Citations (235)
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Francesco Fiorentino, Alessio Nocentini, Dante Rotili, Claudiu T. Supuran & Antonello Mai. (2023) Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Jekaterīna Ivanova, Morteza Abdoli, Alessio Nocentini, Raivis Žalubovskis & Claudiu T. Supuran. (2023) Derivatives of 4-methyl-1,2,3-benzoxathiazine 2,2-dioxide as selective inhibitors of human carbonic anhydrases IX and XII over the cytosolic isoforms I and II. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Doretta Cuffaro, Riccardo Di Leo, Lidia Ciccone, Alessio Nocentini, Claudiu T. Supuran, Elisa Nuti & Armando Rossello. (2023) New isoxazolidinyl-based N-alkylethanolamines as new activators of human brain carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Jekaterina Ivanova, Morteza Abdoli, Alessio Nocentini, Raivis Žalubovskis & Claudiu T. Supuran. (2023) 1,2,3-Benzoxathiazine-2,2-dioxides – effective inhibitors of human carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1, pages 225-238.
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Tingting Liu, Lixia Cao, Tingting Zhang & Huan Fu. (2023) Molecular docking studies, anti-Alzheimer’s disease, antidiabetic, and anti-acute myeloid leukemia potentials of narcissoside. Archives of Physiology and Biochemistry 129:2, pages 405-415.
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Claudiu T. Supuran. (2022) Anti-obesity carbonic anhydrase inhibitors: challenges and opportunities. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 2478-2488.
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Mattia Mori & Claudiu T. Supuran. (2022) Acipimox inhibits human carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 672-679.
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Claudiu T. Supuran. (2021) Multitargeting approaches involving carbonic anhydrase inhibitors: hybrid drugs against a variety of disorders. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 1702-1714.
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Gustavo Provensi, Alessio Nocentini, Maria Beatrice Passani, Patrizio Blandina & Claudiu T. Supuran. (2021) Activation of carbonic anhydrase isoforms involved in modulation of emotional memory and cognitive disorders with histamine agonists, antagonists and derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 719-726.
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Alessio Nocentini, Andrea Angeli, Fabrizio Carta, Jean-Yves Winum, Raivis Zalubovskis, Simone Carradori, Clemente Capasso, William A. Donald & Claudiu T. Supuran. (2021) Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 561-580.
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Andrea Petreni, Viviana De Luca, Andrea Scaloni, Alessio Nocentini, Clemente Capasso & Claudiu T. Supuran. (2021) Anion inhibition studies of the Zn(II)-bound ι-carbonic anhydrase from the Gram-negative bacterium Burkholderia territorii. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 372-376.
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Linda J. Urbański, Andrea Angeli, Vesa P. Hytönen, Anna Di Fiore, Giuseppina De Simone, Seppo Parkkila & Claudiu T. Supuran. (2021) Inhibition of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with sulphonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 330-335.
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Claudiu T Supuran. (2020) Experimental Carbonic Anhydrase Inhibitors for the Treatment of Hypoxic Tumors. Journal of Experimental Pharmacology 12, pages 603-617.
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Claudiu T. Supuran. (2020) Exploring the multiple binding modes of inhibitors to carbonic anhydrases for novel drug discovery. Expert Opinion on Drug Discovery 15:6, pages 671-686.
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Claudiu T. Supuran. (2020) An update on drug interaction considerations in the therapeutic use of carbonic anhydrase inhibitors. Expert Opinion on Drug Metabolism & Toxicology 16:4, pages 297-307.
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Claudiu T. Supuran. (2020) Coumarin carbonic anhydrase inhibitors from natural sources. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1462-1470.
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Patrizio Blandina, Gustavo Provensi, Maria Beatrice Passani, Clemente Capasso & Claudiu T. Supuran. (2020) Carbonic anhydrase modulation of emotional memory. Implications for the treatment of cognitive disorders. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1206-1214.
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Jeremie Brichet, Rodrigo Arancibia, Emanuela Berrino & Claudiu T. Supuran. (2020) Bioorganometallic derivatives of 4-hydrazino-benzenesulphonamide as carbonic anhydrase inhibitors: synthesis, characterisation and biological evaluation. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 622-628.
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Alessio Nocentini & Claudiu T. Supuran. (2019) Advances in the structural annotation of human carbonic anhydrases and impact on future drug discovery. Expert Opinion on Drug Discovery 14:11, pages 1175-1197.
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Sabina Zamanova, Ahmed M Shabana, Utpal K Mondal & Marc A Ilies. (2019) Carbonic anhydrases as disease markers. Expert Opinion on Therapeutic Patents 29:7, pages 509-533.
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Andrea Angeli, Sonia Del Prete, Mariana Pinteala, Stelian S. Maier, William A. Donald, Bogdan C. Simionescu, Clemente Capasso & Claudiu T. Supuran. (2019) The first activation study of the β-carbonic anhydrases from the pathogenic bacteria Brucella suis and Francisella tularensis with amines and amino acids. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1178-1185.
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Sonia Del Prete, Rosa Merlo, Anna Valenti, Rosanna Mattossovich, Mosè Rossi, Vincenzo Carginale, Claudiu T. Supuran, Giuseppe Perugino & Clemente Capasso. (2019) Thermostability enhancement of the α-carbonic anhydrase from Sulfurihydrogenibium yellowstonense by using the anchoring-and-self-labelling-protein-tag system (ASL). Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 946-954.
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Yosselin Huentupil, Luis Peña, Néstor Novoa, Emanuela Berrino, Rodrigo Arancibia & Claudiu T. Supuran. (2019) New sulfonamides containing organometallic-acylhydrazones: synthesis, characterisation and biological evaluation as inhibitors of human carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 451-458.
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Sara Seršen, Katja Traven, Jakob Kljun, Iztok Turel & Claudiu T. Supuran. (2019) Organoruthenium(II) complexes of acetazolamide potently inhibit human carbonic anhydrase isoforms I, II, IX and XII. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 388-393.
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Andrea Angeli, Mariana Pinteala, Stelian S. Maier, Sonia Del Prete, Clemente Capasso, Bogdan C. Simionescu & Claudiu T. Supuran. (2019) Inhibition of bacterial α-, β- and γ-class carbonic anhydrases with selenazoles incorporating benzenesulfonamide moieties. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 244-249.
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Claudiu T. Supuran. (2018) Carbonic anhydrase inhibitors as emerging agents for the treatment and imaging of hypoxic tumors. Expert Opinion on Investigational Drugs 27:12, pages 963-970.
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Claudiu T. Supuran. (2018) Carbonic anhydrase inhibitors and their potential in a range of therapeutic areas. Expert Opinion on Therapeutic Patents 28:10, pages 709-712.
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Claudiu T. Supuran. (2018) Applications of carbonic anhydrases inhibitors in renal and central nervous system diseases. Expert Opinion on Therapeutic Patents 28:10, pages 713-721.
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Claudiu T. Supuran & Clemente Capasso. (2018) Biomedical applications of prokaryotic carbonic anhydrases. Expert Opinion on Therapeutic Patents 28:10, pages 745-754.
