Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 21, Issue 5 (2006)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 21, Issue 5 (2006)

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Research Article

Article
A kinetic, modeling and mechanistic re-analysis of thymidine phosphorylase and some related enzymes
REVIEW ARTICLE
Philip N. Edwards
Pages: 483-518
Published online: 20 Oct 2008
AbstractforA kinetic, modeling and mechanistic re-analysis of thymidine phosphorylase and some related enzymes | Full Text | References | PDF (758.2 KB)
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Article
Synthesis and anticancer activity of certain mononuclear Ru (II) Complexes
Suresh Rathinasamy, Subhas Somalingappa Karki, Shiladitya Bhattacharya, Lakshmanan Manikandan, Senthilkumar G. Prabakaran, Malaya Gupta & Upal Kanti Mazumder
Pages: 501-507
Published online: 04 Oct 2008
AbstractforSynthesis and anticancer activity of certain mononuclear Ru (II) Complexes | Full Text | References | PDF (134.9 KB)
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Article
Detection of sarin in plasma of rats after inhalation intoxication
Lucie Bartosova, Marcela Bielavska & Jiri Bajgar
Pages: 509-514
Published online: 04 Oct 2008
AbstractforDetection of sarin in plasma of rats after inhalation intoxication | Full Text | References | PDF (210 KB)
  • 353 Views
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Article
New group of xylene linker-containing acetylcholinesterase reactivators as antidotes against the nerve agent cyclosarin
Martina Hrabinova, Kamil Musilek, Daniel Jun & Kamil Kuca
Pages: 515-519
Published online: 04 Oct 2008
AbstractforNew group of xylene linker-containing acetylcholinesterase reactivators as antidotes against the nerve agent cyclosarin | Full Text | References | PDF (83.5 KB)
  • 433 Views
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Article
Synthesis, characterization and inhibitory potency of two oxono and thiono analogues of phosphoramidate compounds on acetylcholinesterase
Khodayar Gholivand, Fresia Mojahed, Marjan Salehi, Hossein Naderi-Manesh & Khosro Khajeh
Pages: 521-525
Published online: 04 Oct 2008
AbstractforSynthesis, characterization and inhibitory potency of two oxono and thiono analogues of phosphoramidate compounds on acetylcholinesterase | Full Text | References | PDF (101.7 KB)
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Article
Novel urease inhibitors from Daphne oleoids
MUHAMMAD AYAZ, MUHAMMAD ARIF LODHI, MUHAMMAD RIAZ, AZHAR -UL-HAQ, ABDUL MALIK & M. IQBAL CHOUDHARY
Pages: 527-529
Published online: 04 Oct 2008
AbstractforNovel urease inhibitors from Daphne oleoids | Full Text | References | PDF (106.4 KB)
  • 553 Views
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Article
A New Bacillus pasteurii Urease Inhibitor from Euphorbia decipiens
Muhammad Arif Lodhi, Javid Hussain, Muhammad Athar Abbasi, Amir Reza Jassbi, Muhammad Iqbal Choudhary & Viqar Uddin Ahmad
Pages: 531-535
Published online: 04 Oct 2008
AbstractforA New Bacillus pasteurii Urease Inhibitor from Euphorbia decipiens | Full Text | References | PDF (158 KB)
  • 600 Views
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Article
Inhibition of jack bean urease by tetrachloro-o-benzoquinone and tetrachloro-p-benzoquinone
Mirosława Kot & Wiesława Zaborska
Pages: 537-542
Published online: 04 Oct 2008
AbstractforInhibition of jack bean urease by tetrachloro-o-benzoquinone and tetrachloro-p-benzoquinone | Full Text | References | PDF (162 KB)
  • 600 Views
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Article
Adenosine deaminase in ischemia reperfusion injury in patients with myocardial infarction
Aiki Kaul, M. Chandra & M. K. Misra
Pages: 543-546
Published online: 04 Oct 2008
AbstractforAdenosine deaminase in ischemia reperfusion injury in patients with myocardial infarction | Full Text | References | PDF (64.4 KB)
  • 332 Views
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Article
A fission yeast-based test system for the determination of IC50 values of anti-prostate tumor drugs acting on CYP21
Călin-Aurel Drăgan, Rolf W. Hartmann & Matthias Bureik
Pages: 547-556
Published online: 04 Oct 2008
AbstractforA fission yeast-based test system for the determination of IC50 values of anti-prostate tumor drugs acting on CYP21 | Full Text | References | PDF (277.2 KB)
