Citations (87)
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Anastasija Balašova, Aleksandrs Pustenko, Alessio Nocentini, Daniela Vullo, Claudiu T. Supuran & Raivis Žalubovskis. (2023) Aryl derivatives of 3H-1,2-benzoxaphosphepine 2-oxides as inhibitors of cancer-related carbonic anhydrase isoforms IX and XII. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Alessio Nocentini, Andrea Angeli, Fabrizio Carta, Jean-Yves Winum, Raivis Zalubovskis, Simone Carradori, Clemente Capasso, William A. Donald & Claudiu T. Supuran. (2021) Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 561-580.
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Hamide Salari, Amin Afkhami-Poostchi, Shokouhozaman Soleymanifard, Saeideh Nakhaei-Rad, Elahe Merajifar, Mehrdad Iranshahi, Maryam M. Matin & Fatemeh B. Rassouli. (2020) Coadministration of auraptene and radiotherapy; a novel modality against colon carcinoma cells in vitro and in vivo. International Journal of Radiation Biology 96:8, pages 1051-1059.
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Claudiu T. Supuran. (2020) Exploring the multiple binding modes of inhibitors to carbonic anhydrases for novel drug discovery. Expert Opinion on Drug Discovery 15:6, pages 671-686.
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Alessio Nocentini & Claudiu T. Supuran. (2019) Advances in the structural annotation of human carbonic anhydrases and impact on future drug discovery. Expert Opinion on Drug Discovery 14:11, pages 1175-1197.
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Marta Menicatti, Marco Pallecchi, Silvia Bua, Daniela Vullo, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Fabrizio Carta, Claudiu T. Supuran & Gianluca Bartolucci. (2018) Resolution of co-eluting isomers of anti-inflammatory drugs conjugated to carbonic anhydrase inhibitors from plasma in liquid chromatography by energy-resolved tandem mass spectrometry. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 671-679.
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Claudiu T. Supuran. (2017) Advances in structure-based drug discovery of carbonic anhydrase inhibitors. Expert Opinion on Drug Discovery 12:1, pages 61-88.
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Alessio Nocentini, Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Fatmah A.S. Alasmary, Zeid AlOthman, Clemente Capasso, Fabrizio Carta, Paola Gratteri & Claudiu T. Supuran. (2017) Inhibition of the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa with monothiocarbamates. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1064-1070.
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Chandra Bhushan Mishra, Shikha Kumari, Andrea Angeli, Simona Maria Monti, Martina Buonanno, Amresh Prakash, Manisha Tiwari & Claudiu T. Supuran. (2016) Design, synthesis and biological evaluation of N-(5-methyl-isoxazol-3-yl/1,3,4-thiadiazol-2-yl)-4-(3-substitutedphenylureido) benzenesulfonamides as human carbonic anhydrase isoenzymes I, II, VII and XII inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 31:sup2, pages 174-179.
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F. Zehra Küçükbay, Hasan Küçükbay, Muhammet Tanc & Claudiu T. Supuran. (2016) Synthesis and carbonic anhydrase I, II, IV and XII inhibitory properties of N-protected amino acid – sulfonamide conjugates. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1476-1483.
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Alessio Nocentini, Mariangela Ceruso, Fabrizio Carta & Claudiu T. Supuran. (2016) 7-Aryl-triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrase IX and XII. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1226-1233.
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Lorenzo Di Cesare Mannelli, Laura Micheli, Fabrizio Carta, Andrea Cozzi, Carla Ghelardini & Claudiu T. Supuran. (2016) Carbonic anhydrase inhibition for the management of cerebral ischemia: in vivo evaluation of sulfonamide and coumarin inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 894-899.
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F. Zehra Küçükbay, Hasan Küçükbay, Muhammet Tanc & Claudiu T. Supuran. (2016) Synthesis and carbonic anhydrase inhibitory properties of amino acid – coumarin/quinolinone conjugates incorporating glycine, alanine and phenylalanine moieties. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1198-1202.
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Claudiu T. Supuran. (2016) How many carbonic anhydrase inhibition mechanisms exist?. Journal of Enzyme Inhibition and Medicinal Chemistry 31:3, pages 345-360.
