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Alessandro Bonardi, Seppo Parkkila & Claudiu T. Supuran. (2022) Inhibition studies of the protozoan α-carbonic anhydrase from Trypanosoma cruzi with phenols. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 2417-2422.
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Simone Giovannuzzi, Chad S. Hewitt, Alessio Nocentini, Clemente Capasso, Gabriele Costantino, Daniel P. Flaherty & Claudiu T. Supuran. (2022) Inhibition studies of bacterial α-carbonic anhydrases with phenols. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 666-671.
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Pulala Raghuveer Yadav, Syed Hussain Basha, Sadam D. V. Satyanarayana & Pavan Kumar Pindi. (2022) Microsecond simulation analysis of carbonic anhydrase – II in complex with (+)-cathechin revealed molecular interactions responsible for its amelioration effect on fluoride toxicity. Journal of Biomolecular Structure and Dynamics 40:16, pages 7469-7482.
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Birhanu Geta Meharie & Tewodros Agedew Tunta. (2020) Evaluation of Diuretic Activity and Phytochemical Contents of Aqueous Extract of the Shoot Apex of Podocarpus falcactus. Journal of Experimental Pharmacology 12, pages 629-641.
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Mikhail Krasavin, Raivis Žalubovskis, Aiga Grandāne, Ilona Domračeva, Petr Zhmurov & Claudiu T. Supuran. (2020) Sulfocoumarins as dual inhibitors of human carbonic anhydrase isoforms IX/XII and of human thioredoxin reductase. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 506-510.
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Claudiu T. Supuran. (2017) Advances in structure-based drug discovery of carbonic anhydrase inhibitors. Expert Opinion on Drug Discovery 12:1, pages 61-88.
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P. V. Sri Ramya, Srinivas Angapelly, Andrea Angeli, Chander Singh Digwal, Mohammed Arifuddin, Bathini Nagendra Babu, Claudiu T. Supuran & Ahmed Kamal. (2017) Discovery of curcumin inspired sulfonamide derivatives as a new class of carbonic anhydrase isoforms I, II, IX, and XII inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1274-1281.
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Alessio Nocentini, Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Fatmah A.S. Alasmary, Zeid AlOthman, Clemente Capasso, Fabrizio Carta, Paola Gratteri & Claudiu T. Supuran. (2017) Inhibition of the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa with monothiocarbamates. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1064-1070.
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Mikhail Krasavin, Mikhail Korsakov, Oksana Ronzhina, Tiziano Tuccinardi, Stanislav Kalinin, Muhammet Tanç & Claudiu T. Supuran. (2017) Primary mono- and bis-sulfonamides obtained via regiospecific sulfochlorination of N-arylpyrazoles: inhibition profile against a panel of human carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 920-934.
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Ercan Soydan, Ahmet Güler, Selim Bıyık, Murat Şentürk, Claudiu T. Supuran & Deniz Ekinci. (2017) Carbonic anhydrase from Apis mellifera: purification and inhibition by pesticides. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 47-50.
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Belma Zengin Kurt, Fatih Sönmez, Çiğdem Bilen, Adem Ergun, Nahit Gençer, Oktay Arslan & Mustafa Kucukislamoglu. (2016) Synthesis, antioxidant and carbonic anhydrase I and II inhibitory activities of novel sulphonamide-substituted coumarylthiazole derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 991-998.
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Claudiu T. Supuran, Stanislav Kalinin, Muhammet Tanç, Pakornwit Sarnpitak, Prashant Mujumdar, Sally-Ann Poulsen & Mikhail Krasavin. (2016) Isoform-selective inhibitory profile of 2-imidazoline-substituted benzene sulfonamides against a panel of human carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 31:sup1, pages 197-202.
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Claudiu T. Supuran. (2016) How many carbonic anhydrase inhibition mechanisms exist?. Journal of Enzyme Inhibition and Medicinal Chemistry 31:3, pages 345-360.
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Ramin Ekhteiari Salmas, Murat Senturk, Mine Yurtsever & Serdar Durdagi. (2016) Discovering novel carbonic anhydrase type IX (CA IX) inhibitors from seven million compounds using virtual screening and in vitro analysis. Journal of Enzyme Inhibition and Medicinal Chemistry 31:3, pages 425-433.
