Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 17, Issue 6 (2002)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 17, Issue 6 (2002)

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Research Article

Article
10th Birthday of the European Conferences of GP2A--Nantes 2001
H.J. Smith
Page: 351
Published online: 30 Sep 2008
Citationfor10th Birthday of the European Conferences of GP2A--Nantes 2001 | PDF (34.7 KB)
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Article
Synthesis and Antileishmanial Activity of 3-(α-Azolylbenzyl)indoles
Pascal Marchand, Marc Le Borgne, Young Min Na, Fabrice Pagniez, Hiam Abdala, Guillaume Le Baut & Patrice Le Pape
Pages: 353-358
Published online: 30 Sep 2008
AbstractforSynthesis and Antileishmanial Activity of 3-(α-Azolylbenzyl)indoles | References | PDF (208.5 KB)
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Article
The Chemistry of [1,2,3]Triazolo[1,5- a] pyridines
Belén Abarca-González
Pages: 359-367
Published online: 30 Sep 2008
AbstractforThe Chemistry of [1,2,3]Triazolo[1,5- a] pyridines | References | PDF (374.6 KB)
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Article
Cytotoxic Bis-3,4-dihydro-β-carbolines and Bis-β-carbolines
Wei-Qun Jiang, Catherine Charlet-Fagnère, Janos Sapi, Jean-Yves Laronze, Pierre Renard, Bruno Pfeiffer & Stéphane Léonce
Pages: 369-374
Published online: 30 Sep 2008
AbstractforCytotoxic Bis-3,4-dihydro-β-carbolines and Bis-β-carbolines | References | PDF (150.8 KB)
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Article
Derivatization of (±)-5-[(2-Methylphenoxy)methyl]-2-amino-2-oxazoline, an Imidazoline Binding Sites Ligand, with (+)- (R) -α-Methylbenzyl Isocyanate for Drug Monitoring Purposes
Myriam Matoga, Isabelle Forfar, Corinne Chaimbault, Jean Guillon, Fabienne Péhourcq, Jean-Jacques Bosc, Marie-Claire Rettori & Christian Jarry
Pages: 375-379
Published online: 30 Sep 2008
AbstractforDerivatization of (±)-5-[(2-Methylphenoxy)methyl]-2-amino-2-oxazoline, an Imidazoline Binding Sites Ligand, with (+)- (R) -α-Methylbenzyl Isocyanate for Drug Monitoring Purposes | References | PDF (133 KB)
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Article
Rho-kinase Inhibitors: Pharmacomodulations on the Lead Compound Y-32885
Cédric Logé, Valérie Wallez, Elizabeth Scalbert, Christelle Cario-Tourmaniantz, Gervaise Loirand, Pierre Pacaud & Daniel Lesieur
Pages: 381-390
Published online: 30 Sep 2008
AbstractforRho-kinase Inhibitors: Pharmacomodulations on the Lead Compound Y-32885 | References | PDF (287.9 KB)
  • 244 Views
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Article
Anti-leukemia Activity of 7-hydroxy-2-substituted-methyl-5 H -oxazolo[3,2- a] pyrimidin-5-one Derivatives
Jean Guillon, Maria Mamani-Matsuda, Stephane Massip, Jean-Michel Leger, Denis Thiolat, Djavad Mossalayi & Christian Jarry
Pages: 391-396
Published online: 30 Sep 2008
AbstractforAnti-leukemia Activity of 7-hydroxy-2-substituted-methyl-5 H -oxazolo[3,2- a] pyrimidin-5-one Derivatives | References | PDF (207.7 KB)
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Article
Synthesis and Cytotoxic Evaluation of Novel Thiazolocarbazoles
Christelle Lamazzi, Hadjila Chabane, Valerie Thiery, Alain Pierre, Stephane Leonce, Bruno Pfeiffer, Pierre Renard, Gérald Guillaumet & Thierry Besson
Pages: 397-401
Published online: 30 Sep 2008
AbstractforSynthesis and Cytotoxic Evaluation of Novel Thiazolocarbazoles | References | PDF (147.8 KB)
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Article
Synthesis of New Aromatic Pyrrolo[2,1- c] [1,4]benzodiazepines and Pyrrolo[1,2- a] thieno[3,2- e] [1,4]diazepines as Anti-tumoral Agents
