Citations (47)
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Lisa Sequeira, Simona Distinto, Rita Meleddu, Marco Gaspari, Andrea Angeli, Filippo Cottiglia, Daniela Secci, Alessia Onali, Erica Sanna, Fernanda Borges, Eugenio Uriarte, Stefano Alcaro, Claudiu T. Supuran & Elias Maccioni. (2023) 2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Rita Meleddu, Serenella Deplano, Elias Maccioni, Francesco Ortuso, Filippo Cottiglia, Daniela Secci, Alessia Onali, Erica Sanna, Andrea Angeli, Rossella Angius, Stefano Alcaro, Claudiu T. Supuran & Simona Distinto. (2021) Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 685-692.
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Manuel A. Llanos, María L. Sbaraglini, María L. Villalba, María D. Ruiz, Carolina Carrillo, Catalina Alba Soto, Alan Talevi, Andrea Angeli, Seppo Parkkila, Claudiu T. Supuran & Luciana Gavernet. (2020) A structure-based approach towards the identification of novel antichagasic compounds: Trypanosoma cruzi carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 21-30.
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Simona Distinto, Rita Meleddu, Francesco Ortuso, Filippo Cottiglia, Serenella Deplano, Lisa Sequeira, Claudia Melis, Benedetta Fois, Andrea Angeli, Clemente Capasso, Rossella Angius, Stefano Alcaro, Claudiu T. Supuran & Elias Maccioni. (2019) Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1526-1533.
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Suleyman Akocak, Nabih Lolak, Silvia Bua, Alessio Nocentini & Claudiu T. Supuran. (2019) Activation of human α-carbonic anhydrase isoforms I, II, IV and VII with bis-histamine schiff bases and bis-spinaceamine substituted derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1193-1198.
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Baijayantimala Swain, Andrea Angeli, Srinivas Angapelly, Pavitra S. Thacker, Priti Singh, Claudiu T. Supuran & Mohammed Arifuddin. (2019) Synthesis of a new series of 3-functionalised-1-phenyl-1,2,3-triazole sulfamoylbenzamides as carbonic anhydrase I, II, IV and IX inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1199-1209.
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Pavitra S. Thacker, Pirpasha Shaikh, Andrea Angeli, Mohammed Arifuddin & Claudiu T. Supuran. (2019) Synthesis and biological evaluation of novel 8-substituted quinoline-2-carboxamides as carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1172-1177.
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Andreza R. Garcia, Danielle M. P. Oliveira, Ana Claudia F. Amaral, Jéssica B. Jesus, Ana Carolina Rennó Sodero, Alessandra M. T. Souza, Claudiu T. Supuran, Alane B. Vermelho, Igor A. Rodrigues & Anderson S. Pinheiro. (2019) Leishmania infantum arginase: biochemical characterization and inhibition by naturally occurring phenolic substances. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1100-1109.
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Alessandra Ammazzalorso, Simone Carradori, Andrea Angeli, Atilla Akdemir, Barbara De Filippis, Marialuigia Fantacuzzi, Letizia Giampietro, Cristina Maccallini, Rosa Amoroso & Claudiu T. Supuran. (2019) Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1051-1061.
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Atilla Akdemir, Andrea Angeli, Füsun Göktaş, Pınar Eraslan Elma, Nilgün Karalı & Claudiu T. Supuran. (2019) Novel 2-indolinones containing a sulfonamide moiety as selective inhibitors of candida β-carbonic anhydrase enzyme. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 528-531.
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Rosa Perfetto, Sonia Del Prete, Daniela Vullo, Giovanni Sansone, Carmela M.A. Barone, Mosè Rossi, Claudiu T. Supuran & Clemente Capasso. (2017) Production and covalent immobilisation of the recombinant bacterial carbonic anhydrase (SspCA) onto magnetic nanoparticles. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 759-766.
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Rosa Perfetto, Sonia Del Prete, Daniela Vullo, Giovanni Sansone, Carmela Barone, Mosè Rossi, Claudiu T. Supuran & Clemente Capasso. (2017) Biochemical characterization of the native α-carbonic anhydrase purified from the mantle of the Mediterranean mussel, Mytilus galloprovincialis. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 632-639.
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Articles from other publishers (35)
Yuliya E. Ryzhkova, Varvara M. Kalashnikova, Fedor V. Ryzhkov, Artem N. Fakhrutdinov & Michail N. Elinson. (2023) 4a′-Hydroxy-3′,3′,5,6′,6′,7-hexamethyl-3′,4′,4a′,6′,7′,9a′-hexahydrospiro[indole-3,9′-xanthene]-1′,2,8′(1H,2′H,5′H)-trione. Molbank 2023:3, pages M1721.