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Erdem Aslan, Caglar Guler & Sevki Adem. (2016) In vitro effects of some flavonoids and phenolic acids on human pyruvate kinase isoenzyme M2. Journal of Enzyme Inhibition and Medicinal Chemistry 31:2, pages 314-317.
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Murat Bozdag, Fabrizio Carta, Daniela Vullo, Semra Isik, Zeid AlOthman, Sameh M. Osman, Andrea Scozzafava & Claudiu T. Supuran. (2016) Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase. Journal of Enzyme Inhibition and Medicinal Chemistry 31:1, pages 132-136.
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Namrata Singasane, Prashant S. Kharkar, Mariangela Ceruso, Claudiu T. Supuran & Mrunmayee P. Toraskar. (2015) Inhibition of carbonic anhydrase isoforms I, II, IX and XII with Schiff’s bases incorporating iminoureido moieties. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 901-907.
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Mehmet Arslan, Murat Şentürk, İsmail Fidan, Oktay Talaz, Deniz Ekinci, Sedat Coşgun & Claudiu T. Supuran. (2015) Synthesis of 3,4-dihydroxypyrrolidine-2,5-dione and 3,5-dihydroxybenzoic acid derivatives and evaluation of the carbonic anhydrase I and II inhibition. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 896-900.
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Narasimha Rao Uda, Volker Seibert, Frank Stenner-Liewen, Philipp Müller, Petra Herzig, Gabor Gondi, Reinhard Zeidler, Marc van Dijk, Alfred Zippelius & Christoph Renner. (2015) Esterase activity of carbonic anhydrases serves as surrogate for selecting antibodies blocking hydratase activity. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 955-960.
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Daniela Vullo, Semra Isik, Murat Bozdag, Fabrizio Carta & Claudiu T. Supuran. (2015) 7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring. Journal of Enzyme Inhibition and Medicinal Chemistry 30:5, pages 773-777.
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Claudiu T Supuran. (2015) Nanoparticles for controlled release of anti-biofilm agents WO2014130994 (A1): a patent evaluation. Expert Opinion on Therapeutic Patents 25:8, pages 945-948.
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Ahmed M. Alafeefy, Mariangela Ceruso, Abdul-Malek S. Al-Tamimi, Sonia Del Prete, Claudiu T. Supuran & Clemente Capasso. (2015) Inhibition studies of quinazoline-sulfonamide derivatives against the γ-CA (PgiCA) from the pathogenic bacterium, Porphyromonas gingivalis. Journal of Enzyme Inhibition and Medicinal Chemistry 30:4, pages 592-596.
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Alaa A-M. Abdel-Aziz, Adel S. El-Azab, Deniz Ekinci, Murat Şentürk & Claudiu T. Supuran. (2015) Investigation of arenesulfonyl-2-imidazolidinones as potent carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 30:1, pages 81-84.
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Neslihan Korkmaz, Oday A. Obaidi, Murat Senturk, Demet Astley, Deniz Ekinci & Claudiu T. Supuran. (2015) Synthesis and biological activity of novel thiourea derivatives as carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 30:1, pages 75-80.
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Giuseppina De Simone, Vincenzo Alterio & Claudiu T Supuran. (2013) Exploiting the hydrophobic and hydrophilic binding sites for designing carbonic anhydrase inhibitors. Expert Opinion on Drug Discovery 8:7, pages 793-810.
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Grażyna Kowalska, Salim Bouchentouf, Radosław Kowalski, Jakub Wyrostek, Urszula Pankiewicz, Artur Mazurek, Monika Sujka & Marzena Włodarczyk-Stasiak. (2022) The hop cones (Humulus lupulus L.): Chemical composition, antioxidant properties and molecular docking simulations. Journal of Herbal Medicine 33, pages 100566.
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Atukuri Dorababu. (2021) Pharmacological report of recently designed multifunctional coumarin and coumarin–heterocycle derivatives. Archiv der Pharmazie 355:2, pages 2100345.
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Eva Havránková, Vladimír Garaj, Šárka Mascaretti, Andrea Angeli, Zuzana Soldánová, Miroslav Kemka, Jozef Motyčka, Marie Brázdová, Jozef Csöllei, Josef Jampílek & Claudiu T. Supuran. (2021) Novel 1,3,5-Triazinyl Aminobenzenesulfonamides Incorporating Aminoalcohol, Aminochalcone and Aminostilbene Structural Motifs as Potent Anti-VRE Agents, and Carbonic Anhydrases I, II, VII, IX, and XII Inhibitors. International Journal of Molecular Sciences 23:1, pages 231.
