Citations (460)
Keep up to date with the latest research on this topic with citation updates for this article.
Read on this site (82)
Tuba Tekeli, Suleyman Akocak, Andrea Petreni, Nebih Lolak, Servet Çete & Claudiu T. Supuran. (2023) Potent carbonic anhydrase I, II, IX and XII inhibition activity of novel primary benzenesulfonamides incorporating bis-ureido moieties. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
Read now
Read now
Doretta Cuffaro, Riccardo Di Leo, Lidia Ciccone, Alessio Nocentini, Claudiu T. Supuran, Elisa Nuti & Armando Rossello. (2023) New isoxazolidinyl-based N-alkylethanolamines as new activators of human brain carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
Read now
Read now
Hakan Şahal, Samet Öz, Suat Tekin & Erdal Canpolat. (2023) Synthesis, structural characterizations and in vitro cytotoxic activities of new sulfonamide-based Schiff base derivatives. Journal of Biomolecular Structure and Dynamics 41:10, pages 4361-4367.
Read now
Read now
Hakan Şahal, Samet Öz, Tuba Keskin, Suat Tekin, Erdal Canpolat & Mehmet Kaya. (2023) New sulfa drug derivatives and their zinc(II) complexes: synthesis, spectroscopic properties and in vitro cytotoxic activities. Journal of Biomolecular Structure and Dynamics 0:0, pages 1-14.
Read now
Read now
Hossam Nada, Ahmed Elkamhawy, Magda H. Abdellattif, Andrea Angeli, Chang Hoon Lee, Claudiu T. Supuran & Kyeong Lee. (2022) 4-Anilinoquinazoline-based benzenesulfonamides as nanomolar inhibitors of carbonic anhydrase isoforms I, II, IX, and XII: design, synthesis, in-vitro, and in-silico biological studies. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 994-1004.
Read now
Read now
Kirna Devi & Pamita Awasthi. (2022) Isoleucine with secondary sulfonamide functionality as anticancer, antibacterial and antifungal agents. Journal of Biomolecular Structure and Dynamics 40:15, pages 7052-7069.
Read now
Read now
Rahman Padash, Milad Rabbani Esfahani & Ali Shokuhi Rad. (2021) The computational quantum mechanical study of sulfamide drug adsorption onto X12Y12 fullerene-like nanocages: detailed DFT and QTAIM investigations. Journal of Biomolecular Structure and Dynamics 39:15, pages 5427-5437.
Read now
Read now
Francesco Mincione, Alessio Nocentini & Claudiu T. Supuran. (2021) Advances in the discovery of novel agents for the treatment of glaucoma. Expert Opinion on Drug Discovery 16:10, pages 1209-1225.
Read now
Read now
Chandra Bhushan Mishra, Raj Kumar Mongre, Amresh Prakash, Raok Jeon, Claudiu T. Supuran & Myeong-Sok Lee. (2021) Anti-breast cancer action of carbonic anhydrase IX inhibitor 4-[4-(4-Benzo[1,3]dioxol-5-ylmethyl-piperazin-1-yl)-benzylidene-hydrazinocarbonyl]-benzenesulfonamide (BSM-0004): in vitro and in vivo studies. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 954-963.
Read now
Read now
Paolo Guglielmi, Giulia Rotondi, Daniela Secci, Andrea Angeli, Paola Chimenti, Alessio Nocentini, Alessandro Bonardi, Paola Gratteri, Simone Carradori & Claudiu T. Supuran. (2020) Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1891-1905.
Read now
Read now
Zhuang Hou, Chuanchao Li, Yichuang Liu, Miao Zhang, Yitong Wang, Zhanfang Fan, Chun Guo, Bin Lin & Yang Liu. (2020) Design, synthesis and biological evaluation of carbohydrate-based sulphonamide derivatives as topical antiglaucoma agents through selective inhibition of carbonic anhydrase II. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 383-390.
Read now
Read now
Claudiu T Supuran. (2019) The management of glaucoma and macular degeneration. Expert Opinion on Therapeutic Patents 29:10, pages 745-747.
Read now
Read now
Claudiu T. Supuran. (2019) Agents for the prevention and treatment of age-related macular degeneration and macular edema: a literature and patent review. Expert Opinion on Therapeutic Patents 29:10, pages 761-767.
Read now
Read now
Alessandro Bonardi & Claudiu T Supuran. (2019) Treatment of glaucoma and ocular hypertension using rho kinase inhibitors: patent evaluation of US2018244666 and US2018256595. Expert Opinion on Therapeutic Patents 29:10, pages 753-759.
Read now
Read now
Sabina Zamanova, Ahmed M Shabana, Utpal K Mondal & Marc A Ilies. (2019) Carbonic anhydrases as disease markers. Expert Opinion on Therapeutic Patents 29:7, pages 509-533.
Read now
Read now
Claudiu T. Supuran. (2018) Carbonic anhydrase inhibitors and their potential in a range of therapeutic areas. Expert Opinion on Therapeutic Patents 28:10, pages 709-712.
Read now
Read now
Claudiu T. Supuran. (2018) Applications of carbonic anhydrases inhibitors in renal and central nervous system diseases. Expert Opinion on Therapeutic Patents 28:10, pages 713-721.
Read now
Read now
Sanjay M. Tailor & Urmila H. Patel. (2017) Nickel(II) complex of 4-amino-N-(2-pyrimidinyl)benzenesulfonamide: Synthesis, spectroscopic characterization, antimicrobial activity, crystal structure, and Hirshfeld surface analysis. Inorganic and Nano-Metal Chemistry 47:2, pages 234-243.
Read now
Read now
Parham Taslimi, Afsun Sujayev, Sevgi Mamedova, Pınar Kalın, İlhami Gulçin, Nastaran Sadeghian, Sukru Beydemir, O. Irfan Kufrevioglu, Saleh H. Alwasel, Vagif Farzaliyev & Sabir Mamedov. (2017) Synthesis and bioactivity of several new hetaryl sulfonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 137-145.
Read now
Read now
Manas R Dikhit, Bidyut Purkait, Ruby Singh, Bikash Ranjan Sahoo, Ashish Kumar, Rajiv K Kar, Md Yousuf Ansari, Savita Saini, Kumar Abhishek, Ganesh C Sahoo, Sushmita Das & Pradeep Das. (2016) Activity of a novel sulfonamide compound 2-nitro-N-(pyridin-2-ylmethyl)benzenesulfonamide against Leishmania donovani. Drug Design, Development and Therapy 10, pages 1753-1761.
Read now
Read now
Halise Inci Gul, Mehtap Tugrak, Hiroshi Sakagami, Parham Taslimi, Ilhami Gulcin & Claudiu T. Supuran. (2016) Synthesis and bioactivity studies on new 4-(3-(4-Substitutedphenyl)-3a,4-dihydro-3H-indeno[1,2-c]pyrazol-2-yl) benzenesulfonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1619-1624.
Read now
Read now
Leyla Polat Kose, İlhami Gulcin, Alper Yıldırım, Ufuk Atmaca, Murat Çelik, Saleh H. Alwasel & Claudiu T. Supuran. (2016) The human carbonic anhydrase isoenzymes I and II inhibitory effects of some hydroperoxides, alcohols, and acetates. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1248-1253.
Read now
Read now
Marta Abellán-Flos, Muhammet Tanç, Claudiu T. Supuran & Stéphane P. Vincent. (2016) Multimeric xanthates as carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 946-952.
Read now
Read now
Hulya Gocer, Fevzi Topal, Meryem Topal, Murat Küçük, Dilek Teke, İlhami Gülçin, Saleh H. Alwasel & Claudiu T. Supuran. (2016) Acetylcholinesterase and carbonic anhydrase isoenzymes I and II inhibition profiles of taxifolin. Journal of Enzyme Inhibition and Medicinal Chemistry 31:3, pages 441-447.
Read now
Read now
Parham Taslimi, Ilhami Gulcin, Bunyamin Ozgeris, Suleyman Goksu, Ferhan Tumer, Saleh H. Alwasel & Claudiu T. Supuran. (2016) The human carbonic anhydrase isoenzymes I and II (hCA I and II) inhibition effects of trimethoxyindane derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 31:1, pages 152-157.
Read now
Read now
Andrea Scozzafava, Pınar Kalın, Claudiu T. Supuran, İlhami Gülçin & Saleh H. Alwasel. (2015) The impact of hydroquinone on acetylcholine esterase and certain human carbonic anhydrase isoenzymes (hCA I, II, IX, and XII). Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 941-946.
Read now
Read now
Mehmet Arslan, Murat Şentürk, İsmail Fidan, Oktay Talaz, Deniz Ekinci, Sedat Coşgun & Claudiu T. Supuran. (2015) Synthesis of 3,4-dihydroxypyrrolidine-2,5-dione and 3,5-dihydroxybenzoic acid derivatives and evaluation of the carbonic anhydrase I and II inhibition. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 896-900.