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Claudiu T. Supuran. (2016) Drug interaction considerations in the therapeutic use of carbonic anhydrase inhibitors. Expert Opinion on Drug Metabolism & Toxicology 12:4, pages 423-431.
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Murat Bozdag, Fabrizio Carta, Daniela Vullo, Semra Isik, Zeid AlOthman, Sameh M. Osman, Andrea Scozzafava & Claudiu T. Supuran. (2016) Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase. Journal of Enzyme Inhibition and Medicinal Chemistry 31:1, pages 132-136.
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Joanna Ombouma, Daniela Vullo, Stephan Köhler, Pascal Dumy, Claudiu T. Supuran & Jean-Yves Winum. (2015) N-glycosyl-N-hydroxysulfamides as potent inhibitors of Brucella suis carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 1010-1012.
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Namrata Singasane, Prashant S. Kharkar, Mariangela Ceruso, Claudiu T. Supuran & Mrunmayee P. Toraskar. (2015) Inhibition of carbonic anhydrase isoforms I, II, IX and XII with Schiff’s bases incorporating iminoureido moieties. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 901-907.
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Daniela Vullo, Semra Isik, Murat Bozdag, Fabrizio Carta & Claudiu T. Supuran. (2015) 7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring. Journal of Enzyme Inhibition and Medicinal Chemistry 30:5, pages 773-777.
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Claudiu T Supuran. (2015) Acetazolamide for the treatment of idiopathic intracranial hypertension. Expert Review of Neurotherapeutics 15:8, pages 851-856.
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Ahmed M. Alafeefy, Mariangela Ceruso, Nabila A. Al-Jaber, Seppo Parkkila, Alane Beatriz Vermelho & Claudiu T. Supuran. (2015) A new class of quinazoline-sulfonamides acting as efficient inhibitors against the α-carbonic anhydrase from Trypanosoma cruzi. Journal of Enzyme Inhibition and Medicinal Chemistry 30:4, pages 581-585.
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Articles from other publishers (66)
Claudiu T. Supuran. 2024. Metalloenzymes. Metalloenzymes
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Deepthi S. Manisha, Anandu Kizhakkedath Ratheesh, Sonu Benny & Aneesh Thankappan Presanna. (2023) Heterocyclic and non‐heterocyclic arena of monocarboxylate transporter inhibitors to battle tumorigenesis. Chemical Biology & Drug Design 102:6, pages 1604-1617.
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Satyajit Khatua & Srabani Taraphder. (2023) Dynamics of an inhibitor at and away from an out-of-active site binding location in human carbonic anhydrase II. Chemical Physics Impact 7, pages 100329.
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Claudiu T. Supuran. (2023) A simple yet multifaceted 90 years old, evergreen enzyme: Carbonic anhydrase, its inhibition and activation. Bioorganic & Medicinal Chemistry Letters 93, pages 129411.
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Ashok Aspatwar, Claudiu T. Supuran, Abdul Waheed, William S. Sly & Seppo Parkkila. (2022) Mitochondrial carbonic anhydrase VA and VB: properties and roles in health and disease. The Journal of Physiology 601:2, pages 257-274.
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Claudiu T. Supuran. 2022. Flavonoids and Phenolics. Flavonoids and Phenolics
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Behnam Rasti. (2022) Quantitative Characterization of the Chemical Space Governed by Human Carbonic Anhydrases and selenium-containing derivatives of solfonamides. Brazilian Journal of Pharmaceutical Sciences 58.
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Claudiu T. Supuran. 2021. The Carbonic Anhydrases: Current and Emerging Therapeutic Targets. The Carbonic Anhydrases: Current and Emerging Therapeutic Targets
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Claudiu T. Supuran. 2021. New Trends in Macromolecular and Supramolecular Chemistry for Biological Applications. New Trends in Macromolecular and Supramolecular Chemistry for Biological Applications
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Aiga Grandāne, Alessio Nocentini, Ilona Domračeva, Raivis Žalubovskis & Claudiu T. Supuran. (2020) Development of oxathiino[6,5-b]pyridine 2,2-dioxide derivatives as selective inhibitors of tumor-related carbonic anhydrases IX and XII. European Journal of Medicinal Chemistry 200, pages 112300.