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Giang T. H. Nguyen, Jack L. Bennett, Sherrie Liu, Sarah E. Hancock, Daniel L. Winter, Dominic J. Glover & William A. Donald. (2021) Multiplexed Screening of Thousands of Natural Products for Protein–Ligand Binding in Native Mass Spectrometry. Journal of the American Chemical Society 143:50, pages 21379-21387.
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María Pérez-Jiménez, Carolina Muñoz-González & María Ángeles Pozo-Bayón. (2021) Specificity of Saliva Esterases by Wine Carboxylic Esters and Inhibition by Wine Phenolic Compounds Under Simulated Oral Conditions. Frontiers in Nutrition 8.
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Yang Zhou, Ya-Jiao Wu, Lei Wang, Juan Han, Jia-Cong Wu, Chun-Mei Li & Yun Wang. (2021) Natural deep eutectic solvents as green and biocompatible reaction medium for carbonic anhydrase catalysis. International Journal of Biological Macromolecules 190, pages 206-213.
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Azizah M. Malebari, Tarek S. Ibrahim, Ibrahim M. Salem, Ismail Salama, Ahdab N. Khayyat, Samia M. Mostafa, Osama I. El-Sabbagh & Khaled M. Darwish. (2020) The Anticancer Activity for the Bumetanide-Based Analogs via Targeting the Tumor-Associated Membrane-Bound Human Carbonic Anhydrase-IX Enzyme. Pharmaceuticals 13:9, pages 252.
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Muhammad Imran, Ahmad Irfan, Muhammad Ibrahim, Mohammed A. Assiri, Noreen Khalid, Sami Ullah & Abdullah G. Al-Sehemi. (2020) Carbonic anhydrase and cholinesterase inhibitory activities of isolated flavonoids from Oxalis corniculata L. and their first-principles investigations. Industrial Crops and Products 148, pages 112285.
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Arora, Sharma & Tollefsbol. (2019) Combinatorial Epigenetics Impact of Polyphenols and Phytochemicals in Cancer Prevention and Therapy. International Journal of Molecular Sciences 20:18, pages 4567.
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Saghafi, Taheri, Parkkila & Emameh. (2019) Phytochemicals as Modulators of Long Non-Coding RNAs and Inhibitors of Cancer-Related Carbonic Anhydrases. International Journal of Molecular Sciences 20:12, pages 2939.
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Antonella Di Pizio, Yaron Ben Shoshan-Galeczki, John E. Hayes & Masha Y. Niv. (2019) Bitter and sweet tasting molecules: It's complicated. Neuroscience Letters 700, pages 56-63.
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Mikhail Krasavin, Anton Shetnev, Sergey Baykov, Stanislav Kalinin, Alessio Nocentini, Vladimir Sharoyko, Giulio Poli, Tiziano Tuccinardi, Mikhail Korsakov, Tatiana B. Tennikova & Claudiu T. Supuran. (2019) Pyridazinone-substituted benzenesulfonamides display potent inhibition of membrane-bound human carbonic anhydrase IX and promising antiproliferative activity against cancer cell lines. European Journal of Medicinal Chemistry 168, pages 301-314.
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Mikhail Krasavin, Anton Shetnev, Tatyana Sharonova, Sergey Baykov, Stanislav Kalinin, Alessio Nocentini, Vladimir Sharoyko, Giulio Poli, Tiziano Tuccinardi, Sofia Presnukhina, Tatiana B. Tennikova & Claudiu T. Supuran. (2019) Continued exploration of 1,2,4-oxadiazole periphery for carbonic anhydrase-targeting primary arene sulfonamides: Discovery of subnanomolar inhibitors of membrane-bound hCA IX isoform that selectively kill cancer cells in hypoxic environment. European Journal of Medicinal Chemistry 164, pages 92-105.
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Peter Mikuš, Dominika Krajčiová, Mária Mikulová, Branislav Horváth, Daniel Pecher, Vladimír Garaj, Silvia Bua, Andrea Angeli & Claudiu T. Supuran. (2018) Novel sulfonamides incorporating 1,3,5-triazine and amino acid structural motifs as inhibitors of the physiological carbonic anhydrase isozymes I, II and IV and tumor-associated isozyme IX. Bioorganic Chemistry 81, pages 241-252.