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Emanuela Berrino, Murat Bozdag, Sonia Del Prete, Fatmah A. S. Alasmary, Linah S. Alqahtani, Zeid AlOthman, Clemente Capasso & Claudiu T. Supuran. (2018) Inhibition of α-, β-, γ-, and δ-carbonic anhydrases from bacteria and diatoms with N′-aryl-N-hydroxy-ureas. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 1194-1198.
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Verônica da Silva Cardoso, Alane Beatriz Vermelho, Eduardo Ricci Junior, Igor Almeida Rodrigues, Ana Maria Mazotto & Claudiu T. Supuran. (2018) Antileishmanial activity of sulphonamide nanoemulsions targeting the β-carbonic anhydrase from Leishmania species. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 850-857.
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Andrea Angeli, Fatmah A. S. Alasmary, Sonia Del Prete, Sameh M. Osman, Zeid AlOthman, William A. Donald, Clemente Capasso & Claudiu T. Supuran. (2018) The first activation study of a δ-carbonic anhydrase: TweCAδ from the diatom Thalassiosira weissflogii is effectively activated by amines and amino acids. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 680-685.
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Claudiu T. Supuran. (2018) Carbon- versus sulphur-based zinc binding groups for carbonic anhydrase inhibitors?. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 485-495.
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Andrea Angeli, Sonia Del Prete, Sameh M. Osman, Fatmah A. S. Alasmary, Zeid AlOthman, William A. Donald, Clemente Capasso & Claudiu T. Supuran. (2018) Activation studies with amines and amino acids of the β-carbonic anhydrase encoded by the Rv3273 gene from the pathogenic bacterium Mycobacterium tuberculosis. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 364-369.
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Andrea Angeli, Niccolò Chiaramonte, Dina Manetti, Maria Novella Romanelli & Claudiu T. Supuran. (2018) Investigation of piperazines as human carbonic anhydrase I, II, IV and VII activators. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 303-308.
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Andrea Angeli, Sonia Del Prete, Sameh M. Osman, Fatmah A. S. Alasmary, Zeid AlOthman, William A. Donald, Clemente Capasso & Claudiu T. Supuran. (2018) Activation studies of the α- and β-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae with amines and amino acids. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 227-233.
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Alane Beatriz Vermelho, Verônica da Silva Cardoso, Eduardo Ricci Junior, Elisabete Pereira dos Santos & Claudiu T. Supuran. (2018) Nanoemulsions of sulfonamide carbonic anhydrase inhibitors strongly inhibit the growth of Trypanosoma cruzi. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 139-146.
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Vincenzo Alterio, Davide Esposito, Simona Maria Monti, Claudiu T. Supuran & Giuseppina De Simone. (2018) Crystal structure of the human carbonic anhydrase II adduct with 1-(4-sulfamoylphenyl-ethyl)-2,4,6-triphenylpyridinium perchlorate, a membrane-impermeant, isoform selective inhibitor. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 151-157.
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Daniela Vullo, R. Siva Sai Kumar, Andrea Scozzafava, James G. Ferry & Claudiu T. Supuran. (2018) Sulphonamide inhibition studies of the β-carbonic anhydrase from the bacterial pathogen Clostridium perfringens. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 31-36.
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Claudiu T. Supuran. (2017) Advances in structure-based drug discovery of carbonic anhydrase inhibitors. Expert Opinion on Drug Discovery 12:1, pages 61-88.
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Suleyman Akocak, Nabih Lolak, Daniela Vullo, Mustafa Durgun & Claudiu T. Supuran. (2017) Synthesis and biological evaluation of histamine Schiff bases as carbonic anhydrase I, II, IV, VII, and IX activators. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1305-1312.
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Andrea Angeli, Fabio Vaiano, Francesco Mari, Elisabetta Bertol & Claudiu T. Supuran. (2017) Psychoactive substances belonging to the amphetamine class potently activate brain carbonic anhydrase isoforms VA, VB, VII, and XII. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1253-1259.
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Rajiv Kumar, Vikas Sharma, Silvia Bua, Claudiu T. Supuran & Pawan K. Sharma. (2017) Synthesis and biological evaluation of benzenesulphonamide-bearing 1,4,5-trisubstituted-1,2,3-triazoles possessing human carbonic anhydrase I, II, IV, and IX inhibitory activity. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1187-1194.
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Morteza Abdoli, Andrea Angeli, Murat Bozdag, Fabrizio Carta, Ali Kakanejadifard, Hamid Saeidian & Claudiu T. Supuran. (2017) Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo[d]thiazole-5- and 6-sulfonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 1071-1078.
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Murat Bozdag, Silvia Bua, Sameh M. Osman, Zeid AlOthman & Claudiu T. Supuran. (2017) Carbonic anhydrase I, II, IV and IX inhibition with a series of 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 885-892.
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Marco Bragagni, Fabrizio Carta, Sameh M. Osman, Zeid AlOthman & Claudiu T. Supuran. (2017) Synthesis of an acridine orange sulfonamide derivative with potent carbonic anhydrase IX inhibitory action. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 701-706.
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Erol Licsandru, Muhammet Tanc, Istvan Kocsis, Mihail Barboiu & Claudiu T. Supuran. (2017) A class of carbonic anhydrase I – selective activators. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 37-46.
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Halise Inci Gul, Mehtap Tugrak, Hiroshi Sakagami, Parham Taslimi, Ilhami Gulcin & Claudiu T. Supuran. (2016) Synthesis and bioactivity studies on new 4-(3-(4-Substitutedphenyl)-3a,4-dihydro-3H-indeno[1,2-c]pyrazol-2-yl) benzenesulfonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1619-1624.
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F. Zehra Küçükbay, Hasan Küçükbay, Muhammet Tanc & Claudiu T. Supuran. (2016) Synthesis and carbonic anhydrase I, II, IV and XII inhibitory properties of N-protected amino acid – sulfonamide conjugates. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1476-1483.
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Burak Aday, Pınar Sola, Ferdağ Çolak & Muharrem Kaya. (2016) Synthesis of novel sulfonamide analogs containing sulfamerazine/sulfaguanidine and their biological activities. Journal of Enzyme Inhibition and Medicinal Chemistry 31:6, pages 1005-1010.
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Viviana De Luca, Sonia Del Prete, Daniela Vullo, Vincenzo Carginale, Pietro Di Fonzo, Sameh M Osman, Zeid AlOthman, Claudiu T Supuran & Clemente Capasso. (2016) Expression and characterization of a recombinant psychrophilic γ-carbonic anhydrase (NcoCA) identified in the genome of the Antarctic cyanobacteria belonging to the genus Nostoc. Journal of Enzyme Inhibition and Medicinal Chemistry 31:5, pages 810-817.
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Ozen Ozensoy Guler, Clemente Capasso & Claudiu T. Supuran. (2016) A magnificent enzyme superfamily: carbonic anhydrases, their purification and characterization. Journal of Enzyme Inhibition and Medicinal Chemistry 31:5, pages 689-694.
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Claudiu T. Supuran. (2016) Carbonic anhydrase inhibition and the management of neuropathic pain. Expert Review of Neurotherapeutics 16:8, pages 961-968.
