Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 24, Issue 4 (2009)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 24, Issue 4 (2009)

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Research Article

Article
Effect of a bis-thiazolium compound on the biosynthesis of Plasmodium falciparum phospholipids
Hugues Ahiboh, Allico J Djaman, Félix H Yapi, Angèle Edjeme-Aké, Marie-Laure Hauhouot-Attoungbré, Eric D Yayo & Dagui Monnet
Pages: 911-917
Published online: 22 Jul 2009
AbstractforEffect of a bis-thiazolium compound on the biosynthesis of Plasmodium falciparum phospholipids | Full Text | References | PDF (1,021.5 KB)
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Article
Design, synthesis and pharmacological evaluation of 6-hydroxy-4-methylquinolin-2(1H)-one derivatives as inotropic agents
Hamid Sadeghian, Seyed Mohammad Seyedi, Mohammad Reza Saberi, Reza Shafiee Nick, Azar Hosseini, Mehdi Bakavoli, Seyed Mohammad Taghi Mansouri & Heydar Parsaee
Pages: 918-929
Published online: 08 Apr 2009
AbstractforDesign, synthesis and pharmacological evaluation of 6-hydroxy-4-methylquinolin-2(1H)-one derivatives as inotropic agents | Full Text | References | PDF (2.6 MB)
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Article
Effect of ammonium, sodium, and potassium ions on rabbit muscle phosphofructokinase-1 and adenylate kinase activities
Percy Russell, Anita Williams, Karla Marquez, Tina Hua, Farnaz Ehya, Chanae Hardamon, Traci Tallman & Pierre Valdez
Pages: 930-936
Published online: 07 Apr 2009
AbstractforEffect of ammonium, sodium, and potassium ions on rabbit muscle phosphofructokinase-1 and adenylate kinase activities | Full Text | References | PDF (872.2 KB)
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Article
QSAR of aminopyrido[2,3-d]pyrimidin-7-yl derivatives: Anticancer drug design by computed descriptors
Sisir Nandi & Manish C. Bagchi
Pages: 937-948
Published online: 07 Apr 2009
AbstractforQSAR of aminopyrido[2,3-d]pyrimidin-7-yl derivatives: Anticancer drug design by computed descriptors | Full Text | References | PDF (1.5 MB)
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Article
Synthesis and evaluation of in vitro antiviral activity of 2-[3-(substituted phenyl)-4,5-dihydro-1H-5-pyrazolyl]benzofuran-3-yl chloride derivatives
M. Shahar Yar, M. Mustaqeem Abdullah, A. Husain, M. Afroz Bhakht & Erik De Clercq
Pages: 949-956
Published online: 08 Apr 2009
AbstractforSynthesis and evaluation of in vitro antiviral activity of 2-[3-(substituted phenyl)-4,5-dihydro-1H-5-pyrazolyl]benzofuran-3-yl chloride derivatives | Full Text | References | PDF (869.6 KB)
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Article
Aldose reductase inhibitors from Litchi chinensis Sonn
Sung-Jae Lee, Won-Hwan Park, Sun-Dong Park & Hyung-In Moon
Pages: 957-959
Published online: 07 Apr 2009
AbstractforAldose reductase inhibitors from Litchi chinensis Sonn | Full Text | References | PDF (747.9 KB)
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Article
Design, synthesis and evaluation of some 1,3,5-triazinyl urea and thiourea derivatives as antimicrobial agents
Kishor H Chikhalia & Mayank J Patel
Pages: 960-966
Published online: 08 Apr 2009
AbstractforDesign, synthesis and evaluation of some 1,3,5-triazinyl urea and thiourea derivatives as antimicrobial agents | Full Text | References | PDF (695.5 KB)
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Article
Comparative effect of N-substituted dehydroamino acids and α-tocopherol on rat liver lipid peroxidation activities
Paula M. T. Ferreira, Luis S. Monteiro, T. Coban & S. Suzen
Pages: 967-971
Published online: 08 Apr 2009
AbstractforComparative effect of N-substituted dehydroamino acids and α-tocopherol on rat liver lipid peroxidation activities | Full Text | References | PDF (841.7 KB)
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Article
Synthesis of imidazole-containing analogues of farnesyl pyrophosphate and evaluation of their biological activity on protein farnesyltransferase
Laëtitia Coudray, Renata Marcia de Figueiredo, Stéphanie Duez, Sylvie Cortial & Joëlle Dubois
Pages: 972-985
Published online: 08 Apr 2009
AbstractforSynthesis of imidazole-containing analogues of farnesyl pyrophosphate and evaluation of their biological activity on protein farnesyltransferase | Full Text | References | PDF (1,006.2 KB)
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Article
Synthesis, characterization, antimicrobial activity and structure–activity relationships of new aryldisulfonamides
Saliha Alyar & Nurcan Karacan
Pages: 986-992
Published online: 23 Jun 2009
AbstractforSynthesis, characterization, antimicrobial activity and structure–activity relationships of new aryldisulfonamides | Full Text | References | PDF (638.8 KB)
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Article
Antioxidant phenylpropanoid glycosides from Buddleja davidii
Ijaz Ahmad, Nisar Ahmad & Fanghai Wang
Pages: 993-997
Published online: 23 Jun 2009
AbstractforAntioxidant phenylpropanoid glycosides from Buddleja davidii | Full Text | References | PDF (720.6 KB)
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Article
Alpha glucosidase inhibition by stem extract of Tinospora cordifolia
Ashok D. Chougale, Varsha A. Ghadyale, Shrimant N. Panaskar & Akalpita U. Arvindekar
Pages: 998-1001
Published online: 23 Jun 2009
AbstractforAlpha glucosidase inhibition by stem extract of Tinospora cordifolia | Full Text | References | PDF (1 MB)
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Article
Exploration of QSAR modelling techniques and their combination to rationalize the physicochemical characters of nitrophenyl derivatives towards aldose reductase inhibition
Love Kumar Soni, Arun Kumar Gupta & S. G Kaskhedikar
Pages: 1002-1007
Published online: 10 Jun 2009
AbstractforExploration of QSAR modelling techniques and their combination to rationalize the physicochemical characters of nitrophenyl derivatives towards aldose reductase inhibition | Full Text | References | PDF (934.4 KB)
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Article
Pair wise binding affinity: 3D QSAR studies on a set of triazolo [1, 5-a] quinoxalines as antagonists of AMPA and KA receptors
Ritesh N. Sharma, Hardik M. Thakar, Kamala K. Vasu, Subhash C. Chaturvedi & Shyam S. Pancholi
Pages: 1008-1014
Published online: 23 Jun 2009
AbstractforPair wise binding affinity: 3D QSAR studies on a set of triazolo [1, 5-a] quinoxalines as antagonists of AMPA and KA receptors | Full Text | References | PDF (893.1 KB)
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Research article