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Alexander Sapegin, Stanislav Kalinin, Andrea Angeli, Claudiu T. Supuran & Mikhail Krasavin. (2018) Unprotected primary sulfonamide group facilitates ring-forming cascade en route to polycyclic [1,4]oxazepine-based carbonic anhydrase inhibitors. Bioorganic Chemistry 76, pages 140-146.
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Mikhail Krasavin, Anton Shetnev, Tatyana Sharonova, Sergey Baykov, Tiziano Tuccinardi, Stanislav Kalinin, Andrea Angeli & Claudiu T. Supuran. (2018) Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1,2,4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic hCA II and membrane-bound hCA IX isoforms. Bioorganic Chemistry 76, pages 88-97.
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Abdur Rauf, Muslim Raza, Muhammad Saleem, Ufuk Ozgen, Esen Sezen Karaoglan, Gulin Renda, Erhan Palaska & Ilkay Erdogan Orhan. (2017)
Carbonic Anhydrase and Urease Inhibitory Potential of Various Plant Phenolics Using
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Murat Bozdag, Ahmed Mahmoud Alafeefy, Abdul Malik Altamimi, Fabrizio Carta, Claudiu T. Supuran & Daniela Vullo. (2017) Synthesis of new 3-(2-mercapto-4-oxo-4H-quinazolin-3-yl)-benzenesulfonamides with strong inhibition properties against the tumor associated carbonic anhydrases IX and XII. Bioorganic & Medicinal Chemistry 25:10, pages 2782-2788.
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Sajjad Esmaeili, Mohammad Reza Ashrafi-Kooshk, Hadi Adibi & Reza Khodarahmi. (2017) Captopril/enalapril inhibit promiscuous esterase activity of carbonic anhydrase at micromolar concentrations: An in vitro study. Chemico-Biological Interactions 265, pages 24-35.
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Mikhail Krasavin, Mikhail Korsakov, Zhanna Zvonaryova, Evgenii Semyonychev, Tiziano Tuccinardi, Stanislav Kalinin, Muhammet Tanç & Claudiu T. Supuran. (2017) Human carbonic anhydrase inhibitory profile of mono- and bis-sulfonamides synthesized via a direct sulfochlorination of 3- and 4-(hetero)arylisoxazol-5-amine scaffolds. Bioorganic & Medicinal Chemistry 25:6, pages 1914-1925.
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Yann Le Duc, Erol Licsandru, Daniela Vullo, Mihail Barboiu & Claudiu T. Supuran. (2017) Carbonic anhydrases activation with 3-amino-1H-1,2,4-triazole-1-carboxamides: Discovery of subnanomolar isoform II activators. Bioorganic & Medicinal Chemistry 25:5, pages 1681-1686.
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Rajiv Kumar, Silvia Bua, Sita Ram, Sonia Del Prete, Clemente Capasso, Claudiu T. Supuran & Pawan K. Sharma. (2017) Benzenesulfonamide bearing imidazothiadiazole and thiazolotriazole scaffolds as potent tumor associated human carbonic anhydrase IX and XII inhibitors. Bioorganic & Medicinal Chemistry 25:3, pages 1286-1293.
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Daniela Vullo, Sonia Del Prete, Alessio Nocentini, Sameh M. Osman, Zeid AlOthman, Clemente Capasso, Murat Bozdag, Fabrizio Carta, Paola Gratteri & Claudiu T. Supuran. (2017) Dithiocarbamates effectively inhibit the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa. Bioorganic & Medicinal Chemistry 25:3, pages 1260-1265.
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Murat Bozdag, Ahmed Mahmoud Alafeefy, Abdul Malik Altamimi, Daniela Vullo, Fabrizio Carta & Claudiu T. Supuran. (2017) Coumarins and other fused bicyclic heterocycles with selective tumor-associated carbonic anhydrase isoforms inhibitory activity. Bioorganic & Medicinal Chemistry 25:2, pages 677-683.
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Anastasia Karioti, Fabrizio Carta & Claudiu Supuran. (2016) Phenols and Polyphenols as Carbonic Anhydrase Inhibitors. Molecules 21:12, pages 1649.
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Behnam Rasti, Mohammad H. Karimi-Jafari & Jahan B. Ghasemi. (2016) Quantitative Characterization of the Interaction Space of the Mammalian Carbonic Anhydrase Isoforms I, II, VII, IX, XII, and XIV and their Inhibitors, Using the Proteochemometric Approach. Chemical Biology & Drug Design 88:3, pages 341-353.
