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Simone Giovannuzzi, Viviana De Luca, Alessio Nocentini, Clemente Capasso & Claudiu T. Supuran. (2022) Coumarins inhibit η-class carbonic anhydrase from Plasmodium falciparum. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 680-685.
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Claudiu T. Supuran & Clemente Capasso. (2020) Antibacterial carbonic anhydrase inhibitors: an update on the recent literature. Expert Opinion on Therapeutic Patents 30:12, pages 963-982.
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Mikhail Krasavin, Raivis Žalubovskis, Aiga Grandāne, Ilona Domračeva, Petr Zhmurov & Claudiu T. Supuran. (2020) Sulfocoumarins as dual inhibitors of human carbonic anhydrase isoforms IX/XII and of human thioredoxin reductase. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 506-510.
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Ashok Aspatwar, Milka Hammaren, Mataleena Parikka, Seppo Parkkila, Fabrizio Carta, Murat Bozdag, Daniela Vullo & Claudiu T. Supuran. (2020) In vitro inhibition of Mycobacterium tuberculosis β-carbonic anhydrase 3 with Mono- and dithiocarbamates and evaluation of their toxicity using zebrafish developing embryos. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 65-71.
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Benoit Métayer, Andrea Angeli, Agnès Mingot, Kévin Jouvin, Gwilherm Evano, Claudiu T. Supuran & Sébastien Thibaudeau. (2018) Fluoroenesulphonamides: N-sulphonylurea isosteres showing nanomolar selective cancer-related transmembrane human carbonic anhydrase inhibition. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 804-808.
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Claudiu T. Supuran. (2018) Carbon- versus sulphur-based zinc binding groups for carbonic anhydrase inhibitors?. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 485-495.
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Daniela Vullo, Leo Syrjänen, Marianne Kuuslahti, Seppo Parkkila & Claudiu T. Supuran. (2018) Anion inhibition studies of a beta carbonic anhydrase from the malaria mosquito Anopheles gambiae. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 359-363.
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Alessio Nocentini, Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Fatmah A.S. Alasmary, Zeid AlOthman, Clemente Capasso, Fabrizio Carta, Paola Gratteri & Claudiu T. Supuran. (2017) Inhibition of the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa with monothiocarbamates. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1064-1070.
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Mikhail Krasavin, Mikhail Korsakov, Oksana Ronzhina, Tiziano Tuccinardi, Stanislav Kalinin, Muhammet Tanç & Claudiu T. Supuran. (2017) Primary mono- and bis-sulfonamides obtained via regiospecific sulfochlorination of N-arylpyrazoles: inhibition profile against a panel of human carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 920-934.
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Ashok Aspatwar, Milka Hammarén, Sanni Koskinen, Bruno Luukinen, Harlan Barker, Fabrizio Carta, Claudiu T. Supuran, Mataleena Parikka & Seppo Parkkila. (2017) β-CA-specific inhibitor dithiocarbamate Fc14–584B: a novel antimycobacterial agent with potential to treat drug-resistant tuberculosis. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 832-840.
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Erol Licsandru, Muhammet Tanc, Istvan Kocsis, Mihail Barboiu & Claudiu T. Supuran. (2017) A class of carbonic anhydrase I – selective activators. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 37-46.
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Alessio Nocentini, Mariangela Ceruso, Fabrizio Carta & Claudiu T. Supuran. (2016) 7-Aryl-triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrase IX and XII. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1226-1233.
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Ayşenur Eminoğlu, Daniela Vullo, Aycan Aşık, Dilşat Nigar Çolak, Claudiu T. Supuran, Sabriye Çanakçı & Ali Osman Beldüz. (2016) Cloning, expression and biochemical characterization of a β-carbonic anhydrase from the soil bacterium Enterobacter sp. B13. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1111-1118.
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Claudiu T. Supuran, Stanislav Kalinin, Muhammet Tanç, Pakornwit Sarnpitak, Prashant Mujumdar, Sally-Ann Poulsen & Mikhail Krasavin. (2016) Isoform-selective inhibitory profile of 2-imidazoline-substituted benzene sulfonamides against a panel of human carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 31:sup1, pages 197-202.
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Claudiu T. Supuran. (2016) CA IX stratification based on cancer treatment: a patent evaluation of US2016/0002350. Expert Opinion on Therapeutic Patents 26:10, pages 1105-1109.
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Claudiu T. Supuran. (2016) How many carbonic anhydrase inhibition mechanisms exist?. Journal of Enzyme Inhibition and Medicinal Chemistry 31:3, pages 345-360.
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Claudiu T. Supuran. (2016) Drug interaction considerations in the therapeutic use of carbonic anhydrase inhibitors. Expert Opinion on Drug Metabolism & Toxicology 12:4, pages 423-431.
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Murat Bozdag, Fabrizio Carta, Daniela Vullo, Semra Isik, Zeid AlOthman, Sameh M. Osman, Andrea Scozzafava & Claudiu T. Supuran. (2016) Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase. Journal of Enzyme Inhibition and Medicinal Chemistry 31:1, pages 132-136.
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Clemente Capasso & Claudiu T Supuran. (2015) Bacterial, fungal and protozoan carbonic anhydrases as drug targets. Expert Opinion on Therapeutic Targets 19:12, pages 1689-1704.
