Citations (49)
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Claudiu T. Supuran. (2020) Exploring the multiple binding modes of inhibitors to carbonic anhydrases for novel drug discovery. Expert Opinion on Drug Discovery 15:6, pages 671-686.
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Claudiu T. Supuran. (2017) Advances in structure-based drug discovery of carbonic anhydrase inhibitors. Expert Opinion on Drug Discovery 12:1, pages 61-88.
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Alessio Nocentini, Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Fatmah A.S. Alasmary, Zeid AlOthman, Clemente Capasso, Fabrizio Carta, Paola Gratteri & Claudiu T. Supuran. (2017) Inhibition of the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa with monothiocarbamates. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1064-1070.
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Chandra Bhushan Mishra, Shikha Kumari, Andrea Angeli, Simona Maria Monti, Martina Buonanno, Amresh Prakash, Manisha Tiwari & Claudiu T. Supuran. (2016) Design, synthesis and biological evaluation of N-(5-methyl-isoxazol-3-yl/1,3,4-thiadiazol-2-yl)-4-(3-substitutedphenylureido) benzenesulfonamides as human carbonic anhydrase isoenzymes I, II, VII and XII inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 31:sup2, pages 174-179.
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F. Zehra Küçükbay, Hasan Küçükbay, Muhammet Tanc & Claudiu T. Supuran. (2016) Synthesis and carbonic anhydrase I, II, IV and XII inhibitory properties of N-protected amino acid – sulfonamide conjugates. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1476-1483.
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Serdar Durdagi, Neslihan Korkmaz, Semra Işık, Daniela Vullo, Demet Astley, Deniz Ekinci, Ramin E. Salmas, Murat Senturk & Claudiu T. Supuran. (2016) Kinetic and docking studies of cytosolic/tumor-associated carbonic anhydrase isozymes I, II and IX with some hydroxylic compounds. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1214-1220.
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Claudiu T. Supuran. (2016) How many carbonic anhydrase inhibition mechanisms exist?. Journal of Enzyme Inhibition and Medicinal Chemistry 31:3, pages 345-360.
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Murat Bozdag, Fabrizio Carta, Daniela Vullo, Semra Isik, Zeid AlOthman, Sameh M. Osman, Andrea Scozzafava & Claudiu T. Supuran. (2016) Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase. Journal of Enzyme Inhibition and Medicinal Chemistry 31:1, pages 132-136.
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Joanna Ombouma, Daniela Vullo, Stephan Köhler, Pascal Dumy, Claudiu T. Supuran & Jean-Yves Winum. (2015) N-glycosyl-N-hydroxysulfamides as potent inhibitors of Brucella suis carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 1010-1012.
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Namrata Singasane, Prashant S. Kharkar, Mariangela Ceruso, Claudiu T. Supuran & Mrunmayee P. Toraskar. (2015) Inhibition of carbonic anhydrase isoforms I, II, IX and XII with Schiff’s bases incorporating iminoureido moieties. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 901-907.
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Daniela Vullo, Semra Isik, Murat Bozdag, Fabrizio Carta & Claudiu T. Supuran. (2015) 7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring. Journal of Enzyme Inhibition and Medicinal Chemistry 30:5, pages 773-777.
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Claudiu T Supuran. (2015) Acetazolamide for the treatment of idiopathic intracranial hypertension. Expert Review of Neurotherapeutics 15:8, pages 851-856.
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Ahmed M. Alafeefy, Hatem A. Abdel-Aziz, Daniela Vullo, Abdul-Malek S. Al-Tamimi, Amani S. Awaad, Menshawy A. Mohamed, Clemente Capasso & Claudiu T. Supuran. (2015) Inhibition of human carbonic anhydrase isozymes I, II, IX and XII with a new series of sulfonamides incorporating aroylhydrazone-, [1,2,4]triazolo[3,4-b][1,3,4]thiadiazinyl- or 2-(cyanophenylmethylene)-1,3,4-thiadiazol-3(2H)-yl moieties. Journal of Enzyme Inhibition and Medicinal Chemistry 30:1, pages 52-56.