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Firoj Hassan, Iqbal Azad, Mohd Asif, Deepanjali Shukla, Atif Husain, Abdul Rahman Khan, Mohammad Saquib & Malik Nasibullah. (2023) Isatin Conjugates as Antibacterial Agents: A Brief Review. Medicinal Chemistry 19:5, pages 413-430.
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Yeliz Demir, Cüneyt Türkeş, Muhammet S. Çavuş, Musa Erdoğan, Halit Muğlu, Hasan Yakan & Şükrü Beydemir. (2022) Enzyme inhibition, molecular docking, and density functional theory studies of new thiosemicarbazones incorporating the 4‐hydroxy‐3,5‐dimethoxy benzaldehyde motif. Archiv der Pharmazie 356:4.
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Yuliya E. Ryzhkova, Fedor V. Ryzhkov & Michail N. Elinson. (2023) Triethylammonium 2-(3-Hydroxy-2-oxoindolin-3-yl)-5,5-dimethyl-3-oxocyclohex-1-en-1-olate. Molbank 2023:1, pages M1589.
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T.N. Pashirova, Z.M. Shaihutdinova, A.E. Vandyukov, A.P. Lyubina, S.K. Amerhanova, A.D. Voloshina, A.V. Samorodov, E.B. Souto, V.F. Mironov & A.V. Bogdanov. (2022) Synthesis and structure-activity-toxicity relationships of DABCO-containing ammonium amphiphiles based on natural isatin scaffold. Journal of Molecular Liquids 365, pages 120217.
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Amit Kumar, Kiran Siwach, Claudiu T. Supuran & Pawan K. Sharma. (2022) A decade of tail-approach based design of selective as well as potent tumor associated carbonic anhydrase inhibitors. Bioorganic Chemistry 126, pages 105920.
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Hadi Adibi, Ehsan Beyhaghi, Sonya Hayati, Leila Hosseinzadeh & Niloufar Amin. (2022)
In Vitro
Cytotoxicity and Apoptosis Inducing Evaluation of Novel Halogenated Isatin
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. Anti-Cancer Agents in Medicinal Chemistry 22:13, pages 2439-2447.
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Pınar Eraslan‐Elma, Atilla Akdemir, Emanuela Berrino, Murat Bozdağ, Claudiu T. Supuran & Nilgün Karalı. (2022)
New 1
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. Archiv der Pharmazie 355:8.
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Nilamber A. Mate, Rowan I. L. Meador, Bhaskar D. Joshi & John D. Chisholm. (2022) Alkylation of isatins with trichloroacetimidates. Organic & Biomolecular Chemistry 20:10, pages 2131-2136.
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Ponnusamy Packialakshmi, Perumal Gobinath, Kaliappillai Vijayakumar, Daoud Ali, Saud Alarifi, Balasubramani Ravindran, PitchaiSangan & Radhakrishnan Surendrakumar. (2021) Synthesis of Isatin Derivatives Using Silver Nanoparticles as Green Catalyst: Study of Molecular Docking Interactions in SARS-CoV-2 3c-Like Protease and Determination of Cytotoxic Activities of the Compounds. Journal of Nanomaterials 2021, pages 1-17.
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Hasan YAKAN, M. Serdar ÇAVUŞ, Belma ZENGİN KURT, Halit MUĞLU, Fatih SÖNMEZ & Emre GÜZEL. (2021) A new series of asymmetric bis-isatin derivatives containing urea/thiourea moiety: Preparation, spectroscopic elucidation, antioxidant properties and theoretical calculations. Journal of Molecular Structure 1239, pages 130495.
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Anastasiya S. Sokolova, Kseniya S. Kovaleva, Olga I. Yarovaya, Nikolay I. Bormotov, Larisa N. Shishkina, Olga A. Serova, Alexander A. Sergeev, Alexander P. Agafonov, Rinat A. Maksuytov & Nariman F. Salakhutdinov. (2021) (+)‐Camphor and (−)‐borneol derivatives as potential anti‐orthopoxvirus agents. Archiv der Pharmazie 354:6.
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Anthi Petrou, Maria Fesatidou & Athina Geronikaki. (2021) Thiazole Ring—A Biologically Active Scaffold. Molecules 26:11, pages 3166.
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Sadaf Hashmi, Samra Khan, Zahid Shafiq, Parham Taslimi, Muhamamd Ishaq, Nastaran Sadeghian, Halide Sedef Karaman, Naeem Akhtar, Muhamamd Islam, Asnuzilawati Asari, Habsah Mohamad & İlhami Gulçin. (2021) Probing 4-(diethylamino)-salicylaldehyde-based thiosemicarbazones as multi-target directed ligands against cholinesterases, carbonic anhydrases and α-glycosidase enzymes. Bioorganic Chemistry 107, pages 104554.