Vincent Lisowski, Frédéric Fabis, Alain Pierré, Daniel-Henri Caignard, Pierre Renard & Sylvain Rault
Pages: 403-407
Published online: 30 Sep 2008
AbstractforSynthesis of New Aromatic Pyrrolo[2,1- c] [1,4]benzodiazepines and Pyrrolo[1,2- a] thieno[3,2- e] [1,4]diazepines as Anti-tumoral Agents | References | PDF (152.6 KB)
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Article
Design, Synthesis and In Vitro Evaluation of Novel Derivatives as Serotonin N -Acetyltransferase Inhibitors
N. Beaurain, C. Mésangeau, P. Chavatte, G. Ferry, V. Audinot, J.A. Boutin, P. Delagrange, C. Bennejean & S. Yous
Pages: 409-414
Published online: 30 Sep 2008
AbstractforDesign, Synthesis and In Vitro Evaluation of Novel Derivatives as Serotonin N -Acetyltransferase Inhibitors | References | PDF (148.2 KB)
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Article
New N -pyridinyl(methyl)-indole-2- and 3-(Alkyl)carboxamides and Derivatives Acting as Systemic and Topical Inflammation Inhibitors
Anne Breteche, Muriel Duflos, Alexandra Dassonville, Marie-Renee Nourrisson, Jacques Brelet, Guillaume Le Baut, Nicole Grimaud & Jean-Yves Petit
Pages: 415-424
Published online: 30 Sep 2008
AbstractforNew N -pyridinyl(methyl)-indole-2- and 3-(Alkyl)carboxamides and Derivatives Acting as Systemic and Topical Inflammation Inhibitors | References | PDF (233.8 KB)
  • 280 Views
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Article
In Vitro Activity of a New Antifungal Azolyl-substituted Indole Against Aspergillus fumigatus
Fabrice Pagniez, Marc Le Borgne, Pascal Marchand, Young Min Na, Guillaume Le Baut, Sylvie Robert-Piessard & Patrice Le Pape
Pages: 425-429
Published online: 30 Sep 2008
AbstractforIn Vitro Activity of a New Antifungal Azolyl-substituted Indole Against Aspergillus fumigatus | References | PDF (128.3 KB)
  • 143 Views
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Article
Synthesis and Antimalarial Activity of Some New 1,2-Dioxolane Derivatives
Jean-Jacques Helesbeux, Damien Peyronnet, Mehdi Labaïed, Philippe Grellier, François Frappier, Denis Seraphin, Pascal Richomme & Olivier Duval
Pages: 431-437
Published online: 30 Sep 2008
AbstractforSynthesis and Antimalarial Activity of Some New 1,2-Dioxolane Derivatives | References | PDF (242.6 KB)
  • 343 Views
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Article
A First Cyclopenta [c] thiophene Dimer as a New Bivalent Potent Cytotoxic Derivative
Lan Pham Khanh, Patrick Dallemagne, Henriette Landelle & Sylvain Rault
Pages: 439-442
Published online: 30 Sep 2008
AbstractforA First Cyclopenta [c] thiophene Dimer as a New Bivalent Potent Cytotoxic Derivative | References | PDF (116.4 KB)
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Article
Inhibition of Parasite Protein Kinase C by New Antileishmanial Imidazolidin-2-one Compounds
Nidia Alvarez, Sara Robledo, Ivan Dario Velez, Jean Michel Robert, Guillaume Le Baut & Patrice Le Pape
Pages: 443-447
Published online: 30 Sep 2008
AbstractforInhibition of Parasite Protein Kinase C by New Antileishmanial Imidazolidin-2-one Compounds | References | PDF (165.5 KB)
  • 216 Views
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Article
8-Amino-5-nitro-6-phenoxyquinolines: Potential Non-peptidic Neuropeptide Y Receptor Ligands
Gaetane Wielgosz-collin, Muriel Duflos, Patricia Pinson, Guillaume Le baut, Pierre Renard, Caroline Bennejean, Jean Boutin & Michele Boulanger
Pages: 449-453
Published online: 30 Sep 2008
Abstractfor8-Amino-5-nitro-6-phenoxyquinolines: Potential Non-peptidic Neuropeptide Y Receptor Ligands | References | PDF (136.3 KB)
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