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Leonardo E. Riafrecha, Daniela Vullo, Safia Ouahrani-Bettache, Stephan Köhler, Pascal Dumy, Jean-Yves Winum, Claudiu T. Supuran & Pedro A. Colinas. (2015) Inhibition of β-carbonic anhydrases from Brucella suis with C-cinnamoyl glycosides incorporating the phenol moiety. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 1017-1020.
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Joanna Ombouma, Daniela Vullo, Stephan Köhler, Pascal Dumy, Claudiu T. Supuran & Jean-Yves Winum. (2015) N-glycosyl-N-hydroxysulfamides as potent inhibitors of Brucella suis carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 1010-1012.
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Mehmet Arslan, Murat Şentürk, İsmail Fidan, Oktay Talaz, Deniz Ekinci, Sedat Coşgun & Claudiu T. Supuran. (2015) Synthesis of 3,4-dihydroxypyrrolidine-2,5-dione and 3,5-dihydroxybenzoic acid derivatives and evaluation of the carbonic anhydrase I and II inhibition. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 896-900.
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Daniela Vullo, Semra Isik, Murat Bozdag, Fabrizio Carta & Claudiu T. Supuran. (2015) 7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring. Journal of Enzyme Inhibition and Medicinal Chemistry 30:5, pages 773-777.
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Leonardo E. Riafrecha, Daniela Vullo, Claudiu T. Supuran & Pedro A. Colinas. (2015) C-glycosides incorporating the 6-methoxy-2-naphthyl moiety are selective inhibitors of fungal and bacterial carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 30:5, pages 857-861.
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Erik O. Pettersen, Peter Ebbesen, Roben G. Gieling, Kaye J. Williams, Ludwig Dubois, Philippe Lambin, Carol Ward, James Meehan, Ian H. Kunkler, Simon P. Langdon, Anne H. Ree, Kjersti Flatmark, Heidi Lyng, Maria J. Calzada, Luis del Peso, Manuel O. Landazuri, Agnes Görlach, Hubert Flamm, Jochen Kieninger, Gerald Urban, Andreas Weltin, Dean C. Singleton, Syed Haider, Francesca M. Buffa, Adrian L. Harris, Andrea Scozzafava, Claudiu T. Supuran, Isabella Moser, Gerhard Jobst, Morten Busk, Kasper Toustrup, Jens Overgaard, Jan Alsner, Jacques Pouyssegur, Johanna Chiche, Nathalie Mazure, Ibtissam Marchiq, Scott Parks, Afshan Ahmed, Margaret Ashcroft, Silvia Pastorekova, Yihai Cao, Kasper M. Rouschop, Brad G. Wouters, Marianne Koritzinsky, Hilda Mujcic & Dan Cojocari. (2015) Targeting tumour hypoxia to prevent cancer metastasis. From biology, biosensing and technology to drug development: the METOXIA consortium. Journal of Enzyme Inhibition and Medicinal Chemistry 30:5, pages 689-721.
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Claudiu T Supuran. (2015) Acetazolamide for the treatment of idiopathic intracranial hypertension. Expert Review of Neurotherapeutics 15:8, pages 851-856.
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Claudiu T Supuran. (2015) Nanoparticles for controlled release of anti-biofilm agents WO2014130994 (A1): a patent evaluation. Expert Opinion on Therapeutic Patents 25:8, pages 945-948.
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Ondrej Holas, Pavel Ondrejcek & Martin Dolezal. (2015) Mycobacterium tuberculosis enoyl-acyl carrier protein reductase inhibitors as potential antituberculotics: development in the past decade. Journal of Enzyme Inhibition and Medicinal Chemistry 30:4, pages 629-648.
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Ahmed M. Alafeefy, Mariangela Ceruso, Abdul-Malek S. Al-Tamimi, Sonia Del Prete, Claudiu T. Supuran & Clemente Capasso. (2015) Inhibition studies of quinazoline-sulfonamide derivatives against the γ-CA (PgiCA) from the pathogenic bacterium, Porphyromonas gingivalis. Journal of Enzyme Inhibition and Medicinal Chemistry 30:4, pages 592-596.
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Claudia Palmer & Claudiu T Supuran. (2015) A Key Opinion Leader interview: insight into the research and career of Prof. Claudiu T Supuran. Expert Opinion on Therapeutic Patents 25:4, pages 501-505.
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Daniela Vullo, Mladen Milos, Borivoj Galic, Andrea Scozzafava & Claudiu T. Supuran. (2015) Dipotassium-trioxohydroxytetrafluorotriborate, K2[B3O3F4OH], is a potent inhibitor of human carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 30:2, pages 341-344.
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Jean-Yves Winum & Claudiu T. Supuran. (2015) Recent advances in the discovery of zinc-binding motifs for the development of carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 30:2, pages 321-324.
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Giuseppina De Simone, Vincenzo Alterio & Claudiu T Supuran. (2013) Exploiting the hydrophobic and hydrophilic binding sites for designing carbonic anhydrase inhibitors. Expert Opinion on Drug Discovery 8:7, pages 793-810.
