Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 25, Issue 5 (2010)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 25, Issue 5 (2010)

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Original Article

Article
Some biologically active oxovanadium(IV) complexes of triazole derived Schiff bases: their synthesis, characterization and biological properties
Zahid H. Chohan & Sajjad H. Sumrra
Pages: 599-607
Published online: 30 Apr 2010
AbstractforSome biologically active oxovanadium(IV) complexes of triazole derived Schiff bases: their synthesis, characterization and biological properties | Full Text | References | PDF (814.9 KB)
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Article
RETRACTED: Antioxidant properties of benzylchroman derivatives from Caesalpinia sappan L. against oxidative stress evaluated in vitro
Min-Ja Lee, Hye-Sook Lee, Hyuck Kim, Hyo-Seung Yi, Sun-Dong Park, Hyung-In Moon & Won-Hwan Park
Pages: 608-614
Published online: 27 Jan 2010
AbstractforRETRACTED: Antioxidant properties of benzylchroman derivatives from Caesalpinia sappan L. against oxidative stress evaluated in vitro | Full Text | References | PDF (966.1 KB)
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Article
Synthesis and biological activity of pyrazolo[3,4-d]thiazolo[3,2-a]pyrimidin-4-one derivatives: in silico approach
Chandrahas N. Khobragade, Ragini G. Bodade, Bhaskar S. Dawane, Shankaraiah G. Konda & Namdev T. Khandare
Pages: 615-621
Published online: 09 Dec 2009
AbstractforSynthesis and biological activity of pyrazolo[3,4-d]thiazolo[3,2-a]pyrimidin-4-one derivatives: in silico approach | Full Text | References | PDF (781 KB)
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Article
Acetylcholinesterase and butyrylcholinesterase inhibitory activity of Pinus species essential oils and their constituents
Marco Bonesi, Federica Menichini, Rosa Tundis, Monica R. Loizzo, Filomena Conforti, Nicodemo G. Passalacqua, Giancarlo A. Statti & Francesco Menichini
Pages: 622-628
Published online: 30 Apr 2010
AbstractforAcetylcholinesterase and butyrylcholinesterase inhibitory activity of Pinus species essential oils and their constituents | Full Text | References | PDF (747.1 KB)
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Article
Carbocyclic potential DNA minor groove binders and their biological evaluation
Danuta Drozdowska, Irena Bruzgo & Krystyna Midura-Nowaczek
Pages: 629-634
Published online: 30 Apr 2010
AbstractforCarbocyclic potential DNA minor groove binders and their biological evaluation | Full Text | References | PDF (650.5 KB)
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Article
A common feature-based 3D-pharmacophore model generation and virtual screening: identification of potential PfDHFR inhibitors
Legesse Adane, Prasad V. Bharatam & Vikas Sharma
Pages: 635-645
Published online: 08 Dec 2009
AbstractforA common feature-based 3D-pharmacophore model generation and virtual screening: identification of potential PfDHFR inhibitors | Full Text | References | PDF (1.4 MB)
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Article
Inhibition studies of soybean (Glycine max) urease with heavy metals, sodium salts of mineral acids, boric acid, and boronic acids
Sandeep Kumar & Arvind M. Kayastha
Pages: 646-652
Published online: 16 Dec 2009
AbstractforInhibition studies of soybean (Glycine max) urease with heavy metals, sodium salts of mineral acids, boric acid, and boronic acids | Full Text | References | PDF (728.5 KB)
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Article
Synthesis of new 8(S)-HETE analogs and their biological evaluation as activators of the PPAR nuclear receptors
Mélanie Liutkus, Frédéric Caijo, Anne-Lise Girard, Erwan Ayral, Valérie Audinot, Jean A. Boutin, Pierre Renard, Daniel Henri Caignard, Catherine Dacquet, Alain Ktorza, Paul Mosset & René Grée
Pages: 653-672
Published online: 02 Jun 2010
AbstractforSynthesis of new 8(S)-HETE analogs and their biological evaluation as activators of the PPAR nuclear receptors | Full Text | References | PDF (1.1 MB)
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Research Article

