Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 20, Issue 5 (2005)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 20, Issue 5 (2005)

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Research Article

Article
Synthesis of a novel series of bispyridinium compounds bearing a xylene linker and evaluation of their reactivation activity against chlorpyrifos-inhibited acetylcholinesterase
K. Musilek, K. Kuca, D. Jun, V. Dohnal & M. Dolezal
Pages: 409-415
Published online: 04 Oct 2008
AbstractforSynthesis of a novel series of bispyridinium compounds bearing a xylene linker and evaluation of their reactivation activity against chlorpyrifos-inhibited acetylcholinesterase | Full Text | References | PDF (286.8 KB)
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Article
Evaluation of O3α-, O21-Di-(N1-methyloxycarbonyl-2, 4-dioxo-5-fluoropyrimidinyl)17α-hydroxy-5β-pregnan-20-one as a novel potential antiangiogenic codrug
Michelle Howard-Sparks, Abeer M. Al-Ghananeem, Andrew P. Pearson & Peter A. Crooks
Pages: 417-428
Published online: 04 Oct 2008
AbstractforEvaluation of O3α-, O21-Di-(N1-methyloxycarbonyl-2, 4-dioxo-5-fluoropyrimidinyl)17α-hydroxy-5β-pregnan-20-one as a novel potential antiangiogenic codrug | Full Text | References | PDF (311.5 KB)
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Article
Structure–activity relationship studies of 3-dodecanoylindole-2-carboxylic acid inhibitors of cytosolic phospholipase A2α-mediated arachidonic acid release in intact platelets: variation of the keto moiety
Afshin Ghasemi, Alwine Schulze Elfringhoff & Matthias Lehr
Pages: 429-437
Published online: 04 Oct 2008
AbstractforStructure–activity relationship studies of 3-dodecanoylindole-2-carboxylic acid inhibitors of cytosolic phospholipase A2α-mediated arachidonic acid release in intact platelets: variation of the keto moiety | Full Text | References | PDF (182.1 KB)
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Article
Glutamine analogues containing a keto function – novel inhibitors of fungal glucosamine-6-phosphate synthase
Aleksandra Walkowiak, Roland Wakieć, Maria M. Bontemps-Gracz & Ryszard Andruszkiewicz
Pages: 439-447
Published online: 04 Oct 2008
AbstractforGlutamine analogues containing a keto function – novel inhibitors of fungal glucosamine-6-phosphate synthase | Full Text | References | PDF (338.7 KB)
  • 522 Views
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Article
Violacein cytotoxicity on human blood lymphocytes and effect on phosphatases
N. Bromberg, G. Z. Justo, M. Haun, N. Durán & C. V. Ferreira
Pages: 449-454
Published online: 04 Oct 2008
AbstractforViolacein cytotoxicity on human blood lymphocytes and effect on phosphatases | Full Text | References | PDF (198.4 KB)
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Article
Quantitative structure–activity relationship analysis of 2,3-diaryl indoles as selective cyclooxygenase-2 inhibitors
S. PRASANNA, E. MANIVANNAN & S.C. CHATURVEDI
Pages: 455-461
Published online: 04 Oct 2008
AbstractforQuantitative structure–activity relationship analysis of 2,3-diaryl indoles as selective cyclooxygenase-2 inhibitors | Full Text | References | PDF (103.4 KB)
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Article
In-vitro antibacterial and cytotoxic activity of cobalt (ii), copper (ii), nickel (ii) and zinc (ii) complexes of the antibiotic drug cephalothin (Keflin)
Zahid H. Chohan & Claudiu T. Supuran
Pages: 463-468
Published online: 04 Oct 2008
AbstractforIn-vitro antibacterial and cytotoxic activity of cobalt (ii), copper (ii), nickel (ii) and zinc (ii) complexes of the antibiotic drug cephalothin (Keflin) | Full Text | References | PDF (125.1 KB)
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Article
Inhibition of Na+/K+-ATPase and Mg2+-ATPase by metal ions and prevention and recovery of inhibited activities by chelators
Danijela Krstić, Katarina Krinulović & Vesna Vasić
Pages: 469-476
Published online: 04 Oct 2008
AbstractforInhibition of Na+/K+-ATPase and Mg2+-ATPase by metal ions and prevention and recovery of inhibited activities by chelators | Full Text | References | PDF (178.4 KB)
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Article
Inhibition study of rabbit liver cytosolic reductases involved in daunorubicin toxication
Helena Kaiserová & Eva Kvasničková
Pages: 477-483
Published online: 04 Oct 2008
AbstractforInhibition study of rabbit liver cytosolic reductases involved in daunorubicin toxication | Full Text | References | PDF (382.1 KB)
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Article
Effects of some drugs on the activity of glucose 6-phosphate dehydrogenase from rainbow trout (Oncorhynchus mykiss) erythrocytes in vitro
Mehmet Ciftci
Pages: 485-489
Published online: 04 Oct 2008
AbstractforEffects of some drugs on the activity of glucose 6-phosphate dehydrogenase from rainbow trout (Oncorhynchus mykiss) erythrocytes in vitro | Full Text | References | PDF (150.3 KB)
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Article
In vitro effects of some anaesthetic drugs on lactoperoxidase enzyme activity
Hasan ÖZDEMİR & Metin Tansu UĞUZ
Pages: 491-495
Published online: 04 Oct 2008
AbstractforIn vitro effects of some anaesthetic drugs on lactoperoxidase enzyme activity | Full Text | References | PDF (202.7 KB)
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Article
Effects of nicotine and vitamin E on glucose 6-phosphate dehydrogenase activity in some rat tissues in vivo and in vitro
Kenan Gumustekin, Mehmet Ciftci, Abdulkadir Coban, Sayit Altikat, Omer Aktas, Mustafa Gul, Handan Timur & Senol Dane
Pages: 497-502
Published online: 04 Oct 2008
AbstractforEffects of nicotine and vitamin E on glucose 6-phosphate dehydrogenase activity in some rat tissues in vivo and in vitro | Full Text | References | PDF (147.8 KB)
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Article
Synthesis, antioxidant and radical scavenging activities of novel benzimidazoles
Gülgün Ayhan-KIlcigİl, Canan Kuş, Tülay Çoban, Benay Can-Eke, Süheyla Özbey & Mümtaz Iscan
Pages: 503-514
Published online: 04 Oct 2008
AbstractforSynthesis, antioxidant and radical scavenging activities of novel benzimidazoles | Full Text | References | PDF (328 KB)
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