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Emanuela Masini, Fabrizio Carta, Andrea Scozzafava & Claudiu T Supuran. (2013) Antiglaucoma carbonic anhydrase inhibitors: a patent review. Expert Opinion on Therapeutic Patents 23:6, pages 705-716.
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Articles from other publishers (86)
Ojaswitha Ommi, Niccolò Paoletti, Alessandro Bonardi, Paola Gratteri, Harshada Anil Bhalerao, Shashikanta Sau, Srinivas Nanduri, Arifuddin Mohammed, Nitin Pal Kalia, Rajesh Sonti, Claudiu T. Supuran & Venkata Madhavi Yaddanapudi. (2023) Exploration of 3‐aryl pyrazole‐tethered sulfamoyl carboxamides as carbonic anhydrase inhibitors. Archiv der Pharmazie 356:11.
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Jenna Lanz, Nicholas Biniaz-Harris, Mara Kuvaldina, Samta Jain, Kim Lewis & Brian A. Fallon. (2023) Disulfiram: Mechanisms, Applications, and Challenges. Antibiotics 12:3, pages 524.
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Derya Osmaniye, Cüneyt Türkeş, Yeliz Demir, Yusuf Özkay, Şükrü Beydemir & Zafer A. Kaplancıklı. (2022) Design, synthesis, and biological activity of novel dithiocarbamate‐methylsulfonyl hybrids as carbonic anhydrase inhibitors. Archiv der Pharmazie 355:8.
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Kuo-Ting Chen & Yann Seimbille. (2022) New Developments in Carbonic Anhydrase IX-Targeted Fluorescence and Nuclear Imaging Agents. International Journal of Molecular Sciences 23:11, pages 6125.
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Timothy O. Ajiboye, Titilope T. Ajiboye, Riadh Marzouki & Damian C. Onwudiwe. (2022) The Versatility in the Applications of Dithiocarbamates. International Journal of Molecular Sciences 23:3, pages 1317.
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Eva Havránková, Vladimír Garaj, Šárka Mascaretti, Andrea Angeli, Zuzana Soldánová, Miroslav Kemka, Jozef Motyčka, Marie Brázdová, Jozef Csöllei, Josef Jampílek & Claudiu T. Supuran. (2021) Novel 1,3,5-Triazinyl Aminobenzenesulfonamides Incorporating Aminoalcohol, Aminochalcone and Aminostilbene Structural Motifs as Potent Anti-VRE Agents, and Carbonic Anhydrases I, II, VII, IX, and XII Inhibitors. International Journal of Molecular Sciences 23:1, pages 231.
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Chien Ing Yeo, Edward R. T. Tiekink & Jactty Chew. (2021) Insights into the Antimicrobial Potential of Dithiocarbamate Anions and Metal-Based Species. Inorganics 9:6, pages 48.
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Claudiu T. Supuran & Clemente Capasso. (2021) A Highlight on the Inhibition of Fungal Carbonic Anhydrases as Drug Targets for the Antifungal Armamentarium. International Journal of Molecular Sciences 22:9, pages 4324.
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Cristina Campestre, Viviana De Luca, Simone Carradori, Rossella Grande, Vincenzo Carginale, Andrea Scaloni, Claudiu T. Supuran & Clemente Capasso. (2021) Carbonic Anhydrases: New Perspectives on Protein Functional Role and Inhibition in Helicobacter pylori. Frontiers in Microbiology 12.
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D. C. Onwudiwe, J. O. Adeyemi, R. T. Papane, F. F. Bobinihi & E. Hosten. (2021) SPECTROSCOPIC AND STRUCTURAL CHARACTERIZATION OF Zn(II) BIS(N-ETHYL-N-ETHANOL DITHIOCARBAMATE) AND ITS ADDUCTS WITH N-DONOR LIGANDS. Journal of Structural Chemistry 62:3, pages 412-421.
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Laurine Kaul, Regine Süss, Andrew Zannettino & Katharina Richter. (2021) The revival of dithiocarbamates: from pesticides to innovative medical treatments. iScience 24:2, pages 102092.
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Sangita Dattatray Shinde, Akash P. Sakla & Nagula Shankaraiah. (2020) An insight into medicinal attributes of dithiocarbamates: Bird’s eye view. Bioorganic Chemistry 105, pages 104346.
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Sonia Del Prete, Viviana De Luca, Alessio Nocentini, Andrea Scaloni, Margaret D. Mastrolorenzo, Claudiu T. Supuran & Clemente Capasso. (2020) Anion Inhibition Studies of the Beta-Carbonic Anhydrase from Escherichia coli. Molecules 25:11, pages 2564.
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Hamid Beyzaei, Sedigheh Esmaeilzadeh Bahabadi, Shahla Najafi & Fahime Heidari Sadegh. (2020) Synthesis and Antimicrobial Evaluation of the Potassium Salts of Benzhydrazine Dithiocarbamates. Avicenna Journal of Clinical Microbiology and Infection 7:1, pages 15-21.
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Stanislav Kalinin, Alessio Nocentini, Alexander Kovalenko, Vladimir Sharoyko, Alessandro Bonardi, Andrea Angeli, Paola Gratteri, Tatiana B. Tennikova, Claudiu T. Supuran & Mikhail Krasavin. (2019) From random to rational: A discovery approach to selective subnanomolar inhibitors of human carbonic anhydrase IV based on the Castagnoli-Cushman multicomponent reaction. European Journal of Medicinal Chemistry 182, pages 111642.