Article
Characterisation of hydrazides and hydrazine derivatives as novel aspartic protease inhibitors
Waseem Ahmed, Mubeen Rani, Ishtiaq A. Khan, Asif Iqbal, Khalid M. Khan, M. A. Haleem & M. Kamran Azim
Pages: 673-678
Published online: 11 Jan 2010
AbstractforCharacterisation of hydrazides and hydrazine derivatives as novel aspartic protease inhibitors | Full Text | References | PDF (1.1 MB)
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Article
Quantitative structure-activity relationships (QSARs) for inhibitors and substrates of CYP2B enzymes: importance of compound lipophilicity in explanation of potency differences
David FV Lewis, Yuko Ito & Brian G Lake
Pages: 679-684
Published online: 25 Jan 2010
AbstractforQuantitative structure-activity relationships (QSARs) for inhibitors and substrates of CYP2B enzymes: importance of compound lipophilicity in explanation of potency differences | Full Text | References | PDF (744.2 KB)
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Article
Synthesis and antioxidant properties of diphenylmethane derivative bromophenols including a natural product
Halis Türker Balaydın, İlhami Gülçin, Abdullah Menzek, Süleyman Göksu & Ertan Şahin
Pages: 685-695
Published online: 30 Jan 2010
AbstractforSynthesis and antioxidant properties of diphenylmethane derivative bromophenols including a natural product | Full Text | References | PDF (896 KB)
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Article
QSAR model for predicting the fungicidal action of 1,2,4-triazole derivatives against Candida albicans
Rajeev K Singla & Varadaraj Bhat G
Pages: 696-701
Published online: 30 Apr 2010
AbstractforQSAR model for predicting the fungicidal action of 1,2,4-triazole derivatives against Candida albicans | Full Text | References | PDF (1,004.4 KB)
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Article
Protective effects of luteolin-7-O-β-D-glucuronide methyl ester from the ethyl acetate fraction of Lycopi Herba against pro-oxidant reactive species and low-density lipoprotein peroxidation
Min-Ja Lee, Hye-Sook Lee, Sun-Dong Park, Hyung-In Moon & Won-Hwan Park
Pages: 702-707
Published online: 27 Jan 2010
AbstractforProtective effects of luteolin-7-O-β-D-glucuronide methyl ester from the ethyl acetate fraction of Lycopi Herba against pro-oxidant reactive species and low-density lipoprotein peroxidation | Full Text | References | PDF (711 KB)
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Article
Synthesis, structural characterisation and antibacterial activity of bis(1-phenyl-1,3-butanedionato)non-oxovanadium(IV) hydroxamates
Neeraj Sharma, Meena Kumari, Vijay Kumar & S.C. Chaudhry
Pages: 708-714
Published online: 03 Mar 2010
AbstractforSynthesis, structural characterisation and antibacterial activity of bis(1-phenyl-1,3-butanedionato)non-oxovanadium(IV) hydroxamates | Full Text | References | PDF (728.4 KB)
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Article
Differential effects of some antibiotics on paraoxonase enzyme activity on human hepatoma cells (HepG2) in vitro
Feray Kockar, Selma Sinan, Hatice Yildirim & Oktay Arslan
Pages: 715-719
Published online: 30 Apr 2010
AbstractforDifferential effects of some antibiotics on paraoxonase enzyme activity on human hepatoma cells (HepG2) in vitro | Full Text | References | PDF (714.7 KB)
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Article
Curcumin inhibits TNFα-induced lectin-like oxidised LDL receptor-1 (LOX-1) expression and suppresses the inflammatory response in human umbilical vein endothelial cells (HUVECs) by an antioxidant mechanism
Hye-Sook Lee, Min-Ja Lee, Hyuck Kim, Sung-Kyu Choi, Jai-Eun Kim, Hyung-In Moon & Won-Hwan Park
Pages: 720-729
Published online: 18 Feb 2010
AbstractforCurcumin inhibits TNFα-induced lectin-like oxidised LDL receptor-1 (LOX-1) expression and suppresses the inflammatory response in human umbilical vein endothelial cells (HUVECs) by an antioxidant mechanism | Full Text | References | PDF (966.1 KB)
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Article
Synthesis and antitubercular activity of heterocycle substituted diphenyl ether derivatives
Suvarna G. Kini, Anilchandra Bhat, Zhiqiang Pan & Franck E. Dayan
Pages: 730-736
Published online: 05 May 2010
AbstractforSynthesis and antitubercular activity of heterocycle substituted diphenyl ether derivatives | Full Text | References | PDF (780.1 KB)
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Original Article

Article
Design, synthesis, and biological properties of triazole derived compounds and their transition metal complexes
Zahid H. Chohan & Muhammad Hanif
Pages: 737-749
Published online: 22 Jun 2010
AbstractforDesign, synthesis, and biological properties of triazole derived compounds and their transition metal complexes | Full Text | References | PDF (1.2 MB)
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