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Morteza Abdoli, Alessandro Bonardi, Claudiu T. Supuran & Raivis Žalubovskis. (2023) Investigation of novel alkyl/benzyl (4-sulphamoylphenyl)carbamimidothioates as carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Alessio Nocentini, Andrea Angeli, Fabrizio Carta, Jean-Yves Winum, Raivis Zalubovskis, Simone Carradori, Clemente Capasso, William A. Donald & Claudiu T. Supuran. (2021) Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 561-580.
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Linda J. Urbański, Andrea Angeli, Vesa P. Hytönen, Anna Di Fiore, Giuseppina De Simone, Seppo Parkkila & Claudiu T. Supuran. (2021) Inhibition of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with sulphonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 330-335.
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Yan-Ru Xiao, Yong-Mei Cui, Cheng-Hu Xie, Wei-Qing Qiu & Hai-Xia Lin. (2020) Design, synthesis of novel C-3′-N-sulfonyl modified taxane analogues from 1-deoxybaccatin VI and their impact on anti-HCC activity. Journal of Asian Natural Products Research 22:12, pages 1168-1175.
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Charu Upadhyay, Monika Chaudhary, Ronaldo N. De Oliveira, Aniko Borbas, Prakasha Kempaiah, Poonam S & Brijesh Rathi. (2020) Fluorinated scaffolds for antimalarial drug discovery. Expert Opinion on Drug Discovery 15:6, pages 705-718.
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Sevil Şenkardeş, İhsan Han, Hakan Hançer, Mürüvvet Abbak, Özge Çevik & Ş. Güniz Küçükgüzel. (2019) Synthesis, characterization and biological evaluation of some novel sulfonylthiosemicarbazides. Phosphorus, Sulfur, and Silicon and the Related Elements 194:12, pages 1164-1170.
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Alessio Nocentini & Claudiu T. Supuran. (2019) Advances in the structural annotation of human carbonic anhydrases and impact on future drug discovery. Expert Opinion on Drug Discovery 14:11, pages 1175-1197.
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D. I. Ugwuja, U. C. Okoro, S. S. Soman, R. Soni, S. N. Okafor & D. I. Ugwu. (2019) New peptide derived antimalaria and antimicrobial agents bearing sulphonamide moiety. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1388-1399.
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Andrea Angeli, Sonia Del Prete, Mariana Pinteala, Stelian S. Maier, William A. Donald, Bogdan C. Simionescu, Clemente Capasso & Claudiu T. Supuran. (2019) The first activation study of the β-carbonic anhydrases from the pathogenic bacteria Brucella suis and Francisella tularensis with amines and amino acids. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1178-1185.
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Baijayantimala Swain, Andrea Angeli, Srinivas Angapelly, Pavitra S. Thacker, Priti Singh, Claudiu T. Supuran & Mohammed Arifuddin. (2019) Synthesis of a new series of 3-functionalised-1-phenyl-1,2,3-triazole sulfamoylbenzamides as carbonic anhydrase I, II, IV and IX inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1199-1209.
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Pavitra S. Thacker, Pirpasha Shaikh, Andrea Angeli, Mohammed Arifuddin & Claudiu T. Supuran. (2019) Synthesis and biological evaluation of novel 8-substituted quinoline-2-carboxamides as carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1172-1177.
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Alessio Nocentini, Sameh M. Osman, Igor A. Rodrigues, Veronica S. Cardoso, Fatmah Ali S. Alasmary, Zeid AlOthman, Alane B. Vermelho, Paola Gratteri & Claudiu T. Supuran. (2019) Appraisal of anti-protozoan activity of nitroaromatic benzenesulfonamides inhibiting carbonic anhydrases from Trypanosoma cruzi and Leishmania donovani. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1164-1171.
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Sonia Del Prete, Rosa Merlo, Anna Valenti, Rosanna Mattossovich, Mosè Rossi, Vincenzo Carginale, Claudiu T. Supuran, Giuseppe Perugino & Clemente Capasso. (2019) Thermostability enhancement of the α-carbonic anhydrase from Sulfurihydrogenibium yellowstonense by using the anchoring-and-self-labelling-protein-tag system (ASL). Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 946-954.
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Atilla Akdemir, Andrea Angeli, Füsun Göktaş, Pınar Eraslan Elma, Nilgün Karalı & Claudiu T. Supuran. (2019) Novel 2-indolinones containing a sulfonamide moiety as selective inhibitors of candida β-carbonic anhydrase enzyme. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 528-531.
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Claudiu T. Supuran. (2018) Carbonic anhydrase inhibitors as emerging agents for the treatment and imaging of hypoxic tumors. Expert Opinion on Investigational Drugs 27:12, pages 963-970.
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Claudiu T. Supuran. (2018) Carbonic anhydrase inhibitors and their potential in a range of therapeutic areas. Expert Opinion on Therapeutic Patents 28:10, pages 709-712.
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Claudiu T. Supuran. (2018) Applications of carbonic anhydrases inhibitors in renal and central nervous system diseases. Expert Opinion on Therapeutic Patents 28:10, pages 713-721.
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Claudiu T. Supuran & Clemente Capasso. (2018) Biomedical applications of prokaryotic carbonic anhydrases. Expert Opinion on Therapeutic Patents 28:10, pages 745-754.
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Andrea Angeli & Claudiu T. Supuran. (2018) Treatment of sleep apnea with a combination of a carbonic anhydrase inhibitor and an aldosterone antagonist: a patent evaluation of CA2958110 and IN6616DEN2012. Expert Opinion on Therapeutic Patents 28:10, pages 723-727.
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Andrea Angeli, Fatmah A. S. Alasmary, Sonia Del Prete, Sameh M. Osman, Zeid AlOthman, William A. Donald, Clemente Capasso & Claudiu T. Supuran. (2018) The first activation study of a δ-carbonic anhydrase: TweCAδ from the diatom Thalassiosira weissflogii is effectively activated by amines and amino acids. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 680-685.