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Stanislav Kalinin, Annika Valtari, Marika Ruponen, Elisa Toropainen, Alexander Kovalenko, Alessio Nocentini, Maxim Gureev, Dmitry Dar'in, Arto Urtti, Claudiu T. Supuran & Mikhail Krasavin. (2019) Highly hydrophilic 1,3-oxazol-5-yl benzenesulfonamide inhibitors of carbonic anhydrase II for reduction of glaucoma-related intraocular pressure. Bioorganic & Medicinal Chemistry 27:21, pages 115086.
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Aspatwar, Kairys, Rala, Parikka, Bozdag, Carta, Supuran & Parkkila. (2019) Mycobacterium tuberculosis β-Carbonic Anhydrases: Novel Targets for Developing Antituberculosis Drugs. International Journal of Molecular Sciences 20:20, pages 5153.
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Mikhail Krasavin, Anton Shetnev, Sergey Baykov, Stanislav Kalinin, Alessio Nocentini, Vladimir Sharoyko, Giulio Poli, Tiziano Tuccinardi, Mikhail Korsakov, Tatiana B. Tennikova & Claudiu T. Supuran. (2019) Pyridazinone-substituted benzenesulfonamides display potent inhibition of membrane-bound human carbonic anhydrase IX and promising antiproliferative activity against cancer cell lines. European Journal of Medicinal Chemistry 168, pages 301-314.
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Mikhail Krasavin, Anton Shetnev, Tatyana Sharonova, Sergey Baykov, Stanislav Kalinin, Alessio Nocentini, Vladimir Sharoyko, Giulio Poli, Tiziano Tuccinardi, Sofia Presnukhina, Tatiana B. Tennikova & Claudiu T. Supuran. (2019) Continued exploration of 1,2,4-oxadiazole periphery for carbonic anhydrase-targeting primary arene sulfonamides: Discovery of subnanomolar inhibitors of membrane-bound hCA IX isoform that selectively kill cancer cells in hypoxic environment. European Journal of Medicinal Chemistry 164, pages 92-105.
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Claudiu T. Supuran. 2019. Therapeutic Application of Nitric Oxide in Cancer and Inflammatory Disorders. Therapeutic Application of Nitric Oxide in Cancer and Inflammatory Disorders
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Claudiu T. Supuran & Clemente Capasso. 2019. Carbonic Anhydrases. Carbonic Anhydrases
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417
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Clemente Capasso. 2019. Carbonic Anhydrases. Carbonic Anhydrases
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Peter Mikuš, Dominika Krajčiová, Mária Mikulová, Branislav Horváth, Daniel Pecher, Vladimír Garaj, Silvia Bua, Andrea Angeli & Claudiu T. Supuran. (2018) Novel sulfonamides incorporating 1,3,5-triazine and amino acid structural motifs as inhibitors of the physiological carbonic anhydrase isozymes I, II and IV and tumor-associated isozyme IX. Bioorganic Chemistry 81, pages 241-252.
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Ashok Aspatwar, Jean-Yves Winum, Fabrizio Carta, Claudiu Supuran, Milka Hammaren, Mataleena Parikka & Seppo Parkkila. (2018) Carbonic Anhydrase Inhibitors as Novel Drugs against Mycobacterial β-Carbonic Anhydrases: An Update on In Vitro and In Vivo Studies. Molecules 23:11, pages 2911.
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Carrie L. Lomelino, Jacob T. Andring & Robert McKenna. (2018) Crystallography and Its Impact on Carbonic Anhydrase Research. International Journal of Medicinal Chemistry 2018, pages 1-21.
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Misaki Nakai, Jihne Pan, Kuo-Shyan Lin, John R. Thompson, Alessio Nocentini, Claudiu T. Supuran, Yasuo Nakabayashi & Tim Storr. (2018) Evaluation of 99mTc-sulfonamide and sulfocoumarin derivatives for imaging carbonic anhydrase IX expression. Journal of Inorganic Biochemistry 185, pages 63-70.
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Nabih Lolak, Suleyman Akocak, Silvia Bua, Murat Koca & Claudiu T. Supuran. (2018) Design and synthesis of novel 1,3-diaryltriazene-substituted sulfonamides as potent and selective carbonic anhydrase II inhibitors. Bioorganic Chemistry 77, pages 542-547.
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Eva Havránková, Jozef Csöllei, Daniela Vullo, Vladimír Garaj, Pavel Pazdera & Claudiu T. Supuran. (2018) Novel sulfonamide incorporating piperazine, aminoalcohol and 1,3,5-triazine structural motifs with carbonic anhydrase I, II and IX inhibitory action. Bioorganic Chemistry 77, pages 25-37.
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Alexander Sapegin, Stanislav Kalinin, Andrea Angeli, Claudiu T. Supuran & Mikhail Krasavin. (2018) Unprotected primary sulfonamide group facilitates ring-forming cascade en route to polycyclic [1,4]oxazepine-based carbonic anhydrase inhibitors. Bioorganic Chemistry 76, pages 140-146.