Read now
Read now
Andrea Scozzafava, Maurizio Passaponti, Claudiu T. Supuran & İlhami Gülçin. (2015) Carbonic anhydrase inhibitors: guaiacol and catechol derivatives effectively inhibit certain human carbonic anhydrase isoenzymes (hCA I, II, IX and XII). Journal of Enzyme Inhibition and Medicinal Chemistry 30:4, pages 586-591.
Read now
Read now
Aysegul Sahin, Semra Isık, Oktay Arslan, Claudiu T. Supuran & Ozen Ozensoy Guler. (2015) A new affinity gel for the purification of α-carbonic anhdrases. Journal of Enzyme Inhibition and Medicinal Chemistry 30:2, pages 224-228.
Read now
Read now
Mina Ghiasi & Saeedeh Kamalinahad. (2015) Conformational Analysis of Topiramate and Related Anion in the Solution and Interaction Between the Most Stable Conformer of Topiramate with Active Center of Carbonic Anhydrase Enzyme. Journal of Carbohydrate Chemistry 34:2, pages 80-102.
Read now
Read now
Aamer Saeed, Mariya al-Rashida, Mehwish Hamayoun, Amara Mumtaz & Jamshed Iqbal. (2014) Carbonic anhydrase inhibition by 1-aroyl-3-(4-aminosulfonylphenyl)thioureas. Journal of Enzyme Inhibition and Medicinal Chemistry 29:6, pages 901-905.
Read now
Read now
Cheloufi Hadjer, Berredjem Malika, Boufas Wahida, Bouchareb Fouzia, Djahoudi Abdelghani & Aouf Nour-Eddine. (2014) Efficient Synthesis, Characterization, and Antibacterial Activity of Novel N-Acylsulfonamides and Sulfonylureas. Phosphorus, Sulfur, and Silicon and the Related Elements 189:9, pages 1396-1404.
Read now
Read now
Yasin Çetinkaya, Hülya Göçer, Süleyman Göksu & İlhami Gülçin. (2014) Synthesis and carbonic anhydrase isoenzymes I and II inhibitory effects of novel benzylamine derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 29:2, pages 168-174.
Read now
Read now
Fatma Celik, Mustafa Arslan, Mustafa Oguzhan Kaya, Emre Yavuz, Nahit Gencer & Oktay Arslan. (2014) Synthesis and carbonic anhydrase inhibitory properties of tetrazole- and oxadiazole substituted 1,4-dihydropyrimidinone compounds. Artificial Cells, Nanomedicine, and Biotechnology 42:1, pages 58-62.
Read now
Read now
Fatih Sonmez, Cigdem Bilen, Sinem Sumersan, Nahit Gencer, Semra Isik, Oktay Arslan & Mustafa Kucukislamoglu. (2014) In vitro inhibition effect and structure–activity relationships of some saccharin derivatives on erythrocyte carbonic anhydrase I and II. Journal of Enzyme Inhibition and Medicinal Chemistry 29:1, pages 118-123.
Read now
Read now
Yusuf Akbaba, Akın Akıncıoğlu, Hülya Göçer, Süleyman Göksu, İlhami Gülçin & Claudiu T. Supuran. (2014) Carbonic anhydrase inhibitory properties of novel sulfonamide derivatives of aminoindanes and aminotetralins. Journal of Enzyme Inhibition and Medicinal Chemistry 29:1, pages 35-42.
Read now
Read now
Nahit Gençer, Çiğdem Bilen, Dudu Demir, Alparslan Atahan, Mustafa Ceylan & Mustafa Küçükislamoğlu. (2013) In vitro inhibition effect of some chalcones on erythrocyte carbonic anhydrase I and II. Artificial Cells, Nanomedicine, and Biotechnology 41:6, pages 384-388.
Read now
Read now
Mansoura I. Mohamed, Howida T. Zaky & Nadia G. Kandile. (2013) Microwave-assisted synthesis of antimicrobial agents based on pyridazine moiety. Journal of Enzyme Inhibition and Medicinal Chemistry 28:6, pages 1307-1315.
Read now
Read now
Syed Ovais, Shafiya Yaseen, Rafia Bashir, Pooja Rathore, Mohammed Samim, Surender Singh, Vinod Nair & Kalim Javed. (2013) Synthesis and anti-inflammatory activity of celecoxib like compounds. Journal of Enzyme Inhibition and Medicinal Chemistry 28:5, pages 1105-1112.
Read now
Read now
Emanuela Masini, Fabrizio Carta, Andrea Scozzafava & Claudiu T Supuran. (2013) Antiglaucoma carbonic anhydrase inhibitors: a patent review. Expert Opinion on Therapeutic Patents 23:6, pages 705-716.
Read now
Read now
Andrea Scozzafava, Claudiu T Supuran & Fabrizio Carta. (2013)
Antiobesity carbonic anhydrase inhibitors: a literature and patent review
. Expert Opinion on Therapeutic Patents 23:6, pages 725-735.
Read now
Read now
Fabrizio Carta & Claudiu T Supuran. (2013) Diuretics with carbonic anhydrase inhibitory action: a patent and literature review (2005 – 2013). Expert Opinion on Therapeutic Patents 23:6, pages 681-691.
Read now
Read now
Simone Carradori. (2013) Selective carbonic anhydrase IX inhibitors based on coumarin scaffold as promising antimetastatic agents: WO2012070024. Expert Opinion on Therapeutic Patents 23:6, pages 751-756.
Read now
Read now
Fabrizio Carta, Andrea Scozzafava & Claudiu T Supuran. (2012) Sulfonamides: a patent review (2008 – 2012). Expert Opinion on Therapeutic Patents 22:7, pages 747-758.
Read now
Read now
Rafia Bashir, Shafiya Yaseen, Syed Ovais, Shamim Ahmad, Hinna Hamid, M.S. Alam, Mohammad Samim & Kalim Javed. (2012) Synthesis and biological evaluation of some novel sulfamoylphenyl-pyridazinone as anti-inflammatory agents (Part-II). Journal of Enzyme Inhibition and Medicinal Chemistry 27:1, pages 92-96.
Read now
Read now
Fabrizio Carta, Claudiu T Supuran & Andrea Scozzafava. (2012) Novel therapies for glaucoma: a patent review 2007 – 2011. Expert Opinion on Therapeutic Patents 22:1, pages 79-88.
Read now
Read now
Zahid H. Chohan, Claudiu T. Supuran, Taibi Ben Hadda, Faiz-Ul-Hassan Nasim & Khalid M. Khan. (2009) Metal based isatin-derived sulfonamides: Their synthesis, characterization, coordination behavior and biological activity. Journal of Enzyme Inhibition and Medicinal Chemistry 24:3, pages 859-870.
Read now
Read now
Isao MIYAZAKI, Siro SIMIZU, Harumi ICHIMIYA, Makoto KAWATANI & Hiroyuki OSADA. (2008) Robust and Systematic Drug Screening Method Using Chemical Arrays and the Protein Library: Identification of Novel Inhibitors of Carbonic Anhydrase II. Bioscience, Biotechnology, and Biochemistry 72:10, pages 2739-2749.
Read now
Read now
Claudiu T Supuran, Anna Di Fiore & Giuseppina De Simone. (2008) Carbonic anhydrase inhibitors as emerging drugs for the treatment of obesity. Expert Opinion on Emerging Drugs 13:2, pages 383-392.
Read now
Read now
Ismet Basaran, Selma Sinan, Umit Cakir, Mustafa Bulut, Oktay Arslan & Ozen Ozensoy. (2008) In vitro inhibition of cytosolic carbonic anhydrases I and II by some new dihydroxycoumarin compounds. Journal of Enzyme Inhibition and Medicinal Chemistry 23:1, pages 32-36.
Read now
Read now
Zahid H. Chohan. (2008) Metal-based sulfonamides: Their preparation, characterization and in-vitro antibacterial, antifungal & cytotoxic properties. X-ray structure of 4-[(2-hydroxybenzylidene) amino] benzenesulfonamide. Journal of Enzyme Inhibition and Medicinal Chemistry 23:1, pages 120-130.
Read now
Read now
Gabriela Laura Almajan, Stefania-Felicia Barbuceanu, Alessio innocenti, Andrea Scozzafava & Claudiu T. Supuran. (2008) Carbonic anhydrase inhibitors. Inhibition of the cytosolic and tumor-associated carbonic anhydrase isozymes I, II and IX with some 1,3,4-oxadiazole- and 1,2,4-triazole-thiols. Journal of Enzyme Inhibition and Medicinal Chemistry 23:1, pages 101-107.
Read now
Read now
Muhammad Zareef, Rashid Iqbal, NajimA. Al-Masoudi, JavidH. Zaidi, Muhammad Arfan & SohailA. Shahzad. (2007) Synthesis, Anti–HIV, and Antifungal Activity of New Benzensulfonamides Bearing the 2,5-Disubstituted-1,3,4-Oxadiazole Moiety. Phosphorus, Sulfur, and Silicon and the Related Elements 182:2, pages 281-298.
Read now
Read now
Andrea Scozzafava, Antonio Mastrolorenzo & Claudiu T Supuran. (2006) Carbonic anhydrase inhibitors and activators and their use in therapy. Expert Opinion on Therapeutic Patents 16:12, pages 1627-1664.