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Shalini Singh & Claudiu T. Supuran. (2014) Chemometric modeling of breast cancer associated carbonic anhydrase IX inhibitors belonging to the ureido-substituted benzene sulfonamide class. Journal of Enzyme Inhibition and Medicinal Chemistry 29:6, pages 877-883.
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Aditi Sharma, Meena Tiwari & Claudiu T. Supuran. (2014) Novel coumarins and benzocoumarins acting as isoform-selective inhibitors against the tumor-associated carbonic anhydrase IX. Journal of Enzyme Inhibition and Medicinal Chemistry 29:2, pages 292-296.
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Emanuela Masini, Fabrizio Carta, Andrea Scozzafava & Claudiu T Supuran. (2013) Antiglaucoma carbonic anhydrase inhibitors: a patent review. Expert Opinion on Therapeutic Patents 23:6, pages 705-716.
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Claudiu T. Supuran. (2013) Carbonic anhydrases: from biomedical applications of the inhibitors and activators to biotechnological use for CO2 capture. Journal of Enzyme Inhibition and Medicinal Chemistry 28:2, pages 229-230.
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Claudiu T Supuran. (2012) Amide derivatives of benzene-sulfonanilide, pharmaceutical composition thereof and method for cancer treatment using the same (US20120095092). Expert Opinion on Therapeutic Patents 22:10, pages 1251-1255.
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Articles from other publishers (31)
Mohamed S. Bekheit, Eman Sabry, Hanan A. Mohamed, Ewies F. Ewies, Benson M. Kariuki, Marwa A. Fouad, Daniela Vullo & Claudiu T. Supuran. (2023) Novel sulfonamide‐phosphonate conjugates as carbonic anhydrase isozymes inhibitors. Drug Development Research.
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Eyüp Başaran, Reşit Çakmak, Murat Şentürk & Tugba Taskin‐Tok. (2022)
Biological activity and molecular docking studies of some
N
‐phenylsulfonamides against cholinesterases and carbonic anhydrase isoenzymes
. Journal of Molecular Recognition 35:10.
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Amy C. Dodds, Sabrina Puddu & Andrew Sutherland. (2022) Thioarylation of anilines using dual catalysis: two-step synthesis of phenothiazines. Organic & Biomolecular Chemistry 20:28, pages 5602-5614.
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Oliver M. Griffiths, Henrique A. EstevesYiding ChenKarin Sowa, Oliver S. MayPeter Morse, David C. Blakemore & Steven V. Ley. (2021)
Photoredox-Catalyzed Dehydrogenative Csp
3
–Csp
2
Cross-Coupling of Alkylarenes to Aldehydes in Flow
. The Journal of Organic Chemistry 86:19, pages 13559-13571.
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Ahmet Gokhan Aggul, Parham Taslimi, Muslum Kuzu, Naim Uzun, Sinan Bilginer & Ilhami Gulcin. (2021) Oleuropein and Verbascoside - Their Inhibition Effects on Carbonic Anhydrase and Molecular Docking Studies. Journal of Oleo Science 70:9, pages 1275-1283.
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Claudiu T. Supuran. 2021. The Carbonic Anhydrases: Current and Emerging Therapeutic Targets. The Carbonic Anhydrases: Current and Emerging Therapeutic Targets
221
235
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Chandra B. Mishra, Manisha Tiwari & Claudiu T. Supuran. (2020) Progress in the development of human carbonic anhydrase inhibitors and their pharmacological applications: Where are we today?. Medicinal Research Reviews 40:6, pages 2485-2565.
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Mirian R.C. de Castro, Raquel Ferreira Naves, Aline Bernardes, Cameron Capeletti da Silva, Caridad Noda Perez, Andrea Felinto Moura, Manoel Odorico de Moraes & Felipe Terra Martins. (2020) Tandem chalcone-sulfonamide hybridization, cyclization and further Claisen–Schmidt condensation: Tuning molecular diversity through reaction time and order and catalyst. Arabian Journal of Chemistry 13:1, pages 1345-1354.