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Mikhail Krasavin, Anton Shetnev, Tatyana Sharonova, Sergey Baykov, Tiziano Tuccinardi, Stanislav Kalinin, Andrea Angeli & Claudiu T. Supuran. (2018) Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1,2,4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic hCA II and membrane-bound hCA IX isoforms. Bioorganic Chemistry 76, pages 88-97.
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Srinivas Angapelly, P. V. Sri Ramya, Andrea Angeli, Claudiu T. Supuran & Mohammed Arifuddin. (2017) Sulfocoumarin-, Coumarin-, 4-Sulfamoylphenyl-Bearing Indazole-3-carboxamide Hybrids: Synthesis and Selective Inhibition of Tumor-Associated Carbonic Anhydrase Isozymes IX and XII. ChemMedChem 12:19, pages 1578-1584.
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Mikhail Krasavin, Mikhail Korsakov, Zhanna Zvonaryova, Evgenii Semyonychev, Tiziano Tuccinardi, Stanislav Kalinin, Muhammet Tanç & Claudiu T. Supuran. (2017) Human carbonic anhydrase inhibitory profile of mono- and bis-sulfonamides synthesized via a direct sulfochlorination of 3- and 4-(hetero)arylisoxazol-5-amine scaffolds. Bioorganic & Medicinal Chemistry 25:6, pages 1914-1925.
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Daniela Vullo, Sonia Del Prete, Alessio Nocentini, Sameh M. Osman, Zeid AlOthman, Clemente Capasso, Murat Bozdag, Fabrizio Carta, Paola Gratteri & Claudiu T. Supuran. (2017) Dithiocarbamates effectively inhibit the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa. Bioorganic & Medicinal Chemistry 25:3, pages 1260-1265.
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Dhiman Sankar Pal, Mazharul Abbasi, Dipon Kumar Mondal, Binitha Anu Varghese, Ritama Paul, Shalini Singh & Rupak Datta. (2017)
Interplay between a cytosolic and a cell surface carbonic anhydrase in pH homeostasis and acid tolerance of
Leishmania
. Journal of Cell Science.
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Alex G. Dalecki, Cameron L. Crawford & Frank Wolschendorf. 2017. Microbiology of Metal Ions. Microbiology of Metal Ions
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260
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Behnam Rasti, Mohammad H. Karimi-Jafari & Jahan B. Ghasemi. (2016) Quantitative Characterization of the Interaction Space of the Mammalian Carbonic Anhydrase Isoforms I, II, VII, IX, XII, and XIV and their Inhibitors, Using the Proteochemometric Approach. Chemical Biology & Drug Design 88:3, pages 341-353.
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Claudiu T. Supuran. (2016) Structure and function of carbonic anhydrases. Biochemical Journal 473:14, pages 2023-2032.
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Vito Coviello, Beatrice Marchi, Stefania Sartini, Luca Quattrini, Anna Maria Marini, Francesca Simorini, Sabrina Taliani, Silvia Salerno, Paola Orlandi, Anna Fioravanti, Teresa Di Desidero, Daniela Vullo, Federico Da Settimo, Claudiu T. Supuran, Guido Bocci & Concettina La Motta. (2016) 1,2-Benzisothiazole Derivatives Bearing 4-, 5-, or 6-Alkyl/arylcarboxamide Moieties Inhibit Carbonic Anhydrase Isoform IX (CAIX) and Cell Proliferation under Hypoxic Conditions. Journal of Medicinal Chemistry 59:13, pages 6547-6552.
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Claudiu T Supuran. (2016)
Inhibition of carbonic anhydrase from
Trypanosoma cruzi
for the management of Chagas disease: an underexplored therapeutic opportunity
. Future Medicinal Chemistry 8:3, pages 311-324.
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Ahmed M. Alafeefy, Fabrizio Carta, Mariangela Ceruso, Abdul-Malek S. Al-Tamimi, Abdulla A. Al-Kahtani & Claudiu T. Supuran. (2016) Development of 3-(4-aminosulphonyl)-phenyl-2-mercapto-3H-quinazolin-4-ones as inhibitors of carbonic anhydrase isoforms involved in tumorigenesis and glaucoma. Bioorganic & Medicinal Chemistry 24:6, pages 1402-1407.
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Mustafa Durgun, Hasan Turkmen, Mariangela Ceruso & Claudiu T. Supuran. (2016) Synthesis of 4-sulfamoylphenyl-benzylamine derivatives with inhibitory activity against human carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry 24:5, pages 982-988.
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Elisabetta Barresi, Silvia Salerno, Anna Maria Marini, Sabrina Taliani, Concettina La Motta, Francesca Simorini, Federico Da Settimo, Daniela Vullo & Claudiu T. Supuran. (2016) Sulfonamides incorporating heteropolycyclic scaffolds show potent inhibitory action against carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry 24:4, pages 921-927.
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Maria Luisa Villalba, Pablo Palestro, Mariangela Ceruso, Jose L. Gonzalez Funes, Alan Talevi, Luis Bruno Blanch, Claudiu T. Supuran & Luciana Gavernet. (2016) Sulfamide derivatives with selective carbonic anhydrase VII inhibitory action. Bioorganic & Medicinal Chemistry 24:4, pages 894-901.