Read now
Read now
Brian W Clare & Claudiu T Supuran. (2006) A perspective on quantitative structure–activity relationships and carbonic anhydrase inhibitors. Expert Opinion on Drug Metabolism & Toxicology 2:1, pages 113-137.
Read now
Read now
Jean-Yves Winum, Andrea Scozzafava, Jean-Louis Montero & Claudiu T Supuran. (2006) The sulfamide motif in the design of enzyme inhibitors. Expert Opinion on Therapeutic Patents 16:1, pages 27-47.
Read now
Read now
Zahid H. Chohan, Ali U. Shaikh, Muhammad M. Naseer & Claudiu T. Supuran. (2006) In-vitro antibacterial, antifungal and cytotoxic properties of metal-based furanyl derived sulfonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 21:6, pages 771-781.
Read now
Read now
Muhammad Zareef, Alessio Innocenti, Rashid Iqbal, Javid H. Zaidi, Muhammad Arfan, Andrea Scozzafava & Claudiu T. Supuran. (2006) Carbonic anhydrase inhibitors. Inhibition of human tumor-associated isozymes IX and cytosolic isozymes I and II with some 1,3,4-oxadiazole-thiols. Journal of Enzyme Inhibition and Medicinal Chemistry 21:4, pages 351-359.
Read now
Read now
Franciszek Saczewski, Alessio Innocenti, Zdzisław Brzozowski, Jarosław Sławiński, Elżbieta Pomarnacka, Anita Kornicka, Andrea Scozzafava & Claudiu T. Supuran. (2006) Carbonic anhydrase inhibitors. Selective inhibition of human tumor-associated isozymes IX and XII and cytosolic isozymes I and II with some substituted-2-mercapto-benzenesulfonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 21:5, pages 563-568.
Read now
Read now
Craig
A. Obafemi & D.
A. Akinpelu. (2005) Synthesis and Antimicrobial Activity of Some 2(1H)-quinoxalinone-6-sulfonyl Derivatives. Phosphorus, Sulfur, and Silicon and the Related Elements 180:8, pages 1795-1807.
Read now
Read now
Shin Chung, Kyung Min Lim & Song Seok Shin. (2005) Profiles of COX-2 inhibitors: present and future. Expert Opinion on Therapeutic Patents 15:1, pages 9-32.
Read now
Read now
Jean-Yves Winum, Andrea Scozzafava, Jean-Louis Montero & Claudiu T Supuran. (2004) Therapeutic applications of sulfamates. Expert Opinion on Therapeutic Patents 14:9, pages 1273-1308.
Read now
Read now
Andrea Scozzafava, Antonio Mastrolorenzo & Claudiu T Supuran. (2004) Modulation of carbonic anhydrase activity and its applications in therapy. Expert Opinion on Therapeutic Patents 14:5, pages 667-702.
Read now
Read now
Silvia Pastorekova, Seppo Parkkila, Jaromir Pastorek & Claudiu T. Supuran. (2004) Review Article. Journal of Enzyme Inhibition and Medicinal Chemistry 19:3, pages 199-229.
Read now
Read now
Claudiu T Supuran. (2003) Carbonic anhydrase inhibitors in the treatment and prophylaxis of obesity. Expert Opinion on Therapeutic Patents 13:10, pages 1545-1550.
Read now
Read now
Francesco Abbate, Angela Casini, Andrea Scozzafava & Claudiu T. Supuran. (2003) Carbonic Anhydrase Inhibitors: X-ray Crystallographic Structure of the Adduct of Human Isozyme II with the Perfluorobenzoyl Analogue of Methazolamide. Implications for the Drug Design of Fluorinated Inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 18:4, pages 303-308.
Read now
Read now
Claudiu T Supuran. (2003) Indisulam: an anticancer sulfonamide in clinical development. Expert Opinion on Investigational Drugs 12:2, pages 283-287.
Read now
Read now
. (2002) N-Acylsulfonamide apoptosis promoters. Expert Opinion on Therapeutic Patents 12:10, pages 1571-1573.
Read now
Read now
Angela Casini, Andrea Scozzafava & Claudiu T Supuran. (2002) Sulfonamide derivatives with protease inhibitory action as anticancer, anti-inflammatory and antiviral agents. Expert Opinion on Therapeutic Patents 12:9, pages 1307-1327.
Read now
Read now
Claudiu T Supuran & Andrea Scozzafava. (2002) Applications of carbonic anhydrase inhibitors and activators in therapy. Expert Opinion on Therapeutic Patents 12:2, pages 217-242.
Read now
Read now
. (2001) Benzophenones as inhibitors of reverse transcriptase. Expert Opinion on Therapeutic Patents 11:10, pages 1637-1640.
Read now
Read now
Andrea Scozzafava, Antonio Mastrolorenzo & Claudiu T Supuran. (2001) Agents that target cysteine residues of biomolecules and their therapeutic potential. Expert Opinion on Therapeutic Patents 11:5, pages 765-787.
Read now
Read now
Claudiu T Supuran, Andrea Scozzafava & Antonio Mastrolorenzo. (2001) Bacterial proteases: current therapeutic use and future prospects for the development of new antibiotics. Expert Opinion on Therapeutic Patents 11:2, pages 221-259.
Read now
Read now
Andrea Scozzafava, Antonio Mastrolorenzo & Claudiu T. Supuran. (2001) Antimycobacterial Activity of 3,4-dichlorophenyl-ureas, N,N-diphenyl-ureas and Related Derivatives. Journal of Enzyme Inhibition 16:5, pages 425-432.
Read now
Read now
Andrea Scozzafava, Ioana Saramet, Mircea D. Banciu & Claudiu T. Supuran. (2001) Carbonic Anhydrase Activity Modulators: Synthesis of Inhibitors and Activators Incorporating 2-substituted-thiazol-4-yl-methyl Scaffolds. Journal of Enzyme Inhibition 16:4, pages 351-358.
Read now
Read now
Celine Chazalette, Monique Riviere-Baudet, Andrea Scozzafava, Francesco Abbate, Zahra Ben Maarouf & Claudiu T. Supuran. (2001) Carbonic Anhydrase Inhibitors, Interaction of Boron Derivatives with Isozymes I and II: A New Binding Site for Hydrophobic Inhibitors at the Entrance of the Active Site as shown by Docking Studies. Journal of Enzyme Inhibition 16:2, pages 125-133.
Read now
Read now
Angela Casini, Francesco Mincione, Marc A. Ilies, Luca Menabuoni, Andrea Scozzafava & Claudiu T. Supuran. (2001) Carbonic Anhydrase Inhibitors: Synthesis and Inhibition Against Isozymes I, II and IV of Topically Acting Antiglaucoma Sulfonamides Incorporating cis-5-Norbornene-endo-3-Carboxy-2-Carboxamido Moieties. Journal of Enzyme Inhibition 16:2, pages 113-123.
Read now
Read now
Andrea Scozzafava, Antonio Mastrolorenzo & Claudiu T. Supuran. (2001) Arylsulfonyl-N,N-dialkyl-dithiocarbamates as Tumor Cell Growth Inhibitors: Novel Agents Targeting β-Tubulin?. Journal of Enzyme Inhibition 16:1, pages 55-63.
Read now
Read now
. (2000) Compounds for the treatment of oestrogen-dependent illnesses. Expert Opinion on Therapeutic Patents 10:11, pages 1771-1775.
Read now
Read now
Takashi Owa & Takeshi Nagasu. (2000) Novel sulphonamide derivatives for the treatment of cancer. Expert Opinion on Therapeutic Patents 10:11, pages 1725-1740.
Read now
Read now
. (2000) Novel compounds that interact with zinc finger proteins. Expert Opinion on Therapeutic Patents 10:8, pages 1289-1292.
Read now
Read now
Antonio Mastrolorenzo, Andrea Scozzafava & Claudiu T. Supuran. (2000) Antifungal Activity of Ag(I) and Zn(Ii) Complexes of Aminobenzolamide (5-Sulfanilylamido-1,3,4-Thiadiazole-2-Sulfonamide) Derivatives. Journal of Enzyme Inhibition 15:6, pages 517-531.
Read now
Read now
Articles from other publishers (378)
Ulviye Acar Çevik, Ayşen Işık, Ravikumar Kapavarapu, Kaan Küçükoğlu, Hayrunnisa Nadaroglu, Hayrani Eren Bostancı, Yusuf Özkay & Zafer Asım Kaplancıklı. (2024) Design, synthesis and biological evaluation of novel ketone derivatives containing benzimidazole and 1,3,4-triazole as CA inhibitors. Journal of Molecular Structure 1295, pages 136770.
Crossref
Crossref
Adel S. El-Azab, Alaa A.-M. Abdel-Aziz, Silvia Bua, Alessio Nocentini, Ahmed H. Bakheit, Hamad M. Alkahtani, Mohamed M. Hefnawy & Claudiu T. Supuran. (2023) Design, synthesis, and carbonic anhydrase inhibition activities of Schiff bases incorporating benzenesulfonamide scaffold: Molecular docking application. Saudi Pharmaceutical Journal 31:12, pages 101866.