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Daniela Vullo, Ronny Lehneck, Stefanie Pöggeler & Claudiu T. Supuran. (2018) Sulfonamide inhibition studies of two β-carbonic anhydrases from the ascomycete fungus Sordaria macrospora, CAS1 and CAS2. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 390-396.
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Daniela Vullo, R. Siva Sai Kumar, Andrea Scozzafava, James G. Ferry & Claudiu T. Supuran. (2018) Sulphonamide inhibition studies of the β-carbonic anhydrase from the bacterial pathogen Clostridium perfringens. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 31-36.
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Suleyman Akocak, Nabih Lolak, Daniela Vullo, Mustafa Durgun & Claudiu T. Supuran. (2017) Synthesis and biological evaluation of histamine Schiff bases as carbonic anhydrase I, II, IV, VII, and IX activators. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1305-1312.
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Andrea Angeli, Fabio Vaiano, Francesco Mari, Elisabetta Bertol & Claudiu T. Supuran. (2017) Psychoactive substances belonging to the amphetamine class potently activate brain carbonic anhydrase isoforms VA, VB, VII, and XII. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1253-1259.
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Morteza Abdoli, Andrea Angeli, Murat Bozdag, Fabrizio Carta, Ali Kakanejadifard, Hamid Saeidian & Claudiu T. Supuran. (2017) Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo[d]thiazole-5- and 6-sulfonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1071-1078.
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Alessio Nocentini, Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Fatmah A.S. Alasmary, Zeid AlOthman, Clemente Capasso, Fabrizio Carta, Paola Gratteri & Claudiu T. Supuran. (2017) Inhibition of the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa with monothiocarbamates. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1064-1070.
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Murat Bozdag, Silvia Bua, Sameh M. Osman, Zeid AlOthman & Claudiu T. Supuran. (2017) Carbonic anhydrase I, II, IV and IX inhibition with a series of 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 885-892.
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Marco Bragagni, Fabrizio Carta, Sameh M. Osman, Zeid AlOthman & Claudiu T. Supuran. (2017) Synthesis of an acridine orange sulfonamide derivative with potent carbonic anhydrase IX inhibitory action. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 701-706.
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Claudia Melis, Rita Meleddu, Andrea Angeli, Simona Distinto, Giulia Bianco, Clemente Capasso, Filippo Cottiglia, Rossella Angius, Claudiu T. Supuran & Elias Maccioni. (2017) Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 68-73.
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Erol Licsandru, Muhammet Tanc, Istvan Kocsis, Mihail Barboiu & Claudiu T. Supuran. (2017) A class of carbonic anhydrase I – selective activators. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 37-46.
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Claudiu T. Supuran. (2016) CA IX stratification based on cancer treatment: a patent evaluation of US2016/0002350. Expert Opinion on Therapeutic Patents 26:10, pages 1105-1109.
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Ozen Ozensoy Guler, Clemente Capasso & Claudiu T. Supuran. (2016) A magnificent enzyme superfamily: carbonic anhydrases, their purification and characterization. Journal of Enzyme Inhibition and Medicinal Chemistry 31:5, pages 689-694.
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Claudiu T. Supuran. (2016) Carbonic anhydrase inhibition and the management of neuropathic pain. Expert Review of Neurotherapeutics 16:8, pages 961-968.
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György M. Buzás & Claudiu T. Supuran. (2016) The history and rationale of using carbonic anhydrase inhibitors in the treatment of peptic ulcers. In memoriam Ioan Puşcaş (1932–2015). Journal of Enzyme Inhibition and Medicinal Chemistry 31:4, pages 527-533.
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Claudiu T. Supuran. (2016) How many carbonic anhydrase inhibition mechanisms exist?. Journal of Enzyme Inhibition and Medicinal Chemistry 31:3, pages 345-360.
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Mariangela Ceruso, Sabrina Antel, Andrea Scozzafava & Claudiu T. Supuran. (2016) Synthesis and inhibition potency of novel ureido benzenesulfonamides incorporating GABA as tumor-associated carbonic anhydrase IX and XII inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 31:2, pages 205-211.
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Murat Bozdag, Fabrizio Carta, Daniela Vullo, Semra Isik, Zeid AlOthman, Sameh M. Osman, Andrea Scozzafava & Claudiu T. Supuran. (2016) Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase. Journal of Enzyme Inhibition and Medicinal Chemistry 31:1, pages 132-136.
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Namrata Singasane, Prashant S. Kharkar, Mariangela Ceruso, Claudiu T. Supuran & Mrunmayee P. Toraskar. (2015) Inhibition of carbonic anhydrase isoforms I, II, IX and XII with Schiff’s bases incorporating iminoureido moieties. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 901-907.
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Daniela Vullo, Semra Isik, Murat Bozdag, Fabrizio Carta & Claudiu T. Supuran. (2015) 7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring. Journal of Enzyme Inhibition and Medicinal Chemistry 30:5, pages 773-777.
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Claudiu T Supuran. (2015) Acetazolamide for the treatment of idiopathic intracranial hypertension. Expert Review of Neurotherapeutics 15:8, pages 851-856.
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Mariangela Ceruso, Marco Bragagni, Zeid AlOthman, Sameh M. Osman & Claudiu T. Supuran. (2015) New series of sulfonamides containing amino acid moiety act as effective and selective inhibitors of tumor-associated carbonic anhydrase XII. Journal of Enzyme Inhibition and Medicinal Chemistry 30:3, pages 430-434.
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Claudiu T Supuran & Clemente Capasso. (2015) The η-class carbonic anhydrases as drug targets for antimalarial agents. Expert Opinion on Therapeutic Targets 19:4, pages 551-563.
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Kalyan K. Sethi & Saurabh M. Verma. (2014) A systematic quantitative approach to rational drug design and discovery of novel human carbonic anhydrase IX inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 29:4, pages 571-581.
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Erik R Swenson. (2014) Safety of carbonic anhydrase inhibitors. Expert Opinion on Drug Safety 13:4, pages 459-472.