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Aiga Grandane, Alessio Nocentini, Thomas Werner, Raivis Zalubovskis & Claudiu T. Supuran. (2020) Benzoxepinones: A new isoform-selective class of tumor associated carbonic anhydrase inhibitors. Bioorganic & Medicinal Chemistry 28:11, pages 115496.
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Kartsev, Geronikaki, Bua, Nocentini, Petrou, Lichitsky, Frasinyuk, Leitans, Kazaks, Tars & Supuran. (2019) Extending the Inhibition Profiles of Coumarin-Based Compounds Against Human Carbonic Anhydrases: Synthesis, Biological, and In Silico Evaluation. Molecules 24:19, pages 3580.
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Ana Podolski-Renić, Jelena Dinić, Tijana Stanković, Mirna Jovanović, Amra Ramović, Aleksandrs Pustenko, Raivis Žalubovskis & Milica Pešić. (2019) Sulfocoumarins, specific carbonic anhydrase IX and XII inhibitors, interact with cancer multidrug resistant phenotype through pH regulation and reverse P-glycoprotein mediated resistance. European Journal of Pharmaceutical Sciences 138, pages 105012.
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Murat Bozdag, Giulio Poli, Andrea Angeli, Elena Lucarini, Tiziano Tuccinardi, Lorenzo Di Cesare Mannelli, Silvia Selleri, Carla Ghelardini, Jean-Yves Winum, Fabrizio Carta & Claudiu T. Supuran. (2019) N-aryl-N’-ureido-O-sulfamates: Potent and selective inhibitors of the human Carbonic Anhydrase VII isoform with neuropathic pain relieving properties. Bioorganic Chemistry 89, pages 103033.
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Claudiu T. Supuran. 2019. Therapeutic Application of Nitric Oxide in Cancer and Inflammatory Disorders. Therapeutic Application of Nitric Oxide in Cancer and Inflammatory Disorders
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Claudiu T. Supuran & Andrea Scozzafava. 2019. Carbonic Anhydrases. Carbonic Anhydrases
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Claudiu T. Supuran, Vincenzo Alterio, Anna Di Fiore, Katia D’ Ambrosio, Fabrizio Carta, Simona Maria Monti & Giuseppina De Simone. (2018) Inhibition of carbonic anhydrase IX targets primary tumors, metastases, and cancer stem cells: Three for the price of one. Medicinal Research Reviews 38:6, pages 1799-1836.
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Edita Čapkauskaitė, Audrius Zakšauskas, Virginijus Ruibys, Vaida Linkuvienė, Vaida Paketurytė, Marius Gedgaudas, Visvaldas Kairys & Daumantas Matulis. (2018) Benzimidazole design, synthesis, and docking to build selective carbonic anhydrase VA inhibitors. Bioorganic & Medicinal Chemistry 26:3, pages 675-687.
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Murat Bozdag, Ahmed Mahmoud Alafeefy, Abdul Malik Altamimi, Fabrizio Carta, Claudiu T. Supuran & Daniela Vullo. (2017) Synthesis of new 3-(2-mercapto-4-oxo-4H-quinazolin-3-yl)-benzenesulfonamides with strong inhibition properties against the tumor associated carbonic anhydrases IX and XII. Bioorganic & Medicinal Chemistry 25:10, pages 2782-2788.
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Fabrizio Carta, Alexander Birkmann, Tamara Pfaff, Helmut Buschmann, Wilfried Schwab, Holger Zimmermann, Alfonso Maresca & Claudiu T. Supuran. (2017) Lead Development of Thiazolylsulfonamides with Carbonic Anhydrase Inhibitory Action. Journal of Medicinal Chemistry 60:7, pages 3154-3164.
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Behnam Rasti, Mohsen Namazi, M. H. Karimi-Jafari & Jahan B. Ghasemi. (2017) Proteochemometric Modeling of the Interaction Space of Carbonic Anhydrase and its Inhibitors: An Assessment of Structure-based and Sequence-based Descriptors. Molecular Informatics 36:4, pages 1600102.
