Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 21, Issue 6 (2006)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 21, Issue 6 (2006)

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Research Article

Article
Deriving the rate equations for product inhibition patterns in bisubstrate enzyme reactions
Vladimir Leskovac, Svetlana Trivić, Draginja Peričin & Julijan Kandrač
Pages: 617-634
Published online: 04 Oct 2008
AbstractforDeriving the rate equations for product inhibition patterns in bisubstrate enzyme reactions | Full Text | References | PDF (250.8 KB)
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Article
Competitive and uncompetitive inhibitors simultaneously acting on an autocatalytic zymogen activation reaction
R. Varón, M. A. Minaya-Pacheco, F. García-Molina, E. Arribas, E. Arias, J. Masiá & F. García-Sevilla
Pages: 635-645
Published online: 04 Oct 2008
AbstractforCompetitive and uncompetitive inhibitors simultaneously acting on an autocatalytic zymogen activation reaction | Full Text | References | PDF (414.5 KB)
  • 734 Views
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Article
Modeling of acetylcholinesterase inhibition by tacrine analogues using Bayesian-regularized Genetic Neural Networks and ensemble averaging
Michael Fernández, M Carmo Carreiras, José L Marco & Julio Caballero
Pages: 647-661
Published online: 04 Oct 2008
AbstractforModeling of acetylcholinesterase inhibition by tacrine analogues using Bayesian-regularized Genetic Neural Networks and ensemble averaging | Full Text | References | PDF (276.1 KB)
  • 429 Views
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Article
Potency of new structurally different oximes to reactivate cyclosarin-inhibited human brain acetylcholinesterases
Kamil Kuca, Jiri Cabal, Daniel Jun, Jiri Bajgar & Martina Hrabinova
Pages: 663-666
Published online: 04 Oct 2008
AbstractforPotency of new structurally different oximes to reactivate cyclosarin-inhibited human brain acetylcholinesterases | Full Text | References | PDF (102.8 KB)
  • 448 Views
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Article
N, N –Disubstituted piperazines and homopiperazines: Synthesis and affinities at α4β2* and α7* neuronal nicotinic acetylcholine receptors
JIANHONG CHEN, AGRIPINA G. DEACIUC, LINDA P. DWOSKIN, PETER A. CROOKS & DONGLU BAI
Pages: 667-680
Published online: 04 Oct 2008
AbstractforN, N –Disubstituted piperazines and homopiperazines: Synthesis and affinities at α4β2* and α7* neuronal nicotinic acetylcholine receptors | Full Text | References | PDF (380.9 KB)
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Article
Design, synthesis and pharmacological screening of a series of N1-(substituted)aryl-5,7-dimethyl-2-(substituted)pyrido(2,3-d)pyrimidin-4(3H)-ones as potential histamine H1-receptor antagonists
Bhanubhai N. Suhagia, Mahesh T. Chhabria & Ashlesha G. Makwana
Pages: 681-691
Published online: 04 Oct 2008
AbstractforDesign, synthesis and pharmacological screening of a series of N1-(substituted)aryl-5,7-dimethyl-2-(substituted)pyrido(2,3-d)pyrimidin-4(3H)-ones as potential histamine H1-receptor antagonists | Full Text | References | PDF (143.2 KB)
  • 599 Views
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Article
Synthesis and evaluation of (S)-2-ethoxy-3-phenylpropanoic acid derivatives as insulin-sensitizing agents
Xiaohua Cai, Bing Xie & Hui Guo
Pages: 693-696
Published online: 04 Oct 2008
AbstractforSynthesis and evaluation of (S)-2-ethoxy-3-phenylpropanoic acid derivatives as insulin-sensitizing agents | Full Text | References | PDF (100.9 KB)
  • 268 Views
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Article
Inhibition of jack bean urease by p-benzoquinone: elucidation of the role of thiols and reversibility of the process
Mirosława Kot
Pages: 697-701
Published online: 04 Oct 2008
AbstractforInhibition of jack bean urease by p-benzoquinone: elucidation of the role of thiols and reversibility of the process | Full Text | References | PDF (112.9 KB)
  • 681 Views
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Article
New natural cholinesterase inhibiting and calcium channel blocking quinoline alkaloids
Atta-ur -Rahman, Asaad Khalid, Nighat Sultana, M. Nabeel Ghayur, M. Ahmed Mesaik, M. Riaz Khan, Anwar H. Gilani & M. Iqbal Choudhary
Pages: 703-710
Published online: 04 Oct 2008
AbstractforNew natural cholinesterase inhibiting and calcium channel blocking quinoline alkaloids | Full Text | References | PDF (230.2 KB)