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Asta Zubrienė, Edita Čapkauskaitė, Joana Gylytė, Miglė Kišonaitė, Sigitas Tumkevičius & Daumantas Matulis. (2014) Benzenesulfonamides with benzimidazole moieties as inhibitors of carbonic anhydrases I, II, VII, XII and XIII. Journal of Enzyme Inhibition and Medicinal Chemistry 29:1, pages 124-131.
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Sonia Del Prete, Viviana De Luca, Andrea Scozzafava, Vincenzo Carginale, Claudiu T. Supuran & Clemente Capasso. (2014) Biochemical properties of a new α-carbonic anhydrase from the human pathogenic bacterium, Vibrio cholerae. Journal of Enzyme Inhibition and Medicinal Chemistry 29:1, pages 23-27.
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Romualdo Malagola, Loredana Arrico, Rossella Giannotti & Luigi Pattavina. (2013) Acetazolamide-induced cilio-choroidal effusion after cataract surgery: unusual posterior involvement. Drug Design, Development and Therapy 7, pages 33-36.
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Simona Maria Monti, Claudiu T Supuran & Giuseppina De Simone. (2013) Anticancer carbonic anhydrase inhibitors: a patent review (2008 – 2013). Expert Opinion on Therapeutic Patents 23:6, pages 737-749.
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Fabrizio Carta & Claudiu T Supuran. (2013) Diuretics with carbonic anhydrase inhibitory action: a patent and literature review (2005 – 2013). Expert Opinion on Therapeutic Patents 23:6, pages 681-691.
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Claudiu T Supuran. (2013) Carbonic anhydrase inhibitors: an editorial. Expert Opinion on Therapeutic Patents 23:6, pages 677-679.
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Andrea Scozzafava, Fabrizio Carta & Claudiu T Supuran. (2013) Secondary and tertiary sulfonamides: a patent review (2008 – 2012). Expert Opinion on Therapeutic Patents 23:2, pages 203-213.
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Claudiu T Supuran. (2012) Amide derivatives of benzene-sulfonanilide, pharmaceutical composition thereof and method for cancer treatment using the same (US20120095092). Expert Opinion on Therapeutic Patents 22:10, pages 1251-1255.
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Tuğba Meşeli, Şengül Dilem Doğan, Miyase Gözde Gündüz, Zülbiye Kökbudak, Sanja Skaro Bogojevic, Theresa Noonan, Sandra Vojnovic, Gerhard Wolber & Jasmina Nikodinovic-Runic. (2021) Design, synthesis, antibacterial activity evaluation and molecular modeling studies of new sulfonamides containing a sulfathiazole moiety. New Journal of Chemistry 45:18, pages 8166-8177.
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A. I. Samigullina, I. A. Krutov, E. L. Gavrilova & A. T. Gubaidullin. (2021) Conformational Behavior of N1-(Diphenylphosphoryl)acetyl-N4-phenyl-thiosemicarbazide in Various Crystal Environments. Crystallography Reports 66:3, pages 433-440.
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Chandra Bhushan Mishra, Shikha Kumari, Andrea Angeli, Silvia Bua, Raj Kumar Mongre, Manisha Tiwari & Claudiu T. Supuran. (2021) Discovery of Potent Carbonic Anhydrase Inhibitors as Effective Anticonvulsant Agents: Drug Design, Synthesis, and In Vitro and In Vivo Investigations. Journal of Medicinal Chemistry 64:6, pages 3100-3114.
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Simon Waihenya, Pelin Şenel, Francis J. Osonga, Taner Erdoğan, Filiz Altay, Ayşegül Gölcü & Omowunmi A. Sadik. (2021) Mechanism of Interactions of dsDNA Binding with Apigenin and Its Sulfamate Derivatives Using Multispectroscopic, Voltammetric, and Molecular Docking Studies. ACS Omega 6:8, pages 5124-5137.
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Megan D. Hopkins, Garett L. Ozmer, Ryan C. Witt, Zachary C. Brandeburg, David A. Rogers, Claire E. Keating, Presley L. Petcoff, Robert J. Sheaff & Angus A. Lamar. (2021)
PhI(OAc)
2
and iodine-mediated synthesis of
N
-alkyl sulfonamides derived from polycyclic aromatic hydrocarbon scaffolds and determination of their antibacterial and cytotoxic activities
. Organic & Biomolecular Chemistry 19:5, pages 1133-1144.
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Katia D’Ambrosio, Anna Di Fiore, Martina Buonanno, Shikha Kumari, Manisha Tiwari, Claudiu T. Supuran, Chandra Bhushan Mishra, Simona Maria Monti & Giuseppina De Simone. (2021)
The crystal structures of 2-(4-benzhydrylpiperazin-1-yl)-
N
-(4-sulfamoylphenyl)acetamide in complex with human carbonic anhydrase II and VII provide insights into selective CA inhibitor development
. New Journal of Chemistry 45:1, pages 147-152.
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Anita Bułakowska, Jarosław Sławiński, Kamila Siedlecka-Kroplewska, Grzegorz Stasiłojć, Marcin Serocki & Mateusz Heldt. (2020) Novel N-(aryl/heteroaryl)-2-chlorobenzenesulfonamide derivatives: Synthesis and anticancer activity evaluation. Bioorganic Chemistry 104, pages 104309.
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Andrea Angeli, Fabrizio Carta, Alessio Nocentini, Jean-Yves Winum, Raivis Zalubovskis, Atilla Akdemir, Valentina Onnis, Wagdy M. Eldehna, Clemente Capasso, Giuseppina De Simone, Simona Maria Monti, Simone Carradori, William A. Donald, Shoukat Dedhar & Claudiu T. Supuran. (2020) Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment. Metabolites 10:10, pages 412.
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Vivian Garzón, Rosa-Helena Bustos & Daniel G. Pinacho. (2020) Personalized Medicine for Antibiotics: The Role of Nanobiosensors in Therapeutic Drug Monitoring. Journal of Personalized Medicine 10:4, pages 147.