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Claudiu T. Supuran. (2016) How many carbonic anhydrase inhibition mechanisms exist?. Journal of Enzyme Inhibition and Medicinal Chemistry 31:3, pages 345-360.
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Claudiu T. Supuran. (2016) Drug interaction considerations in the therapeutic use of carbonic anhydrase inhibitors. Expert Opinion on Drug Metabolism & Toxicology 12:4, pages 423-431.
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Murat Bozdag, Fabrizio Carta, Daniela Vullo, Semra Isik, Zeid AlOthman, Sameh M. Osman, Andrea Scozzafava & Claudiu T. Supuran. (2016) Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase. Journal of Enzyme Inhibition and Medicinal Chemistry 31:1, pages 132-136.
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Namrata Singasane, Prashant S. Kharkar, Mariangela Ceruso, Claudiu T. Supuran & Mrunmayee P. Toraskar. (2015) Inhibition of carbonic anhydrase isoforms I, II, IX and XII with Schiff’s bases incorporating iminoureido moieties. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 901-907.
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Daniela Vullo, Semra Isik, Murat Bozdag, Fabrizio Carta & Claudiu T. Supuran. (2015) 7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring. Journal of Enzyme Inhibition and Medicinal Chemistry 30:5, pages 773-777.
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Claudiu T Supuran. (2015) Acetazolamide for the treatment of idiopathic intracranial hypertension. Expert Review of Neurotherapeutics 15:8, pages 851-856.
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Claudia Palmer & Claudiu T Supuran. (2015) A Key Opinion Leader interview: insight into the research and career of Prof. Claudiu T Supuran. Expert Opinion on Therapeutic Patents 25:4, pages 501-505.
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Ahmed M. Alafeefy, Hatem A. Abdel-Aziz, Daniela Vullo, Abdul-Malek S. Al-Tamimi, Amani S. Awaad, Menshawy A. Mohamed, Clemente Capasso & Claudiu T. Supuran. (2015) Inhibition of human carbonic anhydrase isozymes I, II, IX and XII with a new series of sulfonamides incorporating aroylhydrazone-, [1,2,4]triazolo[3,4-b][1,3,4]thiadiazinyl- or 2-(cyanophenylmethylene)-1,3,4-thiadiazol-3(2H)-yl moieties. Journal of Enzyme Inhibition and Medicinal Chemistry 30:1, pages 52-56.
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Antonin Lamaziere, Claude Wolf & Peter J Quinn. (2014) How lipidomics provides new insight into drug discovery. Expert Opinion on Drug Discovery 9:7, pages 819-836.
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Articles from other publishers (173)
Claudiu T. Supuran. 2024. Metalloenzymes. Metalloenzymes
139
156
.
Cüneyt Türkeş. (2023) Carbonic anhydrase inhibition by antiviral drugs in vitro and in silico. Journal of Molecular Recognition 36:12.
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Ahmed Sadiq Sheikh, Reem Altaf, Humaira Nadeem, Muhammad Tariq Khan & Babar Murtaza. (2023) Formation of morpholine-acetamide derivatives as potent anti-tumor drug candidates: Pharmacological evaluation and molecular docking studies. Heliyon 9:11, pages e22183.
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Ebrahim Yarmohammadi, Maryam Khanjani, Zahra Khamverdi, Marzieh Savari & Amir Taherkhani. (2023) Herbal Metabolites as Potential Carbonic Anhydrase Inhibitors: Promising Compounds for Cancer and Metabolic Disorders. Journal of Obesity & Metabolic Syndrome 32:3, pages 247-258.
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Claudiu T. Supuran. (2023) A simple yet multifaceted 90 years old, evergreen enzyme: Carbonic anhydrase, its inhibition and activation. Bioorganic & Medicinal Chemistry Letters 93, pages 129411.
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Mahshid Hesar Shourkabi, Maryam Ghobeh & Hanieh Jafary. (2023) Benzenesulfonamide as a novel, pharmaceutical small molecule inhibitor on Aβ gene expression and oxidative stress in Alzheimer's Wistar rats. Biochemical and Biophysical Research Communications 674, pages 154-161.
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Ben Jabrallah Taha, Chaabani Amal & Belhadj Tahar Noureddine. (2023) Electrochemical determination of sulfaguanidine using COOH‐MWCNT coated GC electrode. Electroanalysis.
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Andrea Angeli, Marta Ferraroni, Carlotta Granchi, Filippo Minutolo, Xiaozhuo Chen, Pratik Shriwas, Emilio Russo, Antonio Leo, Silvia Selleri, Fabrizio Carta & Claudiu T. Supuran. (2023) First-in-Class Dual Targeting Compounds for the Management of Seizures in Glucose Transporter Type 1 Deficiency Syndrome. Journal of Medicinal Chemistry 66:14, pages 10010-10026.
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Kaan Küçükoğlu, Ulviye Acar Çevik, Hayrunnisa Nadaroglu, Ismail Celik, Ayşen Işık, Hayrani Eren Bostancı, Yusuf Özkay & Zafer Asım Kaplancıklı. (2023) Synthesis and Molecular Docking of New N-Acyl Hydrazones-
Benzimidazole as hCA I and II Inhibitors. Medicinal Chemistry 19:5, pages 485-494.
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Andrea Angeli, Niccolò Paoletti & Claudiu T. Supuran. (2023) Five-Membered Heterocyclic Sulfonamides as Carbonic Anhydrase Inhibitors. Molecules 28:7, pages 3220.
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Ashok Aspatwar, Claudiu T. Supuran, Abdul Waheed, William S. Sly & Seppo Parkkila. (2022) Mitochondrial carbonic anhydrase VA and VB: properties and roles in health and disease. The Journal of Physiology 601:2, pages 257-274.
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Laura De Luca, Andrea Angeli, Federico Ricci, Claudiu T. Supuran & Rosaria Gitto. (2022) Structure‐guided identification of a selective sulfonamide‐based inhibitor targeting the human carbonic anhydrase VA isoform. Archiv der Pharmazie 356:1.
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Claudiu T. Supuran. 2022. Flavonoids and Phenolics. Flavonoids and Phenolics
298
329
.
Petr Heneberg. (2022) Lactic Acidosis in Patients with Solid Cancer. Antioxidants & Redox Signaling 37:16-18, pages 1130-1152.
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Shoaib Manzoor, Andrea Angeli, Susi Zara, Simone Carradori, Md Ataur Rahman, Md Kausar Raza, Claudiu T. Supuran & Nasimul Hoda. (2022) Development of benzene and benzothiazole-sulfonamide analogues as selective inhibitors of the tumor-associated carbonic anhydrase IX. European Journal of Medicinal Chemistry 243, pages 114793.
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Baijayantimala Swain, Abrar Khan, Priti Singh, Vaibhav S. Marde, Andrea Angeli, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Simone Carradori, Claudiu T. Supuran & Mohammed Arifuddin. (2022) Design, Synthesis and Biological Assessment of Rhodanine-Linked Benzenesulfonamide Derivatives as Selective and Potent Human Carbonic Anhydrase Inhibitors. Molecules 27:22, pages 8028.
