Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 22, Issue 1 (2007)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 22, Issue 1 (2007)

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Research Article

Article
Quantitative structure-activity relationships (QSARs) in inhibitors of various cytochromes P450: The importance of compound lipophilicity
David F. V. Lewis, Brian G. Lake & Maurice Dickins
Pages: 1-6
Published online: 20 Oct 2008
AbstractforQuantitative structure-activity relationships (QSARs) in inhibitors of various cytochromes P450: The importance of compound lipophilicity | Full Text | References | PDF (84.7 KB)
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Article
HQSAR study of β-ketoacyl‐acyl carrier protein synthase III (FabH) inhibitors
Ali Ashek, Amor A. San Juan & Seung J. Cho
Pages: 7-14
Published online: 04 Oct 2008
AbstractforHQSAR study of β-ketoacyl‐acyl carrier protein synthase III (FabH) inhibitors | Full Text | References | PDF (169.1 KB)
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Article
Quantitative structure-activity relationship study of benzylsulfanyl imidazoles as cytokine release inhibitors
P. Singh & B. K. Sharma
Pages: 15-21
Published online: 04 Oct 2008
AbstractforQuantitative structure-activity relationship study of benzylsulfanyl imidazoles as cytokine release inhibitors | Full Text | References | PDF (94.8 KB)
  • 286 Views
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Article
A quantitative structure-activity relationship study on matrix metalloproteinase inhibitors: Piperidine sulfonamide aryl hydroxamic acid analogs
S. Kumaran & S. P. Gupta
Pages: 23-27
Published online: 04 Oct 2008
AbstractforA quantitative structure-activity relationship study on matrix metalloproteinase inhibitors: Piperidine sulfonamide aryl hydroxamic acid analogs | Full Text | References | PDF (69.3 KB)
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Article
New inhibitors of fungal 17β-hydroxysteroid dehydrogenase based on the [1,5]-benzodiazepine scaffold
Matej Živec, Matej Sova, Mojca Brunskole, Roman Lenaršič, Tea Lanišnik Rižner & Stanislav Gobec
Pages: 29-36
Published online: 04 Oct 2008
AbstractforNew inhibitors of fungal 17β-hydroxysteroid dehydrogenase based on the [1,5]-benzodiazepine scaffold | Full Text | References | PDF (165.6 KB)
  • 587 Views
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Article
Molecular modifications of 2-arylidene-1-indanones leading to increased cytotoxic potencies
Hari N. Pati, Umashankar Das, Erik De Clercq, Jan Balzarini & Jonathan R. Dimmock
Pages: 37-42
Published online: 04 Oct 2008
AbstractforMolecular modifications of 2-arylidene-1-indanones leading to increased cytotoxic potencies | Full Text | References | PDF (118 KB)
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Article
Isolation and characterization of N98-1272 A, B and C, selective acetylcholinesterase inhibitors from metabolites of an actinomycete strain
Zhi-Hui Zheng, Yue-Sheng Dong, Hua Zhang, Xin-Hua Lu, Xiao Ren, Guiyu Zhao, Jian-Gong He & Shu-Yi Si
Pages: 43-49
Published online: 04 Oct 2008
AbstractforIsolation and characterization of N98-1272 A, B and C, selective acetylcholinesterase inhibitors from metabolites of an actinomycete strain | Full Text | References | PDF (267.6 KB)
  • 501 Views
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Article
Synthesis and in vitro anti-HIV activities of didanosine prodrugs
Dhrmarajan Sriram, Perumal Yogeeswari, Nagell Raveendra Babu & Purna Nagashree Kurre
Pages: 51-55
Published online: 04 Oct 2008
AbstractforSynthesis and in vitro anti-HIV activities of didanosine prodrugs | Full Text | References | PDF (82.4 KB)
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Article
Novel benzothiazolyl urea and thiourea derivatives with potential cytotoxic and antimicrobial activities
Hamdy M. Abdel-Rahman & Mohamed A. Morsy
Pages: 57-64
Published online: 04 Oct 2008
AbstractforNovel benzothiazolyl urea and thiourea derivatives with potential cytotoxic and antimicrobial activities | Full Text | References | PDF (652.4 KB)
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Article
Synthesis, characterization and antibacterial properties of some trivalent metal complexes with [(2-hydroxy-1-naphthaldehyde)-3-isatin]-bishydrazone
Balakrishnan Murukan & Kochukittan Mohanan
Pages: 65-70
Published online: 04 Oct 2008
AbstractforSynthesis, characterization and antibacterial properties of some trivalent metal complexes with [(2-hydroxy-1-naphthaldehyde)-3-isatin]-bishydrazone | Full Text | References | PDF (151.3 KB)
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Article
Leishmania amazonensis trypanothione reductase: Evaluation of the effect of glutathione analogs on parasite growth, infectivity and enzyme activity
Denise Barçante Castro-Pinto, Edson L. Silva Lima, Andrea S. Cunha, Marcelo Genestra, Rosa Maria De Léo, Fabiane Monteiro & Leonor L. Leon
Pages: 71-75
Published online: 04 Oct 2008
AbstractforLeishmania amazonensis trypanothione reductase: Evaluation of the effect of glutathione analogs on parasite growth, infectivity and enzyme activity | Full Text | References | PDF (119.9 KB)
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Article
Inhibition by L-aspartol adenylate of a nondiscriminating aspartyl-tRNA synthetase reveals differences between the interactions of its active site with tRNAAsp and tRNAAsn.