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Alessio Nocentini, Daniela Vullo, Gianluca Bartolucci & Claudiu T. Supuran. (2016) N-Nitrosulfonamides: A new chemotype for carbonic anhydrase inhibition. Bioorganic & Medicinal Chemistry 24:16, pages 3612-3617.
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Vito Coviello, Beatrice Marchi, Stefania Sartini, Luca Quattrini, Anna Maria Marini, Francesca Simorini, Sabrina Taliani, Silvia Salerno, Paola Orlandi, Anna Fioravanti, Teresa Di Desidero, Daniela Vullo, Federico Da Settimo, Claudiu T. Supuran, Guido Bocci & Concettina La Motta. (2016) 1,2-Benzisothiazole Derivatives Bearing 4-, 5-, or 6-Alkyl/arylcarboxamide Moieties Inhibit Carbonic Anhydrase Isoform IX (CAIX) and Cell Proliferation under Hypoxic Conditions. Journal of Medicinal Chemistry 59:13, pages 6547-6552.
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Giosuè Costa, Maria Concetta Gidaro, Daniela Vullo, Claudiu T. Supuran & Stefano Alcaro. (2016) Active Components of Essential Oils as Anti-Obesity Potential Drugs Investigated by in Silico Techniques. Journal of Agricultural and Food Chemistry 64:26, pages 5295-5300.
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Daniela Vullo, Sonia Del Prete, Viviana De Luca, Vincenzo Carginale, Marta Ferraroni, Nurcan Dedeoglu, Sameh M. Osman, Zeid AlOthman, Clemente Capasso & Claudiu T. Supuran. (2016) Anion inhibition studies of the β-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae. Bioorganic & Medicinal Chemistry Letters 26:5, pages 1406-1410.
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Ahmed M. Alafeefy, Fabrizio Carta, Mariangela Ceruso, Abdul-Malek S. Al-Tamimi, Abdulla A. Al-Kahtani & Claudiu T. Supuran. (2016) Development of 3-(4-aminosulphonyl)-phenyl-2-mercapto-3H-quinazolin-4-ones as inhibitors of carbonic anhydrase isoforms involved in tumorigenesis and glaucoma. Bioorganic & Medicinal Chemistry 24:6, pages 1402-1407.
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Mustafa Durgun, Hasan Turkmen, Mariangela Ceruso & Claudiu T. Supuran. (2016) Synthesis of 4-sulfamoylphenyl-benzylamine derivatives with inhibitory activity against human carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry 24:5, pages 982-988.
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Elisabetta Barresi, Silvia Salerno, Anna Maria Marini, Sabrina Taliani, Concettina La Motta, Francesca Simorini, Federico Da Settimo, Daniela Vullo & Claudiu T. Supuran. (2016) Sulfonamides incorporating heteropolycyclic scaffolds show potent inhibitory action against carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry 24:4, pages 921-927.
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Maria Luisa Villalba, Pablo Palestro, Mariangela Ceruso, Jose L. Gonzalez Funes, Alan Talevi, Luis Bruno Blanch, Claudiu T. Supuran & Luciana Gavernet. (2016) Sulfamide derivatives with selective carbonic anhydrase VII inhibitory action. Bioorganic & Medicinal Chemistry 24:4, pages 894-901.
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Ylenia Cau, Mattia Mori, Claudiu T. Supuran & Maurizio Botta. (2016) Mycobacterial carbonic anhydrase inhibition with phenolic acids and esters: kinetic and computational investigations. Organic & Biomolecular Chemistry 14:35, pages 8322-8330.
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Daniela Vullo, Avni Bhatt, Brian P. Mahon, Robert McKenna & Claudiu T. Supuran. (2016) Sulfonamide inhibition studies of the α-carbonic anhydrase from the gammaproteobacterium Thiomicrospira crunogena XCL-2, TcruCA. Bioorganic & Medicinal Chemistry Letters 26:2, pages 401-405.
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Adel S. El-Azab, Alaa A.-M. Abdel-Aziz, Rezk R. Ayyad, Mariangela Ceruso & Claudiu T. Supuran. (2016) Inhibition of carbonic anhydrase isoforms I, II, IV, VII and XII with carboxylates and sulfonamides incorporating phthalimide/phthalic anhydride scaffolds. Bioorganic & Medicinal Chemistry 24:1, pages 20-25.