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Mukul Kumar, Deepika Kaushik, Jasjit Kaur, Charalampos Proestos, Fatih Oz, Emel Oz, Prerna Gupta, Priyanka Kundu, Anmol Kaur, Anisha Anisha & Ritika Ritika. (2022) A Critical Review on Obesity: Herbal Approach, Bioactive Compounds, and Their Mechanism. Applied Sciences 12:16, pages 8342.
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Pınar Eraslan‐Elma, Atilla Akdemir, Emanuela Berrino, Murat Bozdağ, Claudiu T. Supuran & Nilgün Karalı. (2022)
New 1
H
‐indole‐2,3‐dione 3‐thiosemicarbazones with 3‐sulfamoylphenyl moiety as selective carbonic anhydrase inhibitors
. Archiv der Pharmazie 355:8.
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Shiyang Zhou & Gangliang Huang. (2022) Some important inhibitors and mechanisms of rheumatoid arthritis. Chemical Biology & Drug Design 99:6, pages 930-943.
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Yun-Fei Bai, Chang Zeng, Miaomiao Jia & Bo Xiao. (2022) Molecular mechanisms of topiramate and its clinical value in epilepsy. Seizure 98, pages 51-56.
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Valeria Poggetti, Silvia Salerno, Emma Baglini, Elisabetta Barresi, Federico Da Settimo & Sabrina Taliani. (2022) Carbonic Anhydrase Activators for Neurodegeneration: An Overview. Molecules 27:8, pages 2544.
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Uğur Güller, Şükrü Beydemir & Ömer İrfan Küfrevioğlu. (2022)
In vitro
and
in silico
interactions of antiulcer, glucocorticoids and urological drugs on human carbonic anhydrase I and II isozymes
. Biopharmaceutics & Drug Disposition 43:2, pages 47-56.
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Pengcheng Lv, Yinyi Cai, Jiayi Luo & Kun Chen. (2022) Recent Advances in the Design and Synthesis of Small Molecule Carbonic
Anhydrase IX Inhibitors. Current Topics in Medicinal Chemistry 22:7, pages 550-560.
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Muhammad Danish, Ayesha Bibi, Arusa Akhtar, Nadia Noreen, Fatima Batool, Nallain Zahra, Muhammad Nadeem Arshad & Abdullah M. Asiri. (2022)
Theoretical and Experimental Investigations of
N
‐ and
O
‐Alkylated Sulfonamides: Density Functional Theory, Hirshfeld Surface Analysis, and Molecular Docking Studies
. ChemistrySelect 7:4.
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Andrea Petreni, Sameh M. Osman, Fatmah A. Alasmary, Tahani M. Almutairi, Alessio Nocentini & Claudiu T. Supuran. (2021) Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. European Journal of Medicinal Chemistry 226, pages 113875.
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Nicole Lemon, Elisa Canepa, Marc A. Ilies & Silvia Fossati. (2021) Carbonic Anhydrases as Potential Targets Against Neurovascular Unit Dysfunction in Alzheimer’s Disease and Stroke. Frontiers in Aging Neuroscience 13.
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Aysha Fatima, Meenakshi Singh, Neha Singh, Sandhya Savita, Indresh Verma, Nazia Siddiqui & Saleem Javed. (2021) Investigations on experimental, theoretical spectroscopic, electronic excitations, molecular docking of Sulfaguanidine (SG): An antibiotic drug. Chemical Physics Letters 783, pages 139049.
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Dandan Su, Yan Zhang, Sébastien Ulrich & Mihail Barboiu. (2021) Constitutional Dynamic Inhibition/Activation of Carbonic Anhydrases. ChemPlusChem 86:11, pages 1500-1510.
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Yağmur HOŞGÖR, Ekrem TUNCA & Metin BÜLBÜL. (2021) C Vitamininin Karbonik Anhidraz İzoenzimleri (hCA I ve II) Üzerine Etkisi. Afyon Kocatepe University Journal of Sciences and Engineering 21:5, pages 1038-1045.
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Michael Kugler, Jan Nekvinda, Josef Holub, Suzan El Anwar, Viswanath Das, Václav Šícha, Klára Pospíšilová, Milan Fábry, Vlastimil Král, Jiří Brynda, Václav Kašička, Marián Hajdúch, Pavlína Řezáčová & Bohumír Grüner. (2021) Inhibitors of CA IX Enzyme Based on Polyhedral Boron Compounds. ChemBioChem 22:18, pages 2741-2761.
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Chi-Ren Huang, Hung-Yi Chuang, Nai-Ching Chen, Shu-Fang Chen, Chung-Yao Hsu & Yao-Chung Chuang. (2021) Zonisamide Therapy Reduces Metabolic Consequences and Diminishes Nonalcoholic Fatty Liver Disease in Patients with Epilepsy. Journal of Clinical Medicine 10:15, pages 3380.
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Mary Sravani Galla, Darshana Bora & Nagula Shankaraiah. (2021)
The Role of Sulphonamides and
N
‐Sulphonyl Ketimines/Aldimines as Directing Groups in the Field of C−H Activation
. Chemistry – An Asian Journal 16:13, pages 1661-1684.
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Asmaa M. Sayed, Nashwa M. Saleh, Mohamed S. A. El‐Gaby, Mohammad R. K. Abdel‐Samad & Fatma A. Taher. (2021)
Synthesis and in vivo evaluation of novel benzimidazole‐sulfonamide hybrids and
Lucilia cuprina
maggots' excretion/secretion topical gels for wound healing
. Journal of the Chinese Chemical Society 68:7, pages 1291-1301.
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Baijayantimala Swain, Kamtam Aashritha, Priti Singh, Andrea Angeli, Abhay Kothari, Dilep K. Sigalapalli, Venkata M. Yaddanapudi, Claudiu T. Supuran & Mohammed Arifuddin. (2021)
Design and synthesis of benzenesulfonamide‐linked imidazo[2,1‐
b
][1,3,4]thiadiazole derivatives as carbonic anhydrase I and II inhibitors
. Archiv der Pharmazie 354:7.
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Ali Irfan, Sajjad Ahmad, Saddam Hussain, Fozia Batool, Haseeba Riaz, Rehman Zafar, Katarzyna Kotwica-Mojzych & Mariusz Mojzych. (2021) Recent Updates on the Synthesis of Bioactive Quinoxaline-Containing Sulfonamides. Applied Sciences 11:12, pages 5702.
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Claudiu T. Supuran. (2021) Emerging role of carbonic anhydrase inhibitors. Clinical Science 135:10, pages 1233-1249.
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Justina Kazokaitė-Adomaitienė, Holger M. Becker, Joana Smirnovienė, Ludwig J. Dubois & Daumantas Matulis. (2021) Experimental Approaches to Identify Selective Picomolar Inhibitors for Carbonic Anhydrase IX. Current Medicinal Chemistry 28:17, pages 3361-3384.
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Chandra Bhushan Mishra, Shikha Kumari, Andrea Angeli, Silvia Bua, Raj Kumar Mongre, Manisha Tiwari & Claudiu T. Supuran. (2021) Discovery of Potent Carbonic Anhydrase Inhibitors as Effective Anticonvulsant Agents: Drug Design, Synthesis, and In Vitro and In Vivo Investigations. Journal of Medicinal Chemistry 64:6, pages 3100-3114.
