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Research Article

Kinetic and in silico analysis of thiazolidin-based inhibitors of α-carbonic anhydrase isoenzymes

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Pages 370-374 | Received 28 Aug 2012, Accepted 17 Sep 2012, Published online: 23 Nov 2012

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Read on this site (6)

Claudiu T. Supuran. (2017) Advances in structure-based drug discovery of carbonic anhydrase inhibitors. Expert Opinion on Drug Discovery 12:1, pages 61-88.
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Chandra Bhushan Mishra, Shikha Kumari, Andrea Angeli, Simona Maria Monti, Martina Buonanno, Amresh Prakash, Manisha Tiwari & Claudiu T. Supuran. (2016) Design, synthesis and biological evaluation of N-(5-methyl-isoxazol-3-yl/1,3,4-thiadiazol-2-yl)-4-(3-substitutedphenylureido) benzenesulfonamides as human carbonic anhydrase isoenzymes I, II, VII and XII inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 31:sup2, pages 174-179.
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F. Zehra Küçükbay, Hasan Küçükbay, Muhammet Tanc & Claudiu T. Supuran. (2016) Synthesis and carbonic anhydrase I, II, IV and XII inhibitory properties of N-protected amino acid – sulfonamide conjugates. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1476-1483.
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Claudiu T. Supuran. (2016) How many carbonic anhydrase inhibition mechanisms exist?. Journal of Enzyme Inhibition and Medicinal Chemistry 31:3, pages 345-360.
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Ramin Ekhteiari Salmas, Murat Senturk, Mine Yurtsever & Serdar Durdagi. (2016) Discovering novel carbonic anhydrase type IX (CA IX) inhibitors from seven million compounds using virtual screening and in vitro analysis. Journal of Enzyme Inhibition and Medicinal Chemistry 31:3, pages 425-433.
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Ahmed M. Alafeefy, Mariangela Ceruso, Abdul-Malek S. Al-Tamimi, Sonia Del Prete, Claudiu T. Supuran & Clemente Capasso. (2015) Inhibition studies of quinazoline-sulfonamide derivatives against the γ-CA (PgiCA) from the pathogenic bacterium, Porphyromonas gingivalis. Journal of Enzyme Inhibition and Medicinal Chemistry 30:4, pages 592-596.
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Articles from other publishers (8)

Ali Atasever. (2023) Molecular docking and inhibition profiles of some antidepressants on human carbonic anhydrase enzymes. Results in Chemistry 6, pages 101174.
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Saad Alghamdi, Mazen M. Almehmadi, Mohammad Asif, Mohammed M. Alshehri & Mehnaz Kamal. (2022) Antimycobacterial Evaluation and Microwave-Assisted Synthesis of N-(5-methyl-4-oxo-2-arylthiazolidin-3-yl) Isonicotinamide Derivatives. Pharmaceutical Chemistry Journal 56:2, pages 215-219.
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Saad Alghamdi, Mehnaz Kamal & Mohammad Asif. (2022) Antimycobacterial Assessment and Microwave-assisted Synthesis of 2-aryl- 3-(4-methylphenylamino)thiazolidin-4-one Derivatives. Letters in Organic Chemistry 19:3, pages 250-255.
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Galal H. Elgemeie, Rasha A. Azzam, Wafaa A. Zaghary, Ashraf A. Aly, Nadia H. Metwally, Mona O. Sarhan, Elshimaa M. Abdelhafez & Rasha E. Elsayed. 2022. N-Sulfonated-N-Heterocycles. N-Sulfonated-N-Heterocycles 113 133 .
Baijayantimala Swain, Kamtam Aashritha, Priti Singh, Andrea Angeli, Abhay Kothari, Dilep K. Sigalapalli, Venkata M. Yaddanapudi, Claudiu T. Supuran & Mohammed Arifuddin. (2021) Design and synthesis of benzenesulfonamide‐linked imidazo[2,1‐ b ][1,3,4]thiadiazole derivatives as carbonic anhydrase I and II inhibitors . Archiv der Pharmazie 354:7, pages 2100028.
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Daniela Vullo, Viviana De Luca, Sonia Del Prete, Vincenzo Carginale, Andrea Scozzafava, Clemente Capasso & Claudiu T. Supuran. (2015) Sulfonamide inhibition studies of the γ-carbonic anhydrase from the Antarctic bacterium Pseudoalteromonas haloplanktis. Bioorganic & Medicinal Chemistry Letters 25:17, pages 3550-3555.
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Murat Güney, Hüseyin Çavdar, Murat Şentürk & Deniz Ekinci. (2015) Synthesis and carbonic anhydrase inhibitory properties of novel uracil derivatives. Bioorganic & Medicinal Chemistry Letters 25:16, pages 3261-3263.
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Süleyman Göksu, Ali Naderi, Yusuf Akbaba, Pınar Kalın, Akın Akıncıoğlu, İlhami Gülçin, Serdar Durdagi & Ramin Ekhteiari Salmas. (2014) Carbonic anhydrase inhibitory properties of novel benzylsulfamides using molecular modeling and experimental studies. Bioorganic Chemistry 56, pages 75-82.
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