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Alessandra Cincinelli, Tania Martellini, Daniela Vullo & Claudiu T. Supuran. (2015) Anion and sulfonamide inhibition studies of an α-carbonic anhydrase from the Antarctic hemoglobinless fish Chionodraco hamatus. Bioorganic & Medicinal Chemistry Letters 25:23, pages 5485-5489.
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Murat Bozdag, Ahmed M. Alafeefy, Daniela Vullo, Fabrizio Carta, Nurcan Dedeoglu, Abdul-Malek S. Al-Tamimi, Nabila A. Al-Jaber, Andrea Scozzafava & Claudiu T. Supuran. (2015) Benzenesulfonamides incorporating bulky aromatic/heterocyclic tails with potent carbonic anhydrase inhibitory activity. Bioorganic & Medicinal Chemistry 23:24, pages 7751-7764.
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Sonia Del Prete, Daniela Vullo, Sameh M. Osman, Zeid AlOthman, Clemente Capasso & Claudiu T. Supuran. (2015) Anion inhibition studies of the dandruff-producing fungus Malassezia globosa β-carbonic anhydrase MgCA. Bioorganic & Medicinal Chemistry Letters 25:22, pages 5194-5198.
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Viviana De Luca, Sonia Del Prete, Vincenzo Carginale, Daniela Vullo, Claudiu T. Supuran & Clemente Capasso. (2015) Cloning, characterization and anion inhibition studies of a γ-carbonic anhydrase from the Antarctic cyanobacterium Nostoc commune. Bioorganic & Medicinal Chemistry Letters 25:21, pages 4970-4975.
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Anastasia Karioti, Mariangela Ceruso, Fabrizio Carta, Anna-Rita Bilia & Claudiu T. Supuran. (2015) New natural product carbonic anhydrase inhibitors incorporating phenol moieties. Bioorganic & Medicinal Chemistry 23:22, pages 7219-7225.
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Alfonso Maresca, Gulay Akyuz, Sameh M. Osman, Zeid AlOthman & Claudiu T. Supuran. (2015) Inhibition of mammalian carbonic anhydrase isoforms I–XIV with a series of phenolic acid esters. Bioorganic & Medicinal Chemistry 23:22, pages 7181-7188.
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Fabrizio Carta, Sameh M. Osman, Daniela Vullo, Zeid AlOthman, Sonia Del Prete, Clemente Capasso & Claudiu T. Supuran. (2015) Poly(amidoamine) dendrimers show carbonic anhydrase inhibitory activity against α-, β-, γ- and η-class enzymes. Bioorganic & Medicinal Chemistry 23:21, pages 6794-6798.
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Alessio Nocentini, Fabrizio Carta, Mariangela Ceruso, Gianluca Bartolucci & Claudiu T. Supuran. (2015) Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII. Bioorganic & Medicinal Chemistry 23:21, pages 6955-6966.
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Cenzo Congiu, Valentina Onnis, Alessandro Deplano, Gianfranco Balboni, Nurcan Dedeoglu & Claudiu T. Supuran. (2015) Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity. Bioorganic & Medicinal Chemistry Letters 25:18, pages 3850-3853.
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Cenzo Congiu, Valentina Onnis, Alessandro Deplano, Gianfranco Balboni, Mariangela Ceruso & Claudiu T. Supuran. (2015) Synthesis and carbonic anhydrase I, II, IX and XII inhibitory activity of sulfamates incorporating piperazinyl-ureido moieties. Bioorganic & Medicinal Chemistry 23:17, pages 5619-5625.
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Mikhail Krasavin, Mikhail Korsakov, Mikhail Dorogov, Tiziano Tuccinardi, Nurcan Dedeoglu & Claudiu T. Supuran. (2015) Probing the ‘bipolar’ nature of the carbonic anhydrase active site: Aromatic sulfonamides containing 1,3-oxazol-5-yl moiety as picomolar inhibitors of cytosolic CA I and CA II isoforms. European Journal of Medicinal Chemistry 101, pages 334-347.
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Murat Güney, Hüseyin Çavdar, Murat Şentürk & Deniz Ekinci. (2015) Synthesis and carbonic anhydrase inhibitory properties of novel uracil derivatives. Bioorganic & Medicinal Chemistry Letters 25:16, pages 3261-3263.
