Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 26, Issue 3 (2011)

Browse this journal
Sample our Bioscience journals, sign in here to start your access, Latest two full volumes FREE to you for 14 days

Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 26, Issue 3 (2011)

See all volumes and issues
Vol 39, 2024 Vol 38, 2023 Vol 37, 2022 Vol 36, 2021 Vol 35, 2020 Vol 34, 2019 Vol 33, 2018 Vol 32, 2017 Vol 31, 2016 Vol 30, 2015 Vol 29, 2014 Vol 28, 2013 Vol 27, 2012 Volume 26, 2011 Vol 25, 2010 Vol 24, 2009 Vol 23, 2008 Vol 22, 2007 Vol 21, 2006 Vol 20, 2005 Vol 19, 2004 Vol 18, 2003 Vol 17, 2002 Vol 16, 2001 Vol 15, 1999-2000 Vol 14, 1998-1999 Vol 13, 1998 Vol 12, 1997 Vol 11, 1996-1997 Vol 10, 1995-1996 Vol 9, 1995 Vol 8, 1994-1995 Vol 7, 1993 Vol 6, 1992-1993 Vol 5, 1991 Vol 4, 1990-1991 Vol 3, 1989-1990 Vol 2, 1987-1989 Vol 1, 1985-1987
Download citations Download PDFs Download issue

Editorial

Editorial
Enzyme Inhibition and more− A Tribute to John Smith
Claudiu T. Supuran
Pages: 301-302
Published online: 27 Apr 2011
CitationforEnzyme Inhibition and more− A Tribute to John Smith | Full Text | PDF (636.6 KB)
  • 422 Views
  • 8 CrossRef citations
  • 0Altmetric
Free Access

Review Article

Article
Kinetic prerequisites of oximes as effective reactivators of organophosphate-inhibited acetylcholinesterase: a theoretical approach
Franz Worek, Nadine Aurbek, Timo Wille, Peter Eyer & Horst Thiermann
Pages: 303-308
Published online: 31 Aug 2010
AbstractforKinetic prerequisites of oximes as effective reactivators of organophosphate-inhibited acetylcholinesterase: a theoretical approach | Full Text | References | PDF (900.9 KB)
  • 727 Views
  • 7 CrossRef citations
  • 0Altmetric
Free Access

Research Article

Article
Urease activity and l-ascorbic acid
Barbara Krajewska & Małgorzata Brindell
Pages: 309-318
Published online: 09 Aug 2010
AbstractforUrease activity and l-ascorbic acid | Full Text | References | PDF (918.5 KB)
  • 2158 Views
  • 9 CrossRef citations
  • 0Altmetric
Free Access
Article
Use of Quantitative Structure–Activity Relationship (QSAR) and ADMET prediction studies as screening methods for design of benzyl urea derivatives for anti-cancer activity
Deepak Lokwani, Shashikant Bhandari, Radha Pujari, Padma Shastri, Ganesh shelke & Vidya Pawar
Pages: 319-331
Published online: 17 Sep 2010
AbstractforUse of Quantitative Structure–Activity Relationship (QSAR) and ADMET prediction studies as screening methods for design of benzyl urea derivatives for anti-cancer activity | Full Text | References | PDF (1,002.8 KB)
  • 1017 Views
  • 7 CrossRef citations
  • 0Altmetric
Free Access
Article
Synthesis and in vitro antimicrobial activity of novel N-(6-chlorobenzo[d]thiazol-2-yl) hydrazine carboxamide derivatives of benzothiazole class
Sadaf J. Gilani, Suroor A. Khan, Nadeem Siddiqui, Suraj P. Verma, Pooja Mullick & Ozair Alam
Pages: 332-340
Published online: 31 Aug 2010
AbstractforSynthesis and in vitro antimicrobial activity of novel N-(6-chlorobenzo[d]thiazol-2-yl) hydrazine carboxamide derivatives of benzothiazole class | Full Text | References | PDF (837.8 KB)
  • 1042 Views
  • 17 CrossRef citations
  • 0Altmetric
Free Access
Article
Design, synthesis and pharmacological evaluation of conformationally restricted N-arylsulfonyl-3-aminoalkoxy indoles as a potential 5-HT6 receptor ligands
Ramakrishna V.S. Nirogia, Ramasastri Kambhampati, Anand V. Daulatabad, Parandhama Gudla, Mohammad Shaikh, Pramod Kumar Achanta, Anil K. Shinde & Pramod Kumar Dubey
Pages: 341-349
Published online: 27 Apr 2011
AbstractforDesign, synthesis and pharmacological evaluation of conformationally restricted N-arylsulfonyl-3-aminoalkoxy indoles as a potential 5-HT6 receptor ligands | Full Text | References | PDF (822.4 KB)
  • 874 Views
  • 8 CrossRef citations
  • 0Altmetric
Free Access