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Daniela Vullo, Avni Bhatt, Brian P. Mahon, Robert McKenna & Claudiu T. Supuran. (2016) Sulfonamide inhibition studies of the α-carbonic anhydrase from the gammaproteobacterium Thiomicrospira crunogena XCL-2, TcruCA. Bioorganic & Medicinal Chemistry Letters 26:2, pages 401-405.
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Adel S. El-Azab, Alaa A.-M. Abdel-Aziz, Rezk R. Ayyad, Mariangela Ceruso & Claudiu T. Supuran. (2016) Inhibition of carbonic anhydrase isoforms I, II, IV, VII and XII with carboxylates and sulfonamides incorporating phthalimide/phthalic anhydride scaffolds. Bioorganic & Medicinal Chemistry 24:1, pages 20-25.
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Claudiu T. Supuran & Clemente Capasso. 2017. Zinc Enzyme Inhibitors. Zinc Enzyme Inhibitors
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133
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Marta Ferraroni, Sonia Del Prete, Daniela Vullo, Clemente Capasso & Claudiu T. Supuran. (2015)
Crystal structure and kinetic studies of a tetrameric type II β-carbonic anhydrase from the pathogenic bacterium
Vibrio cholerae
. Acta Crystallographica Section D Biological Crystallography 71:12, pages 2449-2456.
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Alessandra Cincinelli, Tania Martellini, Daniela Vullo & Claudiu T. Supuran. (2015) Anion and sulfonamide inhibition studies of an α-carbonic anhydrase from the Antarctic hemoglobinless fish Chionodraco hamatus. Bioorganic & Medicinal Chemistry Letters 25:23, pages 5485-5489.
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Murat Bozdag, Ahmed M. Alafeefy, Daniela Vullo, Fabrizio Carta, Nurcan Dedeoglu, Abdul-Malek S. Al-Tamimi, Nabila A. Al-Jaber, Andrea Scozzafava & Claudiu T. Supuran. (2015) Benzenesulfonamides incorporating bulky aromatic/heterocyclic tails with potent carbonic anhydrase inhibitory activity. Bioorganic & Medicinal Chemistry 23:24, pages 7751-7764.
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Sonia Del Prete, Daniela Vullo, Sameh M. Osman, Zeid AlOthman, Clemente Capasso & Claudiu T. Supuran. (2015) Anion inhibition studies of the dandruff-producing fungus Malassezia globosa β-carbonic anhydrase MgCA. Bioorganic & Medicinal Chemistry Letters 25:22, pages 5194-5198.
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Alfonso Maresca, Gulay Akyuz, Sameh M. Osman, Zeid AlOthman & Claudiu T. Supuran. (2015) Inhibition of mammalian carbonic anhydrase isoforms I–XIV with a series of phenolic acid esters. Bioorganic & Medicinal Chemistry 23:22, pages 7181-7188.
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Fabrizio Carta, Sameh M. Osman, Daniela Vullo, Zeid AlOthman, Sonia Del Prete, Clemente Capasso & Claudiu T. Supuran. (2015) Poly(amidoamine) dendrimers show carbonic anhydrase inhibitory activity against α-, β-, γ- and η-class enzymes. Bioorganic & Medicinal Chemistry 23:21, pages 6794-6798.
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Alessio Nocentini, Fabrizio Carta, Mariangela Ceruso, Gianluca Bartolucci & Claudiu T. Supuran. (2015) Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII. Bioorganic & Medicinal Chemistry 23:21, pages 6955-6966.
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Hany S. Ibrahim, Sahar M. Abou-Seri, Muhammet Tanc, Mahmoud M. Elaasser, Hatem A. Abdel-Aziz & Claudiu T. Supuran. (2015) Isatin-pyrazole benzenesulfonamide hybrids potently inhibit tumor-associated carbonic anhydrase isoforms IX and XII. European Journal of Medicinal Chemistry 103, pages 583-593.
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İbrahim Esirden, Ramazan Ulus, Burak Aday, Muhammet Tanç, Claudiu T. Supuran & Muharrem Kaya. (2015) Synthesis of novel acridine bis-sulfonamides with effective inhibitory activity against the carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry 23:20, pages 6573-6580.
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Cenzo Congiu, Valentina Onnis, Alessandro Deplano, Gianfranco Balboni, Nurcan Dedeoglu & Claudiu T. Supuran. (2015) Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity. Bioorganic & Medicinal Chemistry Letters 25:18, pages 3850-3853.
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Cenzo Congiu, Valentina Onnis, Alessandro Deplano, Gianfranco Balboni, Mariangela Ceruso & Claudiu T. Supuran. (2015) Synthesis and carbonic anhydrase I, II, IX and XII inhibitory activity of sulfamates incorporating piperazinyl-ureido moieties. Bioorganic & Medicinal Chemistry 23:17, pages 5619-5625.
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Mikhail Krasavin, Mikhail Korsakov, Mikhail Dorogov, Tiziano Tuccinardi, Nurcan Dedeoglu & Claudiu T. Supuran. (2015) Probing the ‘bipolar’ nature of the carbonic anhydrase active site: Aromatic sulfonamides containing 1,3-oxazol-5-yl moiety as picomolar inhibitors of cytosolic CA I and CA II isoforms. European Journal of Medicinal Chemistry 101, pages 334-347.