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Dmistocles A. Vicente, Danilo Galdino, Marcelo Navarro & Paulo H. Menezes. (2020) Electrochemical synthesis of sulfonamides in a graphite powder macroelectrode. Green Chemistry 22:16, pages 5262-5266.
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Wei Dong, Zemei Ge, Xin Wang, Ridong Li & Runtao Li. (2020) Cu-mediated one-pot three-component synthesis of 3-N-substituted 1,4,2-benzodithiazine 1,1-dioxide derivatives. Tetrahedron 76:30, pages 131354.
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Alexander Ahrens, Julia Schwarz, Danilo M. Lustosa, Raheleh Pourkaveh, Marvin Hoffmann, Frank Rominger, Matthias Rudolph, Andreas Dreuw & A. Stephen K. Hashmi. (2020) Synthesis of Fulvene Vinyl Ethers by Gold Catalysis. Chemistry – A European Journal 26:23, pages 5280-5287.
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Ji-Woo Choi, Seung-Hye Choi, Seung Taek Hong, Mun Seok Kim, Seong Shick Ryu, Yeo Uk Yoon, Kyu Cheol Paik, Man So Han, Taebo Sim & Bong Rae Cho. (2020) Two-photon probes for the endoplasmic reticulum: its detection in a live tissue by two-photon microscopy. Chemical Communications 56:25, pages 3657-3660.
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Daniela Vullo, Ronny Lehneck, William A. Donald, Stefanie Pöggeler & Claudiu T. Supuran. (2020) Sulfonamide Inhibition Studies of the β-Class Carbonic Anhydrase CAS3 from the Filamentous Ascomycete Sordaria macrospora. Molecules 25:5, pages 1036.
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Hongbo Liu, Fusheng Zhang, Jiangdong Dai, Li Chen & Yongsheng Yan. (2019) Optical Recognition of Sulfamethoxazole by a Colored Chiral Nematic Imprinted Film. Analytical Sciences 36:2, pages 221-225.
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Soumajit Ghorai, Sravani Pulya, Kalyan Ghosh, Parthasarathi Panda, Balaram Ghosh & Shovanlal Gayen. (2020) Structure-activity relationship of human carbonic anhydrase-II inhibitors: Detailed insight for future development as anti-glaucoma agents. Bioorganic Chemistry 95, pages 103557.
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Claudiu T. Supuran & Clemente Capasso. 2020. Physiological and Biotechnological Aspects of Extremophiles. Physiological and Biotechnological Aspects of Extremophiles
295
306
.
Marcelo Luís Occhiutto, Raul C. Maranhão, Vital Paulino Costa & Anastasios G. Konstas. (2019) Nanotechnology for Medical and Surgical Glaucoma Therapy—A Review. Advances in Therapy 37:1, pages 155-199.
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Alexey Yu Nikonov, Irina V. Sterkhova, Valeriy Yu Serykh, Nikita A. Kolyvanov & Natalya F. Lazareva. (2019) Synthesis and structural features of N-[(2-(trimethylsilyl)oxy)phenyl]-arylsulfonamides. Journal of Molecular Structure 1198, pages 126782.
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Megan D. Hopkins, Felagot A. Abebe, Kristina A. Scott, Garett L. Ozmer, Alec A. Sheir, Lucas J. Schroeder, Robert J. Sheaff & Angus A. Lamar. (2019)
Synthesis and identification of heteroaromatic
N
-benzyl sulfonamides as potential anticancer agents
. Organic & Biomolecular Chemistry 17:36, pages 8391-8402.
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Renate Melngaile, Arturs Sperga, Kim K. Baldridge & Janis Veliks. (2019) Diastereoselective Monofluorocyclopropanation Using Fluoromethylsulfonium Salts. Organic Letters 21:17, pages 7174-7178.
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Thuy Trang Pham, Ashley C. Lindsay, Xi Chen, Gökalp Gözaydin, Ning Yan & Jonathan Sperry. (2019) Transferring the biorenewable nitrogen present in chitin to several N-functional groups. Sustainable Chemistry and Pharmacy 13, pages 100143.
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Prete, Angeli, Ghobril, Hitce, Clavaud, Marat, Supuran & Capasso. (2019) Anion Inhibition Profile of the β-Carbonic Anhydrase from the Opportunist Pathogenic Fungus Malassezia Restricta Involved in Dandruff and Seborrheic Dermatitis. Metabolites 9:7, pages 147.
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Sonia Del Prete, Daniela Vullo, Cynthia Ghobril, Julien Hitce, Cécile Clavaud, Xavier Marat, Clemente Capasso & Claudiu T. Supuran. (2019) Cloning, Purification, and Characterization of a β-Carbonic Anhydrase from Malassezia restricta, an Opportunistic Pathogen Involved in Dandruff and Seborrheic Dermatitis. International Journal of Molecular Sciences 20:10, pages 2447.
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Silvia Bua, Sameh M. Osman, Sonia Del Prete, Clemente Capasso, Zeid AlOthman, Alessio Nocentini & Claudiu T. Supuran. (2019) Click-tailed benzenesulfonamides as potent bacterial carbonic anhydrase inhibitors for targeting Mycobacterium tuberculosis and Vibrio cholerae. Bioorganic Chemistry 86, pages 183-186.
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Alba Vicente‐Blázquez, Myriam González, Raquel Álvarez, Sara del Mazo, Manuel Medarde & Rafael Peláez. (2018) Antitubulin sulfonamides: The successful combination of an established drug class and a multifaceted target. Medicinal Research Reviews 39:3, pages 775-830.
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Shalini Singh. (2019) 3D-QSAR CoMFA Studies on Benzenesulfonamides with Benzimidazole Moieties as Inhibitors of Carbonic Anhydrases XII as Antitumor Agents. Current Enzyme Inhibition 15:1, pages 69-77.
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Janusz J. PetkowskiWilliam BainsSara Seager. (2019) An Apparent Binary Choice in Biochemistry: Mutual Reactivity Implies Life Chooses Thiols or Nitrogen-Sulfur Bonds, but Not Both. Astrobiology 19:4, pages 579-613.