  • 1037 Views
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Article
The inhibitory effect of benzenethiol on the cresolase and catecholase activities of mushroom tyrosinase
A. A. Saboury, S. Zolghadri, K. Haghbeen & A. A. Moosavi-Movahedi
Pages: 711-717
Published online: 04 Oct 2008
AbstractforThe inhibitory effect of benzenethiol on the cresolase and catecholase activities of mushroom tyrosinase | Full Text | References | PDF (216.8 KB)
  • 816 Views
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Article
Phenolic extracts from various Algerian plants as strong inhibitors of porcine liver carboxylesterase
A. Djeridane, M. Yousfi, B. Nadjemi, S. Maamri, F. Djireb & P. Stocker
Pages: 719-726
Published online: 04 Oct 2008
AbstractforPhenolic extracts from various Algerian plants as strong inhibitors of porcine liver carboxylesterase | Full Text | References | PDF (146.8 KB)
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Article
The kinetics of inhibition of Vigna catjang cotyledon and buffalo liver arginase by L-proline and branched-chain amino acids
Snehal Dabir, Pankaj Dabir & Baburao Somvanshi
Pages: 727-731
Published online: 04 Oct 2008
AbstractforThe kinetics of inhibition of Vigna catjang cotyledon and buffalo liver arginase by L-proline and branched-chain amino acids | Full Text | References | PDF (165.9 KB)
  • 411 Views
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Article
In-vitro Antibacterial, Antifungal and cytotoxic activity of cobalt (II), copper (II), nickel (II) and zinc (II) complexes with furanylmethyl- and thienylmethyl-dithiolenes: [1, 3-dithiole- 2-one and 1,3-dithiole-2-thione]
Zahid H. Chohan, Ali U. Shaikh & Claudiu T. Supuran
Pages: 733-740
Published online: 04 Oct 2008
AbstractforIn-vitro Antibacterial, Antifungal and cytotoxic activity of cobalt (II), copper (II), nickel (II) and zinc (II) complexes with furanylmethyl- and thienylmethyl-dithiolenes: [1, 3-dithiole- 2-one and 1,3-dithiole-2-thione] | Full Text | References | PDF (123.2 KB)
  • 653 Views
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Article
Antibacterial, antifungal and cytotoxic properties of novel N-substituted sulfonamides from 4-hydroxycoumarin
Zahid H. Chohan, Ali U. Shaikh, Abdul Rauf & Claudiu T. Supuran
Pages: 741-748
Published online: 04 Oct 2008
AbstractforAntibacterial, antifungal and cytotoxic properties of novel N-substituted sulfonamides from 4-hydroxycoumarin | Full Text | References | PDF (125.3 KB)
  • 1629 Views
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Article
Some bivalent metal complexes of Schiff bases containing N and S donor atoms
Kiran Singh, D. P. Singh, Manjeet Singh Barwa, Parikshit Tyagi & Yasmin Mirza
Pages: 749-755
Published online: 04 Oct 2008
AbstractforSome bivalent metal complexes of Schiff bases containing N and S donor atoms | Full Text | References | PDF (108.6 KB)
  • 1059 Views
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Article
Effect of calcium on rat intestinal alkaline phosphatase activity and molecular aggregation
Lucas R. M. Brun, María L. Brance, Alfredo Rigalli & Rodolfo C. Puche
Pages: 757-763
Published online: 04 Oct 2008
AbstractforEffect of calcium on rat intestinal alkaline phosphatase activity and molecular aggregation | Full Text | References | PDF (105.2 KB)
  • 602 Views
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Article
Antimicrobial bioassay of colchicum luteum baker
Bashir Ahmad, Haroon Khan, Shumaila Bashir & Murad Ali
Pages: 765-769
Published online: 04 Oct 2008
AbstractforAntimicrobial bioassay of colchicum luteum baker | Full Text | References | PDF (90.5 KB)
  • 883 Views
  • 8 CrossRef citations
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Article
In-vitro antibacterial, antifungal and cytotoxic properties of metal-based furanyl derived sulfonamides
Zahid H. Chohan, Ali U. Shaikh, Muhammad M. Naseer & Claudiu T. Supuran
Pages: 771-781
Published online: 04 Oct 2008
AbstractforIn-vitro antibacterial, antifungal and cytotoxic properties of metal-based furanyl derived sulfonamides | Full Text | References | PDF (142.9 KB)
  • 656 Views
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Article
Inhibition of choline oxidase by quinoid dyes
Özden Tacal & Inci Özer
Pages: 783-787
Published online: 04 Oct 2008
AbstractforInhibition of choline oxidase by quinoid dyes | Full Text | References | PDF (144.5 KB)
  • 546 Views
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