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Joseane A. Mendes, Eduardo J. Salustiano, Carulini de S. Pires, Thaís Oliveira, Julio C.F. Barcellos, Jhonny M.C. Cifuentes, Paulo R.R. Costa, Magdalena N. Rennó & Camilla D. Buarque. (2018) 11a-N-tosyl-5-carbapterocarpans: Synthesis, antineoplastic evaluation and in silico prediction of ADMETox properties. Bioorganic Chemistry 80, pages 585-590.
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Changrui Xu, Zhengxing Wu, Jianzhong Chen, Fang Xie & Wanbin Zhang. (2017) Palladium(II)-catalyzed aerobic intramolecular allylic C H activation for the synthesis of indolines. Tetrahedron 73:14, pages 1904-1910.
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Daniela Vullo, Sonia Del Prete, Alessio Nocentini, Sameh M. Osman, Zeid AlOthman, Clemente Capasso, Murat Bozdag, Fabrizio Carta, Paola Gratteri & Claudiu T. Supuran. (2017) Dithiocarbamates effectively inhibit the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa. Bioorganic & Medicinal Chemistry 25:3, pages 1260-1265.
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Deryanur KILIÇ, Orhan ERDOĞAN & Ömer İrfan KÜFREVİOĞLU. (2017) Effect of mutation in active site residue Trp209 to Val, Leu, Ile and Pro on the catalytic activity and affinity for some benzenesulfonamides of human carbonic anhydrase II. TURKISH JOURNAL OF BIOLOGY 41, pages 835-842.
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Tayfun Arslan, Emir Alper Türkoğlu, Murat Şentürk & Claudiu T. Supuran. (2016) Synthesis and carbonic anhydrase inhibitory properties of novel chalcone substituted benzenesulfonamides. Bioorganic & Medicinal Chemistry Letters 26:24, pages 5867-5870.
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Semra Işık, Daniela Vullo, Serdar Durdagi, Deniz Ekinci, Murat Şentürk, Ahmet Çetin, Esra Şentürk & Claudiu T. Supuran. (2015) Interaction of carbonic anhydrase isozymes I, II, and IX with some pyridine and phenol hydrazinecarbothioamide derivatives. Bioorganic & Medicinal Chemistry Letters 25:23, pages 5636-5641.
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İsmail Fidan, Ramin Ekhteiari Salmas, Mehmet Arslan, Murat Şentürk, Serdar Durdagi, Deniz Ekinci, Esra Şentürk, Sedat Coşgun & Claudiu T. Supuran. (2015) Carbonic anhydrase inhibitors: Design, synthesis, kinetic, docking and molecular dynamics analysis of novel glycine and phenylalanine sulfonamide derivatives. Bioorganic & Medicinal Chemistry 23:23, pages 7353-7358.
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Sonia Del Prete, Daniela Vullo, Sameh M. Osman, Zeid AlOthman, Clemente Capasso & Claudiu T. Supuran. (2015) Anion inhibition studies of the dandruff-producing fungus Malassezia globosa β-carbonic anhydrase MgCA. Bioorganic & Medicinal Chemistry Letters 25:22, pages 5194-5198.
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Murat Güney, Hüseyin Çavdar, Murat Şentürk & Deniz Ekinci. (2015) Synthesis and carbonic anhydrase inhibitory properties of novel uracil derivatives. Bioorganic & Medicinal Chemistry Letters 25:16, pages 3261-3263.
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Nurcan Dedeoglu, Viviana De Luca, Semra Isik, Hatice Yildirim, Feray Kockar, Clemente Capasso & Claudiu T. Supuran. (2015) Cloning, characterization and anion inhibition study of a β-class carbonic anhydrase from the caries producing pathogen Streptococcus mutans. Bioorganic & Medicinal Chemistry 23:13, pages 2995-3001.
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Nurcan Dedeoglu, Viviana DeLuca, Semra Isik, Hatice Yildirim, Feray Kockar, Clemente Capasso & Claudiu T. Supuran. (2015) Sulfonamide inhibition study of the β-class carbonic anhydrase from the caries producing pathogen Streptococcus mutans. Bioorganic & Medicinal Chemistry Letters 25:11, pages 2291-2297.