Original Article

Article
Hyperbolic mixed-type inhibition of acetylcholinesterase by tetracyclic thienopyrimidines
C. M. González Tanarro & M. Gütschow
Pages: 350-358
Published online: 31 Aug 2010
AbstractforHyperbolic mixed-type inhibition of acetylcholinesterase by tetracyclic thienopyrimidines | Full Text | References | PDF (887.9 KB)
  • 873 Views
  • 14 CrossRef citations
  • 0Altmetric
Free Access
Article
Ternary copper(II) complexes of levofloxacin and phenanthroline derivatives: In-vitro antibacterial, DNA interactions, and SOD-like activity
M.N. Patel, Pradhuman Amrutsinh Parmar, Deepen Sureshbhai Gandhi & Vasudev R. Thakkar
Pages: 359-366
Published online: 27 Jan 2011
AbstractforTernary copper(II) complexes of levofloxacin and phenanthroline derivatives: In-vitro antibacterial, DNA interactions, and SOD-like activity | Full Text | References | PDF (783.7 KB) | Supplemental
  • 1085 Views
  • 10 CrossRef citations
  • 0Altmetric
Free Access
Article
Molecular modelling studies on d-annulated benzazepinones as VEGF-R2 kinase inhibitors using docking and 3D-QSAR
Ping Lan, Jun-Rong Sun, Wan-Na Chen, Ping-Hua Sun & Wei-Min Chen
Pages: 367-377
Published online: 17 Sep 2010
AbstractforMolecular modelling studies on d-annulated benzazepinones as VEGF-R2 kinase inhibitors using docking and 3D-QSAR | Full Text | References | PDF (1.1 MB)
  • 461 Views
  • 7 CrossRef citations
  • 0Altmetric
Free Access
Article
Fluorescence, circular dichroism, NMR, and docking studies of the interaction of the alkaloid malbrancheamide with calmodulin
Mario Figueroa, Martín González-Andrade, Alejandro Sosa-Peinado, Abraham Madariaga-Mazón, Federico Del Río-Portilla, María Del Carmen González & Rachel Mata
Pages: 378-385
Published online: 13 Oct 2010
AbstractforFluorescence, circular dichroism, NMR, and docking studies of the interaction of the alkaloid malbrancheamide with calmodulin | Full Text | References | PDF (868.1 KB) | Supplemental
  • 999 Views
  • 18 CrossRef citations
  • 0Altmetric
Free Access
Article
The inhibition study of human UDP-glucuronosyltransferases with cytochrome P450 selective substrates and inhibitors
Yuping Liu, Miaoqin She, Zhicong Wu & Renke Dai
Pages: 386-393
Published online: 13 Oct 2010
AbstractforThe inhibition study of human UDP-glucuronosyltransferases with cytochrome P450 selective substrates and inhibitors | Full Text | References | PDF (813.3 KB)
  • 3314 Views
  • 30 CrossRef citations
  • 0Altmetric
Free Access
Article
Transition metal complexes with N, S donor ligands as synthetic antioxidants: Synthesis, characterization and antioxidant activity
Alka Choudhary, Renu Sharma, Meena Nagar & Mohammed Mohsin
Pages: 394-403
Published online: 13 Oct 2010
AbstractforTransition metal complexes with N, S donor ligands as synthetic antioxidants: Synthesis, characterization and antioxidant activity | Full Text | References | PDF (798.1 KB)
  • 1657 Views
  • 18 CrossRef citations
  • 0Altmetric
Free Access
Article
Chemical composition and protective effect of oregano (Origanum heracleoticum L.) ethanolic extract on oxidative damage and on inhibition of NO in LPS-stimulated RAW 264.7 macrophages
Filomena Conforti, Mariangela Marrelli, Federica Menichini, Rosa Tundis, Giancarlo A. Statti, Umberto Solimene & Francesco Menichini
Pages: 404-411
Published online: 27 Apr 2011
AbstractforChemical composition and protective effect of oregano (Origanum heracleoticum L.) ethanolic extract on oxidative damage and on inhibition of NO in LPS-stimulated RAW 264.7 macrophages | Full Text | References | PDF (712.1 KB)
  • 2780 Views
  • 16 CrossRef citations
  • 0Altmetric
Free Access
Article
A QSAR study on 2-(4-methylpiperazin-1-yl)quinoxalines as human histamine H4 receptor ligands
Brij K. Sharma, Pradeep Pilania, Prithvi Singh & Yenamandra S. Prabhakar
Pages: 412-421
Published online: 13 Oct 2010
AbstractforA QSAR study on 2-(4-methylpiperazin-1-yl)quinoxalines as human histamine H4 receptor ligands | Full Text | References | PDF (832.5 KB)
  • 566 Views
  • 5 CrossRef citations
  • 0Altmetric
Free Access
Article
Evaluation of 3-(4′-(4″-fluorophenyl)-6′-phenylpyrimidin-2′-yl)-2-phenylthiazolidin-4-one for in vivo modulation of biomarkers of chemoprevention in the 7,12-dimethylbenz[a]anthracene-induced hamster buccal pouch carcinogenesis
J. Thanusu, V. Kanagarajan, S. Nagini & M. Gopalakrishnan
Pages: 422-429
Published online: 28 Oct 2010
AbstractforEvaluation of 3-(4′-(4″-fluorophenyl)-6′-phenylpyrimidin-2′-yl)-2-phenylthiazolidin-4-one for in vivo modulation of biomarkers of chemoprevention in the 7,12-dimethylbenz[a]anthracene-induced hamster buccal pouch carcinogenesis | Full Text | References | PDF (646.1 KB)
  • 331 Views
  • 2 CrossRef citations
  • 0Altmetric
Free Access
Article
Synthesis and antimicrobial studies of novel 2,4-diaryl-3-azabicyclo[3.3.1]nonan-9-one 4′-phenylthiosemicarbazones
Seeman Umamatheswari & Senthamaraikannan Kabilan
Pages: 430-439
Published online: 28 Oct 2010
AbstractforSynthesis and antimicrobial studies of novel 2,4-diaryl-3-azabicyclo[3.3.1]nonan-9-one 4′-phenylthiosemicarbazones | Full Text | References | PDF (777.2 KB)
  • 568 Views
  • 3 CrossRef citations
  • 0Altmetric
Free Access