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Zafer Gurel & Nader Sheibani. 2021. The Carbonic Anhydrases: Current and Emerging Therapeutic Targets. The Carbonic Anhydrases: Current and Emerging Therapeutic Targets
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W. Richard Chegwidden. 2021. The Carbonic Anhydrases: Current and Emerging Therapeutic Targets. The Carbonic Anhydrases: Current and Emerging Therapeutic Targets
1
12
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Claudiu T. Supuran. 2021. New Trends in Macromolecular and Supramolecular Chemistry for Biological Applications. New Trends in Macromolecular and Supramolecular Chemistry for Biological Applications
115
131
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Zuhal Alım, Zeynep Köksal & Muhammet Karaman. (2020) Evaluation of some thiophene-based sulfonamides as potent inhibitors of carbonic anhydrase I and II isoenzymes isolated from human erythrocytes by kinetic and molecular modelling studies. Pharmacological Reports 72:6, pages 1738-1748.
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Lilia Clima, Bogdan Florin Craciun, Andrea Angeli, Andrea Petreni, Alessandro Bonardi, Alessio Nocentini, Fabrizio Carta, Paola Gratteri, Mariana Pinteala & Claudiu T. Supuran. (2020)
Synthesis, Computational Studies and Assessment of
in Vitro
Activity of Squalene Derivatives as Carbonic Anhydrase Inhibitors
. ChemMedChem 15:21, pages 2052-2057.
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Shuang Hao, Xue Cheng, Xin Wang, Ran An, Hang Xu, Mengbi Guo, Chuanchao Li, Yitong Wang, Zhuang Hou & Chun Guo. (2020) Design, synthesis and biological evaluation of novel carbohydrate-based sulfonamide derivatives as antitumor agents. Bioorganic Chemistry 104, pages 104237.
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Andrea Angeli, Fabrizio Carta, Alessio Nocentini, Jean-Yves Winum, Raivis Zalubovskis, Atilla Akdemir, Valentina Onnis, Wagdy M. Eldehna, Clemente Capasso, Giuseppina De Simone, Simona Maria Monti, Simone Carradori, William A. Donald, Shoukat Dedhar & Claudiu T. Supuran. (2020) Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment. Metabolites 10:10, pages 412.
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Mert O. Karataş, Samir A. A. Noma, Canbolat Gürses, Sevgi Balcıoğlu, Burhan Ateş, Bülent Alıcı & Ümit Çakır. (2020) Water Soluble Coumarin Quaternary Ammonium Chlorides: Synthesis and Biological Evaluation. Chemistry & Biodiversity 17:9.
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Aiga Grandāne, Alessio Nocentini, Ilona Domračeva, Raivis Žalubovskis & Claudiu T. Supuran. (2020) Development of oxathiino[6,5-b]pyridine 2,2-dioxide derivatives as selective inhibitors of tumor-related carbonic anhydrases IX and XII. European Journal of Medicinal Chemistry 200, pages 112300.
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Aiga Grandane, Alessio Nocentini, Thomas Werner, Raivis Zalubovskis & Claudiu T. Supuran. (2020) Benzoxepinones: A new isoform-selective class of tumor associated carbonic anhydrase inhibitors. Bioorganic & Medicinal Chemistry 28:11, pages 115496.
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Sinan Bilginer, Halise I. Gul, Feyza S. Erdal, Hiroshi Sakagami & Ilhami Gulcin. (2020)
New halogenated chalcones with cytotoxic and carbonic anhydrase inhibitory properties: 6‐(3‐Halogenated phenyl‐2‐propen‐1‐oyl)‐2(3
H
)‐benzoxazolones
. Archiv der Pharmazie 353:6.
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Zuhal ALIM. (2020) Inhibition Effect of Eosin Y on Carbonic Anhydrase (CA) I and II Isoenzymes Purified from Human Erythrocytesİnsan Eritrositlerinden Saflaştırılan Karbonik Anhidraz (CA) I ve II İzoenzimleri Üzerinde Eozin Y'nin İnhibisyon Etkisi. Iğdır Üniversitesi Fen Bilimleri Enstitüsü Dergisi 10:1, pages 338-344.
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Adem ERGÜN & Mert Olgun KARATAŞ. (2020) Synthesis, characterization, and inhibitory properties of novel N-benzylbenzimidazole-silver(I) complexes on carbonic anhydrase and polyphenol oxidase enzymes. Journal of the Institute of Science and Technology, pages 320-327.
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Audrius Zakšauskas, Edita Čapkauskaitė, Linas Jezepčikas, Vaida Linkuvienė, Vaida Paketurytė, Alexey Smirnov, Janis Leitans, Andris Kazaks, Elviss Dvinskis, Elena Manakova, Saulius Gražulis, Kaspars Tars & Daumantas Matulis. (2020) Halogenated and di-substituted benzenesulfonamides as selective inhibitors of carbonic anhydrase isoforms. European Journal of Medicinal Chemistry 185, pages 111825.
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Damiano Tanini, Antonella Capperucci, Marta Ferraroni, Fabrizio Carta, Andrea Angeli & Claudiu T. Supuran. (2020) Direct and straightforward access to substituted alkyl selenols as novel carbonic anhydrase inhibitors. European Journal of Medicinal Chemistry 185, pages 111811.
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Claudiu T. Supuran & Clemente Capasso. 2020. Physiological and Biotechnological Aspects of Extremophiles. Physiological and Biotechnological Aspects of Extremophiles
295
306
.
Justina Kazokaitė, Visvaldas Kairys, Joana Smirnovienė, Alexey Smirnov, Elena Manakova, Martti Tolvanen, Seppo Parkkila & Daumantas Matulis. (2019) Engineered Carbonic Anhydrase VI-Mimic Enzyme Switched the Structure and Affinities of Inhibitors. Scientific Reports 9:1.
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Murat Bozdag, Abdulmalik Saleh Alfawaz Altamimi, Daniela Vullo, Claudiu T. Supuran & Fabrizio Carta. (2019) State of the Art on Carbonic Anhydrase Modulators for Biomedical Purposes. Current Medicinal Chemistry 26:15, pages 2558-2573.
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Mert Ogun KARATAŞ & Adem Ergün. (2019) Synthesis, Characterization, and Carbonic Anhydrase Inhibitory Properties of Silver(I) Complexes of Benzimidazole Derivatives. Journal of the Turkish Chemical Society, Section A: Chemistry, pages 253-260.
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Micheli, Bozdag, Akgul, Carta, Guccione, Bergonzi, Bilia, Cinci, Lucarini, Parisio, Supuran, Ghelardini & Di Cesare Mannelli. (2019) Pain Relieving Effect of-NSAIDs-CAIs Hybrid Molecules: Systemic and Intra-Articular Treatments against Rheumatoid Arthritis. International Journal of Molecular Sciences 20:8, pages 1923.
