Dipotassium-trioxohydroxytetrafluorotriborate, K2[B3O3F4OH], is a potent inhibitor of human carbonic anhydrases
Daniela Vullo, Mladen Milos, Borivoj Galic, Andrea Scozzafava & Claudiu T. Supuran
Pages: 341-344
Published online: 18 Jun 2014
AbstractforDipotassium-trioxohydroxytetrafluorotriborate, K2[B3O3F4OH], is a potent inhibitor of human carbonic anhydrases | Full Text | References | PDF (155.7 KB)
  • 727 Views
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