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Article
Antibacterial Co(II), Ni(II), Cu(II) and Zn(II) Complexes of Schiff bases Derived from Fluorobenzaldehyde and Triazoles
Kiran Singh
Pages: 557-562
Published online: 04 Oct 2008
AbstractforAntibacterial Co(II), Ni(II), Cu(II) and Zn(II) Complexes of Schiff bases Derived from Fluorobenzaldehyde and Triazoles | Full Text | References | PDF (110.9 KB)
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Article
Carbonic anhydrase inhibitors. Selective inhibition of human tumor-associated isozymes IX and XII and cytosolic isozymes I and II with some substituted-2-mercapto-benzenesulfonamides
Franciszek Saczewski, Alessio Innocenti, Zdzisław Brzozowski, Jarosław Sławiński, Elżbieta Pomarnacka, Anita Kornicka, Andrea Scozzafava & Claudiu T. Supuran
Pages: 563-568
Published online: 04 Oct 2008
AbstractforCarbonic anhydrase inhibitors. Selective inhibition of human tumor-associated isozymes IX and XII and cytosolic isozymes I and II with some substituted-2-mercapto-benzenesulfonamides | Full Text | References | PDF (128.8 KB)
  • 432 Views
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Article
WY 14,643 inhibits human aldose reductase activity
Sara Klemin, Richard Y. Calvo, Stephanie Bond, Heather Dingess, Balakrishnan Rajkumar, Rachel Perez, Lucy Chow & Ganesaratnam K. Balendiran
Pages: 569-573
Published online: 04 Oct 2008
AbstractforWY 14,643 inhibits human aldose reductase activity | Full Text | References | PDF (82.3 KB)
  • 467 Views
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Article
Sevoflurane modulates the activity of glyceraldehyde 3-phosphate dehydrogenase
Timothy A. Swearengin, Eugene E. Fibuch & Norbert W. Seidler
Pages: 575-579
Published online: 04 Oct 2008
AbstractforSevoflurane modulates the activity of glyceraldehyde 3-phosphate dehydrogenase | Full Text | References | PDF (151 KB)
  • 307 Views
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Article
Inhibition of human glutathione transferases by multidrug resistance chemomodulators in vitro
Rose Hayeshi, Farai Chinyanga, Shylet Chengedza & Stanley Mukanganyama
Pages: 581-587
Published online: 04 Oct 2008
AbstractforInhibition of human glutathione transferases by multidrug resistance chemomodulators in vitro | Full Text | References | PDF (190 KB)
  • 951 Views
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Article
The extract of leaves of Acer truncatum Bunge: A natural inhibitor of fatty acid synthase with antitumor activity
Wen-Hua Zhao, Jin-Feng Zhang, Zhe-Wang, Ying-Xia Zhang & Wei-Xi Tian
Pages: 589-596
Published online: 04 Oct 2008
AbstractforThe extract of leaves of Acer truncatum Bunge: A natural inhibitor of fatty acid synthase with antitumor activity | Full Text | References | PDF (275.1 KB)
  • 796 Views
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Article
A new fermentation process allows large-scale production of tetra-N-acetyl-chitotetraosyl allosamizoline
Gang-Liang Huang, Xin-Ya Mei, Hou-Cheng Zhang & Peng-George Wang
Pages: 597-599
Published online: 04 Oct 2008
AbstractforA new fermentation process allows large-scale production of tetra-N-acetyl-chitotetraosyl allosamizoline | Full Text | References | PDF (75.3 KB)
  • 246 Views
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Article
Quantitative structure–activity relationship study of new potent and selective antagonists at the 5-HT1A and adrenergic α1d receptors: Derivatives of spiroethyl phenyl(substituted)piperazine
B. K. Sharma, P. Singh & Susheela Sharma
Pages: 601-607
Published online: 04 Oct 2008
AbstractforQuantitative structure–activity relationship study of new potent and selective antagonists at the 5-HT1A and adrenergic α1d receptors: Derivatives of spiroethyl phenyl(substituted)piperazine | Full Text | References | PDF (90.7 KB)
  • 279 Views
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Article
A quantitative structure-activity relationship study for structurally diverse HIV-1 protease inhibitors: contribution of conformational flexibility to inhibitory activity
Keigo Gohda
Pages: 609-615
Published online: 04 Oct 2008
AbstractforA quantitative structure-activity relationship study for structurally diverse HIV-1 protease inhibitors: contribution of conformational flexibility to inhibitory activity | Full Text | References | PDF (94.1 KB)
  • 233 Views
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