Crossref
Crossref
Delal Erzurum, Derya Osmaniye, Begüm Nurpelin Sağlık, Serkan Levent, Yusuf Özkay & Zafer Asım Kaplancıklı. (2023) Design, synthesis, and biological activity studies of carbonic anhydrase inhibitors. Zeitschrift für Naturforschung C 78:11-12, pages 421-432.
Crossref
Crossref
Sachin B. Pandya, Bhavesh N. Socha, Rahul P. Dubey, Urmila H. Patel, R. H. Patel, Bhupesh S. Bhatt, Parth Thakor, Sanjay Bhakhar, Nikhil Vekariya & Jignesh Valand. (2023) Visible light-driven photocatalysts, quantum chemical calculations, ADMET-SAR parameters, and DNA binding studies of nickel complex of sulfadiazine. Scientific Reports 13:1.
Crossref
Crossref
İsmail Çelik, Ulviye Acar Çevik, Kaan Küçükoğlu, Hayrunnisa Nadaroglu, Hayrani Eren Bostancı, Ayşen Işık, Yusuf Özkay & Zafer Asım Kaplancıklı. (2023)
Design, synthesis, and molecular docking studies of benzimidazole‐1,3,4‐triazole hybrids as carbonic anhydrase I and
II
inhibitors
. Chemical Biology & Drug Design.
Crossref
Crossref
Merve Taşcı, Mustafa Arslan, Kübra Çıkrıkcı, Adem Ergun, Nahit Gençer & Oktay Arslan. (2023) Synthesis and Investigation of Carbonic Anhydrase I and II Activity of Dihydrobenzo[h]Quinazolin-2-yl Thiourea Compounds. Pharmaceutical Chemistry Journal 57:6, pages 899-906.
Crossref
Crossref
Serpil Gerni, Cansu Ozturk, Zuleyha Almaz, Cetin Bayrak & Ayse Tan. (2023) Celecoxib Derivatives Containing Pyrazole Linked‐Sulfonamide Moiety: Carbonic Anhydrase I–II and Acetylcholinesterase Inhibition Profiles, Molecular Docking Studies. ChemistrySelect 8:29.
Crossref
Crossref
Krishna K. Chinchilli, Priti Singh, Baijayantimala Swain, Nerella S. Goud, Dilep K. Sigalapalli, Abhishek Choli, Andrea Angeli, Srinivas Nanduri, Venkata M. Yaddanapudi, Claudiu T. Supuran & Mohammed Arifuddin. (2023) Development of Novel Indole-3-sulfonamide-heteroaryl Hybrids as Carbonic
Anhydrase Inhibitors: Design, Synthesis and in-vitro Screening. Anti-Cancer Agents in Medicinal Chemistry 23:11, pages 1225-1233.
Crossref
Crossref
Krishna Kartheek Chinchilli, Ravikumar Akunuri, Shaik Mahammad Ghouse, Devandla Soujanya, Andrea Angeli, Ramulu Parupalli, Mohammed Arifuddin, Venkata Madhavi Yaddanapudi, Claudiu T. Supuran & Srinivas Nanduri. (2023) Design, synthesis, and structure–activity studies of new rhodanine derivatives as carbonic anhydrase II, IX inhibitors. Archiv der Pharmazie.
Crossref
Crossref
Yao Zheng, Cai Chen, Mengli Wang, Ali Shoaib Moawad, Xiaoyan Wang & Chengyi Song. (2023) SINE Insertion in the Pig Carbonic Anhydrase 5B (CA5B) Gene Is Associated with Changes in Gene Expression and Phenotypic Variation. Animals 13:12, pages 1942.
Crossref
Crossref
Hakan Şahal, Önder İdil, Erdal Canpolat & Mustafa Özkan. (2023) Cu(II) Complexes of New Sulfa Drug Schiff Base Ligands: Synthesis, Structural Characterization, Antimicrobial Activities, and Time-Killing Kinetics. Russian Journal of Bioorganic Chemistry 49:3, pages 602-609.
Crossref
Crossref
Ahmad Badreddin Musatat, Alparslan Atahan, Adem Ergün, Kübra Çıkrıkcı, Nahit Gençer, Oktay Arslan & Mustafa Zengin. (2023) Synthesis, enzyme inhibition, and molecular docking studies of a novel chalcone series bearing benzothiazole scaffold. Biotechnology and Applied Biochemistry 70:3, pages 1357-1370.
Crossref
Crossref
T. N. Borodina, V. I. Smirnov, V. Yu. Serykh & I. B. Rozentsveig. (2023) Structural and theoretical study of π-stacking interactions in new complexes based on CuCl2 and 3-sulfonamide-substituted imidazo[2,1-b]thiazoles. Journal of Molecular Modeling 29:5.
Crossref
Crossref
Büşra ÇALIŞKAN, Mine AKSOY, Muhammet Serhat ÖZASLAN & İlknur AKYOL SALMAN. (2023) Investigation of Some Metabolic Enzyme Activities in Samples of Serum and Humor Aqueous of Cataract Cases with Pseudoexfoliation Syndrome. Türk Doğa ve Fen Dergisi 12:1, pages 163-170.
Crossref
Crossref
Kaan Kucukoglu, Nagihan Faydali, Dilek Bul, Hayrunnisa Nadaroglu, Belgin Sever, Mehlika Dilek Altıntop, Bahadır Ozturk & Ilkay Guzel. (2023) Synthesis, in silico and in vitro evaluation of new 3,5-disubstituted-1,2,4-oxadiazole derivatives as carbonic anhydrase inhibitors and cytotoxic agents. Journal of Molecular Structure 1276, pages 134699.
Crossref
Crossref
Ahmed N. Al-Rawahi, Raeid M. M. Abed, Najeeb Ur Rehman, Kashif Rafiq, Ajmal Khan, Abdul L. Khan, Majid Khan, Sobia Ahsan Halim, Fahad Al-Senafi, Huda Mahmoud & Ahmed Al-Harrasi. (2023) New Sulfur-Containing Diketopiperazine from Marine-Derived Bacteria Streptomyces rochei sp. 81 with Potent Carbonic Anhydrase II Inhibition. Chemistry of Natural Compounds 59:2, pages 346-350.
Crossref
Crossref
Feyzi Sinan Tokalı, Zuhal Alım & Ümit Yırtıcı. (2023) Carboxylate‐ and Sulfonate‐Containing Quinazolin‐4(3H)‐one Rings: Synthesis, Characterization, and Carbonic Anhydrase I–II and Acetylcholinesterase Inhibition Properties. ChemistrySelect 8:8.
Crossref
Crossref
Lalit Vats, Kiran Siwach, Andrea Angeli, Prerna Bikal, Jitender Kumar Bhardwaj, Claudiu T. Supuran & Pawan K. Sharma. (2022) Tail approach synthesis of triazolylthiazolotriazole bearing benzenesulfonamides as carbonic anhydrase inhibitors capable of inducing apoptosis. Archiv der Pharmazie 356:2.
Crossref
Crossref
Ashok Aspatwar, Claudiu T. Supuran, Abdul Waheed, William S. Sly & Seppo Parkkila. (2022) Mitochondrial carbonic anhydrase VA and VB: properties and roles in health and disease. The Journal of Physiology 601:2, pages 257-274.
Crossref
Crossref
Claudiu T. Supuran. 2023. Nitric Oxide in Health and Disease. Nitric Oxide in Health and Disease
305
317
.
Arti GuptaViney LatherDushyanth R. VennapuSandeep KumarMallikarjun. B.P.Neerupma DhimanArchana Sharma. (2022) 3D-QSAR, E-pharmacophore and molecular docking to explore substituted sulfonamides as carbonic anhydrase inhibitors in epilepsy. Research Journal of Pharmacy and Technology, pages 5521-5528.
Crossref
Crossref
Pervaiz Ali Channar, Rima D. Alharthy, Syeda Abida Ejaz, Aamer Saeed & Jamshed Iqbal. (2022) Synthesis, Biological Evaluation, and Molecular Dynamics of Carbothioamides Derivatives as Carbonic Anhydrase II and 15-Lipoxygenase Inhibitors. Molecules 27:24, pages 8723.
Crossref
Crossref
Evgenia G. Matveeva, Andrea K. Stoddard, Hui-Hui Zeng, Graham Franke, Leslie Bourne, Carol A. Fierke & Richard B. Thompson. (2022) Ratiometric Zinc Biosensor Based on Bioluminescence Resonance Energy Transfer: Trace Metal Ion Determination with Tunable Response. International Journal of Molecular Sciences 23:23, pages 14936.
Crossref
Crossref
Majid Khan, Syed Raza Shah, Faizullah Khan, Sobia Ahsan Halim, Shaikh Mizanoor Rahman, Mohammad Khalid, Ajmal Khan & Ahmed Al-Harrasi. (2022) Efficient Synthesis with Green Chemistry Approach of Novel Pharmacophores of Imidazole-Based Hybrids for Tumor Treatment: Mechanistic Insights from In Situ to In Silico. Cancers 14:20, pages 5079.