Short Communications

Honey, polen, and propolis extracts show potent inhibitory activity against the zinc metalloenzyme carbonic anhydrase
H. Sahin, R. Aliyazicioglu, O. Yildiz, S. Kolayli, A. Innocenti & C. T. Supuran
Pages: 440-444
Published online: 05 Aug 2010
AbstractforHoney, polen, and propolis extracts show potent inhibitory activity against the zinc metalloenzyme carbonic anhydrase | Full Text | References | PDF (575.4 KB)
  • 1501 Views
  • 37 CrossRef citations
  • 0Altmetric
Free Access
A FLT3-inhibitory constituent from the rhizomes of Anemarrhena asphodeloides
Sun-Young Han & Young-Won Chin
Pages: 445-448
Published online: 17 Sep 2010
AbstractforA FLT3-inhibitory constituent from the rhizomes of Anemarrhena asphodeloides | Full Text | References | PDF (607.9 KB)
  • 573 Views
  • 4 CrossRef citations
  • 0Altmetric
Free Access
Synthesis and biological evaluation of polyhydroxy benzophenone as mushroom tyrosinase inhibitors
Jianlong Wu, Xuesen Hu & Lin Ma
Pages: 449-452
Published online: 13 Oct 2010
AbstractforSynthesis and biological evaluation of polyhydroxy benzophenone as mushroom tyrosinase inhibitors | Full Text | References | PDF (635.5 KB)
  • 1175 Views
  • 8 CrossRef citations
  • 0Altmetric
Free Access

Explore articles

Explore the most recently published articles

The activity of pyrazolo[4,3-e][1,2,4]triazine and pyrazolo[4,3-e]tetrazolo[1,5-b][1,2,4]triazine sulphonamide derivatives in monolayer and spheroid breast cancer cell cultures
Anna Szymanowska et al.
Article | Published online: 3 May 2024
Open Access
Discovery of novel FGFR4 inhibitors through a build-up fragment strategy
Jihyung Kim et al.
Brief Report | Published online: 24 Apr 2024
Open Access
Targeting bacterial growth in biofilm conditions: rational design of novel inhibitors to mitigate clinical and food contamination using QSAR
Maria Galvez-Llompart et al.
Article | Published online: 23 Apr 2024
Open Access
Evaluation of the anticancer effects exerted by 5-fluorouracil and heme oxygenase-1 inhibitor hybrids in HTC116 colorectal cancer cells
Loredana Salerno et al.
Brief Report | Published online: 18 Apr 2024
Open Access