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Nabih Lolak, Suleyman Akocak, Silvia Bua, Rajesh K.K. Sanku & Claudiu T. Supuran. (2019) Discovery of new ureido benzenesulfonamides incorporating 1,3,5-triazine moieties as carbonic anhydrase I, II, IX and XII inhibitors. Bioorganic & Medicinal Chemistry 27:8, pages 1588-1594.
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Nabih Lolak, Suleyman Akocak, Silvia Bua & Claudiu T. Supuran. (2019) Design, synthesis and biological evaluation of novel ureido benzenesulfonamides incorporating 1,3,5-triazine moieties as potent carbonic anhydrase IX inhibitors. Bioorganic Chemistry 82, pages 117-122.
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Claudiu T. Supuran. 2019. Therapeutic Application of Nitric Oxide in Cancer and Inflammatory Disorders. Therapeutic Application of Nitric Oxide in Cancer and Inflammatory Disorders
229
242
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Clemente Capasso & Mihail Barboiu. 2019. Carbonic Anhydrases. Carbonic Anhydrases
495
514
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Silvia Bua, Alessio Nocentini & Claudiu T. Supuran. 2019. Carbonic Anhydrases. Carbonic Anhydrases
287
309
.
Andrey V. Smolobochkin, Ekaterina A. Muravyeva, Liliya I. Vagapova, Irina R. Knyazeva, Julia K. Voronina, Alexander R. Burilov, Michail A. Pudovik, Anastasiya V. Gildebrant, Ivan S. Sazykin, Marina A. Sazykina & Almir S. Gazizov. (2019) Synthesis and Evaluation of Water‐Soluble 2‐Aryl‐1‐Sulfonylpyrrolidine Derivatives as Bacterial Biofilm Formation Inhibitors. Chemistry & Biodiversity 16:1.
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Maksim A. Burkin, Gennady B. Lapa, Inna A. Galvidis, Konstantin M. Burkin, Alexander V. Zubkov & Sergei A. Eremin. (2018) Three steps improving the sensitivity of sulfonamide immunodetection in milk. Analytical Methods 10:48, pages 5773-5782.
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Andrea Angeli, Damiano Tanini, Antonella Capperucci, Gianni Malevolti, Francesca Turco, Marta Ferraroni & Claudiu T. Supuran. (2018) Synthesis of different thio-scaffolds bearing sulfonamide with subnanomolar carbonic anhydrase II and IX inhibitory properties and X-ray investigations for their inhibitory mechanism. Bioorganic Chemistry 81, pages 642-648.
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Jahanzaib Arshad, Muhammad Hanif, Ayesha Zafar, Sanam Movassaghi, Kelvin K. H. Tong, Jóhannes Reynisson, Mario Kubanik, Amir Waseem, Tilo Söhnel, Stephen M. F. Jamieson & Christian G. Hartinger. (2018) Organoruthenium and Organoosmium Complexes of 2-Pyridinecarbothioamides Functionalized with a Sulfonamide Motif: Synthesis, Cytotoxicity and Biomolecule Interactions. ChemPlusChem 83:7, pages 612-619.
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Chandra Bhushan Mishra, Shikha Kumari, Andrea Angeli, Silvia Bua, Manisha Tiwari & Claudiu T. Supuran. (2018) Discovery of Benzenesulfonamide Derivatives as Carbonic Anhydrase Inhibitors with Effective Anticonvulsant Action: Design, Synthesis, and Pharmacological Evaluation. Journal of Medicinal Chemistry 61:7, pages 3151-3165.
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Nabih Lolak, Suleyman Akocak, Silvia Bua, Murat Koca & Claudiu T. Supuran. (2018) Design and synthesis of novel 1,3-diaryltriazene-substituted sulfonamides as potent and selective carbonic anhydrase II inhibitors. Bioorganic Chemistry 77, pages 542-547.
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Halise Inci Gul, Cem Yamali, Hiroshi Sakagami, Andrea Angeli, Janis Leitans, Andris Kazaks, Kaspars Tars, Dilan Ozmen Ozgun & Claudiu T. Supuran. (2018) New anticancer drug candidates sulfonamides as selective hCA IX or hCA XII inhibitors. Bioorganic Chemistry 77, pages 411-419.
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Claudiu Supuran. (2018) Carbonic Anhydrases and Metabolism. Metabolites 8:2, pages 25.
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Janusz J. Petkowski, William BainsSara Seager. (2018) Natural Products Containing a Nitrogen–Sulfur Bond. Journal of Natural Products 81:2, pages 423-446.
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Fusheng Zhang, Enxiu Liu, Xudong Zheng, Longbao Yu & Yongsheng Yan. (2018) A flexible imprinted photonic resin film templated by nanocrystalline cellulose for naked-eye recognition of sulfonamides. Journal of Industrial and Engineering Chemistry 58, pages 172-178.
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Alaaeldin M. F. Galal, Maha M. Soltan, Esam R. Ahmed & Atef G. Hanna. (2018)
Synthesis and biological evaluation of novel 5-chloro-
N
-(4-sulfamoylbenzyl) salicylamide derivatives as tubulin polymerization inhibitors
. MedChemComm 9:9, pages 1511-1528.
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German L. Perlovich & Tatyana V. Volkova. (2018) Sublimation thermodynamics aspects of adamantane and memantine derivatives of sulfonamide molecular crystals. Physical Chemistry Chemical Physics 20:30, pages 19784-19791.
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Shuai Liang, Saad Shaaban, Nai-Wei Liu, Kamil Hofman & Georg Manolikakes. 2018.
135
207
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Hany M Dalloul. (2017) Synthesis and Biological Activities Evaluation of Some New 1,2,4-Triazinone Derivatives Bearing Sulfonamide Moiety. MOJ Bioorganic & Organic Chemistry 1:7.
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Haibo Zhu, Yajing Shen, Qinyue Deng, Zhang-Gao Le & Tao Tu. (2017) Ligand-Free Pd/Cu-Catalyzed Aminosulfonylation of Aryl Iodides for Direct Sulfonamide Syntheses. Asian Journal of Organic Chemistry 6:11, pages 1542-1545.