Article
Synthesis and biological evaluation of new 4-thiazolidinone derivatives
Özlen Güzel & Aydın Salman
Pages: 1015-1023
Published online: 22 Jul 2009
AbstractforSynthesis and biological evaluation of new 4-thiazolidinone derivatives | Full Text | References | PDF (707.8 KB)
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Research Article

Article
Modeling of the growth hormone secretagogue receptor antagonistic activity using chemometric tools
Susheela Sharma, B. K. Sharma, P. Pilania, P. Singh & Y. S. Prabhakar
Pages: 1024-1033
Published online: 23 Jun 2009
AbstractforModeling of the growth hormone secretagogue receptor antagonistic activity using chemometric tools | Full Text | References | PDF (1 MB)
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Article
Effect of some analgesics on Paraoxonase-1 purified from human serum
Deniz EKİNCİ & Şükrü BEYDEMİR
Pages: 1034-1039
Published online: 23 Jun 2009
AbstractforEffect of some analgesics on Paraoxonase-1 purified from human serum | Full Text | References | PDF (806.8 KB)
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Article
A comparison of the reactivating and therapeutic efficacy of newly developed bispyridinium oximes (K250, K251) with commonly used oximes against tabun in rats and mice
Jiri Kassa, Jana Karasova, Jiri Bajgar, Kamil Kuca, Kamil Musilek & Irena Kopelikova
Pages: 1040-1044
Published online: 24 Jun 2009
AbstractforA comparison of the reactivating and therapeutic efficacy of newly developed bispyridinium oximes (K250, K251) with commonly used oximes against tabun in rats and mice | Full Text | References | PDF (615.2 KB)
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Article
Update on biochemical properties of recombinant Pseudomonas diminuta phosphotriesterase
Eugénie Carletti, Lilian Jacquamet, Mélanie Loiodice, Daniel Rochu, Patrick Masson & Florian Nachon
Pages: 1045-1055
Published online: 23 Jun 2009
AbstractforUpdate on biochemical properties of recombinant Pseudomonas diminuta phosphotriesterase | Full Text | References | PDF (1.7 MB)
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Article
Inhibition of protein tyrosine phosphatase 1B by lupeol and lupenone isolated from Sorbus commixta
Minkyun Na, Bo Yeon Kim, Hiroyuki Osada & Jong Seog Ahn
Pages: 1056-1059
Published online: 23 Jun 2009
AbstractforInhibition of protein tyrosine phosphatase 1B by lupeol and lupenone isolated from Sorbus commixta | Full Text | References | PDF (793.5 KB)
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Miscellany

Corrigendum
Page: 1060
Published online: 02 Apr 2009
CitationforCorrigendum | Full Text | PDF (483.9 KB)
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