Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 27, Issue 4 (2012)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 27, Issue 4 (2012)

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Research Article

Article
Inhibition of human carbonic anhydrase isozymes I, II and VI with a series of bisphenol, methoxy and bromophenol compounds
Halis Türker Balaydin, Serdar Durdaği, Deniz Ekinci, Murat Şentürk, Süleyman Göksu & Abdullah Menzek
Pages: 467-475
Published online: 04 Aug 2011
AbstractforInhibition of human carbonic anhydrase isozymes I, II and VI with a series of bisphenol, methoxy and bromophenol compounds | Full Text | References | PDF (1.3 MB)
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Article
Divergent effects of compounds on the hydrolysis and transpeptidation reactions of γ-glutamyl transpeptidase
Stephanie Wickham, Nicholas Regan, Matthew B. West, Vidya Prasanna Kumar, Justin Thai, Pui Kai Li, Paul F. Cook & Marie H. Hanigan
Pages: 476-489
Published online: 24 Aug 2011
AbstractforDivergent effects of compounds on the hydrolysis and transpeptidation reactions of γ-glutamyl transpeptidase | Full Text | References | PDF (1 MB)
  • 701 Views
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Article
Inhibitory alkaloids from Dictamnus dasycarpus root barks on lipopolysaccharide-induced nitric oxide production in BV2 cells
Jeong Seon Yoon, Eun Ju Jeong, Hyekyung Yang, Seung Hyun Kim, Sang Hyun Sung & Young Choong Kim
Pages: 490-494
Published online: 10 Aug 2011
AbstractforInhibitory alkaloids from Dictamnus dasycarpus root barks on lipopolysaccharide-induced nitric oxide production in BV2 cells | Full Text | References | PDF (637.4 KB)
  • 1091 Views
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Article
Evaluation of the inhibition of mushroom tyrosinase and cellular tyrosinase activities of oxyresveratrol: comparison with mulberroside A
Jeong-Keun Kim, Keun-Tae Park, Hyun-Sun Lee, Mijin Kim & Young-Hee Lim
Pages: 495-503
Published online: 10 Aug 2011
AbstractforEvaluation of the inhibition of mushroom tyrosinase and cellular tyrosinase activities of oxyresveratrol: comparison with mulberroside A | Full Text | References | PDF (875.1 KB)
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Article
Synthesis, biological screening and molecular modeling studies of novel 3-chloro-4-substituted-1-(2-(1H-benzimidazol-2-yl)phenyl))-azetidin-2-ones
Santosh S. Chhajed & Chandrashekhar D. Upasani
Pages: 504-508
Published online: 08 Aug 2011
AbstractforSynthesis, biological screening and molecular modeling studies of novel 3-chloro-4-substituted-1-(2-(1H-benzimidazol-2-yl)phenyl))-azetidin-2-ones | Full Text | References | PDF (710 KB)
  • 741 Views
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Article
Synthesis and characterization of novel dioxoacridine sulfonamide derivatives as new carbonic anhydrase inhibitors
Muharrem Kaya, Erhan Basar, Emrah Çakir, Ekrem Tunca & Metin Bülbül
Pages: 509-514
Published online: 16 Aug 2011
AbstractforSynthesis and characterization of novel dioxoacridine sulfonamide derivatives as new carbonic anhydrase inhibitors | Full Text | References | PDF (658.4 KB)
  • 1131 Views
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Article
Synthesis of some N-[4-(benzothiazole-2yl) phenyl]-2-aryloxyacetamide derivatives and their anticancer activities
Funda Tay, Leyla Yurttaş & Şeref Demirayak
Pages: 515-520
Published online: 08 Aug 2011
AbstractforSynthesis of some N-[4-(benzothiazole-2yl) phenyl]-2-aryloxyacetamide derivatives and their anticancer activities | Full Text | References | PDF (606.1 KB)
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Article
Effects of cysteinyl-leukotriene receptors’ antagonism by montelukast on lung mechanics and olfactory system histology in healthy mice
Alessandro Rubini, Michela Bondì & Carla Mucignat-Caretta
Pages: 521-527
Published online: 10 Aug 2011
AbstractforEffects of cysteinyl-leukotriene receptors’ antagonism by montelukast on lung mechanics and olfactory system histology in healthy mice | Full Text | References | PDF (643.7 KB)
  • 453 Views
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Article
Synthesis, inhibitory activity and molecular docking studies of two Cu(II) complexes against Helicobacter pylori urease
Yong-Ming Cui, Xiong-Wei Dong, Wu Chen, Wen-Jun Wang, Yu-Guang Li & Hai-Liang Zhu
Pages: 528-532
Published online: 18 Jul 2012
AbstractforSynthesis, inhibitory activity and molecular docking studies of two Cu(II) complexes against Helicobacter pylori urease | Full Text | References | PDF (711.3 KB) | Supplemental
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Article
Definition of peptide inhibitors from a synthetic peptide library by targeting gelatinase B/matrix metalloproteinase-9 (MMP-9) and TNF-α converting enzyme (TACE/ADAM-17)
Zheng Qiu, Ming Yan, Qian Li, Datao Liu, Philippe E. Van den Steen, Min Wang, Ghislain Opdenakker & Jialiang Hu
Pages: 533-540
Published online: 10 Aug 2011
AbstractforDefinition of peptide inhibitors from a synthetic peptide library by targeting gelatinase B/matrix metalloproteinase-9 (MMP-9) and TNF-α converting enzyme (TACE/ADAM-17) | Full Text | References | PDF (735.2 KB)