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Claudiu Supuran. (2017) Special Issue: Sulfonamides. Molecules 22:10, pages 1642.
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Andrea Angeli, Fabrizio Carta, Gianluca Bartolucci & Claudiu T. Supuran. (2017) Synthesis of novel acyl selenoureido benzensulfonamides as carbonic anhydrase I, II, VII and IX inhibitors. Bioorganic & Medicinal Chemistry 25:13, pages 3567-3573.
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Sonia Del Prete, Daniela Vullo, Sameh M. Osman, Zeid AlOthman, Claudiu T. Supuran & Clemente Capasso. (2017) Sulfonamide inhibition profiles of the β-carbonic anhydrase from the pathogenic bacterium Francisella tularensis responsible of the febrile illness tularemia. Bioorganic & Medicinal Chemistry 25:13, pages 3555-3561.
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Lina Baranauskiene & Daumantas Matulis. (2017)
Herbicide oryzalin inhibits human carbonic anhydrases
in vitro
. Journal of Biochemical and Molecular Toxicology 31:6, pages e21894.
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Elvira Bruno, Maria Rosa Buemi, Anna Di Fiore, Laura De Luca, Stefania Ferro, Andrea Angeli, Roberto Cirilli, Daniele Sadutto, Vincenzo Alterio, Simona Maria Monti, Claudiu T. Supuran, Giuseppina De Simone & Rosaria Gitto. (2017) Probing Molecular Interactions between Human Carbonic Anhydrases (hCAs) and a Novel Class of Benzenesulfonamides. Journal of Medicinal Chemistry 60:10, pages 4316-4326.
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Fabrizio Carta, Daniela Vullo, Sameh M. Osman, Zeid AlOthman & Claudiu T. Supuran. (2017) Synthesis and carbonic anhydrase inhibition of a series of SLC-0111 analogs. Bioorganic & Medicinal Chemistry 25:9, pages 2569-2576.
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Menshawy A. Mohamed, Alaa A.-M. Abdel-Aziz, Helmy M. Sakr, Adel S. El-Azab, Silvia Bua & Claudiu T. Supuran. (2017) Synthesis and human/bacterial carbonic anhydrase inhibition with a series of sulfonamides incorporating phthalimido moieties. Bioorganic & Medicinal Chemistry 25:8, pages 2524-2529.
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Andrea Angeli, Damiano Tanini, Caterina Viglianisi, Lucia Panzella, Antonella Capperucci, Stefano Menichetti & Claudiu T. Supuran. (2017) Evaluation of selenide, diselenide and selenoheterocycle derivatives as carbonic anhydrase I, II, IV, VII and IX inhibitors. Bioorganic & Medicinal Chemistry 25:8, pages 2518-2523.
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Yann Le Duc, Erol Licsandru, Daniela Vullo, Mihail Barboiu & Claudiu T. Supuran. (2017) Carbonic anhydrases activation with 3-amino-1H-1,2,4-triazole-1-carboxamides: Discovery of subnanomolar isoform II activators. Bioorganic & Medicinal Chemistry 25:5, pages 1681-1686.
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Rajiv Kumar, Silvia Bua, Sita Ram, Sonia Del Prete, Clemente Capasso, Claudiu T. Supuran & Pawan K. Sharma. (2017) Benzenesulfonamide bearing imidazothiadiazole and thiazolotriazole scaffolds as potent tumor associated human carbonic anhydrase IX and XII inhibitors. Bioorganic & Medicinal Chemistry 25:3, pages 1286-1293.
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Daniela Vullo, Sonia Del Prete, Alessio Nocentini, Sameh M. Osman, Zeid AlOthman, Clemente Capasso, Murat Bozdag, Fabrizio Carta, Paola Gratteri & Claudiu T. Supuran. (2017) Dithiocarbamates effectively inhibit the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa. Bioorganic & Medicinal Chemistry 25:3, pages 1260-1265.
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A. R. Kaliev, V. Yu. Serykh, G. G. Levkovskaya, V. I. Potkin, S. K. Petkevich & I. B. Rozentsveig. (2017) Reaction of polychloroacetaldehyde arylsulfonylimines with 2-amino-6H-1,3-thiazine-6-thiones and 2-amino-4-phenyl-6H-1,3-thiazin-6-one. Russian Journal of Organic Chemistry 52:11, pages 1670-1673.
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Elvira Bruno, Maria R. Buemi, Laura De Luca, Stefania Ferro, Anna‐Maria Monforte, Claudiu T. Supuran, Daniela Vullo, Giovambattista De Sarro, Emilio Russo & Rosaria Gitto. (2016) In Vivo Evaluation of Selective Carbonic Anhydrase Inhibitors as Potential Anticonvulsant Agents. ChemMedChem 11:16, pages 1812-1818.
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Claudiu T. Supuran. (2016) Structure and function of carbonic anhydrases. Biochemical Journal 473:14, pages 2023-2032.
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Daniela Vullo, Viviana De Luca, Sonia Del Prete, Vincenzo Carginale, Andrea Scozzafava, Sameh M. Osman, Zeid AlOthman, Clemente Capasso & Claudiu T. Supuran. (2016) Sulfonamide inhibition studies of the γ-carbonic anhydrase from the Antarctic bacterium Colwellia psychrerythraea. Bioorganic & Medicinal Chemistry Letters 26:4, pages 1253-1259.
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Pavlo A. Sokolyuk, Ivan S. Kondratov, Olexiy V. Gavrylenko & Andrey A. Tolmachov. (2015) Synthesis of diverse pyrazole-4-sulfonyl chlorides starting from 2-(benzylthio)malonaldehyde. Molecular Diversity 20:1, pages 1-7.
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Ylenia Cau, Mattia Mori, Claudiu T. Supuran & Maurizio Botta. (2016) Mycobacterial carbonic anhydrase inhibition with phenolic acids and esters: kinetic and computational investigations. Organic & Biomolecular Chemistry 14:35, pages 8322-8330.