Crossref
Crossref
Mohammed Hadj Mortada Belhachemi, Abdelmadjid Benmohammed, Halima Saiah, Nourdine Boukabcha, Merzouk Saidj, Necmi Dege, Ayada Djafri & Abdelkader Chouaih. (2022) Synthesis, structural determination, molecular docking and biological activity of 1-(4-fluorobenzyl)-5-bromolindolin-2,3-dione. Journal of Molecular Structure 1265, pages 133342.
Crossref
Crossref
Alfredo Fabrizio Lo Faro, Anastasio Tini, Giulia Bambagiotti, Filippo Pirani, Andrea Faragalli, Flavia Carle, Elena Pacella, Artan Ceka, Marco Moretti, Massimo Gottardi, Nicola Vito Lassandro, Michele Nicolai, Marco Lupidi, Cesare Mariotti, Francesco Paolo Busardò & Jeremy Carlier. (2022) Quantification of Carbonic Anhydrase Inhibitors and Metabolites in Urine and Hair of Patients and Their Relatives. Biology 11:10, pages 1379.
Crossref
Crossref
Md. Nazmul Islam, Md. Fahim Hasan, Aishwarja Dey, Bishwajit Bokshi, Asish Kumar Das, Samir Kumar Sadhu & Nripendra Nath Biswas. (2022) Identification of Potential Diuretic and Laxative Drug Candidates from Avicennia officinalis L. Bark through In Vivo Mice Model Studies and In Vitro Gas Chromatography-Mass Spectrometry and Molecular Docking Analysis. Evidence-Based Complementary and Alternative Medicine 2022, pages 1-14.
Crossref
Crossref
Işıl Nihan Korkmaz, Pınar Güller, Ramazan Kalın, Aykut Öztekin & Hasan Özdemir. (2022) In vitro Inhibition Profiles and Molecular Docking Analysis of Benzohydrazide
Derivatives on Red Blood Cell Carbonic Anhydrases Isozymes. Current Computer-Aided Drug Design 18:5, pages 381-392.
Crossref
Crossref
Khawla Bechlem, Malika Berredjem, Seif Eddine Djouad, Tan Ouk Sothea, Sofiane Bouacida, Christelle Marminon, Taibi Ben Hadda, Jaques Lebreton & Abdeslem Bouzina. (2022) Novel N-acylsulfamoyl-oxazolidin-2ones: Synthesis, antitumor activity, X-ray crystallographic study, molecular docking and POM analyses. Journal of Molecular Structure 1262, pages 132935.
Crossref
Crossref
Francesco P. Busardò, Alfredo F. Lo Faro, Ascanio Sirignano, Raffaele Giorgetti & Jeremy Carlier. (2022) In silico, in vitro, and in vivo human metabolism of acetazolamide, a carbonic anhydrase inhibitor and common “diuretic and masking agent” in doping. Archives of Toxicology 96:7, pages 1989-2001.
Crossref
Crossref
Erbay KALAY. (2022) Synthesis and Characterization of Novel Hybrid Sulfonamide Molecules with Benzothiazole Scaffold. Iğdır Üniversitesi Fen Bilimleri Enstitüsü Dergisi 12:2, pages 899-907.
Crossref
Crossref
Emel Karakılıç, Zuhal Alım, Aslıhan Günel & Arif Baran. (2022) A versatile study of novel A3B-type unsymmetric zinc(II) phthalocyanines containing thiazolidin-4-one: Their, carbonic anhydrase I, II isoenzymes, and xanthine oxidase inhibitors evaluation. Journal of Molecular Structure 1257, pages 132630.
Crossref
Crossref
Nuri YORULMAZ, Hilal ÖZTÜRK & Mustafa DURGUN. (2022) Evaluation of Some Sulfonamide Derivatives as a Potential Inhibitors of The Carbonic Anhydrase IX/XII by ADME and Molecular Docking Method. Adıyaman University Journal of Science.
Crossref
Crossref
Valeria Poggetti, Silvia Salerno, Emma Baglini, Elisabetta Barresi, Federico Da Settimo & Sabrina Taliani. (2022) Carbonic Anhydrase Activators for Neurodegeneration: An Overview. Molecules 27:8, pages 2544.
Crossref
Crossref
Najeeb Ur Rehman, Sobia Ahsan Halim, Ajmal Khan, Majid Khan, Saif Al-Hatmi & Ahmed Al-Harrasi. (2022) Commikuanoids A-C: New cycloartane triterpenoids with exploration of carbonic anhydrase-II inhibition from the resins of Commiphora kua by in vitro and in silico molecular docking. Fitoterapia 157, pages 105125.
Crossref
Crossref
Emel Karakılıç, Zuhal Alım, Mustafa Emirik & Arif Baran. (2021) Some characteristics of new and innovative COX inhibitor derivatives: Potent hCA‐I and hCA‐II inhibitors supported by molecular docking studies. Applied Organometallic Chemistry 36:3.
Crossref
Crossref
Ahmed Elkamhawy, Jiyu Woo, Hossam Nada, Andrea Angeli, Tarek M. Bedair, Claudiu T. Supuran & Kyeong Lee. (2022) Identification of Novel and Potent Indole-Based Benzenesulfonamides as Selective Human Carbonic Anhydrase II Inhibitors: Design, Synthesis, In Vitro, and In Silico Studies. International Journal of Molecular Sciences 23:5, pages 2540.
Crossref
Crossref
Chaofu Yang, Xianyu Sun, Zhan Li, Yunyun Cheng, Yu Lei, Liang Lu, Xuan Liu, Xiaomei Zhuang, Tao Wang & Xinhua He. (2022) The effect of benzenesulfonamide's side chains on their human carbonic anhydrase Ⅰ/Ⅱ inhibitory activities. Journal of Molecular Structure 1250, pages 131927.
Crossref
Crossref
BETÜL AYGÜN, AHMET A. BERBER, MERVE A. DOGANCI, NURCAN BERBER, SELEN ŞEN, ESRA YILDIZ & HÜSEYIN AKSOY. (2022) Genotoxicity evaluation of a new phthalazine substituted β-lactam derivative in human lymphocytes. Anais da Academia Brasileira de Ciências 94:1.
Crossref
Crossref
T.N. Borodina, V.I. Smirnov, V.Yu. Serykh & I.B. Rozentsveig. (2022) π-Stacking interactions in new arylsulphonylamine-substituted derivatives of imidazo[2,1-b]thiazol. Journal of Molecular Structure 1248, pages 131423.
Crossref
Crossref
Aamer Saeed, Shafi Ullah Khan, Maria Saeed, Ghulam Shabir, Abbas Hasan, Rasheed Ahmad Khera, Hesham El‐Seedi, Sobia Ahsan Halim, Ajmal Khan, Ahmed Al‐Harrasi & Jamshed Iqbal. (2021)
Synthesis of novel hybrid pharmacophore of
N
‐((
4‐sulfamoylphenyl
)carbamothioyl)alkanamides as potent carbonic
anhydrase‐II
and
15‐lipoxygenase
inhibitors
. Drug Development Research.
Crossref
Crossref
Xin Wang, Yan-lian Feng, Xiao-yu Zhao, Ran An, Chun Cao, Meng-bi Guo, Rui Zhang, Yuan-xin Wang, Zhuang Hou & Chun Guo. (2021) Discovery of novel aminosaccharide-based sulfonamide derivatives as potential carbonic anhydrase II inhibitors. Bioorganic & Medicinal Chemistry Letters 53, pages 128420.
Crossref
Crossref
Bashistha Kumar Kanth & Seung Pil Pack. (2021) Carbonic Anhydrase as CO2 capturing agent: its Classes and Catalytic Mechanisms. International Journal of Mathematics and Computers in Simulation 15, pages 102-106.
Crossref
Crossref
Madhuri Pandiri, Satheesh Kumar Nukala, Gouthami Dasari, Vinitha Badithapuram & Srinivas Bandari. (2021) Design and Synthesis of Some New N-Phenyl-[1,2,4]triazolo[4,3-a]quinoxaline-1-sulfonamide Derivatives and Their Anti-Cancer Activity. Russian Journal of General Chemistry 91:11, pages 2280-2285.
Crossref
Crossref
Aamer Saeed, Syeda Abida Ejaz, Anwar Ul-Hamid, Hesham R. El-Seedi & Jamshed Iqbal. (2021) Synthesis of and molecular docking studies of azomethine- tethered sulfonamides as carbonic anhydrase II & 15-lipoxygenase inhibitors. Journal of Molecular Structure 1243, pages 130821.
Crossref
Crossref
Zhuang Hou, Qiang Cai & Mao-sheng Cheng. (2021) Novel carbohydrate-based sulfonamide derivatives as selective carbonic anhydrase II inhibitors: Synthesis, biological and molecular docking analysis. Bioorganic & Medicinal Chemistry Letters 51, pages 128291.