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Silvia Bua, Lorenzo Di Cesare Mannelli, Daniela Vullo, Carla Ghelardini, Gianluca Bartolucci, Andrea Scozzafava, Claudiu T. Supuran & Fabrizio Carta. (2017) Design and Synthesis of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs–CAIs) for the Treatment of Rheumatoid Arthritis. Journal of Medicinal Chemistry 60:3, pages 1159-1170.
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Daniela Vullo, Sonia Del Prete, Alessio Nocentini, Sameh M. Osman, Zeid AlOthman, Clemente Capasso, Murat Bozdag, Fabrizio Carta, Paola Gratteri & Claudiu T. Supuran. (2017) Dithiocarbamates effectively inhibit the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa. Bioorganic & Medicinal Chemistry 25:3, pages 1260-1265.
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Murat Bozdag, Ahmed Mahmoud Alafeefy, Abdul Malik Altamimi, Daniela Vullo, Fabrizio Carta & Claudiu T. Supuran. (2017) Coumarins and other fused bicyclic heterocycles with selective tumor-associated carbonic anhydrase isoforms inhibitory activity. Bioorganic & Medicinal Chemistry 25:2, pages 677-683.
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Behnam Rasti, Mohammad H. Karimi-Jafari & Jahan B. Ghasemi. (2016) Quantitative Characterization of the Interaction Space of the Mammalian Carbonic Anhydrase Isoforms I, II, VII, IX, XII, and XIV and their Inhibitors, Using the Proteochemometric Approach. Chemical Biology & Drug Design 88:3, pages 341-353.
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Daniela Vullo, Claudiu T. Supuran, Andrea Scozzafava, Giuseppina De Simone, Simona Maria Monti, Vincenzo Alterio & Fabrizio Carta. (2016) Kinetic and X-ray crystallographic investigations of substituted 2-thio-6-oxo-1,6-dihydropyrimidine–benzenesulfonamides acting as carbonic anhydrase inhibitors. Bioorganic & Medicinal Chemistry 24:16, pages 3643-3648.
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Claudiu T. Supuran. (2016) Structure and function of carbonic anhydrases. Biochemical Journal 473:14, pages 2023-2032.
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Nagwa M. Abdel Gawad, Noha H. Amin, Mohammed T. Elsaadi, Fatma M.M. Mohamed, Andrea Angeli, Viviana De Luca, Clemente Capasso & Claudiu T. Supuran. (2016) Synthesis of 4-(thiazol-2-ylamino)-benzenesulfonamides with carbonic anhydrase I, II and IX inhibitory activity and cytotoxic effects against breast cancer cell lines. Bioorganic & Medicinal Chemistry 24:13, pages 3043-3051.
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Daniela Vullo, Mariaconcetta Durante, Francesco Saverio Di Leva, Sandro Cosconati, Emanuela Masini, Andrea Scozzafava, Ettore Novellino, Claudiu T. Supuran & Fabrizio Carta. (2016) Monothiocarbamates Strongly Inhibit Carbonic Anhydrases in Vitro and Possess Intraocular Pressure Lowering Activity in an Animal Model of Glaucoma. Journal of Medicinal Chemistry 59:12, pages 5857-5867.
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Haydar Göksu, Meryem Topal, Ali Keskin, Mehmet S. Gültekin, Murat Çelik, İlhami Gülçin, Muhammet Tanc & Claudiu T. Supuran. (2016)
9,10-Dibromo-
N
-aryl-9,10-dihydro-9,10-[3,4]epipyrroloanthracene-12,14-diones: Synthesis and Investigation of Their Effects on Carbonic Anhydrase Isozymes I, II, IX, and XII
. Archiv der Pharmazie 349:6, pages 466-474.
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Suleyman Akocak, M. Raqibul Alam, Ahmed M. Shabana, Rajesh Kishore Kumar Sanku, Daniela Vullo, Harry Thompson, Erik R. Swenson, Claudiu T. Supuran & Marc A. Ilies. (2016) PEGylated Bis-Sulfonamide Carbonic Anhydrase Inhibitors Can Efficiently Control the Growth of Several Carbonic Anhydrase IX-Expressing Carcinomas. Journal of Medicinal Chemistry 59:10, pages 5077-5088.