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Raquel L. Bernardino, Tânia R. Dias, Bruno P. Moreira, Mariana Cunha, Alberto Barros, Elsa Oliveira, Mário Sousa, Marco G. Alves & Pedro F. Oliveira. (2019) Carbonic anhydrases are involved in mitochondrial biogenesis and control the production of lactate by human Sertoli cells. The FEBS Journal 286:7, pages 1393-1406.
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Nabih Lolak, Suleyman Akocak, Silvia Bua, Rajesh K.K. Sanku & Claudiu T. Supuran. (2019) Discovery of new ureido benzenesulfonamides incorporating 1,3,5-triazine moieties as carbonic anhydrase I, II, IX and XII inhibitors. Bioorganic & Medicinal Chemistry 27:8, pages 1588-1594.
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Robert J. Gillies, Christian Pilot, Yoshinori Marunaka & Stefano Fais. (2019) Targeting acidity in cancer and diabetes. Biochimica et Biophysica Acta (BBA) - Reviews on Cancer 1871:2, pages 273-280.
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Özgül Karlık, Nahit Gençer, Mert O. Karataş, Adem Ergün, Kübra Çıkrıkcı, Oktay Arslan, Bülent Alıcı, Işın Kılıç‐Cıkla & Namık Özdemir. (2019)
Microwave‐assisted synthesis of 1‐substituted‐1
H
‐benzimidazolium salts: Non‐competitive inhibition of human carbonic anhydrase I and II
. Archiv der Pharmazie 352:4.
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Kerem Buran, Silvia Bua, Giulio Poli, F. Önen Bayram, Tiziano Tuccinardi & Claudiu T. Supuran. (2019) Novel 8-Substituted Coumarins That Selectively Inhibit Human Carbonic Anhydrase IX and XII. International Journal of Molecular Sciences 20:5, pages 1208.
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Nabih Lolak, Suleyman Akocak, Silvia Bua & Claudiu T. Supuran. (2019) Design, synthesis and biological evaluation of novel ureido benzenesulfonamides incorporating 1,3,5-triazine moieties as potent carbonic anhydrase IX inhibitors. Bioorganic Chemistry 82, pages 117-122.
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Ali Akremi & Adel Noubigh. (2019) New organotin(IV) chlorides derived from N-(2-hydroxyphenyl)aryloxy sulfamates. Synthesis, characterization and DSC investigation. Journal of Chemical Sciences 131:2.
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Andrea Angeli, Damiano Tanini, Alessio Nocentini, Antonella Capperucci, Marta Ferraroni, Paola Gratteri & Claudiu T. Supuran. (2019) Selenols: a new class of carbonic anhydrase inhibitors. Chemical Communications 55:5, pages 648-651.
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Chuang Zhao, K.P. Rakesh, L. Ravidar, Wan-Yin Fang & Hua-Li Qin. (2019) Pharmaceutical and medicinal significance of sulfur (SVI)-Containing motifs for drug discovery: A critical review. European Journal of Medicinal Chemistry 162, pages 679-734.
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Nasr Y. Khalil, Haitham K. AlRabiah, Saad S. AL Rashoud, Ahmed Bari & Tanveer A. Wani. 2019. Profiles of Drug Substances, Excipients, and Related Methodology. Profiles of Drug Substances, Excipients, and Related Methodology
333
378
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Claudiu T. Supuran. 2019. Therapeutic Application of Nitric Oxide in Cancer and Inflammatory Disorders. Therapeutic Application of Nitric Oxide in Cancer and Inflammatory Disorders
229
242
.
Clemente Capasso & Mihail Barboiu. 2019. Carbonic Anhydrases. Carbonic Anhydrases
495
514
.
Patrizio Blandina & Claudiu T. Supuran. 2019. Carbonic Anhydrases. Carbonic Anhydrases
477
492
.
Emanuela Berrino & Fabrizio Carta. 2019. Carbonic Anhydrases. Carbonic Anhydrases
311
329
.
Daniela Vullo & Fabrizio Carta. 2019. Carbonic Anhydrases. Carbonic Anhydrases
187
222
.
Alessio Nocentini & Claudiu T. Supuran. 2019. Carbonic Anhydrases. Carbonic Anhydrases
3
16
.
Lina Baranauskienė & Daumantas Matulis. 2019. Carbonic Anhydrase as Drug Target. Carbonic Anhydrase as Drug Target
3
14
.
Anyaporn Sangkaew, Jerapan Krungkrai & Chulee Yompakdee. (2018) Development of a high throughput yeast-based screening assay for human carbonic anhydrase isozyme II inhibitors. AMB Express 8:1.
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Andrea Angeli, Sonia Del Prete, Fatmah A.S. Alasmary, Linah S. Alqahtani, Zeid AlOthman, William A. Donald, Clemente Capasso & Claudiu T. Supuran. (2018) The first activation studies of the η-carbonic anhydrase from the malaria parasite Plasmodium falciparum with amines and amino acids. Bioorganic Chemistry 80, pages 94-98.
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Zuhal Alim. (2018) 1H-indazole molecules reduced the activity of human erythrocytes carbonic anhydrase I and II isoenzymes. Journal of Biochemical and Molecular Toxicology 32:9, pages e22194.
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Audrius Zakšauskas, Edita Čapkauskaitė, Linas Jezepčikas, Vaida Linkuvienė, Miglė Kišonaitė, Alexey Smirnov, Elena Manakova, Saulius Gražulis & Daumantas Matulis. (2018) Design of two-tail compounds with rotationally fixed benzenesulfonamide ring as inhibitors of carbonic anhydrases. European Journal of Medicinal Chemistry 156, pages 61-78.
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Andrea Angeli, Marianne Kuuslahti, Seppo Parkkila & Claudiu T. Supuran. (2018) Activation studies with amines and amino acids of the α-carbonic anhydrase from the pathogenic protozoan Trypanosoma cruzi. Bioorganic & Medicinal Chemistry 26:14, pages 4187-4190.
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Andrea Angeli, William A. Donald, Seppo Parkkila & Claudiu T. Supuran. (2018) Activation studies with amines and amino acids of the β-carbonic anhydrase from the pathogenic protozoan Leishmania donovani chagasi. Bioorganic Chemistry 78, pages 406-410.
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Mam Y. Mboge, Anusha Kota, Robert McKenna & Susan C. Frost. (2018) Biophysical, Biochemical, and Cell Based Approaches Used to Decipher the Role of Carbonic Anhydrases in Cancer and to Evaluate the Potency of Targeted Inhibitors. International Journal of Medicinal Chemistry 2018, pages 1-18.
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Srinivas Angapelly, Andrea Angeli, Arbaj Jabbar Khan, P. V. Sri Ramya, Claudiu T. Supuran & Mohammed Arifuddin. (2018) Synthesis and Biological Evaluation of 4-Sulfamoylphenyl/Sulfocoumarin Carboxamides as Selective Inhibitors of Carbonic Anhydrase Isoforms hCA II, IX, and XII. ChemMedChem 13:12, pages 1165-1171.