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Article
Design, synthesis and biological evaluation of novel quinazoline derivatives as potential anti-cancer agents
Ahmed M. Alafeefy & Abdelkader E. Ashour
Pages: 541-545
Published online: 18 Aug 2011
AbstractforDesign, synthesis and biological evaluation of novel quinazoline derivatives as potential anti-cancer agents | Full Text | References | PDF (634.9 KB)
  • 1255 Views
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Article
Inhibition of Lck: evidence for a novel natural Src family kinase inhibitor
Shudong Zhu, Donald J. Fujita & Jerry H. C. Wang
Pages: 546-552
Published online: 10 Aug 2011
AbstractforInhibition of Lck: evidence for a novel natural Src family kinase inhibitor | Full Text | References | PDF (745.3 KB)
  • 759 Views
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Article
Ranitidine induces inhibition and structural changes in sucrase
Dariush Minai-Tehrani, Mina Ghaffari, Zahra Sobhani-Damavandifar, Saeed Minoui, Sana Alavi, Rahele Osmani & Shiva Ahmadi
Pages: 553-557
Published online: 18 Aug 2011
AbstractforRanitidine induces inhibition and structural changes in sucrase | Full Text | References | PDF (609.6 KB)
  • 1669 Views
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Article
Pharmacophore generation and atom-based 3D-QSAR of novel quinoline-3-carbonitrile derivatives as Tpl2 kinase inhibitors
Mahesh Kumar Teli & G. K. Rajanikant
Pages: 558-570
Published online: 18 Aug 2011
AbstractforPharmacophore generation and atom-based 3D-QSAR of novel quinoline-3-carbonitrile derivatives as Tpl2 kinase inhibitors | Full Text | References | PDF (1.3 MB) | Supplemental
  • 1111 Views
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Article
Predicting subsite interactions of plasmin with substrates and inhibitors through computational docking analysis
Keigo Gohda, Naoki Teno, Keiko Wanaka & Yuko Tsuda
Pages: 571-577
Published online: 12 Oct 2011
AbstractforPredicting subsite interactions of plasmin with substrates and inhibitors through computational docking analysis | Full Text | References | PDF (965.1 KB)
  • 666 Views
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Article
Inhibitory effect of Terminalia chebula Retz. fruit extracts on digestive enzyme related to diabetes and oxidative stress
Indu Sasidharan, A. Sundaresan, V. M. Nisha, Mahesh S. Kirishna, K. G. Raghu & P. Jayamurthy
Pages: 578-586
Published online: 18 Apr 2012
AbstractforInhibitory effect of Terminalia chebula Retz. fruit extracts on digestive enzyme related to diabetes and oxidative stress | Full Text | References | PDF (1 MB)
  • 1729 Views
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Article
Apoptotic, antioxidant and antiradical effects of majdine and isomajdine from Vinca herbacea Waldst. and kit
I˙lhami Gülçi˙n, Şükrü Beydemi˙r, Fevzi Topal, Natia Gagua, Aliko Bakuridze, Recep Bayram & Akçahan Gepdiremen
Pages: 587-594
Published online: 02 Sep 2011
AbstractforApoptotic, antioxidant and antiradical effects of majdine and isomajdine from Vinca herbacea Waldst. and kit | Full Text | References | PDF (750.2 KB)
  • 1229 Views
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Article
Effects of some metals on paraoxonase activity from shark Scyliorhinus canicula
Demet Sayın, Dilek Türker Çakır, Nahit Gençer & Oktay Arslan
Pages: 595-598
Published online: 02 Sep 2011
AbstractforEffects of some metals on paraoxonase activity from shark Scyliorhinus canicula | Full Text | References | PDF (559 KB)
  • 761 Views
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Article
Synthesis, characterization and in vitro antimicrobial evaluation of new compounds incorporating oxindole nucleus
Nadia G. Kandile, Howida T. Zaky, Mansoura I. Mohamed, Hind M. Ismaeel & Nashwa A. Ahmed
Pages: 599-608
Published online: 03 May 2011
AbstractforSynthesis, characterization and in vitro antimicrobial evaluation of new compounds incorporating oxindole nucleus | Full Text | References | PDF (778.9 KB)
  • 1194 Views
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Short Communications

Antiproliferative activity of some 1,4-dimethylcarbazoles on cells that express estrogen receptors: part I
Anna Caruso, Adele Chimento, Hussein El-Kashef, Jean-Charles Lancelot, Antonella Panno, Vincenzo Pezzi, Carmela Saturnino, Maria Stefania Sinicropi, Rosa Sirianni & Sylvain Rault
Pages: 609-613
Published online: 02 Sep 2011
AbstractforAntiproliferative activity of some 1,4-dimethylcarbazoles on cells that express estrogen receptors: part I | Full Text | References | PDF (719.5 KB)
  • 669 Views
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Using C60 fullerenes for photodynamic inactivation of mosquito iridescent viruses
Yu. Rud, L. Buchatskyy, Yu. Prylutskyy, O. Marchenko, A. Senenko, Ch. Schütze & U. Ritter
Pages: 614-617
Published online: 02 Sep 2011
AbstractforUsing C60 fullerenes for photodynamic inactivation of mosquito iridescent viruses | Full Text | References | PDF (658 KB)
  • 858 Views
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