Dominic Bernard, Pierre-Marie Akochy, Stéphane Bernier, Olivier Fisette, Olivier Côté Brousseau, Robert Chênevert, Paul H. Roy & Jacques Lapointe
Pages: 77-82
Published online: 04 Oct 2008
AbstractforInhibition by L-aspartol adenylate of a nondiscriminating aspartyl-tRNA synthetase reveals differences between the interactions of its active site with tRNAAsp and tRNAAsn. | Full Text | References | PDF (136.1 KB)
  • 538 Views
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Article
Tyrosinase inhibitory effects and inhibition mechanisms of nobiletin and hesperidin from citrus peel crude extracts
Chongwei Zhang, Yanhua Lu, Lin Tao, Xinyi Tao, Xiaochun Su & Dongzhi Wei
Pages: 83-90
Published online: 04 Oct 2008
AbstractforTyrosinase inhibitory effects and inhibition mechanisms of nobiletin and hesperidin from citrus peel crude extracts | Full Text | References | PDF (388 KB)
  • 2344 Views
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Article
Tyrosinase inhibitory effects and inhibition mechanisms of nobiletin and hesperidin from citrus peel crude extracts
Chongwei Zhang, Yanhua Lu, Lin Tao, Xinyi Tao, Xiaochun Su & Dongzhi Wei
Pages: 91-98
Published online: 04 Oct 2008
AbstractforTyrosinase inhibitory effects and inhibition mechanisms of nobiletin and hesperidin from citrus peel crude extracts | Full Text | References | PDF (341.5 KB)
  • 3333 Views
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Article
Inhibitory effect on soybean lipoxygenase and docking studies of some secondary metabolites, isolated from Origanum vulgare L. ssp. hirtum
Catherine Koukoulitsa, Dimitra Hadjipavlou–Litina, George D. Geromichalos & Helen Skaltsa
Pages: 99-104
Published online: 04 Oct 2008
AbstractforInhibitory effect on soybean lipoxygenase and docking studies of some secondary metabolites, isolated from Origanum vulgare L. ssp. hirtum | Full Text | References | PDF (3 MB)
  • 842 Views
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Article
Inhibition of carbonyl reductase activity in pig heart by alkyl phenyl ketones
Yorishige Imamura, Rika Narumi & Hideaki Shimada
Pages: 105-109
Published online: 04 Oct 2008
AbstractforInhibition of carbonyl reductase activity in pig heart by alkyl phenyl ketones | Full Text | References | PDF (146 KB)
  • 748 Views
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Article
Identification of a single and non-essential cysteine residue in dextransucrase of Leuconostoc mesenteroides NRRL B-512F
Arun Goyal, D. P. Tyagi & Sarvagya S. Katiyar
Pages: 111-113
Published online: 04 Oct 2008
AbstractforIdentification of a single and non-essential cysteine residue in dextransucrase of Leuconostoc mesenteroides NRRL B-512F | Full Text | References | PDF (58.2 KB)
  • 314 Views
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Article
Purification and characterization of a trypsin inhibitor from seeds of Murraya koenigii
Chandan Shee & Ashwani K. Sharma
Pages: 115-120
Published online: 04 Oct 2008
AbstractforPurification and characterization of a trypsin inhibitor from seeds of Murraya koenigii | Full Text | References | PDF (161.5 KB)
  • 2329 Views
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Article
Arginine deiminases: Therapeutic tools in the etiology and pathogenesis of Alzheimer's disease
Short Communication
Cassandra Louw, Alon Gordon, Nicolette Johnston, Carolyn Mollatt, Graeme Bradley & Chris G. Whiteley
Pages: 121-126
Published online: 04 Oct 2008
AbstractforArginine deiminases: Therapeutic tools in the etiology and pathogenesis of Alzheimer's disease | Full Text | References | PDF (151.6 KB)
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