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Mariangela Ceruso, Fabrizio Carta, Sameh M. Osman, Zeid Alothman, Simona Maria Monti & Claudiu T. Supuran. (2015) Inhibition studies of bacterial, fungal and protozoan β-class carbonic anhydrases with Schiff bases incorporating sulfonamide moieties. Bioorganic & Medicinal Chemistry 23:15, pages 4181-4187.
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Diaa A. Ibrahim, Deena S. Lasheen, Maysoun Y. Zaky, Amany W. Ibrahim, Daniela Vullo, Mariangela Ceruso, Claudiu T. Supuran & Dalal A. Abou El Ella. (2015) Design and synthesis of benzothiazole-6-sulfonamides acting as highly potent inhibitors of carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry 23:15, pages 4989-4999.
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Nurcan Dedeoglu, Viviana De Luca, Semra Isik, Hatice Yildirim, Feray Kockar, Clemente Capasso & Claudiu T. Supuran. (2015) Cloning, characterization and anion inhibition study of a β-class carbonic anhydrase from the caries producing pathogen Streptococcus mutans. Bioorganic & Medicinal Chemistry 23:13, pages 2995-3001.
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Nurcan Dedeoglu, Viviana DeLuca, Semra Isik, Hatice Yildirim, Feray Kockar, Clemente Capasso & Claudiu T. Supuran. (2015) Sulfonamide inhibition study of the β-class carbonic anhydrase from the caries producing pathogen Streptococcus mutans. Bioorganic & Medicinal Chemistry Letters 25:11, pages 2291-2297.
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Aiga Grandane, Muhammet Tanc, Lorenzo Di Cesare Mannelli, Fabrizio Carta, Carla Ghelardini, Raivis Žalubovskis & Claudiu T. Supuran. (2015) 6-Substituted Sulfocoumarins Are Selective Carbonic Anhdydrase IX and XII Inhibitors with Significant Cytotoxicity against Colorectal Cancer Cells. Journal of Medicinal Chemistry 58:9, pages 3975-3983.
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Murat Bozdag, Fabrizio Carta, Daniela Vullo, Atilla Akdemir, Semra Isik, Cecilia Lanzi, Andrea Scozzafava, Emanuela Masini & Claudiu T. Supuran. (2015) Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma action. Bioorganic & Medicinal Chemistry 23:10, pages 2368-2376.
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Dhiman Sankar Pal, Dipon Kumar Mondal & Rupak Datta. (2015) Identification of Metal Dithiocarbamates as a Novel Class of Antileishmanial Agents. Antimicrobial Agents and Chemotherapy 59:4, pages 2144-2152.
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Aiga Grandane, Muhammet Tanc, Raivis Žalubovskis & Claudiu T. Supuran. (2015) Synthesis of 6-aryl-substituted sulfocoumarins and investigation of their carbonic anhydrase inhibitory action. Bioorganic & Medicinal Chemistry 23:7, pages 1430-1436.
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Jekaterina Ivanova, Janis Leitans, Muhammet Tanc, Andris Kazaks, Raivis Zalubovskis, Claudiu T. Supuran & Kaspars Tars. (2015) X-ray crystallography-promoted drug design of carbonic anhydrase inhibitors. Chemical Communications 51:33, pages 7108-7111.
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Alaa A.-M. Abdel-Aziz, Adel S. El-Azab, Mariangela Ceruso & Claudiu T. Supuran. (2014) Carbonic anhydrase inhibitory activity of sulfonamides and carboxylic acids incorporating cyclic imide scaffolds. Bioorganic & Medicinal Chemistry Letters 24:22, pages 5185-5189.
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Claudiu T Supuran & Clemente CapassoFabrizio CartaMurat BozdagMuhammet TancClaudiu T Supuran. 2014. Targeting Carbonic Anhydrases. Targeting Carbonic Anhydrases
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Sonia Del Prete, Daniela Vullo, Gillian M. Fisher, Katherine T. Andrews, Sally-Ann Poulsen, Clemente Capasso & Claudiu T. Supuran. (2014) Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum —The η-carbonic anhydrases. Bioorganic & Medicinal Chemistry Letters 24:18, pages 4389-4396.
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Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Andrea Scozzafava, Zeid Alothman, Claudiu T. Supuran & Clemente Capasso. (2014) Anion inhibition study of the β-class carbonic anhydrase (PgiCAb) from the oral pathogen Porphyromonas gingivalis. Bioorganic & Medicinal Chemistry Letters 24:18, pages 4402-4406.
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Mehri Haeili, Casey Moore, Christopher J. C. Davis, James B. Cochran, Santosh Shah, Tej B. Shrestha, Yaofang Zhang, Stefan H. Bossmann, William H. Benjamin, Olaf Kutsch & Frank Wolschendorf. (2014) Copper Complexation Screen Reveals Compounds with Potent Antibiotic Properties against Methicillin-Resistant Staphylococcus aureus. Antimicrobial Agents and Chemotherapy 58:7, pages 3727-3736.