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Kęstutis Aidas, Kiril Lanevskij, Rytis Kubilius, Liutauras Juška, Daumantas Petkevičius & Pranas Japertas. (2015) Aqueous acidities of primary benzenesulfonamides: Quantum chemical predictions based on density functional theory and SMD. Journal of Computational Chemistry 36:29, pages 2158-2167.
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Sonia Del Prete, Daniela Vullo, Sameh M. Osman, Zeid AlOthman, Clemente Capasso & Claudiu T. Supuran. (2015) Anion inhibition studies of the dandruff-producing fungus Malassezia globosa β-carbonic anhydrase MgCA. Bioorganic & Medicinal Chemistry Letters 25:22, pages 5194-5198.
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Maria Rosa Buemi, Laura De Luca, Stefania Ferro, Elvira Bruno, Mariangela Ceruso, Claudiu T. Supuran, Klára Pospíšilová, Jiří Brynda, Pavlína Řezáčová & Rosaria Gitto. (2015) Carbonic anhydrase inhibitors: Design, synthesis and structural characterization of new heteroaryl-N-carbonylbenzenesulfonamides targeting druggable human carbonic anhydrase isoforms. European Journal of Medicinal Chemistry 102, pages 223-232.
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Rita Meleddu, Elias Maccioni, Simona Distinto, Giulia Bianco, Claudia Melis, Stefano Alcaro, Filippo Cottiglia, Mariangela Ceruso & Claudiu T. Supuran. (2015) New 4-[(3-cyclohexyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII. Bioorganic & Medicinal Chemistry Letters 25:16, pages 3281-3284.
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Wagdy M. Eldehna, Mohamed Fares, Hany S. Ibrahim, Mohamed H. Aly, Suher Zada, Mamdouh M. Ali, Sahar M. Abou-Seri, Hatem A. Abdel-Aziz & Dalal A. Abou El Ella. (2015) Indoline ureas as potential anti-hepatocellular carcinoma agents targeting VEGFR-2: Synthesis, in vitro biological evaluation and molecular docking. European Journal of Medicinal Chemistry 100, pages 89-97.
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Nurcan Dedeoglu, Viviana De Luca, Semra Isik, Hatice Yildirim, Feray Kockar, Clemente Capasso & Claudiu T. Supuran. (2015) Cloning, characterization and anion inhibition study of a β-class carbonic anhydrase from the caries producing pathogen Streptococcus mutans. Bioorganic & Medicinal Chemistry 23:13, pages 2995-3001.
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Dattatraya B. Bagal, Georgiy Kachkovskyi, Matthias Knorn, Thomas Rawner, Bhalchandra M. Bhanage & Oliver Reiser. (2015) Trifluoromethylchlorosulfonylation of Alkenes: Evidence for an Inner-Sphere Mechanism by a Copper Phenanthroline Photoredox Catalyst. Angewandte Chemie International Edition 54:24, pages 6999-7002.
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Dattatraya B. Bagal, Georgiy Kachkovskyi, Matthias Knorn, Thomas Rawner, Bhalchandra M. Bhanage & Oliver Reiser. (2015) Trifluormethylchlorsulfonylierung von Alkenen – Hinweise auf einen Innensphärenmechanismus eines Kupferphenanthrolin‐Photoredoxkatalysators. Angewandte Chemie 127:24, pages 7105-7108.
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Nurcan Dedeoglu, Viviana DeLuca, Semra Isik, Hatice Yildirim, Feray Kockar, Clemente Capasso & Claudiu T. Supuran. (2015) Sulfonamide inhibition study of the β-class carbonic anhydrase from the caries producing pathogen Streptococcus mutans. Bioorganic & Medicinal Chemistry Letters 25:11, pages 2291-2297.
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Özlen Güzel-Akdemir, Atilla Akdemir, Nilgün Karalı & Claudiu T. Supuran. (2015) Discovery of novel isatin-based sulfonamides with potent and selective inhibition of the tumor-associated carbonic anhydrase isoforms IX and XII. Organic & Biomolecular Chemistry 13:23, pages 6493-6499.
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Jinghan Tian, Jialei Bai, Yuan Peng, Zhiwei Qie, Yufeng Zhao, Baoan Ning, Dan Xiao & Zhixian Gao. (2015) A core–shell-structured molecularly imprinted polymer on upconverting nanoparticles for selective and sensitive fluorescence sensing of sulfamethazine. The Analyst 140:15, pages 5301-5307.
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V. Alterio, M. Tanc, J. Ivanova, R. Zalubovskis, I. Vozny, S. M. Monti, A. Di Fiore, G. De Simone & C. T. Supuran. (2015) X-ray crystallographic and kinetic investigations of 6-sulfamoyl-saccharin as a carbonic anhydrase inhibitor. Organic & Biomolecular Chemistry 13:13, pages 4064-4069.
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Katia D'Ambrosio, Simone Carradori, Simona M. Monti, Martina Buonanno, Daniela Secci, Daniela Vullo, Claudiu T. Supuran & Giuseppina De Simone. (2015) Out of the active site binding pocket for carbonic anhydrase inhibitors. Chemical Communications 51:2, pages 302-305.
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Mariangela Ceruso, Sabrina Antel, Daniela Vullo, Andrea Scozzafava & Claudiu T. Supuran. (2014) Inhibition studies of new ureido-substituted sulfonamides incorporating a GABA moiety against human carbonic anhydrase isoforms I–XIV. Bioorganic & Medicinal Chemistry 22:24, pages 6768-6775.
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Busra Sarikaya, Mariangela Ceruso, Fabrizio Carta & Claudiu T. Supuran. (2014) Inhibition of carbonic anhydrase isoforms I, II, IX and XII with novel Schiff bases: Identification of selective inhibitors for the tumor-associated isoforms over the cytosolic ones. Bioorganic & Medicinal Chemistry 22:21, pages 5883-5890.