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Ayşenur Eminoğlu, Daniela Vullo, Aycan Aşık, Dilşat Nigar Çolak, Sabriye Çanakçı, Ali Osman Beldüz & Claudiu T. Supuran. (2016) Sulfonamide inhibition studies of the β-carbonic anhydrase from the newly discovered bacterium Enterobacter sp. B13. Bioorganic & Medicinal Chemistry Letters 26:7, pages 1821-1826.
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Daniela Vullo, Sonia Del Prete, Viviana De Luca, Vincenzo Carginale, Marta Ferraroni, Nurcan Dedeoglu, Sameh M. Osman, Zeid AlOthman, Clemente Capasso & Claudiu T. Supuran. (2016) Anion inhibition studies of the β-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae. Bioorganic & Medicinal Chemistry Letters 26:5, pages 1406-1410.
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Sonia Del Prete, Daniela Vullo, Viviana De Luca, Vincenzo Carginale, Marta Ferraroni, Sameh M. Osman, Zeid AlOthman, Claudiu T. Supuran & Clemente Capasso. (2016) Sulfonamide inhibition studies of the β-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae. Bioorganic & Medicinal Chemistry 24:5, pages 1115-1120.
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Daniela Vullo, Viviana De Luca, Sonia Del Prete, Vincenzo Carginale, Andrea Scozzafava, Sameh M. Osman, Zeid AlOthman, Clemente Capasso & Claudiu T. Supuran. (2016) Sulfonamide inhibition studies of the γ-carbonic anhydrase from the Antarctic bacterium Colwellia psychrerythraea. Bioorganic & Medicinal Chemistry Letters 26:4, pages 1253-1259.
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Benedetta Cornelio, Marie Laronze-Cochard, Mariangela Ceruso, Marta Ferraroni, Graham A. RanceFabrizio Carta, Andrei N. KhlobystovAntonella Fontana, Claudiu T. Supuran & Janos Sapi. (2016) 4-Arylbenzenesulfonamides as Human Carbonic Anhydrase Inhibitors (hCAIs): Synthesis by Pd Nanocatalyst-Mediated Suzuki–Miyaura Reaction, Enzyme Inhibition, and X-ray Crystallographic Studies. Journal of Medicinal Chemistry 59:2, pages 721-732.
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Marta Ferraroni, Fabrizio Carta, Andrea Scozzafava & Claudiu T. Supuran. (2015) Thioxocoumarins Show an Alternative Carbonic Anhydrase Inhibition Mechanism Compared to Coumarins. Journal of Medicinal Chemistry 59:1, pages 462-473.
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Adel S. El-Azab, Alaa A.-M. Abdel-Aziz, Rezk R. Ayyad, Mariangela Ceruso & Claudiu T. Supuran. (2016) Inhibition of carbonic anhydrase isoforms I, II, IV, VII and XII with carboxylates and sulfonamides incorporating phthalimide/phthalic anhydride scaffolds. Bioorganic & Medicinal Chemistry 24:1, pages 20-25.
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Fabrizio Carta, Marta Ferraroni, Andrea Scozzafava & Claudiu T. Supuran. (2016) Fluorescent sulfonamide carbonic anhydrase inhibitors incorporating 1,2,3-triazole moieties: Kinetic and X-ray crystallographic studies. Bioorganic & Medicinal Chemistry 24:2, pages 104-112.
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Murat Bozdag, Ahmed M. Alafeefy, Daniela Vullo, Fabrizio Carta, Nurcan Dedeoglu, Abdul-Malek S. Al-Tamimi, Nabila A. Al-Jaber, Andrea Scozzafava & Claudiu T. Supuran. (2015) Benzenesulfonamides incorporating bulky aromatic/heterocyclic tails with potent carbonic anhydrase inhibitory activity. Bioorganic & Medicinal Chemistry 23:24, pages 7751-7764.
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Sonia Del Prete, Daniela Vullo, Sameh M. Osman, Zeid AlOthman, Clemente Capasso & Claudiu T. Supuran. (2015) Anion inhibition studies of the dandruff-producing fungus Malassezia globosa β-carbonic anhydrase MgCA. Bioorganic & Medicinal Chemistry Letters 25:22, pages 5194-5198.