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Mariangela Ceruso, Fabrizio Carta, Sameh M. Osman, Zeid Alothman, Simona Maria Monti & Claudiu T. Supuran. (2015) Inhibition studies of bacterial, fungal and protozoan β-class carbonic anhydrases with Schiff bases incorporating sulfonamide moieties. Bioorganic & Medicinal Chemistry 23:15, pages 4181-4187.
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Diaa A. Ibrahim, Deena S. Lasheen, Maysoun Y. Zaky, Amany W. Ibrahim, Daniela Vullo, Mariangela Ceruso, Claudiu T. Supuran & Dalal A. Abou El Ella. (2015) Design and synthesis of benzothiazole-6-sulfonamides acting as highly potent inhibitors of carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry 23:15, pages 4989-4999.
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Nurcan Dedeoglu, Viviana De Luca, Semra Isik, Hatice Yildirim, Feray Kockar, Clemente Capasso & Claudiu T. Supuran. (2015) Cloning, characterization and anion inhibition study of a β-class carbonic anhydrase from the caries producing pathogen Streptococcus mutans. Bioorganic & Medicinal Chemistry 23:13, pages 2995-3001.
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Nurcan Dedeoglu, Viviana DeLuca, Semra Isik, Hatice Yildirim, Feray Kockar, Clemente Capasso & Claudiu T. Supuran. (2015) Sulfonamide inhibition study of the β-class carbonic anhydrase from the caries producing pathogen Streptococcus mutans. Bioorganic & Medicinal Chemistry Letters 25:11, pages 2291-2297.
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Murat Bozdag, Fabrizio Carta, Daniela Vullo, Atilla Akdemir, Semra Isik, Cecilia Lanzi, Andrea Scozzafava, Emanuela Masini & Claudiu T. Supuran. (2015) Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma action. Bioorganic & Medicinal Chemistry 23:10, pages 2368-2376.
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Daniela Vullo, Viviana De Luca, Sonia Del Prete, Vincenzo Carginale, Andrea Scozzafava, Clemente Capasso & Claudiu T. Supuran. (2015) Sulfonamide inhibition studies of the γ-carbonic anhydrase from the Antarctic cyanobacterium Nostoc commune. Bioorganic & Medicinal Chemistry 23:8, pages 1728-1734.
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Aiga Grandane, Muhammet Tanc, Raivis Žalubovskis & Claudiu T. Supuran. (2015) Synthesis of 6-aryl-substituted sulfocoumarins and investigation of their carbonic anhydrase inhibitory action. Bioorganic & Medicinal Chemistry 23:7, pages 1430-1436.
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Alaa A.-M. Abdel-Aziz, Adel S. El-Azab, Mariangela Ceruso & Claudiu T. Supuran. (2014) Carbonic anhydrase inhibitory activity of sulfonamides and carboxylic acids incorporating cyclic imide scaffolds. Bioorganic & Medicinal Chemistry Letters 24:22, pages 5185-5189.
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Busra Sarikaya, Mariangela Ceruso, Fabrizio Carta & Claudiu T. Supuran. (2014) Inhibition of carbonic anhydrase isoforms I, II, IX and XII with novel Schiff bases: Identification of selective inhibitors for the tumor-associated isoforms over the cytosolic ones. Bioorganic & Medicinal Chemistry 22:21, pages 5883-5890.
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Ahmed M. Alafeefy, Mariangela Ceruso, Abdul-Malek S. Al-Tamimi, Sonia Del Prete, Clemente Capasso & Claudiu T. Supuran. (2014) Quinazoline–sulfonamides with potent inhibitory activity against the α-carbonic anhydrase from Vibrio cholerae. Bioorganic & Medicinal Chemistry 22:19, pages 5133-5140.
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Sonia Del Prete, Daniela Vullo, Gillian M. Fisher, Katherine T. Andrews, Sally-Ann Poulsen, Clemente Capasso & Claudiu T. Supuran. (2014) Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum —The η-carbonic anhydrases. Bioorganic & Medicinal Chemistry Letters 24:18, pages 4389-4396.
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Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Andrea Scozzafava, Zeid Alothman, Claudiu T. Supuran & Clemente Capasso. (2014) Anion inhibition study of the β-class carbonic anhydrase (PgiCAb) from the oral pathogen Porphyromonas gingivalis. Bioorganic & Medicinal Chemistry Letters 24:18, pages 4402-4406.
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