Crossref
Crossref
Emanuela Berrino, Bastien Michelet, Agnès Martin‐Mingot, Fabrizio Carta, Claudiu T. Supuran & Sébastien Thibaudeau. (2021) Modulating the Efficacy of Carbonic Anhydrase Inhibitors through Fluorine Substitution. Angewandte Chemie International Edition 60:43, pages 23068-23082.
Crossref
Crossref
Emanuela Berrino, Bastien Michelet, Agnès Martin‐Mingot, Fabrizio Carta, Claudiu T. Supuran & Sébastien Thibaudeau. (2021) Modulating the Efficacy of Carbonic Anhydrase Inhibitors through Fluorine Substitution. Angewandte Chemie 133:43, pages 23252-23266.
Crossref
Crossref
Pınar Güller, Ziya Dağalan, Uğur Güller, Ulaş Çalışır & Bilal Nişancı. (2021) Enzymes inhibition profiles and antibacterial activities of benzylidenemalononitrile derivatives. Journal of Molecular Structure 1239, pages 130498.
Crossref
Crossref
Phatsawee Jansook, Hay Marn Hnin, Thorsteinn Loftsson & Einar Stefánsson. (2021) Cyclodextrin-based formulation of carbonic anhydrase inhibitors for ocular delivery – A review. International Journal of Pharmaceutics 606, pages 120955.
Crossref
Crossref
Semih GÜLER, Hatice Gamze SOĞUKÖMEROĞULLARI, Sadin ÖZDEMİR, Mustafa Serkan YALÇIN & Mehmet SÖNMEZ. (2021) New Carboxamid ligand and its metal complexes containing sulfonamide group: Synthesis, Characterization, DNA cleavage and antimicrobial activitySülfonamid Grubu İçeren Yeni Karboksamid Ligand ve Metal Kompleksleri: Sentez, Karakterizasyon, DNA Bölünmesi ve Antimikrobiyal Aktivite. Erzincan Üniversitesi Fen Bilimleri Enstitüsü Dergisi 14:2, pages 724-736.
Crossref
Crossref
Pınar Güller, Ufuk Atmaca, Uğur Güller, Ulaş Çalışır & Feray Dursun. (2021) Antibacterial properties and carbonic anhydrase inhibition profiles of azido sulfonyl carbamate derivatives. Future Medicinal Chemistry 13:15, pages 1285-1299.
Crossref
Crossref
Alexey S. Pospelov, Tommi Ala‐Kurikka, Samu Kurki, Juha Voipio & Kai Kaila. (2021) Carbonic anhydrase inhibitors suppress seizures in a rat model of birth asphyxia. Epilepsia 62:8, pages 1971-1984.
Crossref
Crossref
Musa Erdoğan, Leyla Polat Köse, Selçuk Eşsiz & İlhami Gülçin. (2021) Synthesis and biological evaluation of some 1‐naphthol derivatives as antioxidants, acetylcholinesterase, and carbonic anhydrase inhibitors. Archiv der Pharmazie 354:8, pages 2100113.
Crossref
Crossref
Tuğba Kul Köprülü, Salih Ökten, Vildan Enisoğlu Atalay, Şaban Tekin & Osman Çakmak. (2021) Biological activity and molecular docking studies of some new quinolines as potent anticancer agents. Medical Oncology 38:7.
Crossref
Crossref
Baijayantimala Swain, Kamtam Aashritha, Priti Singh, Andrea Angeli, Abhay Kothari, Dilep K. Sigalapalli, Venkata M. Yaddanapudi, Claudiu T. Supuran & Mohammed Arifuddin. (2021)
Design and synthesis of benzenesulfonamide‐linked imidazo[2,1‐
b
][1,3,4]thiadiazole derivatives as carbonic anhydrase I and II inhibitors
. Archiv der Pharmazie 354:7.
Crossref
Crossref
Marwa F. Ahmed & Eman Y. Santali. (2021) Discovery of pyridine- sulfonamide hybrids as a new scaffold for the development of potential VEGFR-2 inhibitors and apoptosis inducers. Bioorganic Chemistry 111, pages 104842.
Crossref
Crossref
Nadini Thushara, Taniya Darshani, Sameera R. Samarakoon, Inoka C. Perera, Frank R. Fronczek, W. M. C. Sameera & Theshini Perera. (2021) Synthesis, characterization and biological evaluation of dipicolylamine sulfonamide derivatized platinum complexes as potential anticancer agents. RSC Advances 11:29, pages 17658-17668.
Crossref
Crossref
O. V. Kovalchukova, V. P. Kazachenko, V. V. Tkachev, A. N. Utenyshev, N. N. Strakhova & A. N. Proshin. (2021) Crystal Structure and Physicochemical Characteristics of Two Novel Adamantane Derivatives of Sulfonamides. Crystallography Reports 66:3, pages 424-428.
Crossref
Crossref
Farhan M. Khan, Muhammad A. Abbasi, Aziz‐ur‐Rehman, Sabahat Z. Siddiqui, Abdul R. Sadiq Butt, Hussain Raza, Ayesha Zafar, Syed A. Ali Shah, Muhammad Shahid & Sung‐Yum Seo. (2021) Convergent synthesis of carbonic anhydrase inhibiting bi‐heterocyclic benzamides: Structure–activity relationship and mechanistic explorations through enzyme inhibition, kinetics, and computational studies. Journal of Heterocyclic Chemistry 58:5, pages 1089-1103.
Crossref
Crossref
Baijayantimala Swain, Abhay, Priti Singh, Andrea Angeli, Kamtam Aashritha, Narayana Nagesh, Claudiu T. Supuran & Mohammed Arifuddin. (2021) 3-Functionalised benzenesulphonamide based 1,3,4-oxadiazoles as selective carbonic anhydrase XIII inhibitors: Design, synthesis and biological evaluation. Bioorganic & Medicinal Chemistry Letters 37, pages 127856.
Crossref
Crossref
Agnieszka Wróbel & Danuta Drozdowska. (2021) Recent Design and Structure-Activity Relationship Studies on the Modifications of DHFR Inhibitors as Anticancer Agents. Current Medicinal Chemistry 28:5, pages 910-939.
Crossref
Crossref
Shubham Kumar, Sandeep Rulhania, Shalini Jaswal & Vikramdeep Monga. (2021) Recent advances in the medicinal chemistry of carbonic anhydrase inhibitors. European Journal of Medicinal Chemistry 209, pages 112923.
Crossref
Crossref
Sinan Bilginer, Halise I. Gul, Baris Anil, Yeliz Demir & Ilhami Gulcin. (2020) Synthesis and in silico studies of triazene‐substituted sulfamerazine derivatives as acetylcholinesterase and carbonic anhydrases inhibitors. Archiv der Pharmazie 354:1, pages 2000243.
Crossref
Crossref
Muhammad Danish, Muhammad Asam Raza, Hirra Khalid, Umara Iftikhar & Muhammad Nadeem Arshad. (2020) New metal complexes of sulfonamide: Synthesis, characterization, in‐vitro anticancer, anticholinesterase, antioxidant, and antibacterial studies. Applied Organometallic Chemistry 35:1.
Crossref
Crossref
Nurcan Berber, Mustafa Arslan, Fırat Vural, Adem Ergun, Nahit Gençer & Oktay Arslan. (2020)
Synthesis of new series of thiazol‐(2(3
H
)‐ylideneamino)benzenesulfonamide derivatives as carbonic anhydrase inhibitors
. Journal of Biochemical and Molecular Toxicology 34:12.
Crossref
Crossref
Shuang Hao, Xue Cheng, Xin Wang, Ran An, Hang Xu, Mengbi Guo, Chuanchao Li, Yitong Wang, Zhuang Hou & Chun Guo. (2020) Design, synthesis and biological evaluation of novel carbohydrate-based sulfonamide derivatives as antitumor agents. Bioorganic Chemistry 104, pages 104237.
Crossref
Crossref
Chandra B. Mishra, Manisha Tiwari & Claudiu T. Supuran. (2020) Progress in the development of human carbonic anhydrase inhibitors and their pharmacological applications: Where are we today?. Medicinal Research Reviews 40:6, pages 2485-2565.
Crossref
Crossref
Giosuè Costa, Annalisa Maruca, Roberta Rocca, Francesca Alessandra Ambrosio, Emanuela Berrino, Fabrizio Carta, Francesco Mesiti, Alessandro Salatino, Delia Lanzillotta, Francesco Trapasso, Anna Artese, Stefano Alcaro & Claudiu T. Supuran. (2020) In Silico Identification and Biological Evaluation of Antioxidant Food Components Endowed with Human Carbonic Anhydrase IX and XII Inhibition. Antioxidants 9:9, pages 775.
Crossref
Crossref
Satheesh Kumar Dende, Raghu Babu KorupoluKrishnakanth Reddy Leleti. (2020)
Design and Synthesis of Sulfonamide‐Attached 2‐(Isoxazol‐3‐yl)‐1
H
‐imidazoles as Anticancer Agents
. ChemistrySelect 5:26, pages 7919-7922.