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A. V. Bogdanov, A. D. Voloshina, A. S. Sapunova, N. V. Kulik & V. F. Mironov. (2020) Effect of Structure of 1-Substituted Isatins on Direction of Their Reactions with Some Acetohydrazide Ammonium Derivatives. Russian Journal of General Chemistry 90:9, pages 1591-1600.
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Rita Meleddu, Simona Distinto, Filippo Cottiglia, Rossella Angius, Pierluigi Caboni, Andrea Angeli, Claudia Melis, Serenella Deplano, Stefano Alcaro, Francesco Ortuso, Claudiu T. Supuran & Elias Maccioni. (2020) New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII. ACS Medicinal Chemistry Letters 11:5, pages 852-856.
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Riham F. George, Silvia Bua, Claudiu T. Supuran & Fadi M. Awadallah. (2020) Synthesis of some N-aroyl-2-oxindole benzenesulfonamide conjugates with carbonic anhydrase inhibitory activity. Bioorganic Chemistry 96, pages 103635.
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Ya‐Zhou Zhang, Hong‐Zhi Du, Hai‐Lin Liu, Qian‐Song He & Zhi Xu. (2020) Isatin dimers and their biological activities. Archiv der Pharmazie 353:3.
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Mohamed A. Abdelrahman, Wagdy M. Eldehna, Alessio Nocentini, Silvia Bua, Sara T. Al-Rashood, Ghada S. Hassan, Alessandro Bonardi, Abdulrahman A. Almehizia, Hamad M. Alkahtani, Amal Alharbi, Paola Gratteri & Claudiu T. Supuran. (2019) Novel Diamide-Based Benzenesulfonamides as Selective Carbonic Anhydrase IX Inhibitors Endowed with Antitumor Activity: Synthesis, Biological Evaluation and In Silico Insights. International Journal of Molecular Sciences 20:10, pages 2484.
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Rita Meleddu, Vilma Petrikaite, Simona Distinto, Antonella Arridu, Rossella Angius, Lorenzo Serusi, Laura Škarnulytė, Ugnė Endriulaitytė, Miglė Paškevičiu̅tė, Filippo Cottiglia, Marco Gaspari, Domenico Taverna, Serenella Deplano, Benedetta Fois & Elias Maccioni. (2018) Investigating the Anticancer Activity of Isatin/Dihydropyrazole Hybrids. ACS Medicinal Chemistry Letters 10:4, pages 571-576.
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Wagdy M. Eldehna, Mahmoud F. Abo-Ashour, Emanuela Berrino, Daniela Vullo, Hazem A. Ghabbour, Sara T. Al-Rashood, Ghada S. Hassan, Hamad M. Alkahtani, Abdulrahman A. Almehizia, Amal Alharbi, Hatem A. Abdel-Aziz & Claudiu T. Supuran. (2019) SLC-0111 enaminone analogs, 3/4-(3-aryl-3-oxopropenyl) aminobenzenesulfonamides, as novel selective subnanomolar inhibitors of the tumor-associated carbonic anhydrase isoform IX. Bioorganic Chemistry 83, pages 549-558.
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Wagdy M. Eldehna, Mahmoud F. Abo-Ashour, Alessio Nocentini, Radwan S. El-Haggar, Silvia Bua, Alessandro Bonardi, Sara T. Al-Rashood, Ghada S. Hassan, Paola Gratteri, Hatem A. Abdel-Aziz & Claudiu T. Supuran. (2019) Enhancement of the tail hydrophobic interactions within the carbonic anhydrase IX active site via structural extension: Design and synthesis of novel N-substituted isatins-SLC-0111 hybrids as carbonic anhydrase inhibitors and antitumor agents. European Journal of Medicinal Chemistry 162, pages 147-160.
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Marc A. Ilies & Jean-Yves Winum. 2019. Carbonic Anhydrases. Carbonic Anhydrases
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Wagdy M. Eldehna, Alessio Nocentini, Sara T. Al-Rashood, Ghada S. Hassan, Hamad M. Alkahtani, Abdulrahman A. Almehizia, Ahmed M. Reda, Hatem A. Abdel-Aziz & Claudiu T. Supuran. (2018) Tumor-associated carbonic anhydrase isoform IX and XII inhibitory properties of certain isatin-bearing sulfonamides endowed with in vitro antitumor activity towards colon cancer. Bioorganic Chemistry 81, pages 425-432.