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Kęstutis Rutkauskas, Asta Zubrienė, Ingrida Tumosienė, Kristina Kantminienė, Marytė Kažemėkaitė, Alexey Smirnov, Justina Kazokaitė, Vaida Morkūnaitė, Edita Čapkauskaitė, Elena Manakova, Saulius Gražulis, Zigmuntas Beresnevičius & Daumantas Matulis. (2014) 4-Amino-substituted Benzenesulfonamides as Inhibitors of Human Carbonic Anhydrases. Molecules 19:11, pages 17356-17380.
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Claudiu T Supuran & Clemente CapassoJean-Yves Winum. 2014. Targeting Carbonic Anhydrases. Targeting Carbonic Anhydrases
18
33
.
Ahmed M. Alafeefy, Mariangela Ceruso, Abdul-Malek S. Al-Tamimi, Sonia Del Prete, Clemente Capasso & Claudiu T. Supuran. (2014) Quinazoline–sulfonamides with potent inhibitory activity against the α-carbonic anhydrase from Vibrio cholerae. Bioorganic & Medicinal Chemistry 22:19, pages 5133-5140.
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Sonia Del Prete, Daniela Vullo, Gillian M. Fisher, Katherine T. Andrews, Sally-Ann Poulsen, Clemente Capasso & Claudiu T. Supuran. (2014) Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum —The η-carbonic anhydrases. Bioorganic & Medicinal Chemistry Letters 24:18, pages 4389-4396.
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Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Andrea Scozzafava, Zeid Alothman, Claudiu T. Supuran & Clemente Capasso. (2014) Anion inhibition study of the β-class carbonic anhydrase (PgiCAb) from the oral pathogen Porphyromonas gingivalis. Bioorganic & Medicinal Chemistry Letters 24:18, pages 4402-4406.
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Mariangela Ceruso, Sonia Del Prete, Zeid AlOthman, Sameh M. Osman, Andrea Scozzafava, Clemente Capasso & Claudiu T. Supuran. (2014) Synthesis of sulfonamides with effective inhibitory action against Porphyromonas gingivalis γ-carbonic anhydrase. Bioorganic & Medicinal Chemistry Letters 24:16, pages 4006-4010.
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Emiliano Rosatelli, Andrea Carotti, Mariangela Ceruso, Claudiu T. Supuran & Antimo Gioiello. (2014) Flow synthesis and biological activity of aryl sulfonamides as selective carbonic anhydrase IX and XII inhibitors. Bioorganic & Medicinal Chemistry Letters 24:15, pages 3422-3425.
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Cenzo Congiu, Valentina Onnis, Gianfranco Balboni & Claudiu T. Supuran. (2014) Synthesis and carbonic anhydrase I, II, IX and XII inhibition studies of 4-N,N-disubstituted sulfanilamides incorporating 4,4,4-trifluoro-3-oxo-but-1-enyl, phenacylthiourea and imidazol-2(3H)-one/thione moieties. Bioorganic & Medicinal Chemistry Letters 24:7, pages 1776-1779.
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Amrita K. Saluja, Meena Tiwari, Daniela Vullo & Claudiu T. Supuran. (2014) Substituted benzene sulfonamides incorporating 1,3,5-triazinyl moieties potently inhibit human carbonic anhydrases II, IX and XII. Bioorganic & Medicinal Chemistry Letters 24:5, pages 1310-1314.
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Melissa D’Ascenzio, Simone Carradori, Celeste De Monte, Daniela Secci, Mariangela Ceruso & Claudiu T. Supuran. (2014) Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII. Bioorganic & Medicinal Chemistry 22:6, pages 1821-1831.
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Murat Bozdag, Marta Ferraroni, Elisa Nuti, Daniela Vullo, Armando Rossello, Fabrizio Carta, Andrea Scozzafava & Claudiu T. Supuran. (2014) Combining the tail and the ring approaches for obtaining potent and isoform-selective carbonic anhydrase inhibitors: Solution and X-ray crystallographic studies. Bioorganic & Medicinal Chemistry 22:1, pages 334-340.
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Janis Leitans, Agnese Sprudza, Muhammet Tanc, Igor Vozny, Raivis Zalubovskis, Kaspars Tars & Claudiu T. Supuran. (2013) 5-Substituted-(1,2,3-triazol-4-yl)thiophene-2-sulfonamides strongly inhibit human carbonic anhydrases I, II, IX and XII: Solution and X-ray crystallographic studies. Bioorganic & Medicinal Chemistry 21:17, pages 5130-5138.
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Christopher Waldmann, Otmar Schober, Günter Haufe & Klaus Kopka. (2013)
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Ahmed M. Alafeefy, Semra Isik, Nabila A. Al-Jaber, Daniela Vullo, Hatem A. Abdel-Aziz, Abdelkader E. Ashour, Amani S. Awaad, Clemente Capasso & Claudiu T. Supuran. (2013) Carbonic anhydrase inhibitors. Benzenesulfonamides incorporating cyanoacrylamide moieties strongly inhibit Saccharomyces cerevisiae β-carbonic anhydrase. Bioorganic & Medicinal Chemistry Letters 23:12, pages 3570-3575.
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Ahmed M. Alafeefy, Semra Isik, Hatem A. Abdel-Aziz, Abdelkader E. Ashour, Daniela Vullo, Nabila A. Al-Jaber & Claudiu T. Supuran. (2013) Carbonic anhydrase inhibitors: Benzenesulfonamides incorporating cyanoacrylamide moieties are low nanomolar/subnanomolar inhibitors of the tumor-associated isoforms IX and XII. Bioorganic & Medicinal Chemistry 21:6, pages 1396-1403.
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Laszlo Tarko & Claudiu T. Supuran. (2013) QSAR studies of sulfamate and sulfamide inhibitors targeting human carbonic anhydrase isozymes I, II, IX and XII. Bioorganic & Medicinal Chemistry 21:6, pages 1404-1409.
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Peiwen Pan, Alane Beatriz Vermelho, Giseli Capaci Rodrigues, Andrea Scozzafava, Martti E. E. Tolvanen, Seppo Parkkila, Clemente Capasso & Claudiu T. Supuran. (2013)
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