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Viviana De Luca, Sonia Del Prete, Vincenzo Carginale, Daniela Vullo, Claudiu T. Supuran & Clemente Capasso. (2015) Cloning, characterization and anion inhibition studies of a γ-carbonic anhydrase from the Antarctic cyanobacterium Nostoc commune. Bioorganic & Medicinal Chemistry Letters 25:21, pages 4970-4975.
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Alfonso Maresca, Gulay Akyuz, Sameh M. Osman, Zeid AlOthman & Claudiu T. Supuran. (2015) Inhibition of mammalian carbonic anhydrase isoforms I–XIV with a series of phenolic acid esters. Bioorganic & Medicinal Chemistry 23:22, pages 7181-7188.
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Alessio Nocentini, Fabrizio Carta, Mariangela Ceruso, Gianluca Bartolucci & Claudiu T. Supuran. (2015) Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII. Bioorganic & Medicinal Chemistry 23:21, pages 6955-6966.
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İbrahim Esirden, Ramazan Ulus, Burak Aday, Muhammet Tanç, Claudiu T. Supuran & Muharrem Kaya. (2015) Synthesis of novel acridine bis-sulfonamides with effective inhibitory activity against the carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry 23:20, pages 6573-6580.
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Nurcan Dedeoglu, Viviana De Luca, Semra Isik, Hatice Yildirim, Feray Kockar, Clemente Capasso & Claudiu T. Supuran. (2015) Cloning, characterization and anion inhibition study of a β-class carbonic anhydrase from the caries producing pathogen Streptococcus mutans. Bioorganic & Medicinal Chemistry 23:13, pages 2995-3001.
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Nurcan Dedeoglu, Viviana DeLuca, Semra Isik, Hatice Yildirim, Feray Kockar, Clemente Capasso & Claudiu T. Supuran. (2015) Sulfonamide inhibition study of the β-class carbonic anhydrase from the caries producing pathogen Streptococcus mutans. Bioorganic & Medicinal Chemistry Letters 25:11, pages 2291-2297.
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Mustafa Durgun, Hasan Turkmen, Mariangela Ceruso & Claudiu T. Supuran. (2015) Synthesis of Schiff base derivatives of 4-(2-aminoethyl)-benzenesulfonamide with inhibitory activity against carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry Letters 25:11, pages 2377-2381.
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Aiga Grandane, Muhammet Tanc, Lorenzo Di Cesare Mannelli, Fabrizio Carta, Carla Ghelardini, Raivis Žalubovskis & Claudiu T. Supuran. (2015) 6-Substituted Sulfocoumarins Are Selective Carbonic Anhdydrase IX and XII Inhibitors with Significant Cytotoxicity against Colorectal Cancer Cells. Journal of Medicinal Chemistry 58:9, pages 3975-3983.
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Murat Bozdag, Fabrizio Carta, Daniela Vullo, Atilla Akdemir, Semra Isik, Cecilia Lanzi, Andrea Scozzafava, Emanuela Masini & Claudiu T. Supuran. (2015) Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma action. Bioorganic & Medicinal Chemistry 23:10, pages 2368-2376.
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Daniela Vullo, Viviana De Luca, Sonia Del Prete, Vincenzo Carginale, Andrea Scozzafava, Clemente Capasso & Claudiu T. Supuran. (2015) Sulfonamide inhibition studies of the γ-carbonic anhydrase from the Antarctic cyanobacterium Nostoc commune. Bioorganic & Medicinal Chemistry 23:8, pages 1728-1734.
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Aiga Grandane, Muhammet Tanc, Raivis Žalubovskis & Claudiu T. Supuran. (2015) Synthesis of 6-aryl-substituted sulfocoumarins and investigation of their carbonic anhydrase inhibitory action. Bioorganic & Medicinal Chemistry 23:7, pages 1430-1436.
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Murat Boztaş, Yasin Çetinkaya, Meryem Topal, İlhami Gülçin, Abdullah Menzek, Ertan Şahin, Muhammet Tanc & Claudiu T. Supuran. (2014) Synthesis and Carbonic Anhydrase Isoenzymes I, II, IX, and XII Inhibitory Effects of Dimethoxybromophenol Derivatives Incorporating Cyclopropane Moieties. Journal of Medicinal Chemistry 58:2, pages 640-650.