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Ozlem Akgul, Lorenzo Di Cesare Mannelli, Daniela Vullo, Andrea Angeli, Carla Ghelardini, Gianluca Bartolucci, Abdulmalik Saleh Alfawaz Altamimi, Andrea Scozzafava, Claudiu T. Supuran & Fabrizio Carta. (2018) Discovery of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs–CAIs) for the Management of Rheumatoid Arthritis. Journal of Medicinal Chemistry 61:11, pages 4961-4977.
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Morteza Abdoli, Murat Bozdag, Andrea Angeli & Claudiu Supuran. (2018) Benzamide-4-Sulfonamides Are Effective Human Carbonic Anhydrase I, II, VII, and IX Inhibitors. Metabolites 8:2, pages 37.
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Hirotaka Iwaki, Kazutaka Jin, Mayu Fujikawa, Nobukazu Nakasato & Sunao Kaneko. (2018) Topiramate-induced weight loss depends on level of intellectual disability in patients with epilepsy. Epilepsy & Behavior 83, pages 87-91.
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Niccolò Chiaramonte, Maria Romanelli, Elisabetta Teodori & Claudiu Supuran. (2018) Amino Acids as Building Blocks for Carbonic Anhydrase Inhibitors. Metabolites 8:2, pages 36.
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Chandra Bhushan Mishra, Shikha Kumari, Andrea Angeli, Silvia Bua, Manisha Tiwari & Claudiu T. Supuran. (2018) Discovery of Benzenesulfonamide Derivatives as Carbonic Anhydrase Inhibitors with Effective Anticonvulsant Action: Design, Synthesis, and Pharmacological Evaluation. Journal of Medicinal Chemistry 61:7, pages 3151-3165.
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Nabih Lolak, Suleyman Akocak, Silvia Bua, Murat Koca & Claudiu T. Supuran. (2018) Design and synthesis of novel 1,3-diaryltriazene-substituted sulfonamides as potent and selective carbonic anhydrase II inhibitors. Bioorganic Chemistry 77, pages 542-547.
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Andrea Angeli, Sonia Del Prete, William A. Donald, Clemente Capasso & Claudiu T. Supuran. (2018) The γ-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae is potently activated by amines and amino acids. Bioorganic Chemistry 77, pages 1-5.
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Claudiu Supuran. (2018) Carbonic Anhydrases and Metabolism. Metabolites 8:2, pages 25.
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Claudiu T Supuran. (2018) Carbonic anhydrase activators. Future Medicinal Chemistry 10:5, pages 561-573.
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Ramazan Ulus, İbrahim Esirden, Burak Aday, Gurbet Çelik Turgut, Alaattin Şen & Muharrem Kaya. (2017) Synthesis of novel acridine-sulfonamide hybrid compounds as acetylcholinesterase inhibitor for the treatment of alzheimer’s disease. Medicinal Chemistry Research 27:2, pages 634-641.
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Aikaterini Peperidou, Silvia Bua, Murat Bozdag, Dimitra Hadjipavlou-Litina & Claudiu Supuran. (2018) Novel 6- and 7-Substituted Coumarins with Inhibitory Action against Lipoxygenase and Tumor-Associated Carbonic Anhydrase IX. Molecules 23:1, pages 153.
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Vaida Linkuvienė, Asta Zubrienė, Elena Manakova, Vytautas Petrauskas, Lina Baranauskienė, Audrius Zakšauskas, Alexey Smirnov, Saulius Gražulis, John E. Ladbury & Daumantas Matulis. (2018) Thermodynamic, kinetic, and structural parameterization of human carbonic anhydrase interactions toward enhanced inhibitor design. Quarterly Reviews of Biophysics 51.
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Ylenia Cau, Daniela Vullo, Mattia Mori, Elena Dreassi, Claudiu Supuran & Maurizio Botta. (2017) Potent and Selective Carboxylic Acid Inhibitors of Tumor-Associated Carbonic Anhydrases IX and XII. Molecules 23:1, pages 17.
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Srinivas Angapelly, P.V. Sri Ramya, Andrea Angeli, Sonia Del Prete, Clemente Capasso, Mohammed Arifuddin & Claudiu T. Supuran. (2017) Development of sulfonamides incorporating phenylacrylamido functionalities as carbonic anhydrase isoforms I, II, IX and XII inhibitors. Bioorganic & Medicinal Chemistry 25:20, pages 5726-5732.
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Claudiu Supuran. (2017) Special Issue: Sulfonamides. Molecules 22:10, pages 1642.
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Nilgün Karalı, Atilla Akdemir, Füsun Göktaş, Pınar Eraslan Elma, Andrea Angeli, Merih Kızılırmak & Claudiu T. Supuran. (2017) Novel sulfonamide-containing 2-indolinones that selectively inhibit tumor-associated alpha carbonic anhydrases. Bioorganic & Medicinal Chemistry 25:14, pages 3714-3718.
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Fabrizio Carta, Alexander Birkmann, Tamara Pfaff, Helmut Buschmann, Wilfried Schwab, Holger Zimmermann, Alfonso Maresca & Claudiu T. Supuran. (2017) Lead Development of Thiazolylsulfonamides with Carbonic Anhydrase Inhibitory Action. Journal of Medicinal Chemistry 60:7, pages 3154-3164.
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Menshawy A. Mohamed, Alaa A.-M. Abdel-Aziz, Helmy M. Sakr, Adel S. El-Azab, Silvia Bua & Claudiu T. Supuran. (2017) Synthesis and human/bacterial carbonic anhydrase inhibition with a series of sulfonamides incorporating phthalimido moieties. Bioorganic & Medicinal Chemistry 25:8, pages 2524-2529.
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Chandra Bhushan Mishra, Shikha Kumari, Andrea Angeli, Simona Maria Monti, Martina Buonanno, Manisha Tiwari & Claudiu T. Supuran. (2017) Discovery of Benzenesulfonamides with Potent Human Carbonic Anhydrase Inhibitory and Effective Anticonvulsant Action: Design, Synthesis, and Pharmacological Assessment. Journal of Medicinal Chemistry 60:6, pages 2456-2469.
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Alaa A.-M. Abdel-Aziz, Andrea Angeli, Adel S. El-Azab, Mohamed A. Abu El-Enin & Claudiu T. Supuran. (2017) Synthesis and biological evaluation of cyclic imides incorporating benzenesulfonamide moieties as carbonic anhydrase I, II, IV and IX inhibitors. Bioorganic & Medicinal Chemistry 25:5, pages 1666-1671.
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Silvia Bua, Lorenzo Di Cesare Mannelli, Daniela Vullo, Carla Ghelardini, Gianluca Bartolucci, Andrea Scozzafava, Claudiu T. Supuran & Fabrizio Carta. (2017) Design and Synthesis of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs–CAIs) for the Treatment of Rheumatoid Arthritis. Journal of Medicinal Chemistry 60:3, pages 1159-1170.
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Crossref
Ramazan Ulus, Belma Zengin Kurt, Isil Gazioğlu & Muharrem Kaya. (2017) Microwave assisted synthesis of novel hybrid tacrine-sulfonamide derivatives and investigation of their antioxidant and anticholinesterase activities. Bioorganic Chemistry 70, pages 245-255.