Crossref
Crossref
Chaofu Yang, Jing Wang, Yunyun Cheng, Xu Yang, Yan Feng, Xiaomei Zhuang, Zhenwang Li, Wangyu Zhao, Jiwen Zhang, Xianyu Sun & Xinhua He. (2020) N-Quinary heterocycle-4-sulphamoylbenzamides exert anti-hypoxic effects as dual inhibitors of carbonic anhydrases I/II. Bioorganic Chemistry 100, pages 103931.
Crossref
Crossref
Ishaq Yahaya Lawan, Mohammed Muftahu Beli, Mohammed Adamu, Fatima Baba Isah & Maryam Abubakar. (2020) Schiff Base of Metal Complex Derived from Glycine and Benzaldehyde. Earthline Journal of Chemical Sciences, pages 105-114.
Crossref
Crossref
Essam M. Hussein, Munirah M. Al-Rooqi, Amal A. Elkhawaga & Saleh A. Ahmed. (2020) Tailoring of novel biologically active molecules based on N-substituted sulfonamides bearing thiazole moiety exhibiting unique multi-addressable biological potentials. Arabian Journal of Chemistry 13:5, pages 5345-5362.
Crossref
Crossref
Ali Irfan, Laila Rubab, Mishbah Ur Rehman, Rukhsana Anjum, Sami Ullah, Mahwish Marjana, Saba Qadeer & Sadia Sana. (2020) Coumarin sulfonamide derivatives: An emerging class of therapeutic agents. Heterocyclic Communications 26:1, pages 46-59.
Crossref
Crossref
Bahar Yilmaz, Abdullah Tahir Bayrac & Mevlut Bayrakci. (2019) Evaluation of Anticancer Activities of Novel Facile Synthesized Calix[n]arene Sulfonamide Analogs. Applied Biochemistry and Biotechnology 190:4, pages 1484-1497.
Crossref
Crossref
Chaofu Yang, Yan Feng, Xu Yang, Mingxia Sun, Zhenwang Li, Xuan Liu, Liang Lu, Xianyu Sun, Jiwen Zhang & Xinhua He. (2020) Synthesis and evaluation of 4-(1,3,4-oxadiazol-2-yl)-benzenesulfonamides as potent carbonic anhydrase inhibitors. Bioorganic & Medicinal Chemistry Letters 30:2, pages 126874.
Crossref
Crossref
Soumajit Ghorai, Sravani Pulya, Kalyan Ghosh, Parthasarathi Panda, Balaram Ghosh & Shovanlal Gayen. (2020) Structure-activity relationship of human carbonic anhydrase-II inhibitors: Detailed insight for future development as anti-glaucoma agents. Bioorganic Chemistry 95, pages 103557.
Crossref
Crossref
Marcelo Luís Occhiutto, Raul C. Maranhão, Vital Paulino Costa & Anastasios G. Konstas. (2019) Nanotechnology for Medical and Surgical Glaucoma Therapy—A Review. Advances in Therapy 37:1, pages 155-199.
Crossref
Crossref
Maximilian Bremerich, Christian M. Conrads, Tim Langletz & Carsten Bolm. (2019)
Additions to
N
‐Sulfinylamines as an Approach for the Metal‐free Synthesis of Sulfonimidamides:
O
‐Benzotriazolyl Sulfonimidates as Activated Intermediates
. Angewandte Chemie International Edition 58:52, pages 19014-19020.
Crossref
Crossref
Maximilian Bremerich, Christian M. Conrads, Tim Langletz & Carsten Bolm. (2019)
Additions to
N
‐Sulfinylamines as an Approach for the Metal‐free Synthesis of Sulfonimidamides:
O
‐Benzotriazolyl Sulfonimidates as Activated Intermediates
. Angewandte Chemie 131:52, pages 19190-19196.
Crossref
Crossref
Essam M. Hussein, Munirah M. Al-Rooqi, Shimaa M. Abd El-Galil & Saleh A. Ahmed. (2019) Design, synthesis, and biological evaluation of novel N4-substituted sulfonamides: acetamides derivatives as dihydrofolate reductase (DHFR) inhibitors. BMC Chemistry 13:1.
Crossref
Crossref
Aleksandr V. Pavliuk, Yurii V. Bezugly, Vladimir V. Sukhoveev & Vladimir I. Kashkovsky. (2019) A convenient method for efficient synthesis of isoxazole-containing thiadiazepine derivatives. Chemistry of Heterocyclic Compounds 55:12, pages 1274-1277.
Crossref
Crossref
Raquel L. Bernardino, David F. Carrageta, Mário Sousa, Marco G. Alves & Pedro F. Oliveira. (2019) pH and male fertility: making sense on pH homeodynamics throughout the male reproductive tract. Cellular and Molecular Life Sciences 76:19, pages 3783-3800.
Crossref
Crossref
Seyed-Omar Zaraei, Mohammed I. El-Gamal, Zainab Shafique, Sayyeda Tayyeba Amjad, Saifullah Afridi, Sumera Zaib, Hanan S. Anbar, Randa El-Gamal & Jamshed Iqbal. (2019) Sulfonate and sulfamate derivatives possessing benzofuran or benzothiophene nucleus as potent carbonic anhydrase II/IX/XII inhibitors. Bioorganic & Medicinal Chemistry 27:17, pages 3889-3901.
Crossref
Crossref
Vladimir Amirkhanov, Abdur Rauf, Taibi Ben Hadda, Vladimir Ovchynnikov, Viktor Trush, Muhammad Saleem, Muslam Raza, Tayyeba Rehman, Hsaine Zgou, Usama Shaheen & Thoraya A. Farghaly. (2019) Pharmacophores Modeling in Terms of Prediction of Theoretical Physicochemical Properties and Verification by EXPERIMENTAL correlations of Carbacylamidophosphates (CAPh) and Sulfanylamidophosphates (SAPh) Tested as New Carbonic Anhydrase Inhibitors. Mini-Reviews in Medicinal Chemistry 19:12, pages 1015-1027.
Crossref
Crossref
Kübra Demir-Yazıcı, Silvia Bua, Nurgül Mutlu Akgüneş, Atilla Akdemir, Claudiu T. Supuran & Özlen Güzel-Akdemir. (2019) Indole-Based Hydrazones Containing A Sulfonamide Moiety as Selective Inhibitors of Tumor-Associated Human Carbonic Anhydrase Isoforms IX and XII. International Journal of Molecular Sciences 20:9, pages 2354.
Crossref
Crossref
Radivojka Bánová Vulić, Martina Zdurienčíková, Silvia Tyčiaková, Oldřich Benada, Mária Dubrovčáková, Ján Lakota & Ľudovít Škultéty. (2019) Silencing of carbonic anhydrase I enhances the malignant potential of exosomes secreted by prostatic tumour cells. Journal of Cellular and Molecular Medicine 23:5, pages 3641-3655.
Crossref
Crossref
Attique Ahmed, Pervaiz Ali Channar, Aamer Saeed, Markus Kalesse, Mehar Ali Kazi, Fayaz Ali Larik, Qamar Abbas, Mubashir Hassan, Hussain Raza & Sung-Yum Seo. (2019) Synthesis of sulfonamide, amide and amine hybrid pharmacophore, an entry of new class of carbonic anhydrase II inhibitors and evaluation of chemo-informatics and binding analysis. Bioorganic Chemistry 86, pages 624-630.
Crossref
Crossref
Raquel L. Bernardino, Tânia R. Dias, Bruno P. Moreira, Mariana Cunha, Alberto Barros, Elsa Oliveira, Mário Sousa, Marco G. Alves & Pedro F. Oliveira. (2019) Carbonic anhydrases are involved in mitochondrial biogenesis and control the production of lactate by human Sertoli cells. The FEBS Journal 286:7, pages 1393-1406.
Crossref
Crossref
Nabih Lolak, Suleyman Akocak, Silvia Bua, Rajesh K.K. Sanku & Claudiu T. Supuran. (2019) Discovery of new ureido benzenesulfonamides incorporating 1,3,5-triazine moieties as carbonic anhydrase I, II, IX and XII inhibitors. Bioorganic & Medicinal Chemistry 27:8, pages 1588-1594.
Crossref
Crossref
Hongying Ma, Sheng Wang, Guorong Zeng, Jintu Guo, Minghao Guo, Xianggui Dong, Guoying Hua, Yu Liu, Min Wang, Yao Ling, Xiangdong Ding, Chunjiang Zhao & Changxin Wu. (2019) The Origin of a Coastal Indigenous Horse Breed in China Revealed by Genome-Wide SNP Data. Genes 10:3, pages 241.
Crossref
Crossref
Jamaluddin Mahar, Aamer Saeed, Kevin D. Belfield, Fayaz Ali Larik, Pervaiz Ali Channar, Mehar Ali Kazi, Qamar Abbas, Mubashir Hassan, Hussain Raza & Sung-Yum Seo. (2019) 1-(2-Hydroxy-5-((trimethylsilyl)ethynyl)phenyl)ethanone based α,β-unsaturated derivatives an alternate to non-sulfonamide carbonic anhydrase II inhibitors, synthesis via Sonogashira coupling, binding analysis, Lipinsk’s rule validation. Bioorganic Chemistry 84, pages 170-176.