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Fulvio Ratto, Ewa Witort, Francesca Tatini, Sonia Centi, Lorenza Lazzeri, Fabrizio Carta, Matteo Lulli, Daniela Vullo, Franco Fusi, Claudiu T. Supuran, Andrea Scozzafava, Sergio Capaccioli & Roberto Pini. (2015) Plasmonic Particles that Hit Hypoxic Cells. Advanced Functional Materials 25:2, pages 316-323.
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Murat Bozdag, Marta Ferraroni, Fabrizio Carta, Daniela Vullo, Laura Lucarini, Elisabetta Orlandini, Armando Rossello, Elisa Nuti, Andrea Scozzafava, Emanuela Masini & Claudiu T. Supuran. (2014) Structural Insights on Carbonic Anhydrase Inhibitory Action, Isoform Selectivity, and Potency of Sulfonamides and Coumarins Incorporating Arylsulfonylureido Groups. Journal of Medicinal Chemistry 57:21, pages 9152-9167.
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Joanna Ombouma, Daniela Vullo, Claudiu T. Supuran & Jean-Yves Winum. (2014) Ferrier sulfamidoglycosylation of glycals catalyzed by nitrosonium tetrafluoroborate: Towards new carbonic anhydrase glycoinhibitors. Bioorganic & Medicinal Chemistry 22:22, pages 6353-6359.
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Busra Sarikaya, Mariangela Ceruso, Fabrizio Carta & Claudiu T. Supuran. (2014) Inhibition of carbonic anhydrase isoforms I, II, IX and XII with novel Schiff bases: Identification of selective inhibitors for the tumor-associated isoforms over the cytosolic ones. Bioorganic & Medicinal Chemistry 22:21, pages 5883-5890.
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Ahmed M. Alafeefy, Mariangela Ceruso, Abdul-Malek S. Al-Tamimi, Sonia Del Prete, Clemente Capasso & Claudiu T. Supuran. (2014) Quinazoline–sulfonamides with potent inhibitory activity against the α-carbonic anhydrase from Vibrio cholerae. Bioorganic & Medicinal Chemistry 22:19, pages 5133-5140.
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Sonia Del Prete, Daniela Vullo, Gillian M. Fisher, Katherine T. Andrews, Sally-Ann Poulsen, Clemente Capasso & Claudiu T. Supuran. (2014) Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum —The η-carbonic anhydrases. Bioorganic & Medicinal Chemistry Letters 24:18, pages 4389-4396.
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Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Andrea Scozzafava, Zeid Alothman, Claudiu T. Supuran & Clemente Capasso. (2014) Anion inhibition study of the β-class carbonic anhydrase (PgiCAb) from the oral pathogen Porphyromonas gingivalis. Bioorganic & Medicinal Chemistry Letters 24:18, pages 4402-4406.
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Aiga Grandane, Muhammet Tanc, Raivis Zalubovskis & Claudiu T. Supuran. (2014) 6-Triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrases IX and XII. Bioorganic & Medicinal Chemistry Letters 24:5, pages 1256-1260.
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Aiga Grandane, Muhammet Tanc, Raivis Zalubovskis & Claudiu T. Supuran. (2014) Synthesis of 6-tetrazolyl-substituted sulfocoumarins acting as highly potent and selective inhibitors of the tumor-associated carbonic anhydrase isoforms IX and XII. Bioorganic & Medicinal Chemistry 22:5, pages 1522-1528.
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Nihed Draoui, Olivier Schicke, Antony Fernandes, Xavier Drozak, Fady Nahra, Amélie Dumont, Jonathan Douxfils, Emmanuel Hermans, Jean-Michel Dogné, Romu Corbau, Arnaud Marchand, Patrick Chaltin, Pierre Sonveaux, Olivier Feron & Olivier Riant. (2013) Synthesis and pharmacological evaluation of carboxycoumarins as a new antitumor treatment targeting lactate transport in cancer cells. Bioorganic & Medicinal Chemistry 21:22, pages 7107-7117.
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