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Leo Syrjänen, Seppo Parkkila, Andrea Scozzafava & Claudiu T. Supuran. (2014) Sulfonamide inhibition studies of the β carbonic anhydrase from Drosophila melanogaster. Bioorganic & Medicinal Chemistry Letters 24:13, pages 2797-2801.
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Mostafa M. Ghorab, Mansour S. Alsaid, Mariangela Ceruso, Yassin M. Nissan & Claudiu T. Supuran. (2014) Carbonic anhydrase inhibitors: Synthesis, molecular docking, cytotoxic and inhibition of the human carbonic anhydrase isoforms I, II, IX, XII with novel benzenesulfonamides incorporating pyrrole, pyrrolopyrimidine and fused pyrrolopyrimidine moieties. Bioorganic & Medicinal Chemistry 22:14, pages 3684-3695.
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Isao Nishimori, Daniela Vullo, Tomoko Minakuchi, Andrea Scozzafava, Sameh M. Osman, Zeid AlOthman, Clemente Capasso & Claudiu T. Supuran. (2014) Anion inhibition studies of two new β-carbonic anhydrases from the bacterial pathogen Legionella pneumophila. Bioorganic & Medicinal Chemistry Letters 24:4, pages 1127-1132.
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Andrea Scozzafava & Claudiu T. Supuran. 2014. Carbonic Anhydrase: Mechanism, Regulation, Links to Disease, and Industrial Applications. Carbonic Anhydrase: Mechanism, Regulation, Links to Disease, and Industrial Applications
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Robert McKenna & Claudiu T. Supuran. 2014. Carbonic Anhydrase: Mechanism, Regulation, Links to Disease, and Industrial Applications. Carbonic Anhydrase: Mechanism, Regulation, Links to Disease, and Industrial Applications
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Daniela Vullo, R. Siva Sai Kumar, Andrea Scozzafava, Clemente Capasso, James G. Ferry & Claudiu T. Supuran. (2013) Anion inhibition studies of a β-carbonic anhydrase from Clostridium perfringens. Bioorganic & Medicinal Chemistry Letters 23:24, pages 6706-6710.
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Janis Leitans, Agnese Sprudza, Muhammet Tanc, Igor Vozny, Raivis Zalubovskis, Kaspars Tars & Claudiu T. Supuran. (2013) 5-Substituted-(1,2,3-triazol-4-yl)thiophene-2-sulfonamides strongly inhibit human carbonic anhydrases I, II, IX and XII: Solution and X-ray crystallographic studies. Bioorganic & Medicinal Chemistry 21:17, pages 5130-5138.
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Peiwen Pan, Alane Beatriz Vermelho, Andrea Scozzafava, Seppo Parkkila, Clemente Capasso & Claudiu T. Supuran. (2013) Anion inhibition studies of the α-carbonic anhydrase from the protozoan pathogen Trypanosoma cruzi, the causative agent of Chagas disease. Bioorganic & Medicinal Chemistry 21:15, pages 4472-4476.
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Muhammet Tanc, Fabrizio Carta, Murat Bozdag, Andrea Scozzafava & Claudiu T. Supuran. (2013) 7-Substituted-sulfocoumarins are isoform-selective, potent carbonic anhydrase II inhibitors. Bioorganic & Medicinal Chemistry 21:15, pages 4502-4510.
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Fabrizio Carta, Atilla Akdemir, Andrea Scozzafava, Emanuela Masini & Claudiu T. Supuran. (2013) Xanthates and Trithiocarbonates Strongly Inhibit Carbonic Anhydrases and Show Antiglaucoma Effects in Vivo. Journal of Medicinal Chemistry 56:11, pages 4691-4700.
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Daniela Vullo, Worraanong Leewattanapasuk, Fritz A. Mühlschlegel, Antonio Mastrolorenzo, Clemente Capasso & Claudiu T. Supuran. (2013) Carbonic anhydrase inhibitors: Inhibition of the β-class enzyme from the pathogenic yeast Candida glabrata with sulfonamides, sulfamates and sulfamides. Bioorganic & Medicinal Chemistry Letters 23:9, pages 2647-2652.
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Peiwen Pan, Alane Beatriz Vermelho, Giseli Capaci Rodrigues, Andrea Scozzafava, Martti E. E. Tolvanen, Seppo Parkkila, Clemente Capasso & Claudiu T. Supuran. (2013)
Cloning, Characterization, and Sulfonamide and Thiol Inhibition Studies of an α-Carbonic Anhydrase from
Trypanosoma cruzi
, the Causative Agent of Chagas Disease
. Journal of Medicinal Chemistry 56:4, pages 1761-1771.
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Daniela Vullo, Viviana De Luca, Andrea Scozzafava, Vincenzo Carginale, Mosè Rossi, Claudiu T. Supuran & Clemente Capasso. (2012) Anion inhibition studies of the fastest carbonic anhydrase (CA) known, the extremo-CA from the bacterium Sulfurihydrogenibium azorense. Bioorganic & Medicinal Chemistry Letters 22:23, pages 7142-7145.
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Giuseppina De Simone & Claudiu T. Supuran. (2012) (In)organic anions as carbonic anhydrase inhibitors. Journal of Inorganic Biochemistry 111, pages 117-129.
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