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Reuel de Paula, Joyce de Almeida, Samir Cavalcante, Arlan Gonçalves, Alessandro Simas, Tanos Franca, Martin Valis, Kamil Kuca, Eugenie Nepovimova & José Granjeiro. (2018) Molecular Modeling and In Vitro Studies of a Neutral Oxime as a Potential Reactivator for Acetylcholinesterase Inhibited by Paraoxon. Molecules 23:11, pages 2954.
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Rita Meleddu, Simona Distinto, Filippo Cottiglia, Rossella Angius, Marco Gaspari, Domenico Taverna, Claudia Melis, Andrea Angeli, Giulia Bianco, Serenella Deplano, Benedetta Fois, Sonia Del Prete, Clemente Capasso, Stefano Alcaro, Francesco Ortuso, Matilde Yanez, Claudiu T. Supuran & Elias Maccioni. (2018) Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides. ACS Medicinal Chemistry Letters 9:10, pages 1045-1050.
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Mahmoud F. Abo-Ashour, Wagdy M. Eldehna, Alessio Nocentini, Hany S. Ibrahim, Silvia Bua, Sahar M. Abou-Seri & Claudiu T. Supuran. (2018) Novel hydrazido benzenesulfonamides-isatin conjugates: Synthesis, carbonic anhydrase inhibitory activity and molecular modeling studies. European Journal of Medicinal Chemistry 157, pages 28-36.
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Claudiu T. Supuran, Vincenzo Alterio, Anna Di Fiore, Katia D’ Ambrosio, Fabrizio Carta, Simona Maria Monti & Giuseppina De Simone. (2018) Inhibition of carbonic anhydrase IX targets primary tumors, metastases, and cancer stem cells: Three for the price of one. Medicinal Research Reviews 38:6, pages 1799-1836.
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Claudia Melis, Simona Distinto, Giulia Bianco, Rita Meleddu, Filippo Cottiglia, Benedetta Fois, Domenico Taverna, Rossella Angius, Stefano Alcaro, Francesco Ortuso, Marco Gaspari, Andrea Angeli, Sonia Del Prete, Clemente Capasso, Claudiu T. Supuran & Elias Maccioni. (2018) Targeting Tumor Associated Carbonic Anhydrases IX and XII: Highly Isozyme Selective Coumarin and Psoralen Inhibitors. ACS Medicinal Chemistry Letters 9:7, pages 725-729.
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A. V. Bogdanov, I. F. Zaripova, A. D. Voloshina, A. S. Strobykina, N. V. Kulik, S. V. Bukharov & V. F. Mironov. (2018) Isatin Derivatives Containing Sterically Hindered Phenolic Fragment and Water-Soluble Acyl Hydrazones on Their Basis: Synthesis and Antimicrobial Activity. Russian Journal of General Chemistry 88:1, pages 57-67.
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Andrea Angeli, Ghulam Abbas, Sonia Del Prete, Fabrizio Carta, Clemente Capasso & Claudiu T. Supuran. (2017) Acyl selenoureido benzensulfonamides show potent inhibitory activity against carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. Bioorganic Chemistry 75, pages 170-172.
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Giulia Bianco, Rita Meleddu, Simona Distinto, Filippo Cottiglia, Marco Gaspari, Claudia Melis, Angela Corona, Rossella Angius, Andrea Angeli, Domenico Taverna, Stefano Alcaro, Janis Leitans, Andris Kazaks, Kaspars Tars, Claudiu T. Supuran & Elias Maccioni. (2017)
N
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. ACS Medicinal Chemistry Letters 8:8, pages 792-796.
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Nilgün Karalı, Atilla Akdemir, Füsun Göktaş, Pınar Eraslan Elma, Andrea Angeli, Merih Kızılırmak & Claudiu T. Supuran. (2017) Novel sulfonamide-containing 2-indolinones that selectively inhibit tumor-associated alpha carbonic anhydrases. Bioorganic & Medicinal Chemistry 25:14, pages 3714-3718.
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Daniela Vullo, Sonia Del Prete, Pietro Di Fonzo, Vincenzo Carginale, W. Donald, Claudiu Supuran & Clemente Capasso. (2017) Comparison of the Sulfonamide Inhibition Profiles of the β- and γ-Carbonic Anhydrases from the Pathogenic Bacterium Burkholderia pseudomallei. Molecules 22:3, pages 421.
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Sonia Del Prete, Daniela Vullo, Pietro di Fonzo, Vincenzo Carginale, Claudiu T. Supuran & Clemente Capasso. (2017) Comparison of the anion inhibition profiles of the β- and γ-carbonic anhydrases from the pathogenic bacterium Burkholderia pseudomallei. Bioorganic & Medicinal Chemistry 25:6, pages 2010-2015.
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