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Mustafa Durgun, Hasan Turkmen, Mariangela Ceruso & Claudiu T. Supuran. (2015) Synthesis of Schiff base derivatives of 4-(2-aminoethyl)-benzenesulfonamide with inhibitory activity against carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry Letters 25:11, pages 2377-2381.
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Daniela Vullo, Sonia Del Prete, Gillian M. Fisher, Katherine T. Andrews, Sally-Ann Poulsen, Clemente Capasso & Claudiu T. Supuran. (2015) Sulfonamide inhibition studies of the η-class carbonic anhydrase from the malaria pathogen Plasmodium falciparum. Bioorganic & Medicinal Chemistry 23:3, pages 526-531.
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M. Nardi, N. Herrera Cano, P. Costanzo, M. Oliverio, G. Sindona & A. Procopio. (2015) Aqueous MW eco-friendly protocol for amino group protection. RSC Advances 5:24, pages 18751-18760.
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Busra Sarikaya, Mariangela Ceruso, Fabrizio Carta & Claudiu T. Supuran. (2014) Inhibition of carbonic anhydrase isoforms I, II, IX and XII with novel Schiff bases: Identification of selective inhibitors for the tumor-associated isoforms over the cytosolic ones. Bioorganic & Medicinal Chemistry 22:21, pages 5883-5890.
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Ahmed M. Alafeefy, Mariangela Ceruso, Abdul-Malek S. Al-Tamimi, Sonia Del Prete, Clemente Capasso & Claudiu T. Supuran. (2014) Quinazoline–sulfonamides with potent inhibitory activity against the α-carbonic anhydrase from Vibrio cholerae. Bioorganic & Medicinal Chemistry 22:19, pages 5133-5140.
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Sonia Del Prete, Daniela Vullo, Gillian M. Fisher, Katherine T. Andrews, Sally-Ann Poulsen, Clemente Capasso & Claudiu T. Supuran. (2014) Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum —The η-carbonic anhydrases. Bioorganic & Medicinal Chemistry Letters 24:18, pages 4389-4396.
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Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Andrea Scozzafava, Zeid Alothman, Claudiu T. Supuran & Clemente Capasso. (2014) Anion inhibition study of the β-class carbonic anhydrase (PgiCAb) from the oral pathogen Porphyromonas gingivalis. Bioorganic & Medicinal Chemistry Letters 24:18, pages 4402-4406.
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Gihane Nasr, Alina Cristian, Mihail Barboiu, Daniella Vullo, Jean-Yves Winum & Claudiu T. Supuran. (2014) Carbonic anhydrase inhibitors. Inhibition of human cytosolic isoforms I and II with (reduced) Schiff’s bases incorporating sulfonamide, carboxylate and carboxymethyl moieties. Bioorganic & Medicinal Chemistry 22:10, pages 2867-2874.
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Cenzo Congiu, Valentina Onnis, Gianfranco Balboni & Claudiu T. Supuran. (2014) Synthesis and carbonic anhydrase I, II, IX and XII inhibition studies of 4-N,N-disubstituted sulfanilamides incorporating 4,4,4-trifluoro-3-oxo-but-1-enyl, phenacylthiourea and imidazol-2(3H)-one/thione moieties. Bioorganic & Medicinal Chemistry Letters 24:7, pages 1776-1779.
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Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Viviana De Luca, Andrea Scozzafava, Zeid AlOthman, Claudiu T. Supuran & Clemente Capasso. (2014) Sulfonamide inhibition studies of the γ-carbonic anhydrase from the oral pathogen Porphyromonas gingivalis. Bioorganic & Medicinal Chemistry Letters 24:1, pages 240-244.
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Murat Bozdag, Marta Ferraroni, Elisa Nuti, Daniela Vullo, Armando Rossello, Fabrizio Carta, Andrea Scozzafava & Claudiu T. Supuran. (2014) Combining the tail and the ring approaches for obtaining potent and isoform-selective carbonic anhydrase inhibitors: Solution and X-ray crystallographic studies. Bioorganic & Medicinal Chemistry 22:1, pages 334-340.
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Claudiu T. Supuran. (2013) Carbonic anhydrases. Bioorganic & Medicinal Chemistry 21:6, pages 1377-1378.
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