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Murat Bozdag, Ahmed Mahmoud Alafeefy, Abdul Malik Altamimi, Daniela Vullo, Fabrizio Carta & Claudiu T. Supuran. (2017) Coumarins and other fused bicyclic heterocycles with selective tumor-associated carbonic anhydrase isoforms inhibitory activity. Bioorganic & Medicinal Chemistry 25:2, pages 677-683.
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Srinivas Angapelly, P.V. Sri Ramya, Andrea Angeli, Simona Maria Monti, Martina Buonanno, Mallika Alvala, Cladiu T. Supuran & Mohammed Arifuddin. (2017) Discovery of 4-sulfamoyl-phenyl-β-lactams as a new class of potent carbonic anhydrase isoforms I, II, IV and VII inhibitors: The first example of subnanomolar CA IV inhibitors. Bioorganic & Medicinal Chemistry 25:2, pages 539-544.
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Alessio Nocentini, Marta Ferraroni, Fabrizio Carta, Mariangela Ceruso, Paola Gratteri, Cecilia Lanzi, Emanuela Masini & Claudiu T. Supuran. (2016) Benzenesulfonamides Incorporating Flexible Triazole Moieties Are Highly Effective Carbonic Anhydrase Inhibitors: Synthesis and Kinetic, Crystallographic, Computational, and Intraocular Pressure Lowering Investigations. Journal of Medicinal Chemistry 59:23, pages 10692-10704.
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Anastasia Karioti, Fabrizio Carta & Claudiu Supuran. (2016) Phenols and Polyphenols as Carbonic Anhydrase Inhibitors. Molecules 21:12, pages 1649.
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Murat Bozdag, Ahmed M. Alafeefy, Fabrizio Carta, Mariangela Ceruso, Abdul-Malek S. Al-Tamimi, Abdulla A. Al-Kahtani, Fatmah A.S. Alasmary & Claudiu T. Supuran. (2016) Synthesis 4-[2-(2-mercapto-4-oxo-4H-quinazolin-3-yl)-ethyl]-benzenesulfonamides with subnanomolar carbonic anhydrase II and XII inhibitory properties. Bioorganic & Medicinal Chemistry 24:18, pages 4100-4107.
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Leonardo E. Riafrecha, Silvia Bua, Claudiu T. Supuran & Pedro A. Colinas. (2016) Synthesis and carbonic anhydrase inhibitory effects of new N-glycosylsulfonamides incorporating the phenol moiety. Bioorganic & Medicinal Chemistry Letters 26:16, pages 3892-3895.
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Claudiu T. Supuran. (2016) Structure and function of carbonic anhydrases. Biochemical Journal 473:14, pages 2023-2032.
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Giosuè Costa, Maria Concetta Gidaro, Daniela Vullo, Claudiu T. Supuran & Stefano Alcaro. (2016) Active Components of Essential Oils as Anti-Obesity Potential Drugs Investigated by in Silico Techniques. Journal of Agricultural and Food Chemistry 64:26, pages 5295-5300.
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Daniela Vullo, Mariaconcetta Durante, Francesco Saverio Di Leva, Sandro Cosconati, Emanuela Masini, Andrea Scozzafava, Ettore Novellino, Claudiu T. Supuran & Fabrizio Carta. (2016) Monothiocarbamates Strongly Inhibit Carbonic Anhydrases in Vitro and Possess Intraocular Pressure Lowering Activity in an Animal Model of Glaucoma. Journal of Medicinal Chemistry 59:12, pages 5857-5867.
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Osman Tektas, Ebru Akkemik & Haci Baykara. (2016) Investigation of the Effect of Some Optically Active Imine Compounds on the Enzyme Activities of hCA-I and hCA-II under In Vitro Conditions: An Experimental and Theoretical Study. Journal of Biochemical and Molecular Toxicology 30:6, pages 277-286.
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Atilla Akdemir, Özlen Güzel-Akdemir, Nilgün Karalı & Claudiu T. Supuran. (2016) Isatin analogs as novel inhibitors of Candida spp. β-carbonic anhydrase enzymes. Bioorganic & Medicinal Chemistry 24:8, pages 1648-1652.
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D. Haslam. (2016) Weight management in obesity – past and present. International Journal of Clinical Practice 70:3, pages 206-217.
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Ahmed M. Alafeefy, Fabrizio Carta, Mariangela Ceruso, Abdul-Malek S. Al-Tamimi, Abdulla A. Al-Kahtani & Claudiu T. Supuran. (2016) Development of 3-(4-aminosulphonyl)-phenyl-2-mercapto-3H-quinazolin-4-ones as inhibitors of carbonic anhydrase isoforms involved in tumorigenesis and glaucoma. Bioorganic & Medicinal Chemistry 24:6, pages 1402-1407.
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Aistė Kasiliauskaitė, Vida Časaitė, Vaida Juozapaitienė, Asta Zubrienė, Vilma Michailovienė, Jurgita Revuckienė, Lina Baranauskienė, Rolandas Meškys & Daumantas Matulis. (2015) Thermodynamic characterization of human carbonic anhydrase VB stability and intrinsic binding of compounds. Journal of Thermal Analysis and Calorimetry 123:3, pages 2191-2200.
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B. Richichi, V. Baldoneschi, S. Burgalassi, M. Fragai, D. Vullo, A. Akdemir, E. Dragoni, A. Louka, M. Mamusa, D. Monti, D. Berti, E. Novellino, G. De Rosa, C. T. Supuran & C. Nativi. (2015) A Divalent PAMAM‐Based Matrix Metalloproteinase/Carbonic Anhydrase Inhibitor for the Treatment of Dry Eye Syndrome. Chemistry – A European Journal 22:5, pages 1714-1721.
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Marta Ferraroni, Fabrizio Carta, Andrea Scozzafava & Claudiu T. Supuran. (2015) Thioxocoumarins Show an Alternative Carbonic Anhydrase Inhibition Mechanism Compared to Coumarins. Journal of Medicinal Chemistry 59:1, pages 462-473.
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Anna Di Fiore, Giuseppina De Simone, Vincenzo Alterio, Vincenzo Riccio, Jean-Yves Winum, Fabrizio Carta & Claudiu T. Supuran. (2016) The anticonvulsant sulfamide JNJ-26990990 and its S,S-dioxide analog strongly inhibit carbonic anhydrases: solution and X-ray crystallographic studies. Organic & Biomolecular Chemistry 14:21, pages 4853-4858.
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Adel S. El-Azab, Alaa A.-M. Abdel-Aziz, Rezk R. Ayyad, Mariangela Ceruso & Claudiu T. Supuran. (2016) Inhibition of carbonic anhydrase isoforms I, II, IV, VII and XII with carboxylates and sulfonamides incorporating phthalimide/phthalic anhydride scaffolds. Bioorganic & Medicinal Chemistry 24:1, pages 20-25.
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Anastasia Karioti, Mariangela Ceruso, Fabrizio Carta, Anna-Rita Bilia & Claudiu T. Supuran. (2015) New natural product carbonic anhydrase inhibitors incorporating phenol moieties. Bioorganic & Medicinal Chemistry 23:22, pages 7219-7225.
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