Crossref
Crossref
Joydeb Chanda, Pulok K. Mukherjee, Rajarshi Biswas, Sayan Biswas, Amrendra Kumar Tiwari & Ashish Pargaonkar. (2018)
UPLC‐QTOF‐MS analysis of a carbonic anhydrase‐inhibiting extract and fractions of
Luffa acutangula
(L.) Roxb (ridge gourd)
. Phytochemical Analysis 30:2, pages 148-155.
Crossref
Crossref
Ali Akremi & Adel Noubigh. (2019) New organotin(IV) chlorides derived from N-(2-hydroxyphenyl)aryloxy sulfamates. Synthesis, characterization and DSC investigation. Journal of Chemical Sciences 131:2.
Crossref
Crossref
Olexandr V. Pavliuk, Yuriy V. Bezugly & Volodimir I. Kashkovsky. (2019) Ring closing metathesis strategies to isoxazole containing thiadiazepines. French-Ukrainian Journal of Chemistry 7:1, pages 104-112.
Crossref
Crossref
Mariana Rocha, Oscar E. Piro, Gustavo A. Echeverría, Ana C. Pastoriza, Melina A. Sgariglia, José R. Soberón & Diego M. Gil. (2019) Co(II), Ni(II) and Cu(II) ternary complexes with sulfadiazine and dimethylformamide: Synthesis, spectroscopic characterization, crystallographic study and antibacterial activity. Journal of Molecular Structure 1176, pages 605-613.
Crossref
Crossref
Chuang Zhao, K.P. Rakesh, L. Ravidar, Wan-Yin Fang & Hua-Li Qin. (2019) Pharmaceutical and medicinal significance of sulfur (SVI)-Containing motifs for drug discovery: A critical review. European Journal of Medicinal Chemistry 162, pages 679-734.
Crossref
Crossref
Emanuela Berrino & Fabrizio Carta. 2019. Carbonic Anhydrases. Carbonic Anhydrases
311
329
.
Silvia Bua, Alessio Nocentini & Claudiu T. Supuran. 2019. Carbonic Anhydrases. Carbonic Anhydrases
287
309
.
Li Liu, Wanqi Wang, Jin Huang, Zhenjiang Zhao, Honglin Li & Yufang Xu. (2018) Novel benzoyl thioureido benzene sulfonamides as highly potent and selective inhibitors of carbonic anhydrase IX: optimization and bioactive studies. MedChemComm 9:12, pages 2100-2105.
Crossref
Crossref
Anyaporn Sangkaew, Jerapan Krungkrai & Chulee Yompakdee. (2018) Development of a high throughput yeast-based screening assay for human carbonic anhydrase isozyme II inhibitors. AMB Express 8:1.
Crossref
Crossref
Loghman Alaei, Reza Khodarahmi, Vahid Sheikh-Hasani, Nader Sheibani & Ali A. Moosavi-Movahedi. (2018) Mechanistic investigation of sulfonamide ligands as human carbonic anhydrase II inhibitors. International Journal of Biological Macromolecules 120, pages 1198-1207.
Crossref
Crossref
Nesrin Buğday, F. Zehra Küçükbay, Hasan Küçükbay, Silvia Bua, Gianluca Bartolucci, Janis Leitans, Andris Kazaks, Kaspars Tars & Claudiu T. Supuran. (2018) Synthesis of novel dipeptide sulfonamide conjugates with effective carbonic anhydrase I, II, IX, and XII inhibitory properties. Bioorganic Chemistry 81, pages 311-318.
Crossref
Crossref
Shahla Daryadel, Ufuk Atmaca, Parham Taslimi, İlhami Gülçin & Murat Çelik. (2018) Novel sulfamate derivatives of menthol: Synthesis, characterization, and cholinesterases and carbonic anhydrase enzymes inhibition properties. Archiv der Pharmazie 351:11, pages 1800209.
Crossref
Crossref
Danish Idrees, Murtuza Hadianawala, Amarjyoti Das Mahapatra, Bhaskar Datta, Sonam Roy, Shahzaib Ahamad, Parvez Khan & Md. Imtaiyaz Hassan. (2018) Implication of sulfonylurea derivatives as prospective inhibitors of human carbonic anhydrase II. International Journal of Biological Macromolecules 115, pages 961-969.
Crossref
Crossref
Fuat Karakuş, Ergül Eyol, Kadir Yılmaz & Songül Ünüvar. (2018) In vitro effect of carbonic anhydrase inhibitor acetazolamide on cell viability, migration and colony formation of colorectal cancer cells. Biologia 73:6, pages 621-628.
Crossref
Crossref
Andrea K. SteigerYu ZhaoMichael D. Pluth. (2018) Emerging Roles of Carbonyl Sulfide in Chemical Biology: Sulfide Transporter or Gasotransmitter?. Antioxidants & Redox Signaling 28:16, pages 1516-1532.
Crossref
Crossref
Srishti Singh, Carrie Lomelino, Mam Mboge, Susan Frost & Robert McKenna. (2018) Cancer Drug Development of Carbonic Anhydrase Inhibitors beyond the Active Site. Molecules 23:5, pages 1045.
Crossref
Crossref
Saghir Abbas, Hafiza Huma Nasir, Sumera Zaib, Saqib Ali, Tariq Mahmood, Khurshid Ayub, Muhammad Nawaz Tahir & Jamshed Iqbal. (2018) Carbonic anhydrase inhibition of Schiff base derivative of imino-methyl-naphthalen-2-ol: Synthesis, structure elucidation, molecular docking, dynamic simulation and density functional theory calculations. Journal of Molecular Structure 1156, pages 193-200.
Crossref
Crossref
Fatemeh Mohammadipanah & Fatemeh Salimi. (2017) Potential biological targets for bioassay development in drug discovery of Sturge–Weber syndrome. Chemical Biology & Drug Design 91:2, pages 359-369.
Crossref
Crossref
Radivojka Vulic, Silvia Tyciakova, Maria Dubrovcakova, Ludovit Skultety & Jan Lakota. (2018) Silencing of CA1 mRNA in tumour cells does not change the gene expression of the extracellular matrix proteins. Journal of Cellular and Molecular Medicine 22:1, pages 695-699.
Crossref
Crossref
German L. Perlovich & Tatyana V. Volkova. (2018) Sublimation thermodynamics aspects of adamantane and memantine derivatives of sulfonamide molecular crystals. Physical Chemistry Chemical Physics 20:30, pages 19784-19791.
Crossref
Crossref
Alexander P. Voronin, Tatiana V. Volkova, Andrey B. Ilyukhin, Tatiana P. Trofimova & German L. Perlovich. (2018) Structural and energetic aspects of adamantane and memantine derivatives of sulfonamide molecular crystals: experimental and theoretical characterisation. CrystEngComm 20:25, pages 3476-3489.
Crossref
Crossref
Javad Mokhtari, Bahareh Babaii, Abolfath Akbarzadeh & Parnian Ferdowsi. (2017) Synthesis and evaluation of novel antibacterial monoazo disperse dyes based on sulfonamide derivatives on polyester. Pigment & Resin Technology 46:6, pages 440-448.
Crossref
Crossref
Umit M. Kocyigit, Ahmet Şevki Taşkıran, Parham Taslimi, Ahmet Yokuş, Yusuf Temel & İlhami Gulçin. (2017) Inhibitory effects of oxytocin and oxytocin receptor antagonist atosiban on the activities of carbonic anhydrase and acetylcholinesterase enzymes in the liver and kidney tissues of rats. Journal of Biochemical and Molecular Toxicology 31:11.
Crossref
Crossref
Taner Dastan, Umit M. Kocyigit, Sevgi Durna Dastan, Pakize Canturk Kilickaya, Parham Taslimi, Ozge Cevik, Metin Koparir, Cahit Orek, İlhami Gulçin & Ahmet Cetin. (2017) Investigation of acetylcholinesterase and mammalian DNA topoisomerases, carbonic anhydrase inhibition profiles, and cytotoxic activity of novel bis(α‐aminoalkyl)phosphinic acid derivatives against human breast cancer. Journal of Biochemical and Molecular Toxicology 31:11.
Crossref
Crossref
Masoumeh Bavadi, Khodabakhsh Niknam & Omolbanin Shahraki. (2017) Novel pyrrole derivatives bearing sulfonamide groups: Synthesis in vitro cytotoxicity evaluation, molecular docking and DFT study. Journal of Molecular Structure 1146, pages 242-253.
Crossref
Crossref
Mina Ghiasi & Mina Seifi. (2017) Thermodynamic study on the mechanism of carbonic anhydrase XII inhibition with glycosyl coumarin as non-zinc mediated inhibitors: A quantum mechanical investigation. Computational and Theoretical Chemistry 1118, pages 16-25.
Crossref
Crossref
Displaying 200 of 460 citing articles. Use the download link below to view the full list of citing articles.
Download full citations list